Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
04/2002
04/11/2002WO2002028837A1 Metabotropic glutamate receptor antagonists
04/11/2002WO2002028831A1 Inhibitors of prenyl-protein transferase
04/11/2002WO2002028829A2 Peptide deformylase inhibitors
04/11/2002WO2001085671A3 Anthranyl amides and their use as medicaments
04/11/2002WO2001077079A3 Polycyclic aryl and heteroaryl substituted 4-pyridones useful for selective inhibition of the coagulation cascade
04/11/2002WO2001019797A3 HYDROXYALKANOYL AMINOLACTAMS AND RELATED STRUCTURES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
04/11/2002US20020042511 New derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
04/11/2002US20020042501 Antiproliferative and antitumor agents and angiogenesis inhibitors
04/11/2002US20020042430 Novel esters of 1, 4-disubstituted piperidine derivatives
04/11/2002US20020042398 Novel lactam metalloprotease inhibitors
04/11/2002US20020042397 4-hydroxycinnoline-3-carboxyamides as antiviral agents
04/11/2002US20020042396 Amino acid derivatives
04/11/2002US20020042377 Rotamase enzyme activity inhibitors
04/11/2002CA2424870A1 Agents for promoting the proliferation or differentiation of stem cells or neural progenitor cells
04/11/2002CA2424222A1 Inhibitors of prenyl-protein transferase
04/11/2002CA2421782A1 Quinoline and quinolinone derivatives as metabotropic glutamate receptor antagonists
04/10/2002EP1194427A1 Thiophene-ethyl thiourea compounds and use in the treatment of hiv
04/10/2002EP1194426A2 Benzofurane derivatives
04/10/2002EP1194418A1 Bicyclic heterocycles, medicaments containing these compounds, their use and methods for the production thereof
04/10/2002EP1194417A1 Phenoxy fluoropyrimidines
04/10/2002EP1194416A1 Halopyrimidines
04/10/2002EP1194411A1 Benzoylpyridazines
04/10/2002EP1194410A1 Benzimidazole derivatives and pharmaceutical compositions comprising these compounds
04/10/2002EP1194144A1 Antibacterial compounds
04/10/2002EP1112261B1 2-ethyl-2,3-dihydrobenzofuran-carboxylic acid ester derivative, preparation method and use for preparing efaroxan derivatives
04/10/2002EP1087662B1 Composition for keeping away vermin
04/10/2002EP0950046B1 3,4-disubstituted azetidin-2-one derivatives useful as cysteine proteinase regulators
04/10/2002EP0797573B1 4-heteroaryl-1,2,4-triazole derivatives with herbicidal properties
04/10/2002EP0734387B1 Hiv protease inhibitors
04/10/2002CN1344266A Novel compounds
04/10/2002CN1344265A Piperidine, tetrahydropyridine and piperazine derivatives, their prepn. and use
04/10/2002CN1344264A Tetrahydropyran derivatives and their use as therapeutic agents
04/10/2002CN1344261A 2,4-diamino-1,3,5-triazines, method for producing them and their use as herbicides and plant growth regulators
04/10/2002CN1344256A (Hetero) aryl-bicyclic heteroaryl derivatives, their prepn. and their use as protease inhibitors
04/10/2002CN1344160A Heterocyclic aromatic compounds useful as growth hormone secretagogues
04/09/2002USRE37650 Aryl and heteroaryl quinazoline compounds which inhibit CSF-1R receptor tyrosine kinase
04/09/2002US6369100 Method for inhibiting gene expression promoted by AP1 protein with RARβ selective retinoids and method for treatment of diseases and conditions with such retinoids
04/09/2002US6369086 Substituted oxidole derivatives as protein tyrosine and as protein serine/threonine kinase inhibitors
04/09/2002US6369083 2-methoxyimino-2 (pyrinyloxymethyl) phenyl acetamides with polyether derivatives on the pyridine ring
04/09/2002US6369077 Protease inhibitors
04/09/2002US6369075 7[4′-trifluoromethyl-biphenyl-2-carbonyl)amino]-quinoline-3-carboxylic acid amides, and method of inhibiting the secretion of apolipoprotein B
04/09/2002US6369068 Amino substituted pyrimidine containing compounds
04/09/2002US6369057 Quinoxalines, processes for their preparation and their use
04/09/2002CA2229000C 1-biphenylimidazole derivatives, their preparation and their therapeutic use
04/09/2002CA2171675C Aromatic heterocyclic compounds; pharmaceutical and cosmetic compositions containing the same and their uses
04/09/2002CA2071224C Quinoline derivatives, their production and use
04/09/2002CA2024185C Substituted 4,5-diamino-1,2,4-triazol-3-(thi)ones
04/04/2002WO2002026734A1 PIPERAZIN-2-ONE AMIDES AS INHIBITORS OF FACTOR Xa
04/04/2002WO2002026706A2 17-beta-hydroxysteroid dehydrogenase-ii inhibitors
04/04/2002WO2002026228A1 Benzimidazolone antiviral agents
04/04/2002WO2002026227A1 Lactone integrin antagonists
04/04/2002WO2002026220A2 Taxoid conjugates as antimitotic and antitumor agents
04/04/2002WO2002026216A1 Pharmaceutical oxan preparation
04/04/2002WO2001089451A3 Protease inhibitors
04/04/2002WO2001081308A3 Aminopiperidines for use as glyt-1 inhibitors
04/04/2002US20020040155 Radiosensitizing taxanes and their pharmaceutical preparations
04/04/2002US20020040147 Novel catechols as antimicrobial agents
04/04/2002US20020040146 Useful as inhibitors of metalloproteases, e.g. zinc proteases, and which are effective in therapy of disease states associated with vasoconstriction
04/04/2002US20020040144 For therapy of thrombotic disease, asthma, emphysema, cirrhosis, arthritis, carcinoma, melanoma, restenois, atheroma, trauma, shock and reperfusion injury
04/04/2002US20020040048 (2S,4R)-4-Mercapto-1-(naphthalene-2-sulfonyl)-pyrrolidine-2 -carboxylic acid N'-isobutyl-N'-(4-methyl-benzenesulfonyl)-hydrazide, for example; inhibitors of metalloproteases, e.g. zinc proteases; vasodilators
04/04/2002US20020040038 Administering donepezil or its hydrochloride salt
04/04/2002US20020040028 2-amine substituted quinoline or quinozoline derivatives useful for treating benign prostatic hyperplasia
04/04/2002DE10044091A1 Chromanonderivate Chromanone
04/04/2002CA2424949A1 Pharmaceutical oxan preparation
04/04/2002CA2423483A1 Taxoid conjugates as antimitotic and antitumor agents
04/04/2002CA2423434A1 Lactone integrin antagonists
04/04/2002CA2422873A1 Piperazin-2-one amides as inhibitors of factor xa
04/03/2002EP1193265A2 A process for the preparation of 4-[2-(aryl or heterocyclo)-1H-imidazol-1-yl]benzenesulfonamides
04/03/2002EP1192152A1 Novel fluorinated imidazoline benzodioxane, preparation and therapeutic uses thereof
04/03/2002EP1192151A1 Anilinoquinazolines as protein tyrosine kinase inhibitors
04/03/2002EP1192148A1 Thiochroman derivatives resisting neurological disorders
04/03/2002EP1192146A1 Chroman derivatives resisting neurological disorders
04/03/2002EP1192135A2 Serine protease inhibitors
04/03/2002EP1192133A1 N-cyclopentyl modulators of chemokine receptor activity
04/03/2002EP1192132A2 Serine protease inhibitors
04/03/2002EP1162201A9 Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives
04/03/2002EP1161240A4 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
04/03/2002EP1158980A4 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
04/03/2002EP1156807A4 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
04/03/2002EP1140087A4 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
04/03/2002EP0999838B1 Self-emulsifying formulation for lipophilic compounds
04/03/2002EP0873331B1 Benzofuran carboxamides and sulphonamides
04/03/2002EP0865440B1 Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives
04/03/2002EP0859774B1 Substituted sulphonylamino (thio)carbonyl compounds as herbicides
04/03/2002CN1343207A Benzofuran-2-ones as colorants for organic materials
04/03/2002CN1343201A Bicyclic heterocycles, pharmaceutical compositions containing these compounds, and processes for preparing them
04/03/2002CN1082049C Sulfoaminomethyl acid radical compound
04/02/2002US6365652 Trisaryl-1,3,5-triazine ultraviolet light absorbers
04/02/2002US6365620 Trifluoromethylpyrrolcarboxamides
04/02/2002US6365613 Fungicidal mixtures
04/02/2002US6365600 For therapy of condition associated with smooth muscle cell proliferation in a warm-blooded animal which comprises administering imidazol-5-yl-methyl-2-quinolinone derivatives
04/02/2002US6365599 For therapy of benign prostatic hyperplasia
04/02/2002US6365588 Tricyclic amide and urea compounds useful for inhibition of G-protein function and for treatment of proliferative diseases
04/02/2002US6365584 For prophylaxis and therapy of inflammatory and/or allergic diseases, lung fibrosis, fibrosing alveolitis and scarring, collagenoses such as lupus erythematodes and sclerodermia as well as arteriosclerosis, psoriasis and neoplasm
04/02/2002US6365552 Substituted 3-phenylpyrazoles
04/02/2002US6365068 Heterocyclic aromatic anion salts, and their uses as ionic conducting materials
04/02/2002CA2223574C Biphenyl-2-carboxylic acid-tetrahydro-isoquinolin-6-yl amide derivatives, their preparation and their use as inhibitors of microsomal triglyceride transfer protein and/or apolipoprotein b (apo b) secretion
04/02/2002CA2178130C Method of producing 2-naphthamide derivative, and compounds for producing 2-naphthamide derivative
03/2002
03/28/2002WO2002024693A1 A process for producing 3,4-dihydro naphthyridinone analogs
03/28/2002WO2002024687A1 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinolinone derivatives