Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
01/2002
01/24/2002CA2415673A1 Tetrazole derivatives
01/24/2002CA2415665A1 Pyrrolidine-2-carboxylic acid hydrazide derivatives for use as metalloprotease inhibitors
01/24/2002CA2415331A1 Beta3 adrenergic agonists
01/24/2002CA2415126A1 Substituted 1-(4-aminophenyl)indoles and their use as anti-inflammatory agents
01/24/2002CA2384041A1 Selective melanin concentrating hormone-1 (mch1) receptor antagonists and uses thereof
01/23/2002EP1173441A1 6-alkenyl-, 6-alkinyl- and 6-epoxy-epothilone derivatives, process for their production, and their use in pharmaceutical preparations
01/23/2002EP1173429A1 Protease inhibitors
01/23/2002EP1173421A2 Indole derivatives as anti-inflammation agents
01/23/2002EP1173212A1 Contraceptive compositions contaning indolone derivatives and progestational agents
01/23/2002EP1173170A1 Pyrrolidine modulators of chemokine receptor activity
01/23/2002EP1173164A2 Estrogen receptor-beta ligands
01/23/2002EP0904269B1 3,4-diaryl-2-hydroxy-2,5-dihydrofurans as prodrugs to cox-2 inhibitors
01/23/2002CN1332747A 2'-fluoronucleosides
01/23/2002CN1332742A Epothilone derivatives and their use as antitumor agents
01/23/2002CN1332174A Optical information gene material and its application in gene chip technology
01/23/2002CN1078210C Watersoluble azole antifungals
01/22/2002US6340759 Fused pyridine derivatives
01/22/2002US6340704 Cell differentiation inducing amide derivatives, their production and use
01/22/2002US6340700 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same
01/22/2002US6340694 Diarylbenzopyran derivatives as cyclooxygenase-2 inhibitors
01/22/2002US6340684 Phthalazine derivatives as phosphodiesterase 4 inhibitors
01/22/2002US6340681 Useful as analgesics in mammals
01/22/2002US6340678 4,4-difluoro-2,3,4,5-tetrahydro-1H-1-benzoazepine derivatives and drug compositions containing them
01/22/2002CA2237971C Substituted 4-(1h-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases
01/17/2002WO2002004444A2 Heterocycle carboxamides as antiviral agents
01/17/2002WO2002004443A2 Heterocycle carboxamides as antiviral agents
01/17/2002WO2002004440A1 Composition and antiviral activity of substituted indoleoxoacetic piperazine derivatives
01/17/2002WO2002004429A1 Pyrimidine derivatives
01/17/2002WO2002004427A1 Phenylpyridazine derivatives and drugs containing the same
01/17/2002WO2002004425A2 Viral polymerase inhibitors
01/17/2002WO2002004424A1 Pyrazole derivatives
01/17/2002WO2002004422A2 Heterocycle carboxamides as antiviral agents
01/17/2002WO2002004420A1 Piperidine coumpounds for use as ccr-3 inhibitors
01/17/2002WO2002004416A2 Lactam metalloprotease inhibitors
01/17/2002WO2002003991A2 Use of substituted indole compounds for increasing nitric oxide synthase activity
01/17/2002WO2001062726A3 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
01/17/2002WO2001055107A3 Aromatic amines and amides acting on the melanocortin receptors
01/17/2002US20020007065 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
01/17/2002US20020007062 Enyme inhibitors for treating neurodegenerative diseases; inhibition of lipidic peroxidation and nitrogen oxide synthase in warm-blooded animal; for treatment of cardiovascular/brain disorders
01/17/2002US20020006948 Central nervous system disorders; antiinflammatory agents
01/17/2002US20020006943 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
01/17/2002US20020006936 Anticancer agents; restenosis
01/17/2002US20020006635 Stereoselectively hydrolyzing an anomeric mixture of 2-benzoyloxydioxolanecarboxylate with an enzyme; separating product; replacing carboxylate by reaction with a purine or pyrimidinyl derivative
01/17/2002DE10031809A1 Neue Flavonoide und ihre Verwendung in kosmetischen und dermatologischen Zubereitungen New flavonoids and their use in cosmetic and dermatological preparations
01/17/2002DE10005302A1 Substituierte 1,2,3,4-Tetrahydrochinolin-2-carbonsäurederivate Substituted 1,2,3,4-tetrahydroquinoline-2-carboxylic acid derivatives
01/17/2002CA2415505A1 Lactam metalloprotease inhibitors
01/17/2002CA2415492A1 Pyrazole derivatives
01/17/2002CA2414111A1 Use of substituted indole compounds for increasing nitric oxide synthase activity
01/17/2002CA2413044A1 Composition and antiviral activity of substituted indoleoxoacetic piperazine derivatives
01/17/2002CA2413042A1 Phenylpyridazine derivatives and drugs containing the same
01/16/2002EP1172106A2 Use of fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles as substance P receptor antagonists
01/16/2002EP1171437A1 Pesticidal indazole or benzotriazole derivatives
01/16/2002EP1171436A1 Process for the preparation of (pyridinylidene)-phthalides
01/16/2002EP1171435A2 Pyrimidine-2-one derivatives as integrin receptor ligands
01/16/2002EP1171422A1 Mmp inhibitor
01/16/2002EP0983237B1 Chemical process for the reduction of 1-substituted -3-hydroxymethyl-4- (4-fluorophenyl)tetrahydropyridines
01/16/2002EP0880517B1 Quinazoline compounds
01/16/2002CN1331691A Piperidines as CCR5 modulators
01/16/2002CN1331690A 4-(caminomethyl)-piperidine benzamides for treating gastrointestinal disorders
01/16/2002CN1331689A 4-and 5-alkynyloxindoles and 4-and 5-alkenyloxindoles
01/16/2002CN1331688A Aminopyrazole derivatives
01/16/2002CN1331680A N-aryl (thio) anthranilic acid amide derivatives, their prepn. and their use as VEGF receptor tyrosine kinase inhibitors
01/16/2002CN1331679A 3-azabicyclo [3.1.0] hexane derivatives as opiate receptors ligands
01/16/2002CN1331677A Pyrrolidine derivatives-CCR-3 receptor antagonists
01/16/2002CN1331674A Sulfonamide hydroxamates
01/16/2002CN1331591A Piperidines as CCR5 modulators
01/16/2002CN1331076A Condensed pyrazole compound, composition containing it and its application
01/16/2002CN1077889C Piperazine derivatives and their use as 5-HT1A antagonists
01/16/2002CN1077888C Benzopyrans and pharmaceutical compsn. contg. same
01/16/2002CN1077886C Amidino derivatives useful as nitric oxide synthase inhibitors
01/15/2002US6339155 Process for producing 3-phenyluracil compounds
01/15/2002US6339099 Guanidine mimics as factor Xa inhibitors
01/15/2002US6339097 N-phenylamide and N-pyridylamide derivatives, method of preparing them and pharmaceutical compositions containing them
01/15/2002US6339094 2-acylaminopropanamines as tachykinin receptor antagonists
01/15/2002US6339089 Antihypoxic agents; chronic obstructive pulmonary disease; vasoconstriction; reduces blood partial pressure of carbon dioxide; respiratory disorders; under oxygen inhalation treatment
01/15/2002US6339082 Tricyclic compounds, preparation method and said method intermediates, application as medicines and pharmaceutical compositions containing same
01/15/2002US6339046 Pyrazde herbicides
01/10/2002WO2002002553A1 Pharmaceutical compositions for treatment of diabetic nephropathy
01/10/2002WO2002002552A1 Quinazoline ditosylate salt compounds
01/10/2002WO2002002550A1 Novel pyrazinone derivatives
01/10/2002WO2002002548A1 Coumarin derivatives with comt inhibiting activity
01/10/2002WO2002002547A1 Pyrones as inhibitors of cyclooxygenase-2
01/10/2002WO2002002546A1 EPOXYCARBOXYLIC ACID AMIDES, AZIDES AND AMINO ALCOHOLS AND PROCESSES FOR PREPARATION OF α-KETO AMIDES BY USING THEM
01/10/2002WO2002002539A1 Aryl phenylheterocyclyl sulfide derivatives and their use as cell adhesion-inhibiting anti-inflammatory and immune-suppressive agents
01/10/2002WO2002002533A1 Propane-1,3-dione derivatives
01/10/2002WO2002002525A2 N-ureidoheterocycloaklyl-piperidines as modulators of chemokine receptor activity
01/10/2002WO2001056993A3 Pyrazole compositions useful as inhibitors of erk
01/10/2002US20020004518 Pyrazolyl compound; anticoagulants, antiproliferative agent
01/10/2002US20020004513 Azacyclic compounds
01/10/2002US20020004503 Viricides
01/10/2002US20020004501 Therapy for muscular disorders, urogenital disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002US20020004494 Muscular disorders, gastrointestinal disorders, respiratory system disorders
01/10/2002US20020004198 Detecting viricides; mix polypeptide samples, incubate with modulator of protein activity, monitor sample viricidal activity
01/10/2002CA2414461A1 Aryl phenylheterocyclyl sulfide derivatives and their use as cell adhesion-inhibiting anti-inflammatory and immune-suppressive agents
01/10/2002CA2413245A1 N-ureidoheterocycloaklyl-piperidines as modulators of chemokine receptor activity
01/10/2002CA2413002A1 Novel pyrazinone derivatives
01/10/2002CA2412874A1 Pyrones as inhibitors of cyclooxygenase-2
01/09/2002EP1170296A2 Process for the preparation of 3-aryl-benzofuran-2-ones
01/09/2002EP1170290A2 Compounds having ultra-violet absorption properties
01/09/2002EP1170289A2 Retroviral protease inhibiting compounds