Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
02/2000
02/03/2000WO2000005222A1 Dihydrotriazolone derivatives as pesticides
02/03/2000WO2000005219A1 Phthalazine derivatives as phosphodiesterase 4 inhibitors
02/03/2000WO2000005218A1 Phthalazine derivatives phosphodiesterase 4 inhibitors
02/03/2000WO2000005217A1 Imidazole compounds and their use as adenosine deaminase inhibitors
02/03/2000WO2000005214A2 Isoquinolines as urokinase inhibitors
02/03/2000WO2000005208A1 Amino-aldehyde solid support, linker therefor and methods of preparation and use thereof
02/03/2000WO2000005204A1 MONOCYCLIC β-LACTAM COMPOUNDS AND CHYMASE INHIBITORS CONTAINING THE SAME
02/03/2000WO2000005198A1 Anthranilic acid derivatives
02/03/2000WO2000004900A1 Substituted benzimidazole antiviral agents
02/03/2000WO2000004893A2 Imidazoline receptor binding compounds
02/03/2000WO2000004892A2 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
02/03/2000WO1999063929A3 Multibinding inhibitors of microsomal triglyceride transferase protein
02/03/2000DE19834751A1 Disubstituierte bicyclische Heterocyclen, ihre Herstellung und ihre Verwendung als Arzneimittel Disubstituted bicyclic heterocycles, their preparation and their use as medicaments
02/03/2000CA2338305A1 Imidazole compounds
02/03/2000CA2338279A1 Imidazoline receptor binding compounds
02/03/2000CA2338147A1 Substituted benzimidazole antiviral agents
02/03/2000CA2338044A1 Phthalazine derivatives phosphodiesterase 4 inhibitors
02/03/2000CA2337954A1 Phthalazine derivatives as phosphodiesterase 4 inhibitors
02/03/2000CA2337247A1 Isquinolines as urokinase inhibitors
02/03/2000CA2335062A1 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
02/03/2000CA2332589A1 Dihydrotriazolone derivatives as pesticides
02/02/2000EP0976747A2 Use of 5HT-1F receptor antagonists for treating anxiety disorders
02/02/2000EP0976746A1 5-HT1F antagonists
02/02/2000EP0976745A1 4-tetrahydropyridylpyrimidine derivatives
02/02/2000EP0976737A1 Pyrazole derivatives, process for preparing the same, intermediates, and pest control agent containing the same as active ingredient
02/02/2000EP0976735A1 Process for producing piperidinecarboxylic acid amides
02/02/2000EP0976734A2 Selective inhibitors of viral or bacterial neuraminidase
02/02/2000EP0976732A1 1,4-substituted cyclic amine derivatives
02/02/2000EP0975624A1 Thermogenic composition and benzazepine thermogenics
02/02/2000EP0975621A1 Cell differentiation inducing amide derivatives, their production and use
02/02/2000EP0975614A1 A bicyclic aryl or a bicyclic heterocyclic ring containing compounds having a combined 5ht1a, 5ht1b and 5ht1d receptor antagonistic activity
02/02/2000EP0975600A1 Heterocyclic derivatives and their use as antithrombotic agents
02/02/2000EP0975593A1 Indole derivatives having combined 5ht1a, 5ht1b and 5ht1d receptor antagonist activity
02/02/2000CN1243513A Quinoline and quinozoline compounds useful in therapy, particularly in the theatment of begnin prostatic hyperplasia
02/02/2000CN1243126A Method for preparing asymmetric lactone
02/02/2000CN1048982C Method for semi-synthesis of taxalkane derivative with metal alkane oxide and beta-lactum
02/01/2000US6020519 Diphenyl-cyclopropenes as selective K-agonists
02/01/2000US6020488 Small molecule inhibition of RNA/ligand binding
02/01/2000US6020366 Butyric acid matrix metalloproteinase inhibitors
02/01/2000US6020362 Glycoprotein IIB IIIA antagonists
02/01/2000US6020348 Endothelin receptor antagonists
02/01/2000US6020345 Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine
02/01/2000US6020343 (Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitors
02/01/2000US6020339 Aryl furan derivatives as PDE IV inhibitors
02/01/2000US6020336 Indole and indazole compounds
02/01/2000US6020334 Piperazinones, their production and use
02/01/2000CA2093798C Pyridine and pyridine n-oxide derivatives of diaryl methyl piperidines or piperazines, and compositions and methods of use thereof
02/01/2000CA2012514C Stabilizers derived from n-hydroxy hindered amines by michael addition reactions
01/2000
01/27/2000WO2000004015A1 1-4-dihydropyridines with benzodioxo carbonyl group as calcium blockers
01/27/2000WO2000004011A1 Cyclic compounds useful in the treatment of dyslipidaemia, atherosclerosis and diabetes, pharmaceutical compositions and preparation process
01/27/2000WO2000004000A1 Piperazinone derivatives and their uses
01/27/2000WO2000003990A1 Pharmaceutical compositions comprising 2-quinolones
01/27/2000WO2000003986A1 Bispiperidines as antithrombotic agents
01/27/2000WO2000003697A1 Pellets having a core coated with an antifungal and a polymer
01/27/2000WO2000003681A2 Process for the synthesis of benzopyran derivatives
01/27/2000WO1999061599A3 Recombinant narbonolide polyketide synthase
01/27/2000WO1999058527A3 Benzofuran derivatives, pharmaceutical composition containing the same, and a process for the preparation of the active ingredient
01/27/2000DE19918588A1 Piperidinverbindung Piperidine
01/27/2000CA2337776A1 Bispiperidines as antithrombotic agents
01/27/2000CA2337481A1 Cyclic compounds useful in the treatment of dyslipidaemia, atherosclerosis and diabetes, pharmaceutical compositions and preparation process
01/27/2000CA2337115A1 Pharmaceutical compositions comprising 2-quinolones
01/26/2000EP0974590A1 Process for the preparation of chiral lactones by asymetrical hydrogenation
01/26/2000EP0974584A1 Fused ring compounds, process for producing the same and use thereof
01/26/2000EP0974583A1 Phenylpiperidine derivatives
01/26/2000EP0973778A1 4,5,6,7-TETRAHYDRO-THIENO 3,2-c]PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE
01/26/2000EP0973768A1 Azole compounds, their production and their use
01/26/2000EP0973767A1 Indazoles of cyclic ureas useful as hiv protease inhibitors
01/26/2000EP0973765A1 Substituted aryluracils
01/26/2000EP0973763A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same
01/26/2000EP0973761A1 RED COLOURING HYPERCHROMIC 3$i(H)-NAPHTHO 2,1-$i(b)]PYRANS
01/26/2000EP0973753A2 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinones useful as hiv reverse transcriptase inhibitors
01/26/2000EP0973752A1 Heterocyclically substituted aromatic amino compounds with a herbicidal effect
01/26/2000EP0973751A1 Phenyl-amino-sulfonyl-urea derivatives as fungicides and pesticides
01/26/2000EP0973750A1 Substituted benzimidazoles and their use for treating retroviral infection
01/26/2000EP0973748A1 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses
01/26/2000EP0973747A1 Pesticidal 1-arylpyrazoles
01/26/2000EP0973705A1 Chromatographic enantiomer separation of lactones
01/26/2000EP0973392A1 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
01/26/2000EP0650484B1 Endothelin receptor antagonists
01/26/2000CN1242772A Pyridin-2-yl-methylamine derivatives, method of preparing and application as medicine
01/26/2000CN1242770A Cyclic ketone derivative and pharmaceutical use thereof
01/26/2000CN1242367A Spiro [Piperidine-4,1'-pyrrolo[3,4-c] pyrrole]
01/26/2000CN1048725C Nicotinic acid derivatives and herbicide
01/25/2000US6018073 Tricyclic taxanes having an alkoxy, alkenoxy or aryloxy substituted side-chain and pharmaceutical compositions containing them
01/25/2000US6018054 Intermediate compounds for preparing novel quinolone and naphthyridone derivatives which are substituted in the 7-position by a partially hydrogenated isoindolinyl ring, use as antibacterial agents and as feed additives
01/25/2000US6018052 Fungicidal optically active 1-(mono-or substituted amino)-2-substituted-4,4-disubstituted-2-imidazolin-5-ones and 5- thiones corresponding
01/25/2000US6017956 N,N-disubstituted amic acid derivatives
01/25/2000US6017954 Angiogenesis inhibitors for treating and preventing angiogenesis-dependent tumors, especially kaposi's sarcoma, breast cancer, colon cancer
01/25/2000US6017952 Endothelin receptor antagonists
01/25/2000US6017951 Butenolide endothelin antagonists
01/25/2000US6017945 Useful in the treatment of restenosis, renal failure and pulmonary hypertension
01/25/2000US6017941 Method of combatting infectious diseases using dicationic bis-benzimidazoles
01/25/2000US6017935 7-sulfur substituted paclitaxels
01/25/2000US6017916 Nonpeptide endothelin antagonists I
01/25/2000US6017915 Heterocyclic compounds
01/20/2000WO2000002877A2 New pharmaceutically active compounds
01/20/2000WO2000002867A1 Substituted acylamino phenyl uracils
01/20/2000WO2000002865A1 Pharmaceutical agents
01/20/2000WO2000002860A1 2-aminopyridine erivatives, their use as medicines and pharmaceutical compositions containing them
01/20/2000WO2000002836A1 Method for preparing 2-disubstituted 2,3-dihydrobenzofuran derivatives