Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
09/1999
09/08/1999CN1228082A Synthesis of bisindolylmalimides
09/07/1999US5948914 Preparing 4-(4-fluorophenyl)-3-hydroxymethylpiperidine by optically resolving with o-chlorotartranilic acid; chemical intermediate for drugs
09/07/1999US5948907 Synthesis of bisindolylmaleimides
09/07/1999US5948813 Method of preventing allograft rejection
09/07/1999US5948806 Treatment of Parkinson's disease with (+)2-(ethyl-2,3-dihydrobenzofuranyl)-2-Imidazoline (dexefaroxan or (+) efaroxan)
09/07/1999US5948794 Enterokinetic benzamide
09/07/1999US5948792 Fluorine-containing 1,4-disubstituted piperidine derivatives
09/07/1999US5948791 Quinoline derivatives for treating malaria
09/07/1999US5948786 Blocking tumor necrosis factor
09/07/1999US5948782 Antiinflammatory agent; rheumatic diseases
09/07/1999US5948624 Methods for the detection and isolation of biomolecules
09/07/1999US5948600 Method and material for the formation of a heat mode image
09/07/1999CA2168563C Benzopyrans and pharmaceutical compositions containing them
09/07/1999CA2098944C Novel pyrazole derivatives, method of preparing them and pharmaceutical compositions in which they are present
09/07/1999CA2016646C Arylsulphonamides
09/07/1999CA2014008C Benzimidazoles, medicaments containing these compounds and processes for their preparation
09/02/1999WO1999043691A1 2'-fluoronucleosides
09/02/1999WO1999043672A1 Inhibitors of phospholipase a2
09/02/1999WO1999043663A1 N-[(substituted five-membered di- or triaza diunsaturated ring)carbonyl] guanidine derivatives for the treatment of ischemia
09/02/1999WO1999043661A2 Substituted cycloalkyl-4-oxonicotinic carboxamides; gaba brain receptor ligands
09/02/1999WO1999043658A1 Heterocyclic substituted aniline calcium channel blockers
09/02/1999WO1999043657A1 2-arylethyl-(piperidin-4-ylmethyl)amine derivatives as muscarinic receptor antagonists
09/02/1999WO1999043654A2 Inhibitors of phospholipase enzymes
09/02/1999WO1999043651A2 Inhibitors of phospholipase enzymes
09/02/1999WO1999043649A1 Arylphenyl-substituted cyclic keto-enols
09/02/1999WO1999024460A3 Dipeptide nitriles
09/02/1999CA2322167A1 Substituted cycloalkyl-4-oxonicotinic carboxamides; gaba brain receptor ligands
09/02/1999CA2322163A1 Inhibitors of phospholipase a2
09/02/1999CA2322162A1 Inhibitors of phospholipase enzymes
09/02/1999CA2322161A1 Inhibitors of phospholipase enzymes
09/02/1999CA2321642A1 N-¬(substituted five-membered di- or triaza diunsaturated ring)carbonyl|guanidine derivatives for the treatment of ischemia
09/01/1999EP0939135A1 Substantially pure hetero-bicyclic alcohol enantiomers
09/01/1999EP0938487A2 2$i(R),4$i(S),$i(R),$i(S)- AND 2$i(S),4$i(R),$i(R),$i(S)-HYDROXYITRACONAZOLE- AND HYDROXYSAPERCONAZOLE DERIVATIVES
09/01/1999EP0938484A1 2r,4s,r,r- and 2s,4r,r,r-hydroxyitraconazole
09/01/1999EP0938483A2 Muscarinic antagonists
09/01/1999EP0938482A1 5-substituted and 5,5-disubstituted-3,4-dihydroxy-2(5h)-furanones and methods of use therefor
09/01/1999EP0938479A1 Quaternary nitrogen heterocycles, method for their production and their use as pesticides
09/01/1999EP0938478A1 Quaternary nitrogen heterocycles, method for their production and their use as pesticides
09/01/1999EP0938476A1 Process for substituted pyridines
09/01/1999EP0938474A2 Cyclopropylindole compounds and their use as prodrugs
09/01/1999EP0938471A1 The preparation and use of ortho-sulfonamido aryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
09/01/1999EP0938311A2 Use of efaroxan for producing medicine for treating huntington disease
09/01/1999CN1227547A Arylalkanoyl pyridazines
09/01/1999CN1227546A Substituted 1-(3-pyrazolyl)-pyrazoles with herbicide activity and intermediate for its preparation
09/01/1999CN1227545A 3-cyanoaryl pyrazoles and use thereof as herbicides
09/01/1999CN1227099A Novel treatment agent
09/01/1999CN1044911C Method for preparing prodrug
08/1999
08/31/1999US5945430 Benzo(5,6)cycloheptapyridine compounds that inhibit ras function, use for treating tumor cells expressing an activated ras oncogene in mammals
08/31/1999US5945423 For agriculture
08/31/1999US5945418 Administering to the mammal to inhibit a mammalian protein kinase p38 which causes cell proliferation, cell death and response to extracellular stimuli
08/31/1999US5945413 Treating human immunodeficiency virus infections
08/31/1999CA2165318C 4-amino-2-quinolinone derivatives
08/27/1999CA2242794A1 2,4-bis[(4-aminidino)phenyl]furans as anti-pneumocystis carini agents
08/26/1999WO1999042463A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
08/26/1999WO1999042461A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
08/26/1999WO1999042458A1 Histamine h3 receptor ligands
08/26/1999WO1999042457A2 Substituted alxoxycarbonyl compounds
08/26/1999WO1999042453A1 5-substituted pyrimidine-2-yloxy carboxylic acid derivatives, the production of the same and their utilization as endothelin antagonists
08/26/1999WO1999042450A1 Solid phase synthesis of 1-aminohydantoins
08/26/1999WO1999042442A1 Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof
08/26/1999WO1999042100A1 Cell death inhibitors
08/26/1999WO1999033825A8 N-phenylamide and n-pyridylamide derivatives, method of preparing them and pharmaceutical compositons containing them
08/26/1999WO1999031060A3 Piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides as cytostatics and immunesuppressants
08/26/1999DE19844192A1 New substituted alkoxycarbonyl compounds
08/26/1999CA2321460A1 Substituted alxoxycarbonyl compounds
08/26/1999CA2321182A1 5-substituted pyrimidine-2-yloxy carboxylic acid derivatives, the production of the same and their utilization as endothelin antagonists
08/26/1999CA2321085A1 Solid phase synthesis of 1-aminohydantoins
08/26/1999CA2318836A1 Histamine h3 receptor ligands
08/26/1999CA2316944A1 Aminoguanidinehydrazone derivative, production and use thereof
08/25/1999EP0937722A1 Benzimidazole derivatives as cyclooxygenase-2 inhibitors
08/25/1999EP0937458A2 Pyrrolidine and piperidine derivatives
08/25/1999EP0937152A2 Screening for and use of an esterase for a stereospecific resolution
08/25/1999EP0937071A1 2r,4s,s,s- and 2s,4r,s,s-hydroxyitraconazole
08/25/1999EP0937070A1 Benzoheterocyclic distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agents
08/25/1999EP0937064A1 Substituted oximes derivatives useful as neurokinin antagonists
08/25/1999EP0937048A1 HETEROCYCLE DERIVATIVES WHICH INHIBIT FACTOR Xa
08/25/1999EP0937046A2 Substituted 3-benzylpyrazoles and their use as herbicides and for lowering the sugar content in blood
08/25/1999EP0937042A1 Heteroaryl succinamides and their use as metalloproteinase inhibitors
08/25/1999EP0936912A1 Inhibitors of cysteine protease
08/25/1999EP0805626B1 Crop protection products
08/25/1999CN1226895A Amino acid derivatives and their use as thrombin inhibitors
08/25/1999CN1226888A Fluorinated 1,4-disubstituted piperidine derivatives
08/25/1999CN1044809C Herbicidal aryl and heteroaryl pyrimidines
08/24/1999US5942622 Novel compounds for treating illness resulting from abnormal stimulation of endothelial receptors; for example: 4-((6-chloro-1,3-benzodioxol-5-yl)methyl)-1-(cyclohexylmethyl) -3-(2-pyridinyl)-1h-pyrazole-5-carboxylate
08/24/1999US5942619 Quinoline-4-one derivatives with optional alkyl groups at positions 1 and 3, 2-substituted with a branched unsaturated alkyl optionally substituted with hydroxyl or ether; treating ulcers; biosynthesis
08/24/1999US5942547 2-Deoxystreptamine derivatives, pharmaceutical compositions thereof and therapeutic methods using same
08/24/1999US5942536 Useful for treating migraine
08/24/1999US5942532 Inhibitors of histidine protein kinase; bacteria resistant to other antibiotics
08/24/1999US5942522 1-benzyl-3-ethoxycarbonyl-4-dimethylaminoethoxy-6-methyl-2-(1h) -quinolinone; antiviral against dna containing viruses, such as herpes group viruses
08/24/1999US5942517 Antagonist of alpha(1c) receptors; treatment of benign prostatic hyperplasia
08/24/1999US5942516 Endothelin receptor antagonists
08/24/1999US5942509 2-(triazinyloxy(or thio)phenyl)-substituted methyl 3-methoxy-2-propenoate
08/24/1999US5942506 1- 2-(substituted vinyl)!-5H-2,3-benzodiazepine derivatives
08/24/1999CA2176974C Phenyl heterocycles as cyclooxygenase-2 inhibitors
08/24/1999CA2141969C Cardio-protective agent
08/19/1999WO1999041367A1 Heteroaromatic oligoamides as affinity ligands
08/19/1999WO1999041248A1 Condensed heterocyclic system derivatives, preparation, pharmaceutical compositions containing them
08/19/1999WO1999041240A1 3,4-dihydroquinoline derivatives as nitrogen monoxide synthase (nos) inhibitors
08/19/1999WO1999041231A1 Amidino derivatives and drugs containing the same as the active ingredient
08/19/1999WO1999040931A1 Cyclic dipeptides and azetidinone compounds and their use in treating cns injury and neurodegenerative disorders