Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
11/1999
11/25/1999WO1999059570A1 Protease inhibitors
11/25/1999WO1999059526A2 Protease inhibitors
11/25/1999WO1999040068A3 2-aminoquinoline derivatives having d4-agonistic activity
11/25/1999DE3943678C2 New isoquinoline:sulphonamide and naphthalene:sulphonamide cpds.
11/25/1999DE19822245A1 New diphenylpyrrole derivatives useful for control of animal pests, e.g. in protection of plants, goods and materials and in veterinary medicine
11/25/1999CA2332531A1 Protease inhibitors
11/25/1999CA2332522A1 2-(2-methylphenyl)-3,4-dihydro-2h-pyrrol derivatives
11/25/1999CA2332492A1 Protease inhibitors
11/25/1999CA2332352A1 Substituted 6-aryl-3-thioxo-5-(thi)oxo-2,3,4,5-tetrahydro-1,2,4-triazines
11/25/1999CA2332316A1 Tetraisoquinololine derivatives as modulators of dopamine d3 receptors
11/25/1999CA2332239A1 Fused tricyclic compounds which inhibit parp activity
11/25/1999CA2331875A1 Imidazolidine derivatives, the production thereof, their use and pharmaceutical preparations containing the same
11/25/1999CA2329530A1 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole in combination with estrogens
11/24/1999EP0959076A1 Heteroarylperidines and piperazines and their use as antipsychotics and analgetics
11/24/1999EP0959075A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
11/24/1999EP0959073A1 Sulfonamide derivative and process for preparing the same
11/24/1999EP0959072A1 Sulfonamide derivative and process for preparing the same
11/24/1999EP0958293A1 Nanomolar, non-peptide inhibitors of cathepsin d
11/24/1999EP0958292A1 4-(3-heterocyclyl-1-benzoyl)pyrazoles and their use as herbicides
11/24/1999EP0958289A1 Amino acid ester containing azole antifungals
11/24/1999EP0957913A1 N-linked sulfonamides of heterocyclic thioesters
11/24/1999EP0901480A4 Process for preparing oxiranemethanamine derivatives
11/24/1999EP0729461B1 Fungicidal cyclic amides
11/24/1999EP0495091B1 Aica riboside analogs
11/24/1999CN1236366A Amino acid ester containing azole antifungals
11/24/1999CN1236364A Substituted benzocycloheptapyridine derivatives useful for inhibition of Farnesyl protein transferase
11/24/1999CN1235973A Sidechain-bearing taxanes
11/24/1999CN1235969A Intermediates used in preparing dihydrobenzolfuran derivatives
11/24/1999CN1046727C HIV protease inhibitors
11/24/1999CN1046715C Process for making HIV protease inhibitors
11/24/1999CN1046713C Tetrahydroisoquinoline compound, pharmaceutical composition containing them and its producing method and use
11/23/1999US5990319 Synthesis of bisindolylmaleimides
11/23/1999US5990156 Viricides for the influenza virus; neuraminidase inhibitors; also parainfluenza, mumps, newcastle disease virus and sendai virus; myxovirus
11/23/1999US5990142 Antiinflammatory agents and antiallergens having good oral adsorption and bioavailability; cardiotonic and antiischemic agents
11/23/1999US5990135 For treating a retroviral infection such as hiv infection; for example 5s-n-((2-pyridinyl)methoxycarbonyl)valinylamino-2-((n-3 -pyridinyl)methoxycarbonyl)amino-4s-hydroxy-1,6-diphenyl-2-azahexane and other compounds of given formula
11/23/1999US5990133 Indole derivatives as 5-HT receptor antagonist
11/23/1999US5990132 Polycyclic systems, and derivatives thereof, as neurotransmitter release enhancers useful in the treatment of cognitive disorders
11/23/1999US5990128 Administering an antagonist that binds to a human alpha-1c adrenergic receptor with a binding affinity at least 691-fold higher than the binding affinity with which the antagonist binds to a human alpha-1b adrenergic receptor
11/23/1999US5990126 Quinolinic sulfide derivatives acting as NMDA receptor antagonists and process for preparation thereof
11/23/1999US5990093 Treating hepatitis b virus (hbv) infections by administering a 5'-phospholipid prodrug of beta-l-2',3'-dideoxyadenosine 5'-monophosphate of given structure optionally with other anti-hbv agents, such as carbovir or 3tc
11/18/1999WO1999058530A1 Water soluble azoles as broad-spectrum antifungals
11/18/1999WO1999058529A1 Water soluble azoles as broad-spectrum antifungals
11/18/1999WO1999058528A1 Substituted aryl hydroxamic acids as metalloproteinase inhibitors
11/18/1999WO1999058527A2 Benzofuran derivatives, pharmaceutical composition containing the same, and a process for the preparation of the active ingredient
11/18/1999WO1999058526A1 Novel 2,5-pyridinedicarboxylic acid derivatives
11/18/1999WO1999058518A2 Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
11/18/1999WO1999058503A1 Novel 1,5 and 3-o-substituted 1h-indazoles with anti-asthmatic, anti-allergic, anti-inflammatory, immuno-modulating and neuro-protective effect, method for the production and use thereof as medicaments
11/18/1999WO1999058496A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
11/18/1999WO1999058495A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
11/18/1999WO1999058487A1 New compounds, their preparation and use
11/18/1999WO1999058486A1 New compounds, their preparation and use
11/18/1999WO1999058116A2 Novel formulation containing paroxetine
11/18/1999WO1999058113A2 Novel formulation containing paroxetine
11/18/1999DE19821483A1 New imidazolidine derivatives useful as leukocyte adhesion and migration inhibitors and/or VLA-4 receptor antagonists for treating E.G. inflammatory and allergic disorders
11/18/1999DE19821002A1 New indazole derivatives useful as antiasthmatic, antiallergic, neuroprotective agents and for treatment of inflammation and immune disorders
11/18/1999CA2332275A1 Benzofuran derivatives, pharmaceutical composition containing the same, and a process for the preparation of the active ingredient
11/18/1999CA2331871A1 Novel formulation containing paroxetine
11/18/1999CA2331849A1 Novel formulation containing paroxetine
11/18/1999CA2330557A1 Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
11/18/1999CA2330095A1 Substituted aryl hydroxamic acids as metalloproteinase inhibitors
11/17/1999EP0957109A2 Novel processes for preparing intermediates of inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof
11/17/1999EP0957102A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
11/17/1999EP0957101A1 Water soluble azoles as broad-spectrum antifungals
11/17/1999EP0957092A1 Ring-closed dihydropyridines and their use in the preparation of pharmaceutical compositions
11/17/1999EP0956283A1 Substituted phenyltriazolin(thi)ones and their use as herbicides
11/17/1999EP0956021A1 L-$g(b)-DIOXOLANE URIDINE ANALOGS AND METHODS FOR TREATING AND PREVENTING VIRUS INFECTIONS
11/17/1999EP0738273B1 Monohydrate of (e)-2'-deoxy-2'-(fluoromethylene)cytidine
11/17/1999EP0707477B1 Use of efaxoran and its derivatives for the production of drugs for treating neurodegenerative diseases
11/17/1999CN1235603A N-substituted azaheterocyclic compounds
11/17/1999CN1235598A Pyrimidinyloxyalkanoic amide derivatives and fungicides for agricultural and horticultural use
11/17/1999CN1235597A Heterocycle derivatives inhibiting factor Xa
11/17/1999CN1235156A New benzothiophene, benzofuran and indole compounds, process for their preparation and pharmaceutical compounds containing them
11/17/1999CN1046513C Substituted pyrazolyl-pyrozole derivatives, preparation thereof and use as herbicidals
11/17/1999CN1046508C (Tetrahydro-3-furyl) methylamine derivatives, insecticide containing the same and its intermediate
11/17/1999CN1046507C Heterocyclic compounds for treatment of CNS and cardiovasular disorders
11/16/1999US5986103 2-alkyl-1H-imidazole-5-carboxylic acids
11/16/1999US5986101 Reaction product of hindered amine with epoxy group for stabilizers for heat and light
11/16/1999US5986096 Reaction of hydrogen iodide with chloro-5-bromopyrimidine
11/16/1999US5986076 A conjugate is formed by bonding a bioreactive agent to the therapeutic agent with a bond that is selectively cleavable with electromagnetic radiation; useful for controlled release of drugs to treat the disorder
11/16/1999US5985919 Insecticides and fungicides
11/16/1999US5985905 Useful for the treatment and/or prophylaxis of diseases associated with loss of bone mass, such as osteoporosis and related osteopenic diseases, paget's disease, hyperparathyroidism and related diseases, also antitumor
11/16/1999US5985900 Treating tumor growth, invasion or metastasis, osteoarthritis, rheumatoid arthritis, osteoporosis, periodontitis, gingivitis, chronic dermal wounds, corneal ulceration, degenerative skin disorders, multiple sclerosis, stroke, atherosclerosis,
11/16/1999US5985896 Piperidine and morpholine derivatives and their use as therapeutic agents
11/16/1999US5985886 Endothelin receptor antagonists
11/16/1999US5985885 Useful in the treatment of hypertension, congestive heart failure, prostate hypertrophy, various urinary tract disorders and pathological symptoms caused by hyperactivity or disfunctioning of the noradrenergic neural system
11/16/1999US5985879 Compounds useful for inhibition of farnesyl protein transferase
11/16/1999US5985869 Benzoheterocyclic compounds
11/16/1999US5985867 Treating hiv infection
11/16/1999US5985334 Contacting test compound to receptor from rat brain tissue that binds 6-acetyl-4-benzamido-3-hydroxy-2,2-dimethylbenzopyran derivatives
11/16/1999US5985306 (+)-enantiomers of cis-3,4-chroman derivatives useful in prevention or treatment of estrogen diseases or syndromes
11/16/1999CA1340821C Heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components
11/11/1999WO1999057117A2 Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
11/11/1999WO1999057115A1 Novel benzimidazoles and benzoxazoles
11/11/1999WO1999057114A1 Heterocyclic carboxamide derivatives as inhibitors of nitric oxide production
11/11/1999WO1999057113A1 Heterocyclic derivatives which inhibit factor xa
11/11/1999WO1999057101A1 Pyrazole derivatives as p-38 map kinase inhibitors
11/11/1999WO1999056765A1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME
11/11/1999WO1999042457A3 Substituted alxoxycarbonyl compounds
11/11/1999WO1998004528A3 Substituted pyridines and biphenyls as anti-hypercholesterinemic, anti-hyperlipoproteinemic and anti-hyperglycemic agents
11/11/1999DE19838506A1 Indolderivate und deren Verwendung zur Behandlung von malignen und anderen, auf pathologischen Zellproliferationen beruhenden Erkrankungen The indole derivatives and their use for the treatment of malignant and other diseases based on pathological cell proliferations