Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
01/2006
01/31/2006CA2119261C Novel sidechain-bearing taxanes and intermediates thereof
01/26/2006WO2006010095A2 Oxime derivative substituted hydroxyethylamine aspartyl protease inhibitors
01/26/2006WO2006009653A1 Amino-5,5-diphenylimidazolone derivatives for the inhibition of beta-secretase
01/26/2006WO2006008644A1 Antidiabetic compounds
01/26/2006WO2005116009B1 Substituted 2-quinolyl-oxazoles useful as pde4 inhibitors
01/26/2006WO2005111020A3 Pyrimidine hydantoin analogues which inhibit leukocyte adhesion mediated by vla-4
01/26/2006WO2005097134A3 Quinazoline based protein kinase inhibitors
01/26/2006WO2005085234A3 Bycyclic anthranilamide derivatives useful as insecticides
01/26/2006WO2005077922A3 Process for the preparation of substituted triazole compounds
01/26/2006WO2005077463A3 Ligand for a monoamine receptor or transporter for treating addiction or dependence
01/26/2006WO2005069981A3 Method of preparation of benzofuran-2-carboxylic acid {(s)-3-methyl-1-[(4s, 7r)-7methyl-3-oxo-1-(pyridine-2-sulfonyl)-azepan-4-ylcarbamoyl]-butyl}-amide
01/26/2006WO2004096798A3 Derivatives of 2-acylamino-4-phenylthiazole, preparation method thereof and use of same as chemokine antagonists
01/26/2006US20060020138 E.g., 3-arylmethyl-7-hydroxy-coumarins as intermediates; affects both the Tumor Necrosis Factor alpha level and transcription activity of NuclearFactor kappa Beta; antiimmunoinflammatory agents and autoimmune properties; antiarthritis agents; rheummatic diseases; osteoporosis; leukemia
01/26/2006US20060020133 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
01/26/2006US20060020016 5-Ethoxy-4-(1-(benzyloxycarbonyl)-2-pyrrolidinylcarbonylamino)-5H-furan-2-one; purification by chromatography, selectively crystallization, or dynamic crystallization; useful for preparing caspase inhibitors
01/26/2006US20060020012 Pyrazole derivatives
01/26/2006US20060020011 Diseases mediated by tachykinins and for seritonin reuptake transporter protein as reuptake inhibitors
01/26/2006US20060020008 Compounds, compositions and methods
01/26/2006US20060020003 Biphenyloxy-acids
01/26/2006US20060019996 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
01/26/2006US20060019974 4-Amino-quinazolines
01/26/2006US20060019953 Pyridine inhibitors of ERK2 and uses thereof
01/26/2006US20060019948 Methylidene-D-xylopyranosyl- and oxo-D-xylopyranosyl-substituted phenyl derivatives, medicaments containing such compounds, their use and process for their manufacture
01/26/2006US20060019947 Therapeutic chromone compounds
01/26/2006US20060019906 Useful as an anti-HIV agent that particularly shows an anti-HIV action based on an integrase inhibitory activity; for treatment or prophylaxis of AIDS; for example, 6-(2,3-dichlorobenzyl)-1-(2-hydroxyethyl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
01/26/2006US20060019831 1-(3-trifluoromethyl)phenyl-3-(N-methyl)carboxamido-2-pyrrolidinone; herbicides; high compatibility with crop plants is desirable; no adverse effect on the chlorophyll synthesis in crop plants; crop protection compositions
01/26/2006US20060018846 Animo substituted hydroxyphenyl benzophenone derivatives
01/26/2006DE10223908B4 Verfahren zur Herstellung von substituierten Pyridinen A process for the preparation of substituted pyridines
01/26/2006CA2579724A1 Amino-5,5-diphenylimidazolone derivatives for the inhibition of beta-secretase
01/26/2006CA2574217A1 Diamine derivative, process of preparation thereof, and fungicide comprising diamine derivative as an active ingredient
01/26/2006CA2573210A1 Viral polymerase inhibitors
01/26/2006CA2573138A1 Oxime derivative substituted hydroxyethylamine aspartyl protease inhibitors
01/25/2006EP1619183A2 1-amido-3-(2-hydroxyphenoxy)-2-propanol derivatives and a process for preparing 2-amidomethyl-1, 4-benzodioxane derivatives
01/25/2006EP1618105A1 Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disorders
01/25/2006EP1618094A1 Substituted heteroaryls as inhibitors of protein tyrosine phosphatases
01/25/2006EP1618093A2 Indazole derivatives as jnk inhibitors
01/25/2006EP1618092A1 Aryl-substituted pyrazole-amide compounds useful as kinase inhibitors
01/25/2006EP1617841A1 Amino cyclobutylamide modulators of chemokine receptor activity
01/25/2006EP1617840A2 Pyrazole-amide compounds useful as kinase inhibitors
01/25/2006EP1617807A2 Substituted 1,4-diazepines and uses thereof
01/25/2006EP1495040A4 Method for synthesizing beta-l-fluoro-2',3'didehydcytidine (beta-l-fd4c)
01/25/2006CN1726211A Imidazole deriviatives and their use as peripherally-selective inhibitors of dopamine-beta-hydroxylase
01/25/2006CN1726207A Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivatives and their use as neurokinin antagonists
01/25/2006CN1726205A 2-substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators
01/25/2006CN1726201A Substituted piperazines,(1,4) diaszepines, and 2,5-diazabicyclo (2.2.1)iieptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists
01/25/2006CN1726196A Pyrazine-based tubulin inhibitors
01/25/2006CN1726194A Novel compounds
01/25/2006CN1724521A New quinazoline hind derivative, medicinal composition containing same and their use
01/25/2006CN1238353C Amino acid ester containing azole antifungal agent
01/25/2006CN1238347C Heterocyclic derivatives
01/25/2006CN1238343C Pyrimidine derivatives and herbicides containing the same
01/24/2006US6989452 Anticancer agents
01/24/2006US6989449 Containing nitroxide or hydroxylamine moieties; use stabilizing pulp or paper against yellowing and discoloration due to light
01/24/2006US6989398 Benzanilides as potassium channel openers
01/24/2006US6989397 Iron chelators and uses thereof
01/24/2006US6989395 TNF inhibitors
01/24/2006US6989392 2-Aminoquinolines as melanin concentrating hormone receptor antagonists
01/24/2006US6989385 Pyrazole compounds useful as protein kinase inhibitors
01/24/2006US6989384 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
01/24/2006CA2292984C Ccr5 modulators
01/24/2006CA2205757C Pyridazinone derivatives and their use as inhibitors of prostaglandin g/h synthase i and ii(cox i and ii)
01/24/2006CA2191832C Block oligomers containing 2,2,6,6-tetramethyl-4-piperidyl groups as stabilizers for organic materials
01/19/2006WO2006006573A1 Filter and cyanine compound
01/19/2006WO2006005915A1 2, 4, 6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer
01/19/2006WO2005115981A3 A process for the preparation of 1-(9h-carbazol-4-yloxy)-3-2-(-methoxyphenoxy)-ethyl amino-propan-2-ol
01/19/2006WO2005113514A3 Substituted pyrimidines as inhibitors of bacterial type iii protein secretion systems
01/19/2006WO2005097746A3 2-propene-1-ones as hsp 70 inducers
01/19/2006WO2005095357A3 Pyrimidine derivatives and methods of treatment related to the use thereof
01/19/2006WO2005092307A3 Pharmaceutical dosage forms and compositions of 5-ht1a receptor antagonists
01/19/2006WO2005075458A8 Pyrimidine derivatives as orexin receptors antagonists
01/19/2006US20060014950 Combining a strong base with a phenyl isonicotinamide in aprotic solvents to form a solutions, then reacting with a cyclohexanone carboxylic acid or ester and water, and acidifying the solution to obtain chemical intermediates for neuropeptide Y antagonists used for treating bulimia, obesity or diabetes
01/19/2006US20060014948 e.g 1-[3,5-bis(trifluoromethyl)benzoyl]-2-[3-[(2-methoxyethoxy)-methoxy]-4-methylbenzyl]-4-[2-[(3R)-3-methoxymethyl-morpholino]ethyl]piperazine; treating or preventing Tachykinin-mediated diseases in humans or animals
01/19/2006US20060014836 e.g. 1-(Benzofuran-2-carbonyl-3-(3-phenoxy-phenyl)-thiourea;viricides; hepatitis virus
01/19/2006US20060014827 3-(Cyclopenten-1-yl)-benzyl-or 3-(cyclopenten-1-yl)-heteroarylmethyl-amine derivatives and use thereof as medicines for treating schizophrenia
01/19/2006US20060014817 CCK-1 receptor modulators
01/19/2006US20060014796 Epothilone derivatives
01/19/2006US20060014792 Heterocyclo inhibitors of potassium channel function
01/19/2006US20060014789 Phenyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatment of pain or gastrointestinal disorders
01/19/2006US20060014787 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
01/19/2006US20060014785 Bicyclic, substituted triazoles as modulators of ppar and methods of their preparation
01/19/2006US20060014780 Nicotinamide derivatives useful as PDE4 inhibitors
01/19/2006US20060014768 Antiproliferative, anticancer, antitumor agents; rheumatism; N-{3-[3-cyclopropyl-5-(2-fluoro-4-iodo-phenylamino)-6,8-dimethyl-2,4,7-trioxo-3,4,6,7-tetrahydro-2H-pyrido[4,3-d]pyrimidin-1-yl]-phenyl}-acetamide; a p15, and/or a protein inducing action, and/or an MEK inhibitory action; side effect reduction
01/19/2006US20060014756 Benzimidazoles
01/19/2006US20060014755 17 Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
01/19/2006US20060014749 (R)-2-{4-[(1H-Indol-2-ylmethyl)-amino]-piperidin-1-yl}-1-(6-methoxyquinolin-4-yl)-ethanol; effective against both gramnegative and grampositive bacteria
01/19/2006US20060014747 Ortho-substituted anthranilic acid amides and their use as pharmaceutical agents
01/19/2006US20060013860 Anticancer agents; side effect reduction
01/19/2006DE19748440B4 6,7-Difluor-1,2,3,4-tetrahydronaphthalin-Derivate und ihre Verwendung in flüssigkristallinen Mischungen, diese enthaltende Flüssigkristallmischungen sowie ferroelektrische Schalt- und/oder Anzeigevorrichtungen 6,7-difluoro-1,2,3,4-tetrahydronaphthalene derivatives and their use in liquid crystalline mixtures, liquid crystal mixtures containing them, as well as ferroelectric switching and / or display devices
01/19/2006DE102004031323A1 Substituierte Pyridazincarboxamide und Derivate hiervon And derivatives thereof substituted Pyridazincarboxamide
01/19/2006DE102004023332A1 Chinoxalin-2-on-derivate, diese enthaltende nutzpflanzenschützende Mittel und Verfahren zu ihrer Herstellung und deren Verwendung Quinoxalin-2-one derivatives, useful-plant-protecting compositions containing them and processes for their preparation and their use
01/19/2006CA2571750A1 2, 4, 6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer
01/18/2006EP1616569A1 Medicinal composition
01/18/2006EP1615914A2 Cgrp receptor antagonists
01/18/2006EP1615909A1 Piperazine derivatives and their use for the treatment of neurological and psychiatric diseases
01/18/2006EP1615906A1 Compositions useful as inhibitors of protein kinases
01/18/2006EP1615905A2 Benzopyran compounds useful for treating inflammatory conditions
01/18/2006EP1615899A1 Alpha-substituted carboxylic acids as ppar modulators
01/18/2006EP1615894A2 3-azabicyclo 3.2.1 octane derivatives
01/18/2006EP1615890A1 Piperidine derivatives as renin inhibitors for the treatment of hypertension
01/18/2006EP1615889A2 Biphenyl derivatives having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity