Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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09/01/2005 | US20050192286 Ligands of melanocortin receptors and compositions and methods related thereto |
09/01/2005 | US20050192279 Pyridazinones as antagonists of alpha4 integrins |
09/01/2005 | US20050192277 Histamine-3 receptor antagonists; 4-(2-{2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl}-1-benzofuran-4-yl)benzonitrile; acute myocardial infarction, asthma, psychological disorders, gastrointestinal disorders, inflammation, jet lag, cancer, septic shock, Tourette's syndrome, neurodegenerative disorders |
09/01/2005 | CA2557433A1 Quinazoline derivatives and therapeutic use thereof |
09/01/2005 | CA2556268A1 Acetylinic piperazine compounds and their use as metabotropic glutamate receptor antagonists |
09/01/2005 | CA2555970A1 Therapeutic amide derivatives |
09/01/2005 | CA2555402A1 Bipyridyl amides as modulators of metabotropic glutamate receptor-5 |
09/01/2005 | CA2555073A1 Amino heterocyclic modulators of chemokine receptor activity |
09/01/2005 | CA2554774A1 Novel heterocyclic compound |
09/01/2005 | CA2554686A1 Compounds |
09/01/2005 | CA2498644A1 Anti-inflammatory and analgesic heterocyclic amidines that inhibit nitrogen oxide (no) production |
08/31/2005 | EP1568693A1 Process for producing quinolinecarbaldehyde |
08/31/2005 | EP1568692A1 (pyridin-4-yl)alkyl-amides as TNF-alpha production inhibitors |
08/31/2005 | EP1568367A1 Compounds effecting glucokinase |
08/31/2005 | EP1567518A2 Oxime ester photoinitiators with heteroaromatic groups |
08/31/2005 | EP1567511A1 Substituted piperazines, (1,4) diaszepines, and 2,5-diazabicyclo (2.2.1) heptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists |
08/31/2005 | EP1567506A2 Cyanoguanidines and cyanoamidines as erbb2 and egfr inhibitors |
08/31/2005 | EP1567504A1 Antibacterial agents |
08/31/2005 | EP1567502A1 Substituted dihydrophenanthridinesul fonamides |
08/31/2005 | EP1567496A1 Phenyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatment of pain or gastrointestinal disorders |
08/31/2005 | EP1567493A1 Phenyl substituted piperidine compounds for use as ppar activators |
08/31/2005 | EP1567489A1 Pyrrolidin-2-one derivatives as inhibitors of thrombin and factor xa |
08/31/2005 | EP1567488A1 Hydroxyethylamine derivatives for the treatment of alzheimer's disease |
08/31/2005 | EP1567151A1 3-(2-hydroxy-phenyl)-1h-pyrazole-4-carboxylic acid amide derivatives as hsp90 inhibitors for the treatment of cancer |
08/31/2005 | EP1395576B1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders |
08/31/2005 | EP1268445B1 4-amino-5-cyano-2-anilino-pyrimidine derivatives and their use as inhibitors of cell-cycle kinases |
08/31/2005 | EP1237875B1 Substituted imidazole neuropeptide y y5 receptor antagonists |
08/31/2005 | EP1182200B1 Tricyclic fused heterocycle compounds, process for preparing the same and use thereof |
08/31/2005 | EP1095020B1 2-aminopyridine erivatives, their use as medicines and pharmaceutical compositions containing them |
08/31/2005 | EP0882718B1 Benzimidazole derivatives |
08/31/2005 | CN1662527A Pyrrolidinium derivatives as antagonists of M3 muscarinic receptors |
08/31/2005 | CN1662525A Preparation for the production of 1, 2, 4-triazolymethyl-oxiranes |
08/31/2005 | CN1662524A Indole derivatives useful as histamine h3 antagonists |
08/31/2005 | CN1662519A Heterocyclic compounds as glycine transport inhibitors |
08/31/2005 | CN1662518A Processes for producing epoxytriazole derivative and intermediate therefor |
08/31/2005 | CN1662508A Compounds, compositions and methods |
08/31/2005 | CN1662505A Quinoline derivatives as caspase-3 inhibitor, preparation for producing the same and pharmaceutical composition comprising the same |
08/31/2005 | CN1662504A 2, 5-disubstituted 3-mercaptopentanoic acid |
08/31/2005 | CN1662498A Novel tetrahydropyridine derivatives as renin inhibitors |
08/31/2005 | CN1662496A Cannabinoid receptor agonists |
08/31/2005 | CN1662236A Inhibitors of histone deacetylase |
08/31/2005 | CN1660841A Itraconazole hydrochloride, oral solid combination and preparation method |
08/31/2005 | CN1660839A Chemical compounds |
08/31/2005 | CN1660821A Oxodiethylenediamine derivative and light stabilized composition |
08/31/2005 | CN1660818A Process for the manufacture of organic compounds |
08/31/2005 | CN1660815A Cyclic amine derivatives and their use as drugs |
08/31/2005 | CN1660811A Compound of 1, 4-substituted benzenes and preparing method and application |
08/30/2005 | US6936720 Method for preparing benzisoxazole methane sulfonyl chloride and its amidation to form zonisamide |
08/30/2005 | US6936633 Pyrrolidinone derivatives |
08/30/2005 | US6936626 Retinoic acid mimetic anilides |
08/30/2005 | US6936616 Pyrimidine matrix metalloproteinase inhibitors |
08/30/2005 | US6936613 for treatment of central nervous system diseases and disorders, which are responsive to modulation of the Gamma amminobutyric acid (GABA) receptor complex, and for inducing and maintaining anesthesia, sedation and muscle relaxation |
08/30/2005 | US6936610 Heterocyclic derivatives |
08/30/2005 | US6936602 Benzazepine derivatives, process for the preparation of the same and uses thereof |
08/30/2005 | US6936600 Oxidoreductase enzyme inhibitors such as (R)-1-[4-(2-methyl-4-phenyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-pyrimidin-2-yl-ethanol, used as antidiabetic agents |
08/30/2005 | US6936325 Optical recording medium |
08/30/2005 | CA2133152C Piperidines and piperazines with affinity for 5-ht receptors |
08/25/2005 | WO2005077944A1 Pyrimidine derivatives for use as vanilloid receptor ligands and their use in the treatment of pain |
08/25/2005 | WO2005077943A1 1 , 3 - dioxane derivatives and analogues thereof useful in the treatment of i.a. obesity and diabetes |
08/25/2005 | WO2005077942A1 Process for preparing substituted benzopyran compounds |
08/25/2005 | WO2005077940A1 Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof |
08/25/2005 | WO2005077937A1 Substituted hydroxamic acid derivatives as tnf inhibitors |
08/25/2005 | WO2005077932A2 Chemokine receptor antagonists |
08/25/2005 | WO2005077922A2 Process for the preparation of substituted triazole compounds |
08/25/2005 | WO2005077918A1 Pth agonists |
08/25/2005 | WO2005077915A1 Pyridazinones as antagonists of a4 integrins |
08/25/2005 | WO2005077914A1 PYRIDAZINONE UREAS AS ANTAGONISTS OF α4 INTEGRINS |
08/25/2005 | WO2005077900A1 Bicyclic amide derivatives |
08/25/2005 | WO2005077896A1 Substituted azetidine compounds as cyclooxygenase-1-cyclooxygenase-2 inhibitors, and their preparation and use as medicaments |
08/25/2005 | WO2005077463A2 Ligand for a monoamine receptor or transporter for treating addiction or dependence |
08/25/2005 | WO2005077361A1 Novel, sustained-action beta-2-agonists and their use as medicaments |
08/25/2005 | WO2005077344A2 Hydantoin derivatives as inhibitors of cellular necrosis |
08/25/2005 | US20050187390 Bicyclic heteroaryl derivatives |
08/25/2005 | US20050187387 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor |
08/25/2005 | US20050187291 use of 2-(urea or thiourea)tetralins as analgesic or to treat pulmonary dysfunction |
08/25/2005 | US20050187284 Integrin receptor inhibitors |
08/25/2005 | US20050187279 Indazole derivatives useful for the treatment of eating disorders, weight gain, obesity, abnormalities in reproduction and sexual behavior, thyroid hormone secretion, diuresis and water/electrolyte homeostasis, sensory processing, memory, sleeping, arousal, anxiety, depression, seizure etc. |
08/25/2005 | US20050187275 Preterm labor, premature birth, dysmenorrhea, inappropriate secretion of vasopressin, congestive heart failure, arterial hypertension, liver cirrhosis, nephrotic syndrome and ocular hypertension; 3-(5-((3-chlorobenzyl)sulfanyl)-4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl)-N-(2-methoxybenzyl)propanamide |
08/25/2005 | US20050187272 Enzyme inhibitor on NO-synthase enzymes; treating STROKE, NEURODEGENERATIVE DISEASES, preventing ISCHEMIC OR HEMORRAGIC CARDIAC OR CEREBRAL INFARCTIONS; inhibiting lipidic peroxidation |
08/25/2005 | US20050187270 16-Halogen-epothilone derivatives, method for producing them and their pharmaceutical use |
08/25/2005 | US20050187266 2-Methyl-2-{3-[({[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]carbonyl}amino)methyl]phenoxy}propanoic acid; polycystic ovarian syndrome; polycystic obesity; dietetics; hypoglycemic agents; antilipemic and - cholesterol agents; hypertriglyceridemia; insulin resistance; metabolic disorders; PPAR modulators |
08/25/2005 | US20050187264 2-Cyano-N-[4-(methoxymethoxy)phenethyl]-3-(3-pyridyl)-2-propenamide: generic derivatives described in WO 99/05109; asthma; bronchitis; rhinitis; vision defects; antiarthritic agents; antiallergens; sepsis; inflammatory bowel disease; bipolar disordes; schizophrenia; Crohn's disease; degenerative joints |
08/25/2005 | US20050187261 For hepatitis C; histone deacetylase inhibitors, anticarcinogenic agents; N-hydroxy-4-{[(benzofuran-, benzothiophen-, or indol-)-2-ylcarbonylamino]alkoxy}benzamides; amidation of a benzoic acid, benzoate, benzoyl halide with hydroxyamine |
08/25/2005 | US20050187257 Methods of treating sepsis |
08/25/2005 | US20050187238 Benzofuran derivatives, their production and use |
08/25/2005 | US20050187236 Nitrogen-containing aromatic derivatives |
08/25/2005 | US20050187231 4-aminoquinazolines e.g. 4-(4-phenylbutylamino)quinazoline; antiproliferative agents; antitumor agents; hyperproliferative disorders, including tumors, such as breast, brain, and kidney tumors |
08/25/2005 | US20050187222 Therapy for impotency, erectile dysfuction; benign prostatic hyperplasia; hypotensive agents; congestive heart failure; vision defects; neurodegenerative disorders; incotinence; cognition activators |
08/25/2005 | US20050187217 Sodium channel modulators; pain relievers; treating epilepsy, neurodegenerative disorders, psychiatric disorders, arrhythmia, movement disorders, autoimmune diseases, and incontinence; fused ring 4-aminopyrimidines e.g. 4-amino-5,6,7,8-tetrahydroquinazolines |
08/25/2005 | US20050186630 Extended tethering approach for rapid identification of ligands |
08/25/2005 | CA2556398A1 Substituted azetidine compounds as cyclooxygenase-1-cyclooxygenase-2 inhibitors, and their preparation and use as medicaments |
08/25/2005 | CA2555825A1 Process for the preparation of substituted triazole compounds |
08/25/2005 | CA2555817A1 1 , 3 - dioxane derivatives and analogues thereof useful in the treatment of i.a. obesity and diabetes |
08/25/2005 | CA2555685A1 Pyrimidine derivatives for use as vanilloid receptor ligands and their use in the treatment of pain |
08/25/2005 | CA2555594A1 Pyridazinones as antagonists of a4 integrins |
08/25/2005 | CA2555227A1 Pyridazinone ureas as antagonists of .alpha.4 integrins |
08/25/2005 | CA2554378A1 Bicycloamide derivative |
08/25/2005 | CA2553630A1 Dehydrophenylahistins and analogs thereof and the synthesis of dehydrophenylahistins and analogs thereof |
08/25/2005 | CA2552871A1 Novel, sustained-action beta-2-agonists and their use as medicaments |
08/25/2005 | CA2536622A1 Inhibitors of cellular necrosis |