Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
08/2002
08/08/2002WO2002044142A3 Piperazine derivatives, their preparation and their use for treating central nervous system (cns) disorders
08/08/2002WO2002034716A3 Pyrrolidine modulators of ccr5 chemokine receptor activity
08/08/2002WO2002024650A3 Pyridinone and pyridinethione derivatives having hiv inhibiting properties
08/08/2002WO2002010140A3 Imidazolyl derivatives
08/08/2002WO2002000631A3 Benzhydryl derivatives
08/08/2002WO2001098268A3 Piperidine amides as modulators of chemokine receptor activity
08/08/2002WO2001081334A3 Cyclic amidine compounds and their use as alpha4beta2 nicotinic acetylcholine receptor ligands
08/08/2002WO2001009090A3 Hydantoin, thiohydantoin, pyrimidinedione and thioxopyrimidinone derivatives, preparation method and use as medicines
08/08/2002US20020107400 Cyanoguanidines as cell proliferation inhibitors
08/08/2002US20020107397 Provide polymeric resin products having low polydispersity.
08/08/2002US20020107392 Quinolinone derivatives
08/08/2002US20020107391 Involving a Grignard addition, such as 6-bromo-2,3-dihydrobenzofuran, and cyclization using a tetrasubstituted phosphordiamidic chloride
08/08/2002US20020107255 Potent and selective inhibitors of chemokine binding to its receptor CCR1 found on inflammatory and immunomodulatory cells (preferably leukocytes and lymphocytes).
08/08/2002US20020107254 P-substituted-N-(2-(4-(2,3-dihydro-benzo(1,4)dioxin-5-yl) -piperazin-1-yl)-propyl)-N-pyridin-2-yl-benzamide,
08/08/2002US20020107225 Use of nucleoside analogues (cytosine or 5-fluorocytosine containing compound) useful for acute or chronic myelogenous leukemia
08/08/2002US20020106338 Galenical formulation
08/08/2002CA2672805A1 Pyrimidine derivatives
08/08/2002CA2436774A1 Sulfonamide lactam inhibitors of factor xa
08/08/2002CA2436544A1 Ether derivatives useful as inhibitors of pde4 isozymes
08/08/2002CA2436535A1 Nicotinamide biaryl derivatives useful as inhibitors of pde4 isozymes
08/08/2002CA2436487A1 Methods of inhibiting kinases
08/08/2002CA2432783A1 Potassium channel inhibitors
08/08/2002CA2432642A1 Substituted aryl compounds as novel cyclooxygenase-2 selective inhibitors, compositions and methods of use
08/08/2002CA2432369A1 Cyclic derivatives as modulators of chemokine receptor activity
08/07/2002EP1229035A1 Imine intermediates for the preparation of trisubstituted imidazole compounds with multiple therapeutic properties
08/07/2002EP1229034A1 Nicotinamide derivatives and their mimetics as inhibitors of PDE4 isozymes
08/07/2002EP1229010A1 Novel diarylamide derivatives and use thereof as medicines
08/07/2002EP1228760A2 5-membered heterocycle derivatives, production thereof and use thereof as medicaments
08/07/2002EP1228759A2 Pharmaceutical compositions containing a taxane having a furyl or thienyl substituted side-chain
08/07/2002EP1228068A1 Polymorphic form of a tachykinin receptor antagonist
08/07/2002EP1228067A1 5-membered n-heterocyclic compounds with hypogylcemic and hypolipidemic activity
08/07/2002EP1228066A2 Sulfonamide derivatives
08/07/2002EP1228063A2 Substituted pyridines and pyridazines with angiogenesis inhibiting activity
08/07/2002EP1228060A1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof
08/07/2002EP1228059A1 Novel cyclopropanes as cgrp antagonists, medicaments containing said compounds and method for the production thereof
08/07/2002EP1228046A1 Phthalazinone derivatives as pde 4 inhibitors
08/07/2002EP1228041A2 Indole derivatives and their use as 5ht2a ligands
08/07/2002EP1227847A2 Inhibitors of the endothelin signalling pathway and alphavbeta3 integrin receptor antagonists for combination therapy
08/07/2002EP1227805A2 Mediators of hedgehog signaling pathways, compositions and uses related thereto
08/07/2002EP1227721A1 Novel substituted succinic acid metallo-beta-lactamase inhibitors and their use in treating bacterial infections
08/07/2002EP1077976B1 Water soluble azoles as broad-spectrum antifungals
08/07/2002EP0912529B1 Triazolyl disulphides
08/07/2002EP0888336B1 Novel substituted n-methyl-n-(4-(4-(1h-benzimidazol-2-yl-amino)p iperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases
08/07/2002EP0874843B1 Substituted 4-(1h-benzimidazol-2-yl) 1,4]diazepanes useful for the treatment of allergic diseases
08/07/2002EP0801649B1 Hydroxylamine derivatives useful for enhancing the molecular chaperon production and the preparation thereof
08/07/2002CN1362959A C10 carbamoyloxy substituted taxanes as antitumor agents
08/07/2002CN1362958A C7 carbonate substituted taxanes as antitumor agents
08/07/2002CN1362957A C17 heterosubustituted acetate taxanes as antitumor agents
08/07/2002CN1362956A C7 carbamoyloxy substituted taxanes as antitumor agents
08/07/2002CN1362955A C7 ester substituted taxanes as antitumor agents
08/07/2002CN1362954A Sulfamato hydroxamic acid metalloprotease inhibitor
08/07/2002CN1362953A Pyrazole compositions useful as inhibitors of ERK
08/07/2002CN1362947A N-cyanomethylamides as protease inhibitors
08/07/2002CN1362876A C10 heterosubstituted acetate taxanes as antitumor agents
08/07/2002CN1362397A Dialkoyl-halogen phenyl substituted keto-enol
08/06/2002US6429213 Cyclic hydroxamic acids as metalloproteinase inhibitors
08/06/2002US6429205 Anticoagulants
08/06/2002US6428667 Multichromophore fluorescent probes using DNA intercalation complexes
08/06/2002CA2223237C 1-phenyl-pyrazole derivatives and their use as parasiticidal agents
08/06/2002CA2208682C Fibrinogen receptor antagonists having substituted .beta.-amino acid residues and pharmaceutical compositions comprising the same
08/01/2002WO2002059117A1 Piperazine- and piperidine-derivatives as melanocortin receptor agonists
08/01/2002WO2002059116A2 Antimicrobial quinolone derivatives and use of the same to treat bacterial infections
08/01/2002WO2002059114A1 Lfa-1 antagonist compounds
08/01/2002WO2002059113A1 2h-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof
08/01/2002WO2002059112A2 Pyrazole compounds useful as protein kinase inhibitors
08/01/2002WO2002059111A2 Pyrazole compounds useful as protein kinase inhibitors
08/01/2002WO2002059108A1 Melanocortin receptor agonists
08/01/2002WO2002059106A1 Isoindole-imide compounds, compositions, and uses thereof
08/01/2002WO2002059089A2 Process for the preparation of heterocyclic indene analogs
08/01/2002WO2002059088A1 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
08/01/2002WO2002059087A1 Preparation of non-crystalline atorvastatin calcium
08/01/2002WO2002059086A1 Carboxamides as fungicides in agriculture
08/01/2002WO2002059084A2 Inhibitors of adp-ribosyl transferases, cyclases, and hydrolases, and uses thereof
08/01/2002WO2002058702A1 Urotensin-ii receptor antagonists
08/01/2002WO2002058695A1 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
08/01/2002WO2002058690A2 Methods for the treatment of diseases using malonyl-coa decarbox ylase inhibitors
08/01/2002WO2002036832A3 Atropisomers of asymmetric xanthene fluorescent dyes and methods of dna sequencing and fragment analysis
08/01/2002WO2002032285A3 Hydrophilic light absorbing compositions for determination of physiological function in critically ill patients
08/01/2002WO2002022572A3 Ligands for monoamine receptors and transporters, and methods of use thereof (neurotransmission)
08/01/2002WO2002011766A3 Use of 5ht4 receptor antagonists in the manufacture of a medicament for the prophylaxis or treatment of atrial fibrillation
08/01/2002US20020103381 Useful in pharmaceutical industry, such as antiinflammatory or antiarthritic agents; solid phase synthesis; esterification of a hydroxylated solid support, treating wtih trimethylsilyldiazomethane, deprotecting
08/01/2002US20020103256 Contacting helminth, nematode, insect or acarid pests or parasites or their food supply, habitat or breeding grounds with a nitroethyl derivative
08/01/2002US20020103245 1-aryl or heteroaryl substituted 5-amino-4 carbonylpyrazole derivatives; antiinflammatory agents
08/01/2002US20020103239 Such as N-hydroxy-2-(((4-phenoxyphenyl)-sulfonyl)methyl) benzamide which inhibits matrix metalloprotease activity
08/01/2002US20020103234 Heterocycl-containing carboxylic acid derivative and drug containing the same
08/01/2002US20020103229 Indazole derivatives as JNK inhibitors and compositions and methods related thereto
08/01/2002US20020103227 Nitric oxide synthase inhibitors such as 6(4'-(4-phenethyl-piperazin-1-ylmethyl)-biphenyl-4-yl)-pyridin-2-ylamine for treatment and prevention of central nervous system disorders
08/01/2002US20020103226 Substituted 8-arylquinoline phosphodiesterase-4 inhibitors
08/01/2002US20020103220 Such as N-(4-chlorobenzyl)-6-(4-morpholinylmethyl)-4-oxo-1-phenyl-1,4- dihydro-3-quinolinecarboxamide for treatment of herpes virus; viral DNA polymerase inhibitors
08/01/2002US20020103208 Useful in treatment of anxiety disorders, affective disorders such as depression, psychosis and schizophrenia, Parkinson's disease
08/01/2002US20020103205 Muscarinic antagonists
08/01/2002US20020103203 For treating cancer and other disease states associated with unwanted angiogenesis and/or cellular proliferation such as diabetic retinopathy, neovascular glaucoma, rheumatoid arthritis, psoriasis
08/01/2002US20020103185 Pyrazole derivatives
08/01/2002US20020102608 Library of indolinone compounds for use in the treatment of cancer
08/01/2002US20020102380 Ionic compounds in which the anionic load has been delocalized; ionic conducting materials, electronic conducting materials, colorant, and the catalysis of various chemical reactions including polymerization
08/01/2002CA2435775A1 2h-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof
08/01/2002CA2435566A1 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
08/01/2002CA2433819A1 Carboxamides as fungicides in agriculture
08/01/2002CA2432985A1 Piperazine- and piperidine-derivatives as melanocortin receptor agonists
08/01/2002CA2431996A1 Melanocortin receptor agonists