Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
06/1999
06/30/1999EP0925289A1 Matrix metalloproteinase inhibitors
06/30/1999EP0925287A1 Heterocyclic metalloprotease inhibitors
06/30/1999EP0699198B1 N-benzoylmethyl substituted paroxetine derivatives
06/30/1999CN1221408A Substituted pyrazolyl-pyrazole derivatives and their use as herbicides
06/30/1999CN1221407A Aminoisoquinolines and aminothienopyridine derivatives and their use as anti-inflammatory agents
06/30/1999CN1220991A Tetrahydro-3-furanyl methylamine
06/30/1999CN1043888C Fungicidal and herbicidal triazoles
06/30/1999CN1043887C Chemopreventive compound and preparation method and use thereof
06/30/1999CN1043886C Substituted pyrimidine, there process of preparation and use as sectivide and fungicide thereof
06/30/1999CN1043884C New substituted azacylobutanone, preparation method and medicinal use thereof
06/29/1999US5917047 Heterocyclic compounds
06/29/1999US5917046 Method for producing 2-naphthamide derivative, and compounds for producing 2-naphthamide derivative
06/29/1999US5917042 Process for the preparation of 2,5-diamino-4,6-dichloropyrimidine
06/29/1999US5917041 Amination and cyclization reaction with amine to make2-aminopurine nucleosides
06/29/1999US5917034 Antithrombotic n-amidinopiperidine and benzamidine derivatives
06/29/1999US5916908 Pharmaceutical pyrazole compositions useful as inhibitors of protein kinases
06/29/1999US5916901 Heterocyclic compounds
06/29/1999US5916889 1,4-disubstituted piperazines
06/24/1999WO1999031090A1 Dihydrobenzofurans
06/24/1999WO1999031088A1 Triazine angiogenesis inhibitors
06/24/1999WO1999031081A1 Ph sensitive photochromic dyes
06/24/1999WO1999031075A1 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031074A2 ((cyclo)alkyl substituted)-.gamma.-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031073A1 Novel pyrimidine-5-carboxamide derivatives
06/24/1999WO1999031070A1 Substituted phenylpyrazolones, method and intermediate products for the production thereof, and their utilization for combating parasitic fungi and animal parasites
06/24/1999WO1999031068A1 Substituted isoquinoline derivatives and their use as anticonvulsants
06/24/1999WO1999031066A1 Pyridones as src family sh2 domain inhibitors
06/24/1999WO1999031064A1 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic and immunosuppressive agents
06/24/1999WO1999031063A1 New piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides
06/24/1999WO1999031060A2 Piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides as cytostatics and immunesuppressants
06/24/1999WO1999031057A1 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031037A1 Apoptosis inhibitors
06/24/1999WO1999030696A1 A method for the prevention and treatment of stunned myocardium
06/24/1999DE19756115A1 Substituierte Phenylpyrazolone, Verfahren und Zwischenprodukte zu ihrer Herstellung und ihre Verwendung zur Bekämpfung von Schadpilzen und tierischen Schädlingen Substituted phenylpyrazolones, processes and intermediates for their preparation and their use for controlling harmful fungi and animal pests
06/24/1999CA2315079A1 Substituted isoquinoline derivatives and their use as anticonvulsants
06/24/1999CA2314954A1 Apoptosis inhibitors
06/24/1999CA2314111A1 Dihydrobenzofurans
06/24/1999CA2313776A1 Triazine angiogenesis inhibitors
06/24/1999CA2311932A1 A method for the prevention and treatment of stunned myocardium
06/23/1999EP0924209A1 Hypoglycemic imidazoline compounds
06/23/1999EP0924202A1 Imidazole derivative and medicine comprising the same as active ingredient
06/23/1999EP0924201A1 Tricyclic-substituted pyrazolyl benzenesulfonamides and their use as cyclooxygenase II inhibitors
06/23/1999EP0923933A1 Substituted pyrazolyl benzenesulfonamides for use in the treatment of inflammation
06/23/1999EP0923575A1 Cyclic ether compounds as sodium channel modulators
06/23/1999EP0923570A1 Pyridyl alkene- and pyridyl alkine- acid amides as cytostatics and immunosuppressives
06/23/1999EP0923569A1 Butyric acid matrix metalloproteinase inhibitors
06/23/1999EP0923568A1 Novel benzofuran-4-carboxamides
06/23/1999EP0923563A1 1,4-heterocyclic metallprotease inhibitors
06/23/1999EP0923558A1 Substituted 1-(3-pyrazolyl)-pyrazoles
06/23/1999EP0923557A1 Stereoselective deoxygenation reaction
06/23/1999EP0923556A1 An asymmetric conjugate addition reaction
06/23/1999EP0923555A1 Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders
06/23/1999EP0923554A1 N-benzylpiperidine and tetrahydropyridine derivatives
06/23/1999EP0671915B1 Use of idazoxan and derivatives thereof in preparing a drug for treating parkinson's disease and its development
06/23/1999CN1220664A Process for producing phenoxy propionic acid derivatives
06/23/1999CN1220265A New piperazine and piperidine compounds
06/22/1999US5914406 Azepanes and their ring homologues having protein kinase inhibiting activity
06/22/1999US5914400 Method and compositions for the synthesis of BCH-189 and related compounds
06/22/1999US5914342 2-imidazolinylamino heterocyclic compounds useful as alpha-2 adrenoceptor agonists
06/22/1999US5914332 Retroviral protease inhibiting compounds
06/22/1999US5914331 Antiviral activity and resolution of 2-hydroxymethyl-5-(5-fluorocytosin-1-yl)-1,3-oxathiolane
06/22/1999US5914263 Enzymatic process for the stereoselective preparation of a hetero-bicyclic alcohol enantiomer
06/22/1999CA2151674C Methods of administering crf antagonists
06/22/1999CA2147893C Enantiomerically pure .beta.-d-dioxolane nucleosides with selective anti-hepatitis .beta. virus activity
06/21/1999EP0954522A4 Novel substituted naphthopyrans
06/17/1999WO1999029687A1 (benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
06/17/1999WO1999029685A1 (e)-3-[1-n-butyl- 5-[2-(2-carboxyphenyl)methoxy- 4-chlorophenyl]-1h- pyrazol-4-yl]-2-[(5- methoxy-2,3- dihydrobenzofuran-6-yl)methyl]- prop-2-enoic acid monoargininyl salt
06/17/1999WO1999029677A1 Substituted 2,4-diamino-1,3,5-triazines
06/17/1999WO1999029674A1 Retinoic acid mimetic anilides
06/17/1999WO1999029673A1 SELECTIVE β3 ADRENERGIC AGONISTS
06/17/1999WO1999029667A1 Hydroxamic acid derivatives as matrix metalloprotease (mmp) inhibitors
06/17/1999DE19755016A1 Substituierte 2,4-Diamino-1,3,5-triazine Substituted 2,4-diamino-1,3,5-triazines
06/17/1999CA2314334A1 Substituted 2,4-diamino-1,3,5-triazines
06/17/1999CA2312987A1 Selective .beta.3 adrenergic agonists
06/17/1999CA2312965A1 (e)-3-¬1-n-butyl-5-¬2-(2-carboxyphenyl)methoxy-4-chlorophenyl|-1h-pyrazol-4-yl|-2-¬(5-methoxy-2,3-dihydrobenzofuran-6-yl)methyl|-prop-2-enoic acid monoargininyl salt
06/17/1999CA2312720A1 Retinoic acid mimetic anilides
06/16/1999EP0922703A1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds
06/16/1999EP0922697A1 Substituted Pyrazolyl benzenesulfonamides and their use as cyclooxygenase II inhibitors
06/16/1999EP0922043A1 Pesticidal 3-(substituted phenyl)-5-(thienyl or furyl)-1,2,4-triazoles
06/16/1999EP0922036A1 Arylalkanoyl pyridazines
06/16/1999EP0922035A1 Tetrahydroisoquinoline derivatives and their pharmaceutical use
06/16/1999EP0922029A1 Ether muscarinic antagonists
06/16/1999EP0922028A1 Inhibitors of phospholipase enzymes
06/16/1999EP0753003B1 Aziridine derivatives, their production and use
06/16/1999EP0752424B1 Nicotinic acid derivative and herbicide
06/16/1999CN1219932A Aromatic amidine derivatives useful as selective thrombin inhibitors
06/16/1999CN1219841A DNA-binding indole derivatives, their prodrugs and immunoconjugates as anticancer agents
06/16/1999CA2255337A1 Imidazole derivative and medicine comprising the same as active ingredient
06/15/1999US5912357 Enzyme inhibitors
06/15/1999US5912342 Synthesis of combinatorial libraries by computer controlled robot
06/15/1999US5912264 Taxane derivatives as antitumor agents
06/15/1999US5912262 Heterocyclic compounds
06/15/1999US5912247 Quinazoline compound and anti-tumor agent containing said compound as an active ingredient
06/15/1999US5912244 Muscle disorders, breathing disorders and urinary incontinence
06/15/1999CA2164949C Photochromic naphthopyran compounds
06/15/1999CA2155664C Oxindole 1-[n-(alkoxycarbonyl)]carboxamides and 1-(n-carboxamido)carboxamides as antiinflammatory agents
06/10/1999WO1999028315A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof
06/10/1999WO1999028307A1 Alicyclic acylated heterocyclic derivatives
06/10/1999WO1999028303A1 Process of preparing substituted pyrimidinones
06/10/1999WO1999028300A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors