Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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12/21/2005 | EP1606267A1 Pyrazine compounds as transforming growth factor (tgf) inhibitors |
12/21/2005 | EP1606266A2 Chemical compounds |
12/21/2005 | EP1606265A1 2, 4- di (phenylamino) pyrimidines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders |
12/21/2005 | EP1606255A2 Cyclic derivatives as modulators of chemokine receptor activity |
12/21/2005 | EP1606251A2 Inhibitors of the binding of chemokines i-tac or sdf-1 to the ccxckr2 receptor |
12/21/2005 | EP1558582B1 Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of disorders related thereto |
12/21/2005 | EP1432701B1 Heterocyclic compounds for use in the treatment of disorders of the urinary tract |
12/21/2005 | EP1395558B1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders |
12/21/2005 | EP1395555B1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derativatives and their use for the treatment of pain, anxiety or gastrointestinal disorders |
12/21/2005 | EP1363897B1 Antagonists of mcp-1 function and methods of use thereof |
12/21/2005 | EP1362039B1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands |
12/21/2005 | EP1307445B1 Benzofuran derivatives and their use as antibacterial agents |
12/21/2005 | EP1178973B1 Pyrazinyl-piperazine- compounds, their use and preparation |
12/21/2005 | CN1711249A Quinazolinone derivatives useful as anti-hyperalgesic agents |
12/21/2005 | CN1711081A Proline derivatives having affinity for the calcium channel alpha-2-delta subunit |
12/21/2005 | CN1232519C Method for producing 5-(1-piperazinyl)-benzofuran-2-carboxamide by transition metal-catalyzed amination |
12/21/2005 | CN1232518C Bi-heterocyclic compounds with antitumour and chemosensitising activity |
12/21/2005 | CN1232509C Novel diamino pyrazole derivatives and dyes containing said compounds |
12/21/2005 | CN1232505C Substituted sulfamide (thio) carbonyl compounds |
12/20/2005 | US6977268 Diacid isoindoleine amide derivative |
12/20/2005 | US6977266 Pyridone derivatives having affinity for cannabinoid 2-type receptor |
12/20/2005 | US6977264 For therapy and prophylaxis of obesity, diabetes |
12/20/2005 | US6977263 Chemical compounds |
12/20/2005 | US6977258 Antiinflammatory agents; cardiotonic agents; rheumatic diseases |
12/20/2005 | CA2338206C High affinity ligands for nociceptin receptor orl-1 |
12/20/2005 | CA2324324C Treatment of pulmonary hypertension |
12/20/2005 | CA2233560C Sulfonamide inhibitors of matrix metalloproteinases |
12/20/2005 | CA2176962C N-substituted azabicycloheptane derivatives, their preparation and use |
12/20/2005 | CA2114007C Substituted beta-lactam compounds useful as hypocholesterolemic agents and processes for the preparation thereof |
12/15/2005 | WO2005118577A1 Novel saperconazole crystalline forms and related processes, pharmaceutical compositions and methods |
12/15/2005 | WO2005118576A1 Constrained himbacine analogs as thrombin receptor antagonists |
12/15/2005 | WO2005118575A1 Non nucleoside reverse transcriptase inhibitors |
12/15/2005 | WO2005118574A1 Mercaptoimidazoles as ccr2 receptor antagonists |
12/15/2005 | WO2005118556A1 Propane-1,3-dione derivative or its salt |
12/15/2005 | WO2005118547A1 Tetrahydroisoquinoline sulfonamide derivatives, the preparation thereof, and the use of the same in therapeutics |
12/15/2005 | WO2005118544A2 Cycloalkyl substituted pyrimidinediamine compounds and their uses |
12/15/2005 | WO2005118543A1 Kinase inhibitor and use thereof |
12/15/2005 | WO2005118535A1 Substituted pyrrolidine-2-ones |
12/15/2005 | WO2005118531A1 Aminomethyl-azacycle derivatives as inhibitors of monoamine uptake |
12/15/2005 | WO2005117908A2 Triheterocyclic compounds compositions, and methods for treating cancer or viral diseases |
12/15/2005 | WO2005117894A1 Leptomycin compounds |
12/15/2005 | WO2005117882A2 Hydroxamic acid derivatives as metalloprotease inhibitors |
12/15/2005 | WO2005117876A1 Dual small molecule inhibitors of cancer and angiogenesis |
12/15/2005 | WO2005087751A3 Substituted hydroxyethylamine aspartyl protease inhibitors |
12/15/2005 | US20050277685 peroxisome proliferator activated receptor agonist such as (2R)-2-(3-{[3-(4-chlorophenoxy)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl}phenoxy)butanoic acid, used for treatment and control of metabilic disorders |
12/15/2005 | US20050277673 such as 4-{[4-({[(3-isopropyl-2-oxo-2,3-dihydro-1H-benzimidazol-1-yl)carbonyl]amino}methyl)piperidin-1-yl]methyl}tetrahydro-2H-pyran-4-carboxylic acid; serotonin receptor agonist; antidepressant, anxiolytic agent, analgesic, cognition activator; less toxicity, good absorption, and metabolic stability |
12/15/2005 | US20050277672 such as 1-{[4-({[(3-isopropyl-2-oxo-2,3-dihydro-1H-benzimidazol-1-yl)carbonyl]amino}methyl)piperidin-1-yl]methyl}cyclopentanecarboxylic acid; serotonin receptor agonist; antidepressant, anxiolytic agent, analgesic, cognition activator; less toxicity, good absorption, and metabolic stability |
12/15/2005 | US20050277671 Benzimidazolone carboxylic acid derivatives |
12/15/2005 | US20050277669 Preparation of paroxetine involving novel intermediates |
12/15/2005 | US20050277663 3-Aryl-3-hydroxy-and 3-aryl-3-oxopropionic acid esters as fungicides |
12/15/2005 | US20050277660 Novel tetrahydroquinoline derivatives |
12/15/2005 | US20050277658 Such as aurora-2 kinase or c-kit kinase; anticancer agents; based on benzo(4,5)furo(3,2-d)pyrimidine, 9-thia-1,5,7-triazafluorene, or pyrimido(5,4-b)indole rings; e.g. 6,7-dimethoxy-4-(4-(benzodioxol-5-ylmethylaminothiocarbonyl)-piperazin-1-yl)-5H-Pyrimido(5,4-b)indole |
12/15/2005 | US20050277654 4,5-Disubstituted-2-aryl pyrimidines |
12/15/2005 | US20050277653 Compositions and treatments for inhibiting kinase and/or HMG-CoA reductase |
12/15/2005 | US20050277646 N-[4-({5-(4-fluorophenyl)-4-[4-(trifluoromethyl)phenyl]pyridin-2-yl}oxy)-1,3-benzothiazol-2-yl]acetamide; vanilloid (capsaicin) receptor antagonist/agonist; antiinflammatory, analgesic, antiarthritis, antirheumatic; diseases involving sensory nerve function |
12/15/2005 | US20050277642 Pyrimidine kinase inhibitors |
12/15/2005 | US20050277640 Pyrimidine derivatives for treatment of hyperproliferative disorders |
12/15/2005 | US20050277638 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor |
12/15/2005 | US20050277637 Arylindenopyridines and related therapeutic and prophylactic methods |
12/15/2005 | US20050277631 Vanilloid receptor ligands and their use in treatments |
12/15/2005 | DE102004025791A1 Chromanol-Derivate, ein Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer Chromanol derivatives, a process for their preparation and their use as anti-inflammatories |
12/15/2005 | CA2568622A1 Dual small molecule inhibitors of cancer and angiogenesis |
12/15/2005 | CA2568341A1 Leptomycin compounds |
12/15/2005 | CA2566531A1 Cycloalkyl substituted pyrimidinediamine compounds and their uses |
12/15/2005 | CA2565689A1 Substituted pyrrolidine-2-ones |
12/15/2005 | CA2565280A1 Mercaptoimidazoles as ccr2 receptor antagonists |
12/14/2005 | EP1604979A1 2-oxo-1-pyrrolidine derivative and its pharmaceutical uses |
12/14/2005 | EP1603912A1 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators |
12/14/2005 | EP1603911A1 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators |
12/14/2005 | EP1603906A2 Process for synthesising useful intermediates for the preparation of alpha v beta 3 receptor antagonists |
12/14/2005 | EP1603901A1 Tetrahydropyran compounds as tachykinin antagonists |
12/14/2005 | EP1603897A1 Pyrazole compounds useful in the treatment of inflammation |
12/14/2005 | EP1603893A1 Ep4 receptor antagonists |
12/14/2005 | EP1603886A1 4-substituted-5-cyano-1h-pyrimidin-6-(thi)ones as gsk-3 inhibitors |
12/14/2005 | EP1603885A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors |
12/14/2005 | EP1603883A2 Quinoline-derived amide modulators of vanilloid vr1 receptor |
12/14/2005 | EP1603882A2 Urea and thiourea derivatives |
12/14/2005 | EP1603880A1 Quinolinone/benzoxazinone derivatives and uses thereof |
12/14/2005 | EP1603879A2 Substituted pyridine derivatives useful in the treatment of cancer and other disorders |
12/14/2005 | EP1603874A2 G-lactam derivatives as prostaglandin agonists |
12/14/2005 | EP1603572A1 Lactam-containing cyclic diamines and derivatives as factor xa inhibitors |
12/14/2005 | EP1603570A2 Aminoheteroaryl compounds as protein kinase inhibitors |
12/14/2005 | EP1326858B1 Piperidine compounds as anti-allergic |
12/14/2005 | EP1224165B1 Novel compounds |
12/14/2005 | EP1200411B1 Process for synthesis of heteroaryl-substituted urea compounds |
12/14/2005 | CN1708560A Beta-isoindigo coloring agent |
12/14/2005 | CN1708491A N-benzodioxolyl, N-benzodioxanyl and N-benzodioxepinyl arylcarbonxamide derivatives, and pharmaceutical compositions comprising them |
12/14/2005 | CN1708481A N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones as antimicrobials |
12/14/2005 | CN1708306A Quinazolinone compounds as calcilytics |
12/14/2005 | CN1231762C Method for directly identifying candidate compound |
12/14/2005 | CN1231476C Substd. pyridine herbicides |
12/14/2005 | CN1231473C Substituted arylpyrazines |
12/14/2005 | CN1231471C 4-amino-5-cyano-2-anilino-pyrimidine derivatives and their use as inhbitors of cell-cycle kinases |
12/14/2005 | CN1231470C N-alkoxy-4, 4-dioxy-polyalkyl-piperidines as polymerisation in hibitors |
12/14/2005 | CN1231467C High affinity ligands for nociceptin receptor ORL-1 |
12/14/2005 | CN1231466C New piperidine derivatives |
12/14/2005 | CN1231215C (Imidazol-5-yl) methyl-2-quinolinone derivatives as inhibitors of smooth muscle cell proliferation |
12/13/2005 | US6974826 such as 3-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydro-2-naphthyl)-4-methoxybenzylidene-2,4-thiazolidinedione; Hodgkin's disease |
12/13/2005 | US6974813 For therapy of perioperative myocardial ischemic injury in mammals, including humans |
12/13/2005 | US6974812 such as 2-chloro-N-(1-hydroxy-cycloheptylmethyl)-5-[4-(2-hydroxy-3-methoxy-propyl)-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl]-benzamide; purinergic receptors (P2x7 E); for treatment of interleukin-1 associated disorders (rheumatoid arthritis) |