Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
04/2006
04/11/2006US7026349 Sulfonamides
04/11/2006US7026346 Anticancer agents
04/11/2006US7026336 4-pyridinylimidazol-2-ylhydrocarbyl amine, (thio)urea, carbamic acid or sulfonamide derivatives, e.g., (2-(4-(4-Chloro-3-methoxy-phenyl)-5-pyridin-4-yl-1H-imidazol-2-yl)-2-methyl-propyl)-carbamic acid tert-butyl ester; Raf kinase inhibitors for the treatment of neurotraumatic diseases
04/11/2006US7026325 pyrazinoylguanidine compounds, e.g., 4-{4-[N-(3,5-diamino-6-chloropyrazine-2-carbonyl)guanidino]butyl}-N-(2-aminoethyl)benzamide hydrochloride; are absorbed less rapidly from mucosal surfaces, especially airway surfaces; rehydration of mucosal surfaces; reducing blood pressure
04/11/2006US7026324 Amide containing a pyridinone or pyrazinone compound as serine protease enzyme inhibitors
04/11/2006US7026323 N-(naphth-2-ylaminocarbonylacetyl)- or N-(naphth-2-ylcarbonylamino- acetyl)- piperazine derivatives, e.g., 2-[((4-(ethoxycarbonyl)piperazin-1-yl)carbonylmethyl)carbonyl]aminonaphthalene; useful as antithrombotic agents
04/11/2006US7026320 Serotonergic agents
04/11/2006US7026314 Psychological disorders, antidepressants, anxiolytic agents, eating disorders; serotonin receptors antagonist
04/11/2006CA2281702C (4-piperidinyl)-1h-2-benzopyran derivatives useful as antipsychotic agents
04/11/2006CA2199117C Compounds and methods for the treatment of cancer
04/11/2006CA2187030C Improved anti-dandruff shampoo
04/06/2006WO2006037117A1 Substituted heterocyclic compounds and methods of use
04/06/2006WO2006036994A2 Modulators of crth2, cox-2 and faah
04/06/2006WO2006036527A1 Substituted dipiperdine ccr2 antagonists
04/06/2006WO2006036507A1 4-(heteroaryl-methyl and substituted heteroaryl-methyl)-imidazole-2-thiones acting as alpha2 adrenergic agonists
04/06/2006WO2006036497A2 4-(condensed cyclicmethyl)-imidazole-2-thiones acting as alpha2 adrenergic agonists
04/06/2006WO2006036404A1 4-(substituted cycloalkylmethyl) imidazole-2-thones, 4-(substituted cycloalkenylmethyl) imidazole-2-thiones, 4-(substituted cyloalkylmethyl) imidazol-2-ones, 4-(substituted cycloalkenylmethyl) imidazol-2-ones and related compounds
04/06/2006WO2006036024A1 Proton pump inhibitors
04/06/2006WO2006035770A1 Process for synthesis of derivatives, compound library, method for making the mase, and screening method
04/06/2006WO2006035303A1 Muscarinic receptor antagonists
04/06/2006WO2006035068A2 Hiv inhibiting 5-carbo- or heterocyclic substituted pyrimidines
04/06/2006WO2006035067A2 Hiv inhibiting 5-heterocyclyl pyrimidines
04/06/2006WO2005102335A3 Methods of treating sleep disorders
04/06/2006US20060074245 Reacting a 5-( beta -ketoalkyl)-3-substituted-1,2,4-oxadiazoles compound with hydrazine
04/06/2006US20060074244 Pyridinyl substituted (1,2,3,)triazoles as inhibitors of the tgf-beta signalling pathway
04/06/2006US20060074243 Hydroxamic acid and amide compounds and their use as protease inhibitors
04/06/2006US20060074238 Asymmetric process for the preparation of diarylethylpiperazines derivatives and novel asymmetric diarylmethylamines as intermediates
04/06/2006US20060074128 Substituted 2-phenyl benzofurans as estrogenic agents
04/06/2006US20060074123 Cyclic AMP-specific phosphodiesterase inhibitors
04/06/2006US20060074122 e.g., N-butyl-6-chloro-5-phenyl-1H-indazol-3-amine; kinase inhibitor; obesity and stroke; diseases involving phosphorylation of the tau protein such as Alzheimer's disease, Parkinson's disease, frontoparietal dementia
04/06/2006US20060074116 3-(Heteroarylamino)methylene-1, 3-dihydro-2H-indol-2-ones as kinase inhibitors
04/06/2006US20060074112 N-aryl (thio) anthranilic acid amide derivatives, their preparation and their use as VEGF receptor tyrosine kinase inhibitors
04/06/2006US20060074096 anti-cell prolifertive agents; 4-(1,2-diethylimidazol-5-yl)-2-{4-[N-(2-ethoxyethyl)sulphamoyl]anilino}pyrimidine; cancers, solid tumours, leukemias, psoriasis, rheumatoid arthritis, Kaposi's sarcoma, hemangioma, nephropathies, atheroma, atherosclerosis, restenosis, autoimmune diseases, inflammation
04/06/2006US20060074084 Inhibitors of soluble adenylate cyclase
04/06/2006US20060074083 Cyclic and acyclic propenones for treating CNS disorders
04/06/2006US20060074069 e.g. (2R-trans) [4-(4-azetidin-3-yl-piperazin-1-yl)-2-benzyl-piperidin-1-yl]-(3,5-bis-trifluoromethyl-phenyl)-methanone;tachykinins, substance P inhibitor; antidepressant, anxiolytic, antiinflammatory agent, cognition activator; neurodegenerative diseases; addiction, sleep, eating disorders
04/06/2006US20060074068 Chemical compounds with dual activity, processes for their preparation and pharmaceutical compositions
04/06/2006CA2582777A1 Proton pump inhibitors
04/06/2006CA2582225A1 Substituted dipiperdine ccr2 antagonists
04/06/2006CA2581828A1 4-(heteroaryl-methyl and substituted heteroaryl-methyl)-imidazole-2-thiones acting as alpha2 adrenergic agonists
04/06/2006CA2581823A1 4-(condensed cyclicmethyl)-imidazole-2-thiones acting as alpha2 adrenergic agonists
04/06/2006CA2581375A1 Specific kinase inhibitors
04/06/2006CA2581254A1 Method for synthesizing derivative, compound library and method for constructing the same, and method for screening
04/06/2006CA2580838A1 Substituted heterocyclic compounds and methods of use
04/06/2006CA2577467A1 Hiv inhibiting 5-heterocyclyl pyrimidines
04/06/2006CA2573976A1 Hiv inhibiting 5-carbo- or heterocyclic substituted pyrimidines
04/05/2006EP1642895A2 Novel substituted naphthopyrans
04/05/2006EP1641785A2 Benzofuranyl-and benzothienyl-piperazinyl quinolines as serotonin reuptake inhibitors
04/05/2006EP1641784A1 4-(aminomethyl)-piperidine benzamides as 5ht4 -antagonists
04/05/2006EP1641783A1 Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists
04/05/2006EP1641782A1 Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists
04/05/2006EP1641780A1 Processes for the preparation of 1- [(benzoimidazole-1yl) quinolin-8-yl] piperidin-4-ylamine derivatives
04/05/2006EP1641764A1 5-membered heterocycle-based p38 kinase inhibitors
04/05/2006EP1641762A2 Cck-1 receptor modulators
04/05/2006EP1641758A2 Diphenylpyridine derivatives, preparation and therapeutic application thereof
04/05/2006EP1300398B1 Propane-1,3-dione derivatives
04/05/2006EP1140846B1 Aspartic protease inhibitors
04/05/2006EP1140192B1 Use of the cyclooxygenase-2 inhibitor celecoxib and capecitabine for combination therapy in neoplasia
04/05/2006EP1019372B1 Fused pyrrolecarboxamides; a new class of gaba brain receptor ligands
04/05/2006CN1756756A Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholesterolemia
04/05/2006CN1756755A Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholesterolemia
04/05/2006CN1756754A Arylvinylazacycloalkane compounds and methods of preparation and use thereof
04/05/2006CN1756753A Benzofuran derivative
04/05/2006CN1756746A 6-substituted nicotinamide derivatives as opioid receptor antagonists
04/05/2006CN1754880A Process for preparing 2-iminopyrrolidine derivatives
04/05/2006CN1249058C Perfluoroalkyl-containing complexes with sugar radicals, process for their production and their use
04/05/2006CN1249057C Chromenylmethyl pyrimidinediamines as antibacterial agents
04/05/2006CN1249052C Pyrazole derivatives as HIV reverse transcriptase inhibitors
04/05/2006CN1249051C Muscarinic agonists
04/05/2006CN1249044C Chromanone derivatives
04/05/2006CN1249043C New heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them
04/05/2006CN1249036C Iron chelators and use thereof
04/04/2006US7022733 Estrogen receptor modulators for treating or inhibiting endometriosis
04/04/2006US7022732 6-substituted 2,3-dihydro-1,4-benzodioxine, 2-position substituted with carboxy, or (C1 C6)alkoxycarbonyl; diabetes, obesity; 6-[2-(R)-[2-(S)-hydroxy-3-(4-hydroxy-3-methanesulfonamido-phenoxy)propylamino]propyl]-2,3-dihydro-1,4-benzodioxine-2-(R)-carboxylic acid; B3 andrenergic receptor agonist
04/04/2006US7022731 Cardiovascular disorders; thrombosis; anticoagulants
04/04/2006US7022730 Protein tyrosine phosphatases inhibitors
04/04/2006US7022723 Heterocyclic compounds
04/04/2006US7022718 Pyridine and pyrimidine derivatives
04/04/2006US7022716 Cyclic amine phenyl beta-3 adrenergic receptor agonists
04/04/2006US7022715 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
04/04/2006US7022707 such as S-4-[(2-propylamino)carbonyl]oxybenzyl piperazine-1-thiocarboxylate for treatment of obesity and/or diabetes
04/04/2006US7022696 Treatment of airway disorders
04/04/2006US7022492 Ecstasy haptens and immunogens
04/04/2006CA2256492C Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
04/04/2006CA2241787C Substituted aza- and diazacycloheptane and cyclooctane compounds and their use
04/04/2006CA2235133C Esters of 3-hydroxy-piperidinemethanol derivatives
04/04/2006CA2198266C Novel benzimidazole derivatives
04/04/2006CA2193039C Indol-2-one derivatives
04/04/2006CA2166315C Process for the preparation of thalidomide
04/04/2006CA2043976C Substituted phthalides and heterocyclic phthalides
03/2006
03/30/2006WO2006034234A1 Crystalline form 3 of atrasentan hydrochloride
03/30/2006WO2006034116A1 Diaminotriazole compounds useful as protein kinase inhibitors
03/30/2006WO2006034094A1 Crystalline form 1 of atrasentan hxdrochloride
03/30/2006WO2006034085A1 Crystalline form of atrasentan hydrochloride
03/30/2006WO2006034084A1 Crystalline form 2 of atrasentan hydrochloride
03/30/2006WO2006033631A1 Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof i
03/30/2006WO2006033630A1 Compounds, compositions containing them, preparation thereof and uses thereof iii
03/30/2006WO2006033627A1 Compounds, compositions containing them, preparation thereof and uses thereof iiii
03/30/2006WO2006033620A1 New heterocyclic amides
03/30/2006WO2006033002A1 4-amino substituted-2-substituted-1,2,3,4-tetrahydroquinoline compounds