Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
03/2002
03/07/2002WO2002018374A1 Substituted pyrimidines as selective cyclooxygenase-2 inhibitors
03/07/2002WO2002018373A1 Quinazoline derivatives, medicaments containing these compounds, their use, and methods for the production thereof
03/07/2002WO2002018370A1 Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
03/07/2002WO2002018368A1 Tricyclic antitumor compounds being farnesyl protein transferase inhibitors
03/07/2002WO2002018348A2 Quinazoline derivatives as alpha-1 adrenergic antagonists
03/07/2002WO2002018346A1 Pyrazole derivatives and their use as protein kinase inhibitors
03/07/2002WO2002018321A2 Amino(oxo)acetic acid protein tyrosine phosphatase inhibitors
03/07/2002WO2002017924A1 Method of treatment
03/07/2002WO2002017912A1 Endothelin antagonists
03/07/2002WO2001089457A3 Thrombopoietin mimetics
03/07/2002WO2001077100A3 Benzoamide piperidine compounds as substance p antagonists
03/07/2002WO2001062765A3 Small molecule modulators of g protein-coupled receptor six
03/07/2002WO2001057022A3 Pyrazole compositions useful as inhibitors of erk
03/07/2002WO2001055131A3 Prodigiosin-derivatives as neoplastic and anti-viral agents
03/07/2002US20020028943 For lowering serum lipid, cholesterol and/or triglyceride levels; treating atherosclerosis
03/07/2002US20020028942 Freeze-dried form of paroxetine hydrochloride suitable for parenteral administration; treatment and prophylaxis of depression, obsessive compulsive disorder and panic disorders
03/07/2002US20020028938 Prostaglandin endoperoxide H synthase biosynthesis inhibitors
03/07/2002US20020028836 Potassium channel openers
03/07/2002US20020028835 Cyclic amine phenyl beta-3 adrenergic receptor agonists
03/07/2002US20020028831 Phenylpyridine derivatives useful as phosphodiesterase inhibitors
03/07/2002US20020028826 HMG-CoA reductase inhibitors and method
03/07/2002US20020028819 Piperazinedione compounds
03/07/2002DE10042064A1 Chinazoline, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Quinazolines, medicaments containing these compounds, their use and process for their preparation
03/07/2002DE10042061A1 Bicyclische Heterocyclen,diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
03/07/2002DE10042060A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
03/07/2002DE10042059A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
03/07/2002DE10042058A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
03/07/2002DE10041574A1 Chromenonderivate Chromenonderivate
03/07/2002CA2420673A1 Tricyclic antitumor compounds being farnesyl protein transferase inhibitors
03/07/2002CA2420363A1 Pyrazole derivatives and their use as protein kinase inhibitors
03/07/2002CA2419255A1 Compounds containing a bicyclic ring system useful as alpha v beta 3 antagonists
03/07/2002CA2417042A1 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for preparing them
03/06/2002EP1184379A1 Chromene compound
03/06/2002EP1184374A1 Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders
03/06/2002EP1184373A1 Tricyclic compounds
03/06/2002EP1183253A1 C7 ester substituted taxanes as antitumor agents
03/06/2002EP1183251A1 Indolylpiperidine derivatives as antihistaminic and antiallergic agents
03/06/2002EP1183242A2 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
03/06/2002EP1183241A1 Spiroimidazolidine derivatives, their preparation, their use and pharmaceutical preparations comprising them
03/06/2002EP1183240A1 Beta2-adrenoceptor agonists
03/06/2002EP1183239A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
03/06/2002EP1183238A1 Metabotropic glutamate receptor antagonists
03/06/2002EP1183229A1 Glucagon antagonists/inverse agonists
03/06/2002EP1183019A2 Ace-2 inhibiting compounds and methods of use thereof
03/06/2002EP1070062B1 Oxidation process using tempo
03/06/2002EP0994865B1 Triazole compounds and the use thereof as dopamine-d 3-ligands
03/06/2002EP0883403A4 Method for treating sexual dysfunctions
03/06/2002EP0819122B1 1,3-dihydro-1-(phenylalkyl)-2h-imidazol-2-one derivatives having pdeiv and cytokine activity
03/06/2002EP0728748B1 Benzodiazepine derivatives
03/06/2002EP0695295B1 3-(hetero)aryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation
03/06/2002CN1338958A The use of 4-H-1-benzopyran-4-one derivatives as inhibitors of smooth muscle cell proliferation
03/06/2002CN1080263C Method and compositions for the synthesis of dioxolane nucleosides with 'beta'-configuration
03/06/2002CN1080262C Novel substituted 4-(1H-benzimidazol-2-YL)[1,4] diazepanes useful for the treatment of allergic diseases
03/06/2002CA2356545A1 Pharmaceutical combinations for the treatment of stroke and traumatic brain injury
03/05/2002US6353116 Endothelin receptor antagonists
03/05/2002US6353110 Key intermediate in the synthesis of an endothelin antagonist; arylation of a 3-oxopropylpyridine with lithium 1,3 benzenedioxole then hydrolysis
03/05/2002US6353107 1-alkoxy-polyallkyl-piperidine derivatives and their use as polymerization regulators
03/05/2002US6353008 Serotonin reuptake inhibitor as antidepressants
03/05/2002US6353007 Substituted 1-(4-aminophenyl)indoles and their use as anti-inflammatory agents
03/05/2002US6352989 Nitrogenous heterocyclic derivatives and medicine thereof
03/05/2002US6352985 Benzimidazole compounds
03/05/2002US6352981 Treat disorders which respond to dopamine d.sub.3 ligands such as schistosomiasis, schizophrenia, depression, neuroses or psychoses
03/05/2002US6352958 Pre- and post-emergence herbicides
03/05/2002CA2272138C Pyrazolopyrimidine and pyrazolopyridine compounds having crf antagonist activity
03/05/2002CA2207574C Esters and amides of non-steroidal anti-inflammatory carboxylic acids which may be used as anti-oxidants, 5-lipoxygenase inhibitors and non-steroidal anti-inflammatory products
02/2002
02/28/2002WO2002016361A2 Nitrogenous heterocyclic compounds
02/28/2002WO2002016353A1 Bicyclic heteroaromatic derivatives for the treatment of immune and inflammatory disorders
02/28/2002WO2002016352A1 Quinazoline derivatives
02/28/2002WO2002016349A1 4-, 5-, 6- and 7-indole derivatives useful for the treatment of cns disorders
02/28/2002WO2002016344A1 Tetrahydropyran derivatives as nk-1 receptor antagonists
02/28/2002WO2002016343A1 Tetrahydropyran derivatives as nk-1 receptor antagonists
02/28/2002WO2002016340A1 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
02/28/2002WO2002016339A1 Aminoalkylbenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
02/28/2002WO2002016338A1 Aminoalkenylbenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
02/28/2002WO2002016313A2 Integrin receptor inhibitors
02/28/2002WO2001079167A3 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
02/28/2002WO2001077080A3 Pyrazole compounds having anti proliferative activity
02/28/2002WO2001056989A3 Inhibitors of factor xa
02/28/2002WO2001017614A3 Methods and compositions containing succinimide or maleimide derivatives of antineoplastic agents
02/28/2002WO2000067746A8 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors
02/28/2002US20020026052 Antineoplastic agents, agents for treatment of osteoporosis and polycystic kidney disease
02/28/2002US20020026050 Thrombin receptor antagonists
02/28/2002US20020025965 Antiserotonine agents
02/28/2002US20020025963 Novel guanidine mimics as factor Xa inhibitors
02/28/2002US20020025961 Platelet ADP receptor inhibitors
02/28/2002US20020025960 Heterocycle carboxamides as antiviral agents
02/28/2002US20020025957 Anticoagulants, cardiovascular disorders
02/28/2002US20020025301 Novel flavonoids and their use in cosmetic and dermatological preparations
02/28/2002DE10041470A1 New 6-substituted 12,13-(cyclopropyl or azacyclopropyl)-epothilone derivatives, useful as cell division regulators for treating e.g. malignant tumors, psoriasis or arthritis
02/28/2002DE10040527A1 New 4-tert. butoxycarbonylamino-quinazoline derivatives, useful as intermediates for tyrosine kinase-mediated signal transduction inhibitors
02/28/2002DE10040525A1 New 6-acylamino-4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors or respiratory or gastrointestinal diseases
02/28/2002CA2419580A1 Integrin receptor inhibitors
02/28/2002CA2419266A1 4-, 5-, 6- and 7-indole derivatives useful for the treatment of cns disorders
02/28/2002CA2415852A1 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
02/28/2002CA2415846A1 Aminoalkenylbenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
02/27/2002EP1182202A1 Aminomethylpyrrolidine derivatives having aromatic substituents
02/27/2002EP1182200A1 Tricyclic fused heterocycle compounds, process for preparing the same and use thereof
02/27/2002EP1182195A1 Cyclic compounds and uses thereof
02/27/2002EP1182193A1 Remedies for neuropathic pain
02/27/2002EP1182192A1 4-hydroxypiperidine derivatives having antiarrhythmic effect