Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
06/1999
06/10/1999WO1999028297A1 Substituted indoles, having a thrombin inhibiting effect
06/10/1999DE19753522A1 Substituierte Indole, ihre Herstellung und ihre Verwendung als Arzneimittel Substituted indoles, their preparation and their use as medicaments
06/10/1999CA2312770A1 Alicyclic acylated heterocyclic derivatives
06/10/1999CA2312338A1 Process of preparing substituted pyrimidinones
06/10/1999CA2312334A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
06/10/1999CA2310629A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof
06/09/1999EP0921120A1 Selective beta 3 adrenergic agonists
06/09/1999EP0921119A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them
06/09/1999EP0920456A1 Phosgenated oxime resins and their preparation
06/09/1999EP0920427A1 Process for the preparation of benzopyran compounds
06/09/1999EP0920425A1 Substituted 4-(1h-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases
06/09/1999EP0920424A1 Non-peptide bombesin receptor antagonists
06/09/1999EP0920419A1 Compounds, compositions and methods for treating influenza
06/09/1999EP0920416A1 Naphtholactams and lactones as bone morphogenetic protein active agents
06/09/1999EP0920415A1 Substituted 2-phenylpyridine as herbicide
06/09/1999EP0920312A1 Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents
06/09/1999CN1219172A Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
06/09/1999CN1219171A Benzofuran carboxamides and their therapeutic use
06/09/1999CN1218801A Tri-substituted imidazoles, and process of their preparation and using the same and having their pharmic composition
06/03/1999WO1999026943A1 Thrombin receptor antagonists
06/03/1999WO1999026941A1 Substituted amidinoaryl derivatives and their use as anticoagulants
06/03/1999WO1999026935A1 Trisaryl-1,3,5-triazine ultraviolet light absorbers
06/03/1999WO1999026932A1 By amidino group substituted heterocyclic derivatives and their use as anticoagulants
06/03/1999WO1999026931A1 Pyrazolylpyrazoles substituted by 1-methyl-5- alkylsulphonyl, 1-methyl-5- alkylsuphinyl and 1-methyl-5- alkylthio, methods for preparing them and use as herbicides
06/03/1999WO1999026930A2 Benzylidene pyrazolones and use as herbicide
06/03/1999WO1999026921A1 SUBSTITUTED β-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS
06/03/1999WO1999005096A3 Urokinase inhibitors
06/03/1999CA2311538A1 Trisaryl-1,3,5-triazine ultraviolet light absorbers
06/03/1999CA2310087A1 Benzylidene pyrazolones and use as herbicide
06/03/1999CA2309341A1 Substituted .beta.-alanine derivatives as cell adhesion inhibitors
06/03/1999CA2309210A1 1-methyl-5-alkylsulfonyl-, 1-methyl-5-alkylsulfinyl- and 1-methyl-5-alkylthiosubstituted pyrazolylpyrazoles, processes for their preparation and their use as herbicides
06/02/1999EP0918768A1 Aromatic amidine derivatives useful as selective thrombin inhibitors
06/02/1999EP0918767A1 Pharmaceutical for treating of neurological and neuropsychiatric disorders
06/02/1999EP0918752A2 Dna-binding indole derivatives, their prodrugs and immunoconjugates as anticancer agents
06/02/1999EP0739341B1 Herbicidal aryl and heteroaryl pyrimidines
06/02/1999EP0581939B1 N-sulphonyl-2-oxoindole derivatives having affinity for vasopressin and/or ocytocin receptors
06/02/1999CN1218467A Sulphur derivatives comprising amide bond, method for preparing same, use thereof as drugs, and pharmaceutical compositions containing such derivatives
06/02/1999CN1218466A 2,4-diaminopyrimidine derivatives as dopamine d4 receptor antagonists
06/02/1999CN1218465A 2,4-diaminopyrimidine derivatives
06/02/1999CN1218464A 2,3 disulbstituted-4 (3H)-quinazolinones
06/02/1999CN1218463A Asymmetric synthesis of R-'alpha'-propyl-piperonyl amine and its analogs
06/02/1999CN1218462A Crystalline (-)-3R, 4R-trans-7-methoxy-2,2-dimetnyl-3-phenyl-4-{4-[2-(pyrrolidin-1-yl) ethoxy] phenyl} chromane, hydrogen fumarate
06/02/1999CN1218460A Substituted 4-hydroxy-phenylalcanoic acid derivatives with activity to ppar-'gamma'
06/02/1999CN1218457A Triazolyl disulphides
06/02/1999CN1218052A New indole and indazole compounds, process for their preparation and pharmaceutical compositions containing them
06/02/1999CN1218051A New 2,3-dioxide, indanol compounds, process for their preparation and pharmaceutical compositions containing them
06/02/1999CN1218050A Sulfonamide-substituted benzopyran derivates processes for their preparation, their use as medicament, and pharmaceutical preparations comprising them
06/02/1999CN1218047A Novel imidazolidine derivatives, their preparation, their use and pharmaceutical preparations comprising them
06/01/1999US5908934 Chemical intermediate for kinase inhibitors
06/01/1999US5908860 4-carbonylamino-substituted-2,2-dimethyl-3,4-dihydrobenzopyran -3-ols
06/01/1999CA2065699C Dry analytical element for lithium assay
06/01/1999CA1340574C Method and compositions providing enhanced chemiluminescence from 1,2-dioxetanes
06/01/1999CA1340567C Heterocyclic amide derivatives
05/1999
05/27/1999WO1999025715A1 Preparation of terazosin hydrochloride dihydrate
05/27/1999WO1999025714A1 Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance p antagonists
05/27/1999WO1999025713A1 2-methoxyimino-2-phenyl acetamides containing a ketal- or dialkoxy substituted pyridine moiety, their preparation and their use as fungicides
05/27/1999WO1999025700A1 Triazole derivatives, intermediates for the production thereof, processes for producing the both, and herbicides containing the derivatives as the active ingredient
05/27/1999WO1999025688A1 Process for the preparation of 1,4-dihydropyridines and compounds used in this process
05/27/1999WO1999025687A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
05/27/1999WO1999025686A1 Cyclic amine derivatives and their use as drugs
05/27/1999WO1999025684A1 Method of synthesis of pyrrole amides
05/27/1999WO1999018099B1 Aryl thiophene derivatives as pde iv inhibitors
05/27/1999DE19751943A1 New pyrazolyl-pyrazole derivatives are pre- and post-emergent herbicides
05/27/1999CA2310095A1 Method of synthesis of pyrrole amides
05/27/1999CA2309829A1 Preparation of terazosin hydrochloride dihydrate
05/27/1999CA2306460A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
05/26/1999EP0918059A1 Substituted imidazoline derivatives, their preparation, their use, and pharmaceutical compositions containing them
05/26/1999EP0917462A1 Cell adhesion inhibitors
05/26/1999EP0823907B1 PROCESS FOR PREPARING (-)-TRANS-N-p-FLUOROBENZOYLMETHYL-4-(p-FLUOROPHENYL)-3-[[3,4-(METHYLENEDIOXY)PHENOXY]METHYL]-PIPERIDINE
05/26/1999EP0817769B1 Borneol esters, process for their preparation and their pharmaceutical use
05/26/1999EP0777663B1 Use of substituted 6-amino-4h-pyrans
05/26/1999EP0752991B1 IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZIN-4-ONES ANTAGONISTS OF AMPA AND NMDA RECEPTORS
05/26/1999EP0686625B1 Anthranilic acid derivative
05/26/1999CN1217719A Novel benzofuranone derivative and process for producing same
05/26/1999CN1217717A Acyl mercapto-triazolyl derivative and use thereof as microbiocides
05/26/1999CN1217335A Method for preparing precursor medicine
05/26/1999CN1217327A D-proline derivative
05/25/1999US5907041 Process for preparing pyrazole derivatives
05/25/1999US5907038 Azepanes
05/20/1999WO1999024870A2 Compound, composition and use
05/20/1999WO1999024460A2 Dipeptide nitriles
05/20/1999WO1999024426A1 N-hydroxyurea derivative and medicine containing the same
05/20/1999WO1999024420A1 Pyrimidinone compounds and pharmaceutical compositions containing them
05/20/1999WO1999024406A1 Phenyl-alkyl-imidazoles as h3 receptor antagonists
05/20/1999WO1999024404A1 Substituted pyridine compounds as anti-inflammatory agents
05/20/1999WO1999024399A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
05/20/1999WO1999024398A2 Urea derivatives and their use as integrin inhibitors
05/20/1999DE19751200A1 New epothilone derivatives
05/20/1999CA2309823A1 Compound, composition and use
05/20/1999CA2309177A1 Pyrimidinone compounds and pharmaceutical compositions containing them
05/20/1999CA2309121A1 Phenyl-alkyl-imidazoles as h3 receptor antagonists
05/20/1999CA2308716A1 Urea derivatives and their use as integrin inhibitors
05/20/1999CA2308359A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
05/19/1999EP0916668A1 Chemokine receptor antagonists
05/19/1999EP0915935A1 4,7-dichlororhodamine dyes
05/19/1999EP0915873A1 Substituted pyrazolyl-pyrazole derivatives, process for their preparation and their use as agents with a herbicidal effect
05/19/1999EP0915869A1 Novel tricyclic n-cyanoimines useful as inhibitors of farnesyl-protein transferase
05/19/1999EP0915855A1 Novel compounds with analgesic effect
05/19/1999EP0915853A1 Substituted 3-phenyl pyrazoles
05/19/1999EP0915848A1 1,2-diarylindole as cox-2 inhibitors