Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
05/2002
05/02/2002EP1201650A2 Ionic malonitril derivatives and their uses
05/02/2002EP1201235A1 Neuropathy improvers containing nitrogenous compounds as the active ingredient
05/02/2002EP1200432A1 Amido spiropiperidines promote the release of growth hormone
05/02/2002EP1200430A1 Thiourea and isothiourea derivatives for inhibiting ras-transformed cell growth
05/02/2002EP1200427A2 Small molecule modulators of g protein-coupled receptor six (gpr6)
05/02/2002EP1200424A1 C7 heterosubstituted acetate taxanes as antitumor agents
05/02/2002EP1200423A1 Substituted phenyl uracils
05/02/2002EP1200422A2 Pyrazole compositions useful as inhibitors of erk
05/02/2002EP1200415A1 Diamino-1,2,4-triazole-carboxylic acid derivatives as gsk-3 inhibitors
05/02/2002EP1200413A1 Trifluoromethylpyri(mi)dine carboxamides
05/02/2002EP1200411A2 Novel process for synthesis of heteroaryl-substituted urea compounds
05/02/2002EP1200404A2 Process for the preparation of spiro[(4-cyclohexanone)- [3h] indol-2'[1'h]-one derivatives
05/02/2002EP1200086A2 Methods for treating or preventing pain and anxiety
05/02/2002EP0615448B1 Sex steroid activity inhibitors
05/02/2002CA2425908A1 Mammalian metabolites of a tachykinin receptor antagonist
05/02/2002CA2425288A1 Pyrrolidine modulators of ccr5 chemokine receptor activity
05/02/2002CA2421796A1 Chemokine receptor binding heterocyclic compounds
05/01/2002CN1347414A Triazole compounds with dopamine-D3-receptor affinity
05/01/2002CN1347326A BAFF, inhibitors thereof and their use in modulation of B-cell response
05/01/2002CN1346830A Novel 2,4-dioxopyrrolidone and 2,4-dioxotetrahydro-furan derivs. and medicine contg. them as active component
05/01/2002CN1083838C Novel imidazole derivs., method for preparing same, use as medicine, and pharmaceutical compositions contg. same
04/2002
04/30/2002US6380396 Chemical intermediates for antiinflammatory agents
04/30/2002US6380394 Anticancer agents
04/30/2002US6380258 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
04/30/2002US6380246 For combating pests and weeds
04/30/2002US6380242 For diagnosis and therapy of central nervous system conditions
04/30/2002US6380241 For therapy of coronary angina, cerebral vasospasm, acute and chronic renal failure, gastric ulceration, cyclosporin-induced nephrotoxicity, endotoxin-induced toxicity, asthma, lpl-related lipoprotein disorders, proliferative diseases
04/30/2002US6380218 For therapy of respiratory, allergic, and inflammatory disorders comprising asthma, chronic obstructive pulmonary disease, acute respiratory disease syndrome, pulmonary hypersensitivity, and allergic rhinitis in a mammal
04/30/2002US6380215 For prevention and/or treatment of diseases caused by thrombus formation such as arterial thrombosis, arterial sclerosis, ischemic heart diseases
04/30/2002US6380210 Heteroaryl fused aminoalkyl-imidazole derivatives: selective modulators of GABAa receptors
04/30/2002US6380205 2-cyclohexyl quinazoline NMDA/NR2B antagonists
04/30/2002US6380201 Methods of treating or ameliorating the symptoms of common cold or allergic rhinitis with serotonin 5-HT1F agonists
04/30/2002US6380197 For treating and preventing a plethora of diseases including diabetes
04/30/2002US6380196 Bronchial therapeutics, bronchial dilators
04/30/2002US6380195 Including (methylenedioxyphenyl)cyclopenteno(1,2-b)pyridine derivatives
04/30/2002US6380194 For treatment of subjects suffering from hiv infection
04/30/2002US6379655 For protection of human skin and/or hair against the damaging effects of ultraviolet irradiation
04/30/2002CA2246994C Novel substituted n-methyl-n-(4-(4-(1h-benzimidazol-2-yl)¬1,4|diazepan-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases
04/30/2002CA2241827C Novel substituted 4-(1h-benzimidazol-2-yl)¬1,4|diazepanes useful for the treatment of allergic diseases
04/25/2002WO2002032920A2 Modified nucleosides for treatment of viral infections and abnormal cellular proliferation
04/25/2002WO2002032893A2 Piperidine compounds as anti-allergic
04/25/2002WO2002032891A1 Flavan compounds, their preparation and their use in therapy
04/25/2002WO2002032889A1 Aromatic and heterocyclic thiazolyl thiourea compounds and use
04/25/2002WO2002032886A1 A process for the preparation of bis-benzazolyl compounds
04/25/2002WO2002032880A1 New derivatives of cyano-aryl (or cyanoheteroaryl)-carbonyl-piperazinyl-pyrimidines, their preparation and application as medication
04/25/2002WO2002032879A1 Dihydropyrimidine derivatives as cysteine protease inhibitors
04/25/2002WO2002032874A2 Substituted heterocyclic compounds for treating multidrug resistance
04/25/2002WO2002032872A1 Nitrogenous aromatic ring compounds
04/25/2002WO2002032871A2 Compounds and methods for treating multidrug resistance
04/25/2002WO2002032870A1 Process of the preparation of 3-substituted-4-aryl piperidine compounds
04/25/2002WO2002032869A2 Substituted heterocyclic compounds for treating multidrug resistance
04/25/2002WO2002032868A2 2-substituted heterocyclic compounds and their use in treating multidrug resistance
04/25/2002WO2002032860A2 Dynamic organ function monitoring agents
04/25/2002WO2002032465A1 Tissue-specific exogenous optical agents
04/25/2002WO2002032377A2 Estrogen receptor modulators
04/25/2002WO2002032285A2 Hydrophilic light absorbing compositions for determination of physiological function in critically ill patients
04/25/2002WO2002010137A3 Indazole derivatives as JNK inhibitors
04/25/2002WO2001081341A3 9-oxa-epothilon derivatives, method for the production and use thereof in pharmaceutical preparations
04/25/2002WO2001058891A3 Piperazine and piperidine derivatives for treatment or prevention of neuronal damage
04/25/2002WO2001056990A3 Pyridine derivates as potentiators of glutamate receptors
04/25/2002WO2001002369A3 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
04/25/2002US20020049329 Novel human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
04/25/2002US20020049322 Quinoline and quinazoline compounds useful in therapy
04/25/2002US20020049231 S(-)-3-aminothalidomide; treating wide variety of diseases including diabetic retinopathy
04/25/2002US20020049229 Agents for treating neuropathic pain
04/25/2002US20020049223 Quinoline and naphthyridine carboxylic acid antibacterials
04/25/2002US20020049221 Analogs of deoxypreussomerin, palmarumycin CPI and related naphthoquinone spiroketals; inhibit thioredoxin-thioredoxin reductase system
04/25/2002US20020049220 Substituted azoles
04/25/2002US20020049210 Heteroaryl amines as novel acetylcholinesterase inhibitors
04/25/2002US20020049209 Dopamine D4 ligands for the treatment of novelty-seeking disorders
04/25/2002US20020049201 Sulfonamide inhibitors of aspartyl protease
04/25/2002US20020049197 Aminoquinazolines and their use as medicaments
04/25/2002US20020049195 Urea compounds that are muscarinic receptor antagonists and agonists, administering to the mammal the urea compound to treat urinary incontinence, chronic pulmonary obstructive disease, asthma, hyper salivation, blurred vision etc.
04/25/2002US20020049194 A benzoazepin or benzodiazepin derivatives, shows excellent anti-vasopressin activity, vasopressin agonistic activity and oxytocin antagonistic activity, and are useful as antagonist
04/25/2002US20020049193 Inhibitors of the enzyme activity associated with immunophilin proteins, particularly peptidyl-prolyl isomerase, or rotamase, enzyme activity.
04/25/2002DE10051321A1 New 2-(4-amino-piperidin-1-yl)-2-aryl-N-(phenylalkyl)-acetamides, are potent neurokinin antagonists, useful e.g. for treating allergic, inflammatory or central nervous system diseases
04/25/2002DE10051320A1 New 2-(4-amino-piperidin-1-yl)-2-aryl-N-(phenylalkyl)-acetamides, are neurokinin antagonists having a long duration of action, useful e.g. for treating allergic, inflammatory or central nervous system diseases
04/25/2002DE10050492A1 New butenolide or pentenolide amide derivatives, useful as kinase inhibitors for treating inflammatory and autoimmune diseases, e.g. rheumatoid arthritis, asthma, Alzheimer's disease or osteoarthritis
04/25/2002DE10050490A1 New butenolide or pentenolide amide derivatives, useful as kinase inhibitors for treating inflammatory and autoimmune diseases, e.g. rheumatoid arthritis, asthma, Alzheimer's disease or osteoarthritis
04/25/2002CA2426271A1 Dihydropyrimidine derivatives as cysteine protease inhibitors
04/25/2002CA2426148A1 Aromatic and heterocyclic thiazolyl thiourea compounds and use
04/25/2002CA2426097A1 New derivatives of cyano-aryl (or cyanoheteroaryl)-carbonyl-piperazinyl-pyrimidines, their preparation and application as medication
04/25/2002CA2425718A1 Dynamic organ function monitoring agents
04/25/2002CA2425698A1 Hydrophilic light absorbing compositions for determination of physiological function in critically ill patients
04/25/2002CA2424729A1 Estrogen receptor modulators
04/24/2002EP1199070A2 Use of PDE V inhibitors for improved fecundity in mammals
04/24/2002EP1198463A2 Compounds for use in treatment of neurological disorders
04/24/2002EP1198456A2 Potassium channel openers
04/24/2002EP1198234A2 Bicyclic aromatic compounds for treating drug addiction
04/24/2002EP0991646B1 An itraconazole exhibiting an improved solubility, a method of preparing the same and a pharmaceutical composition for oral administration comprising the same
04/24/2002EP0686149B1 Use of 2-mercapto-imidazole derivatives substituted in position 4 (or 5) as antioxidizing agents, method of preparation and applications in the pharmaceutical, cosmetic or food industries
04/24/2002CN1346355A Novel inhibitors of farnesyl-protein transferase
04/24/2002CN1346353A Farnesy transferase inhibitors having a pyrrole structure and process for preparation thereof
04/24/2002CN1346350A Compound which inhibiti leukocyte adhesion mediated by VLA-4
04/24/2002CN1346348A Amide compounds and medicinal use thereof
04/24/2002CN1346282A Use of a cyclooxygenase-2 inhibitor and one or more antineoplastic agents as combination therapy method in treating neoplasia
04/24/2002CN1346271A Quinazoline derivatives as angiogenesis inhibitors
04/24/2002CN1083451C Process for synthesizing doxazosin mesylate
04/24/2002CN1083450C Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
04/24/2002CN1083439C 2-amino-4-bicyclomino-1,3,5-triazines as herbicides and plant growth regulators