Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
03/2002
03/20/2002EP1188747A1 Phenoxypropylamine compounds
03/20/2002EP1188732A2 Combinatorial synthesis of a chemical library involving the separation of a zwitterionic compound by precipitation
03/20/2002EP1188439A2 Cell differentiation induction with mevalonate and mevalonolactone derivatives
03/20/2002EP1187831A1 Pyrrolidinyl, piperidinyl or homopiperidinyl substituted (benzodioxan, benzofuran or benzopyran) derivatives
03/20/2002EP1187830A1 Process for the preparation of paroxetine and structurally related compounds
03/20/2002EP1187829A1 Aminoalkyl substituted (benzodioxan, benzofuran or benzopyran) derivatives
03/20/2002EP1187821A1 Benzofuranylsulfonates
03/20/2002EP1187810A2 Heterocyclic analgesic compounds and their use
03/20/2002EP1187614A1 Substituted piperidines as melanocortin-4 receptor agonists
03/20/2002EP1156040A4 2,4-dioxo-5-arylidenimino-1,3-pyrimidines
03/20/2002EP0970074B1 Method and compositions for the synthesis of dioxolane nucleosides with beta-configuration
03/20/2002CN1341115A 16-halogen-epothilone derivatives, process for producing them and their pharmaceutical use
03/20/2002CN1341113A Process for production of paroxetine
03/20/2002CN1341104A 4-amino-quinazoline and quinoline derivatives having an inhibitory effect on signal transduction mediated by tyrosine kinases
03/20/2002CN1341102A Dopamine D1 receptor agonist compounds
03/19/2002US6359154 Exceptional utility as antitumor agents; bioavailability and nontoxic; oral administration; e.g., 10-hydroxy-10-deacetyl baccatin iii; anticarcinogenic agents
03/19/2002US6359151 Use as pesticides.
03/19/2002US6359148 For polymer, lubricants; heat, oxidation resistance, photostability
03/19/2002US6359145 Imidazole compounds
03/19/2002US6359138 4-hydroxy-piperidine derivatives
03/19/2002US6359134 Sulfonamide derivatives, their production and use
03/19/2002US6358995 Carboxylic acid derivatives having fused rings
03/19/2002US6358994 2-acylaminopropanamines as tachykinin receptor antagonists
03/19/2002US6358993 Pharmaceutically active nitrogen ring compounds and methods of use thereof
03/19/2002US6358990 Method for treating Alzheimer's disease
03/19/2002US6358984 For therapy of hypertension and/or diseases such as heart and renal diseases
03/19/2002US6358979 N-cyclopentyl modulators of chemokine receptor activity
03/19/2002US6358972 5-HT1F agonists
03/19/2002US6358961 Farnesyltransferase inhibiting quinazolinones
03/19/2002US6358960 For therapy of intravascular coagulation, coronary thrombosis, cerebral infarction, cerebral embolism, transient ischemic attack, cerebrovascular disorders, pulmonary vascular diseases, deep venous thrombosis, etc.
03/19/2002US6358956 Inhibitors of prenyl-protein transferase
03/19/2002US6358945 Compounds useful as anti-inflammatory agents
03/19/2002US6358886 Pre- and post-emergence herbicides for use on crops such as corn and sunflowers; affects both mono- and dicotyledonous weeds including foxtail; optically active (r,r) and (r,s)-diastereomers; high selectivity
03/19/2002US6358883 Pesticidal and parasiticidal use of 1-aryl-1-(substituted thio, sulfinyl and sulfonyl)-2-nitroethane compounds
03/19/2002US6358689 Detection of markers in nascent proteins
03/14/2002WO2002020514A1 Multivalent neuraminidase inhibitor conjugates
03/14/2002WO2002020513A1 Oxindole derivatives
03/14/2002WO2002020512A1 Imidazolo-5-yl-2-anilino-pyrimidines as agents for the inhibition of the cell proliferation
03/14/2002WO2002020509A2 Medicaments against viral infections
03/14/2002WO2002020500A2 Materials and methods to potentiate cancer treatment
03/14/2002WO2002020495A2 Inhibitors of glycogen synthase kinase 3
03/14/2002WO2002020489A2 QUINOLINE INHIBITORS OF cGMP PHOSPHODIESTERASE
03/14/2002WO2002020485A1 Spiroheterocyclic nitriles useful as reversible inhibitors of cysteine proteases
03/14/2002WO2002020484A1 Chemical compounds
03/14/2002WO2002020483A1 Piperidine derivatives for use 2,3-oxidosqualene-lanosterol cyclase inhibitors
03/14/2002WO2002020437A2 Basic compounds containing tertiary amides with activity on tachykinin receptors, and pharmaceutical compositions containing them
03/14/2002WO2002020436A2 Methods for forming combinatorial libraries combining amide bond formation with epoxide opening
03/14/2002WO2002020008A1 Inhibitors of nadh:ubiquinone oxidoreductase
03/14/2002WO2001070734A3 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
03/14/2002WO2001070692A3 Heterocyclic acylsulfimides, a method for their production, agents containing the same and their use as pesticides
03/14/2002WO2001070673A3 CYCLIC β-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-$g(a)
03/14/2002WO2001055130A3 Novel 1,3-dihydro-2h-indol-2-one derivatives and their use as ligands for v1b and v1a arginine-vasopressin receptors
03/14/2002WO2001051486A3 Process and intermediates for the preparation of imidazopyridines
03/14/2002US20020032339 Aryl borates
03/14/2002US20020032328 Heterocyclic acylsulfimides, processes for their preparation, compositions comprising them and their use as pesticides
03/14/2002US20020032325 4-amino-3-mercapto-1,2,4-triazoles
03/14/2002US20020032219 Use of alpha-1c specific compounds to treat benign prostatic hyperplasia
03/14/2002US20020032207 2-Cyclohexyl quinazoline NMDA/NR2B antagonists
03/14/2002US20020032205 An alkyl amine substituted isobenzofuran compound useful for certain psychiatric and neurological disorders; potently binding to the 5-HT1A receptor
03/14/2002US20020032202 Administering a pharmaceutically effective dose of the heterocycle-containing carboxylic acid derivative or salt to a patient suffering form acute promyelocytic leukemia
03/14/2002US20020032199 5-HT7 receptor antagonists
03/14/2002US20020032195 An mono or polycyclic aromatic or heteroaromatic carbamate or urea or thiacarbamoyl derivatives; inhibit production of cytokines involved in inflammatory processes
03/14/2002US20020032191 6-phenylpyridyl-2-amine derivatives useful as NOS inhibitors
03/14/2002US20020032184 For therapy of human immunodeficiency viral (HIV) , or genetically related retroviral, infection or a resulting acquired immunodeficiency syndrome (AIDS)
03/14/2002US20020032174 Polycyclic aryl and heteroaryl substituted 4-pyridones useful for selective inhibition of the coagulation cascade
03/14/2002US20020031816 Method of inhibition of human glycogen phosphorylase
03/14/2002DE10065434A1 Indole Indoles
03/14/2002DE10043791A1 Antiviral medicaments containing new or known chroman-4-one or chroman-4-one derivatives, especially effective against hepatitis B virus infections
03/14/2002DE10042696A1 New 3-(amino-methylene)-2-indolinone derivatives are kinase inhibitors and cell proliferation inhibitors useful e.g. for treating tumors, metastasis, rheumatoid arthritis or psoriasis
03/14/2002DE10041402A1 Neue Verbindungen, die Faktor Xa-Aktivität inhibieren Novel compounds which inhibit factor Xa activity
03/14/2002DE10023486C1 Ortho substituierte Anthranilsäureamide und deren Verwendung als Arzneimittel Ortho-substituted anthranilic acid amides and their use as medicaments
03/14/2002CA2417177A1 Spiroheterocyclic nitriles useful as reversible inhibitors of cysteine proteases
03/14/2002CA2416336A1 Multivalent neuraminidase inhibitor conjugates
03/13/2002EP1186604A1 Benzazepine derivatives, process for the preparation of the same and uses thereof
03/13/2002EP1186603A2 Processes for preparing endothelin antagonists
03/13/2002EP1186601A1 Novel isoquinoline derivatives or salts thereof
03/13/2002EP1186599A1 Novel processes for the preparation of substituted propenone derivatives
03/13/2002EP1186304A2 Pharmaceutical combinations for the treatment of stroke and traumatic brain injury
03/13/2002EP1185528A1 Inhibitors of il-12 production
03/13/2002EP1185275A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors
03/13/2002EP1185272A2 Novel use of 1-[4-(5-cyanoindol-3yl)butyl]-4-(2-carbamoylbenzofuran-5-yl)piperazine and its physiological acceptable salts
03/13/2002EP0977749B1 Bi-aromatic compounds and pharmaceutical and cosmetic compositions containing same
03/13/2002EP0948483B1 Farnesyl transferase inhibitors
03/13/2002EP0869957B1 3(2h)-pyridazinone derivatives and pharmaceutical compositions containing these compounds
03/13/2002CN1340053A Epothilon derivatives, method for the production and the use as pharmaceuticals
03/13/2002CN1340052A Process for the production of tert-butyl (E)-(6[2-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino] pyrimidin 5-yl] (4R,6S)-2,2-dimethyl [1,3] dioxan-4-yl) acetate
03/13/2002CN1340049A 4-heterocyclylsulfonamide)-5-methoxy-6-(2-methoxyphenoxy)-2-phenyl-or-pyridylpyrimidines as endothelin receptor antagonists
03/13/2002CN1340045A 5-HTIF agonists
03/12/2002US6355813 Intermediates useful in preparing these compounds
03/12/2002US6355804 Process for producing piperidinecarboxylic acid amide derivatives
03/12/2002US6355799 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
03/12/2002US6355726 Multicomponent ugi reaction; antisense agents, antigens; diagnosis; controlling gene expression by polymeric peptide nucleic acids
03/12/2002US6355664 Phenylpyrrolidines, phenylimidazolidines, 3-phenyl-1,3-oxizolidines and 3-phenyl-1,3-thiazolidines and their use in the treatment of inflammatory disease
03/12/2002US6355662 Peptide and nonpeptides autoimmune diseases, antiinflammatory agents
03/12/2002US6355660 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/12/2002US6355658 Coumarin derivatives, methods of preparation and application as medicines
03/12/2002US6355652 Drugs for sodium channel regulators and antiarrythmia agents
03/12/2002CA2187214C Aminostilbazole derivative and medicine
03/12/2002CA2055947C Condensed heterocyclic compounds, their production and use
03/07/2002WO2002018377A1 Compounds containing a bicyclic ring system useful as alpha v beta 3 antagonists