Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
08/2002
08/01/2002CA2431904A1 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
08/01/2002CA2429353A1 Lfa-1 antagonist compounds
08/01/2002CA2424402A1 Antimicrobial quinolone derivatives and use of the same to treat bacterial infections
07/2002
07/31/2002EP1227093A2 Beta-lactams useful for preparation of taxanes having furyl or thienyl substituted side-chain
07/31/2002EP1227092A2 Isonitrile intermediates for the preparation of tri-substituted imidazole compounds with multiple therapeutic properties
07/31/2002EP1227091A2 Formamide intermediates for the preparation of tri-substituted imidazole compounds with multiple therapeutic properties
07/31/2002EP1226146A2 Quinoline and naphthyridine carboxylic acid antibacterials
07/31/2002EP1226141A1 Heterocyclic substituted pyrazolones
07/31/2002EP1226140A1 Novel indole compounds
07/31/2002EP1226138A1 Fab i inhibitors
07/31/2002EP1226136A2 Tyrosine kinase inhibitors
07/31/2002EP1226129A1 Methods and compositions utilizing quinazolinones
07/31/2002EP1226128A1 New pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical agents containing these compounds
07/31/2002EP1226126A1 Pyrimidine derivatives
07/31/2002EP1226120A2 Benz[f]indoles for use in the treatment of 5ht receptor related disorders
07/31/2002EP1225894A1 Fab i inhibitors
07/31/2002EP0880500B1 Esters of 3-hydroxy-piperidinemethanol derivatives
07/31/2002CN1361777A Substituted phenyl uracils
07/31/2002CN1361776A Novel fluorinated imidazoline Benzodioxane, preparation and therapeutic uses thereof
07/31/2002CN1361775A Novel diphenyl-piperidine derivate
07/31/2002CN1361770A Heteroaromatic ring compounds
07/31/2002CN1361769A Substituted 2-aryl-1,2,4-triazine-3,5-di(thi) one
07/31/2002CN1361692A Novel use of 1-[4-(5-cyanoindol-3-yl) butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts
07/31/2002CN1361687A Phosphate transport inhibitors
07/31/2002CN1088459C 1,4-disubstituted piperazines
07/31/2002CA2369462A1 Nicotinamide acids, amides, and their mimetics active as inhibitors of pde4 isozymes
07/30/2002US6426413 Inhibitors of caspases
07/30/2002US6426360 Antiarthritic agents
07/30/2002US6426354 Certain heteroaryl substituted thiol inhibitors of endothelin-converting enzyme
07/30/2002US6426318 3-aryl-1,2,4-triazone derivatives with herbicidal properties
07/30/2002CA2344707C N-substituted cycloalkyl and polycycloalkyl alpha-substituted trp-phe- and phenethylamine derivatives
07/30/2002CA2054342C Azolylmethylspiro [2.5] octanols and fungicides containing these
07/25/2002WO2002057259A2 Pyrazole compounds useful as protein kinase inhibitors
07/25/2002WO2002057250A1 Tetrahydropyran derivatives as neurokinin receptor antagonists
07/25/2002WO2002057249A1 Cyclic 2-carbonylaminoketones as inhibitors of cruzipain and other cysteine proteases
07/25/2002WO2002057248A2 Inhibitors of cruzipain and other cysteine proteases
07/25/2002WO2002057240A1 Substituted triazole diamine derivatives as kinase inhibitors
07/25/2002WO2002057238A1 Substituted quinolines for the treatment of protozoan and retrovirus co-infections
07/25/2002WO2002057233A1 Mch antagonists and their use in the treatment of obesity
07/25/2002WO2002057224A2 Synthesis and antimicrobial activityof novel dicationic 'reversed amidines'
07/25/2002WO2002056887A1 New combination of active ingredients containing alfuzosine and apomorphine
07/25/2002WO2002056882A1 Quinolines and nitrogenated derivaive thereof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents
07/25/2002WO2002050061A8 Piperazine derivatives for treatment of bacterial infections
07/25/2002WO2002042268A3 Ep4 receptor selective agonists in the treatment of osteoporosis
07/25/2002WO2002039988A3 Novel uses of combined selective dopamine d2 receptor antagonists and 5-ht1a receptor agonists
07/25/2002WO2002038107A3 Stat modulators
07/25/2002WO2002032874A3 Substituted heterocyclic compounds for treating multidrug resistance
07/25/2002WO2002008177A3 N-substituted-1-amino-1,1-dialkylcarboxylic acid derivatives
07/25/2002US20020099224 Hydrolysis of [R (R*, R*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid esters with calcium hydroxide
07/25/2002US20020099223 Cyclocarbonylating acetic acid (or benzoic acid)-1-(1-benzenesulfonyl-1H-indol-2-yl)-allyl ester to obtain 9-benzenesulfonyl-9H-carbazol-4-yl ester; saponifying
07/25/2002US20020099219 Piperidine compounds and process for providing the same
07/25/2002US20020099215 For therapy and prophylaxis of P-glycoprotein-mediated multidrug resistance
07/25/2002US20020099214 For prophylaxis and therapy of pruritus
07/25/2002US20020099212 Sulfonamide compounds and pharmaceutical use thereof
07/25/2002US20020099205 Cyclization of (2-Oxo-4-(2-oxo-2-(tetrahydrofuran-2-yl)-ethylsulfanyl)-3-phenylacetylamino -azetidin-1-yl)-(trimethyl- alpha -phosphanylidene)-acetic acid 4-nitro-benzyl ester; reacting with acid
07/25/2002US20020099202 Compoound for use in the sequencing of nucleic acids
07/25/2002US20020099089 Administering compounds such as trans-3-(naphth-2-yl)-but-2-enoic acid-N-(2-carboxy-phenyl)-amide or like for therapy of conditions associated with increased telomerase activity, e.g. tumour diseases
07/25/2002US20020099084 Pharmaceutically active compounds and methods of use
07/25/2002US20020099071 Protein tyrosine kinase and protein serin/threonine kinase inhibitory activity; anticancer agents; treating chemotherapy induced alopecia
07/25/2002US20020099050 E.g., 1-(1,4-benzodioxan-5-ylcarbonyl)-1,2,3,6-tetrahydro-pyridine), 1-(1,3-benzodioxol-5-ylcarbonyl)-piperidine); and 1-(1,3-benzodioxol-5-ylcarbonyl)-1,2,3,6-tetrahydropyridine
07/25/2002US20020099035 Method for preparing alpha-sulfonyl hydroxamic acid derivatives
07/25/2002US20020099007 And the prenylation of the oncogene protein Ras; peptidomimetic macrocyclic compounds
07/25/2002DE10130830A1 Indol-Derivate Indole derivatives
07/25/2002CA2435117A1 Cyclic 2-carbonylaminoketones as inhibitors of cruzipain and other cysteine proteases
07/25/2002CA2433835A1 Tetrahydropyran derivatives as neurokinin receptor antagonists
07/25/2002CA2432870A1 Substituted triazole diamine derivatives as kinase inhibitors
07/25/2002CA2425135A1 Synthesis and antimicrobial activity of novel dicationic "reversed amidines"
07/24/2002EP1225171A1 Substituted cyanophenyluracils
07/24/2002EP1224933A1 New combination of active ingredients containing alfuzosine and apomorphine
07/24/2002EP1224197A1 Hygromycin derivatives
07/24/2002EP1224195A1 C-aryl glucoside sglt2 inhibitors
07/24/2002EP1224183A2 Heterocyclic sodium/proton exchange inhibitors and method
07/24/2002EP1224182A1 N-substituted 1-(lactone) isoquinolones for treating nervous disorders
07/24/2002EP1224180A2 Substituted azoles
07/24/2002EP1224175A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
07/24/2002EP1224174A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
07/24/2002EP1224171A1 Beta disubstituted metalloprotease inhibitors
07/24/2002EP1224170A1 6-position substituted indoline, production and use thereof as a medicament
07/24/2002EP1224165A1 Novel compounds
07/24/2002EP1223933A2 5-membered heterocycle derivatives, production thereof and use thereof as medicaments
07/24/2002EP1223932A1 Compounds and methods
07/24/2002EP0989114B1 N,n-disubstituted amic acid derivatives
07/24/2002EP0934527B1 Non radioactive receptor assay suitable for quantitative and qualitative analysis of trace amounts of receptor binding analyte
07/24/2002EP0889041B1 Novel iridoid derivatives and neovascularization inhibitors containing the same as active ingredient
07/24/2002EP0814804B1 Substituted benzopyrans
07/24/2002EP0804431B1 GLYCOPROTEIN IIb/IIIa ANTAGONISTS
07/24/2002EP0689463B1 Imidazole based nitrogen-sulfur ligands useful in radiographic imaging agents
07/24/2002EP0684945B1 Pyrazole- or isoxazole-substituted alkyl amide acat inhibitors
07/24/2002CN1360605A Thermoplastic polymer having polar group, use thereof, and unsaturated compounds having polar group
07/24/2002CN1360583A Novel compounds, their use and preparation
07/24/2002CN1360581A Benzoylpyridazines
07/24/2002CN1360577A Hydroxamic acid derivs. as matrix metalloprotease inhibitors
07/24/2002CN1360576A Process for preparation of spiro [(4-cyclohexanone)-[3H] indol]-2'[iH]-one derivs.
07/24/2002CN1359900A Metal protease inhibitor, preparing process thereof and pharmaceutical composition contg. same
07/23/2002US6423847 Reacting a-tocopherol with a nicotinic compound; therapy for vision disorders
07/23/2002US6423840 Forming n-acylamino compound
07/23/2002US6423723 Oral bioavailability
07/23/2002US6423716 Nitrogenous heterocyclic compounds
07/23/2002US6423713 Substituted pyrazoles as p38 kinase inhibitors
07/23/2002US6423712 2,4-Substituted imidazolidine derivatives, their preparation, their use and pharmaceutical preparations comprising them