Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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11/24/2005 | WO2005109987A2 3-(((4-phenyl)-piperazine-1-yl)-alkyl)-3-alkyl-1, 3-dihydro-2h-indol-2-one derivatives and related compounds for the treatment of central nervous system disorders |
11/24/2005 | WO2005085198A3 Amino cyclopropane carboxamide derivatives as bradykinin antagonists |
11/24/2005 | WO2005046604A3 Heteroaryl-hydrazone compounds |
11/24/2005 | US20050261502 2-Amino-4-(1,3-benzodioxol-5-yl)-6-benzyloxy-3,5-pyridinedicarbonitrile, acting as adenosine-receptor-selective ligands, for the prophylaxis and/or treatment of cardiovascular disorders |
11/24/2005 | US20050261501 e.g. 1-({[9-(hydroxymethyl)-3-oxaspiro[5.5]undec-9-yl]amino}acetyl)-2-pyrrolidinecarbonitrile; dipeptidyl-peptidase IV inhibitor; antidiabetic, hypoglycemic agent; non-insulin dependent diabetes, obesity |
11/24/2005 | US20050261496 3-(Morpholin-4-ylsulfonyl)-5-(1,3-thiazol-2-yl)-1H-indole-2-carboxamide; inhibiting, modulating and/or regulating signal transduction of both receptor and non-receptor tyrosine kinases; anticarcinogenic, -diabetic, -arhtritic, -inflammatory agents; psoriasis; angiogenesisinhibitors; liver cirrhosis |
11/24/2005 | US20050261361 Novel crystal forms of atorvastatin hemi-calcium and processes for their preparation as well as novel processes for preparing other forms |
11/24/2005 | US20050261360 Dissolving the crystalline form in acetone, allowing to convert to amorphous form and then precipitating it out |
11/24/2005 | US20050261359 Novel processes for preparing amorphous atorvastatin hemi-calcium |
11/24/2005 | US20050261353 Acylsemicarbazides as cyclin dependent kinase inhibitors useful as anti-cancer and anti-proliferative agents |
11/24/2005 | US20050261343 Anthranilamides and their use as pharmaceutical agents |
11/24/2005 | US20050261339 Jun N-terminal kinase inhibitors; neurodegenerative diseases; Alzheimer's disease; amyotrophic lateral sclerosis; multiple sclerosis; spinocerebellar ataxia |
11/24/2005 | US20050261330 Derivatives of 2,2,4-trisubstituted tetrahydrofuran an antifungal agents |
11/24/2005 | US20050261324 Pyrimidine hydantoin analogues which inhibit leukocyte adhesion mediated by VLA-4 |
11/24/2005 | US20050261320 Compounds and methods for the treatment of cancer |
11/24/2005 | US20050261319 Novel 2-amino-4-quinazolinones and 2-amino-4-oxoquinazolones as LXR nuclear receptor binding compounds with partial agonistic properties |
11/24/2005 | US20050261318 Protein kinase inhibitors |
11/24/2005 | US20050261315 tyrosine kinase inhibitors such as N-(3-tert-butylisoxazol-5-yl)-2-(4-(benzyloxy)phenyl)acetamide, used for treating and preventing conditions and diseases, such as cancer, hematologic malignancies, cardiovascular disease, inflammation or multiple sclerosis |
11/24/2005 | US20050261313 For angiogenesis mediated diseases; cancer; acylation, cyclization and Heck-type reduction |
11/24/2005 | US20050261308 1-(2-Chloro-6-piperazin-1-yl-pyrimidin-4-ylmethyl)-3,4-dihydro-1H-quinolin-2-one; substituted benzoxazinone compounds; 5-HT6 modulators/antagonists; Parkinson's disease, Huntington's disease, manic depression, psychoses, Alzheimer's disease and memory disorders |
11/24/2005 | US20050261301 e,g, 1,5-bis(5-acetyl-4,7-dimethoxybenzofuran-6-yloxy)pentane;potassium channel modulator; antiinflammatory agent, autoimmune diseases; immunosuppressant; multiple sclerosis, rejection of foreign organ transplants |
11/24/2005 | US20050261299 e.g. 4-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1(3)H-imidazol-2-yl)methyl)benzamide; transforming growth factor- beta (TGF- beta ) type I receptor (ALK5) and/or the activin type I receptor (ALK4) antagonist; wound healing agent, antidiabetic, anticarcinogenic, antiinflmmatory agent |
11/24/2005 | US20050261293 Compounds which inhibit leukocyte adhesion mediated by VLA-4 |
11/24/2005 | US20050261291 1-Cyclopropylmethyl-4-[2-(3,3,5,5-tetramethylcyclohexyl)phenyl]piperazine or a salt or hydrate; exhibit excellent cell adhesion inhibitory action or cell infiltration inhibitory action; for treating inflammatory diseases and autoimmune diseases such as inflammatory bowel diseases and rheumatoid arthritis |
11/24/2005 | US20050261290 Novel compounds of proline and morpholine derivatives |
11/24/2005 | US20050261285 Tetrahydropyran derivatives and their use as therapeutic agents |
11/24/2005 | US20050261279 antipsychotic agents; phenylsulfonyl compounds; 7-Methoxy-8-(3-phenoxy-benzenesulfonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine; schizophrenia |
11/24/2005 | US20050261273 Substituted urea and carbamate, phenacyl-2-hydroxy-3-diaminoalkane, and benzamide-2-hydroxy-3-diaminoalkane aspartyl-protease inhibitors |
11/24/2005 | US20050261244 Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions |
11/24/2005 | US20050261242 nitroso derivatives of drugs such as antiinflammatory agents, antibiotics, expectorants, mucolytic agents, antidiabetics, antitumor, viricides, enzyme inhibitors bronchodilators and antiulcer agents; oxidative and endothelial stress dysfunction; free radicals scavenger |
11/24/2005 | CA2566707A1 Pyrimidine derivatives for the treatment of abnormal cell growth |
11/24/2005 | CA2565953A1 Piperidine derivatives as nk1 and nk3 antagonists |
11/24/2005 | CA2565514A1 3-(((4-phenyl)-piperazine-1-yl)-alkyl)-3-alkyl-1, 3-dihydro-2h-indol-2-one derivatives and related compounds for the treatment of central nervous system disorders |
11/24/2005 | CA2565238A1 Amido compounds and their use as pharmaceuticals |
11/24/2005 | CA2565211A1 Amino-tetrazoles analogues and methods of use |
11/24/2005 | CA2564517A1 1-aryl-4-substituted isoquinolines |
11/24/2005 | CA2564489A1 Tetrahydropyranyl cyclopentyl 1-substituted and 1,1-disubstituted tetrahydroisoquinoline modulators of chemokine receptor activity |
11/24/2005 | CA2564325A1 Substituted pyrazolyl urea derivatives useful in the treatment of cancer |
11/24/2005 | CA2563607A1 4,5-disubstituted-2-aryl pyrimidines |
11/23/2005 | EP1598350A1 Pyrrolidines and thiazolidines derivatives, their preparation and their use in the treatment of hyperglycaemia and of type II Diabetis |
11/23/2005 | EP1598345A1 Benzopyran compounds, process for preparing the same and their use |
11/23/2005 | EP1598340A1 1-(4-piperidinyl)-1,3-dihydro-2h-benzoxazole-2-one derivatives and related compounds as nociceptin analogs and orl1 ligands for the treatment of pain |
11/23/2005 | EP1598339A1 1-(4-amino-cyclohexyl)-1,3-dihydro-2h-benzimidazole-2-one derivatives and related compounds as nociceptin analogs and orl1 ligands for the treatment of pain |
11/23/2005 | EP1598338A1 1-(4-piperidinyl)-1,3-dihydro-2h-indole-2-one derivatives and related compounds as nociceptin analogs and orl1 ligands for the treatment of pain |
11/23/2005 | EP1597257A1 Oxazole-derivatives as ppar agonists |
11/23/2005 | EP1597254A1 Indole-derivative modulators of steroid hormone nuclear receptors |
11/23/2005 | EP1597253A2 Compounds and methods of treating cell proliferative diseases, retinopathies and arthritis |
11/23/2005 | EP1597252A1 Pyridine derivatives as fungicidal compounds |
11/23/2005 | EP1597251A2 Pyrimidine compounds |
11/23/2005 | EP1597249A1 Anthelmintic agents and insecticidal compositions |
11/23/2005 | EP1597246A2 Inhibitors of hepatitis c virus rna-dependent rna polymerase, and compositions and treatments using the same |
11/23/2005 | EP1597240A1 Bicyclic heterocycles, medicaments containing said compounds, use thereof, and method for the production thereof |
11/23/2005 | EP1597233A1 Benzyl urea and thiourea derivatives useful as androgen antagonists |
11/23/2005 | EP1597228A2 Substituted n-arylheterocycles, method for production and use thereof as medicaments |
11/23/2005 | EP1597223A2 Hydroxyl compounds and compositions for cholesterol management and related uses |
11/23/2005 | EP1597084A2 Imaging system |
11/23/2005 | EP1596656A2 Pyrazoles and methods of making and using the same |
11/23/2005 | EP1320522B1 Compositions and methods of the use thereof achiral analogues of cc-1065 and the duocarmycins |
11/23/2005 | EP1280777B1 Tetrahydroisoquinoline analogs useful as growth hormone secretagogues |
11/23/2005 | EP1066261B1 Pyridine derivative and pharmaceutical containing the same |
11/23/2005 | EP0938474B1 Cyclopropylindole compounds and their use as prodrugs |
11/23/2005 | EP0811007B1 Pyrazol-4-yl-benzoyl derivatives and their use as herbicides |
11/23/2005 | CN1701068A Novel compounds and their use |
11/23/2005 | CN1699350A Processes and intermediates for preparing anti-cancer compounds |
11/23/2005 | CN1699347A Substituted pyrazolyl benzenesulfonamides for the treatment of inflamation |
11/23/2005 | CN1228338C Imidazole derivatives or salts thereof and drugs contg. derivatives or salts |
11/22/2005 | US6967249 Photochromic 3H-naphtho[2,1-b]-pyran compounds and photochromic articles produced therewith |
11/22/2005 | US6967205 Compounds with antibacterial and antiparasitic properties |
11/22/2005 | US6967201 Benzofurylpiperazines and benzofurylhomopiperazines: serotonin agonists |
11/22/2005 | US6967079 Pyrimidine derivatives for labeled binding partners |
11/22/2005 | CA2180445C Chemical switching of taxo-diterpenoids between low solubility active forms and high solubility inactive forms |
11/22/2005 | CA2068066C Herpesvirus particles and vaccine |
11/17/2005 | WO2005108393A1 Pyrrole or imidazole amides for treating obesity |
11/17/2005 | WO2005108389A1 Indole derivatives having piperidine rings |
11/17/2005 | WO2005108384A1 3- or 4-monosubstituted phenol and thiophenol derivatives useful as h3 ligands |
11/17/2005 | WO2005108370A1 Benzene compounds |
11/17/2005 | WO2005108369A1 Phenyl compounds and their use in the treatment of conditions mediated by the action of pge2 at the ep1 receptor |
11/17/2005 | WO2005108364A1 Piperazine derivatives of alkyl oxindoles |
11/17/2005 | WO2005108360A1 Pyrrolidin-2-one and piperidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors |
11/17/2005 | WO2005108359A1 Novel compounds of proline and morpholine derivatives |
11/17/2005 | WO2005107742A1 Novel antiviral helioxanthin analogs |
11/17/2005 | WO2005091752A3 Acrylonitrile derivatives for inflammation and immune-related uses |
11/17/2005 | WO2005090334A3 Processes and intermediates for the preparation of aspartic acetal caspase inhibitors |
11/17/2005 | WO2005085177A3 Biaryl amino acids and their use in dna binding oligomers |
11/17/2005 | WO2005058834A3 Quinolines useful in treating cardiovascular disease |
11/17/2005 | WO2004074281A8 Benzofuran oxyethylamines serving as antidepressant drugs and anxiolytic drugs |
11/17/2005 | US20050256315 1h-benzo{f}indazol-5-yl derivatives as selective glucocorticoid receptor modulators |
11/17/2005 | US20050256311 Pyrimidine compounds |
11/17/2005 | US20050256309 Tri-and bi-cyclic heteroaryl histamine-3 receptor ligands |
11/17/2005 | US20050256185 Spiro and dispiro 1,2,4-trioxolane antimalarials |
11/17/2005 | US20050256180 drugs such as 1 -[4-(aminosulfonyl)phenyl]-8-{[(trifluoromethyl)sulfonyl]amino}-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide, used as antiinflammatory agents, antiarthritic agents, antipyretics or analgesics |
11/17/2005 | US20050256170 EP receptor (for which the endogenous ligand is prostaglandin E2, PGE2); e.g. (4-[(5-Phenyl-furan-2-carbonyl)-amino]-phenyl)-acetic acid or 5-Phenyl-furan-2-carboxylic acid [3-(1H-tetrazol-5-yl)-phenyl]-amide; dysmenorrhoea, preterm labour, glaucoma, immune disorders, inflammatory disorders |
11/17/2005 | US20050256167 Preparation and use of imidazole derivatives for treatment of obesity |
11/17/2005 | US20050256166 Nitrogen-containing compounds |
11/17/2005 | US20050256164 NK1 and NK3 antagonists |
11/17/2005 | US20050256160 Beta-alanine derivatives and the use thereof |
11/17/2005 | US20050256159 1,4-disubstituted piperidine derivatives and their use as 11,betahsd1 inhibitors |
11/17/2005 | US20050256158 PGD2 receptor antagonists for the treatment of inflammatory diseases |
11/17/2005 | US20050256145 Pyrimidine derivatives for the treatment of abnormal cell growth |
11/17/2005 | US20050256137 Pyridone compounds as inhibitors of bacterial type III protien secreation systems |