Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
02/2006
02/22/2006CN1738798A Indole derivatives as somatostatin agonists or antagonists
02/22/2006CN1738797A Substituted aryl thioureas and related compounds; inhibitors of viral replication
02/22/2006CN1738618A Pharmaceutical compositions and their uses
02/22/2006CN1242995C Novel compounds, their use and preparation
02/21/2006US7002022 treatment of neoplastic diseases that respond to inhibition of the vascular endothelial growth factor receptor tyrosine kinase activity; tumors, retinopathy, macular degeneration
02/21/2006US7002017 Enantioselective hydrogenation of intermediates in the synthesis of tipranavir
02/21/2006US7001916 Epothilon derivatives, method for the production and the use thereof as pharmaceuticals
02/21/2006US7001906 Pyrrolo (2,3-B) pyridine derivatives containing Pyran ring, useful as anticancer compounds
02/21/2006US7001904 Guanidine derivatives quinazoline and quinoline for use in the treatment of autoimmune diseases
02/21/2006US7001899 7-member ring N-heterocycles that have a cysteine trap substitution; treating osteoarthritis
02/21/2006US7001895 Pyridazinones; selective inhibitors of the induced isozyme PGHS-2 (Title) and cyclooxygenase 2 (COX-2); side effect reduction; analgesics; antipyretics; antiinflamation, -arthritic and -carcinogenic agents; rheumatic diseases;
02/21/2006CA2250347C Piperazine and piperidine compounds with high affinity for dopamine-d2 and serotonin-5ht1a receptors
02/16/2006WO2006016178A1 Enantioselective process
02/16/2006WO2006015986A1 Mercaptoimidazoles as ccr2 receptor antagonists
02/16/2006WO2006015860A2 Pyrazole derivatives for treating conditions mediated by activation of the adenosine a2b or a3 receptor
02/16/2006WO2005121097A3 Pyrazole derivatives, compositions containing such compounds and methods of use
02/16/2006WO2005118544A3 Cycloalkyl substituted pyrimidinediamine compounds and their uses
02/16/2006WO2005110409A3 Tetrahydropyranyl cyclopentyl 1-substituted and 1,1-disubstituted tetrahydroisoquinoline modulators of chemokine receptor activity
02/16/2006WO2005097137A3 Advanced quinazoline based protein kinase inhibitors
02/16/2006WO2005080352A3 Quinazoline derivatives and therapeutic use thereof
02/16/2006WO2005080317A3 Therapeutic amide derivatives
02/16/2006WO2005055941A3 Novel m3 muscarinic acetylcholine receptor antagonists
02/16/2006US20060036096 Process for producing quinolinecarbaldehyde
02/16/2006US20060036092 making 4(R)-[-2,6-diamino-purin-9-yl)-[1,3]-dioxolan-2(R)-yl]-methanol ( beta -D-DAPD); esterification, cyclization, selective reduction, purification
02/16/2006US20060035948 e.g. 6-nitro-4-[N-(4-chlorophenyl)-N-(2-methyl-2H-tetrazol-5-ylmethyl)amino]-3-hydroxy-2-methyl-2-dimethoxymethyl-3,4-dihydro-2H-1-benzopyran; protecting neuronal cells from oxidative stress induced cell death by iron or by hydrogen peroxide; antihypoxic agent, neuroprotectant
02/16/2006US20060035945 Prevent reproduction, infection of virus; antitumor agents
02/16/2006US20060035932 N-aryl piperidine compounds
02/16/2006US20060035930 4-(2,4-dichloro-5-methoxyphenyl)amino-6-methoxy-7-{[5-substituted -amino)methyl]-3-furyl}-3-quinolinecarbonitriles as kinase inhibitors
02/16/2006US20060035925 Substituted 4h-chromenes and analogs as activators of caspases and inducers of apoptosis and the use thereof
02/16/2006US20060035916 2,4-Pyrimidinediamine compounds and their uses
02/16/2006US20060035891 (1S, 2R)-N4-(2-Aminocarbonylcyclopent-1-yl)-5-fluoro-N2-[4-(4-methylpiperazin-1-yl)-3-methylphenyl]-2,4-pyrimidinediamine, having antiproliferative activity, used to inhibit cellular proliferation and to treat proliferate diseases such as cancers
02/16/2006US20060035884 N-cyclic sulfonamido inhibitors of gamma secretase
02/16/2006US20060035870 Carboxylic acid derivatives as IP antagonists
02/16/2006US20060035865 Lipid-rich plaque regressing agents
02/16/2006US20060035295 Method for determination of thymidine kinase 1 activity and the use thereof
02/16/2006CA2576581A1 Substituted indole compounds, their preparation and use in medicaments
02/16/2006CA2573066A1 Mercaptoimidazoles as ccr2 receptor antagonists
02/16/2006CA2572752A1 Pyrazole derivatives for treating conditions mediated by activation of the adenosine a2b or a3 receptor
02/15/2006EP1626050A1 Sulfur-containing naphthoylimide derivatives
02/15/2006EP1626044A1 Novel piperidine derivative
02/15/2006EP1625121A1 Pyrimidine derivatives for the treatment of abnormal cell growth
02/15/2006EP0994871B1 Novel substituted naphthopyrans
02/15/2006CN1735608A Substituted benzoyl derivatives as herbicides
02/15/2006CN1735596A Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
02/15/2006CN1735595A Substituted alkyl amido piperidines
02/15/2006CN1735593A Novel CB1 receptour inverse agonists
02/15/2006CN1735592A Hydroxyethylamine derivatives for the treatment of alzheimer's disease
02/15/2006CN1735416A Therapeutic combination
02/15/2006CN1733725A Process for preparing 2-iminopyrrolidine derivatives
02/15/2006CN1733722A Bis-heterocyclic compounds with antitumour and chemosensitising activity
02/15/2006CN1241926C Novel intermediate for preparing camptothecin derivative (CPT-11) and correlated compound and method thereof
02/15/2006CN1241924C Method for preparing enkephalinase and angiotensin-converting enzyme inhibitor intermediate and its intermediate
02/15/2006CN1241916C Novel acardite compound, its preparation method and medicinal composition containing said compound
02/15/2006CN1241909C Carboxylic acid derivatives as IP antagonists
02/14/2006US6998416 Cyclic AMP-specific phosphodiesterase inhibitors
02/14/2006US6998414 Substituted arylamides as IP antagonists
02/14/2006US6998412 Heterocyclic compounds
02/14/2006US6998407 For prophylaxis and therapy of chronic or acute inflammatory or autoimmune diseases, those associated with aberrant lymphocyte or monocyte accumulation such as arthritis, asthma, atherosclerosis, diabetic nephropathy, inflammatory bowel disease
02/14/2006US6998256 Methods of obtaining epothilone D using crystallization and /or by the culture of cells in the presence of methyl oleate
02/14/2006US6998233 Methods for ligand discovery
02/14/2006CA2374643C 1-trifluoromethyl-4-hydroxy-7-piperidinylaminomethylchroman derivatives as substance p antagonists
02/14/2006CA2263167C Ether muscarinic antagonists
02/14/2006CA2241186C Benzimidazole derivatives
02/14/2006CA2218945C 4-aminoquinazoline derivatives
02/14/2006CA2192645C Tri-substituted phenyl derivatives useful as pde iv inhibitors
02/14/2006CA2192644C Tri-substituted phenyl derivatives useful as pde iv inhibitors
02/14/2006CA2192643C Tri-substituted phenyl derivatives useful as pde iv inhibitors
02/14/2006CA2180155C Naphthylamides as central nervous system agents
02/14/2006CA2135926C Substituted hexahydrobenzo[a]phenanthridines
02/14/2006CA2105666C New centrally acting substituted phenylazacycloalkanes
02/09/2006WO2006014665A2 Arylpyrrolidine derivatives as nk-1/ssri antagonists
02/09/2006WO2006014136A1 Piperidine derivatives as histamine h3 receptor ligands
02/09/2006WO2006013393A2 Quinoline derivatives as neurokinin receptor antagonists
02/09/2006WO2005095409A3 Tetrahydroquinoline derivatives and a process for preparing the same
02/09/2006US20060030713 N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for its preparation
02/09/2006US20060030709 PNA monomer and precursor
02/09/2006US20060030673 Oxygen-containing heterocyclic fused naphthopyrans
02/09/2006US20060030618 Vanilloid receptor ligands and their use in treatments
02/09/2006US20060030605 Pharmaceutical compounds
02/09/2006US20060030580 Contacting phenolic piperidines with opioid receptors; analgesics, anticonvulsants, antitussive agents; diarrhea, drug addiction
02/09/2006US20060030576 Anilinopyrimidine derivatives as IKK inhibitors and compositions and methods related thereto
02/09/2006US20060030565 Amide derivatives and nociceptin antagonists
02/09/2006US20060030561 2-Benzyl-2-hydroxy-4-methyl-4-phenylpentanoic acid (1-oxo-1,3-dihydroisobenzofuran-5-yl)amide for example; treating type II diabetes, obesity, hypertension, arteriosclerosis, or glaucoma
02/09/2006US20060030560 Pyrimidine compounds
02/09/2006US20060030557 Substituted pyridines having antiangiogenic activity
02/09/2006US20060030553 Cell adhesion inhibitors
02/09/2006US20060030548 Methods of using ryanodine antagonists in treating neural injury
02/09/2006US20060030543 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease
02/09/2006DE69717294C5 Chinazolin derivate und diese enthaltende pharmazeutische zusammenstellungen Quinazoline derivatives and those containing pharmaceutical assortments
02/09/2006CA2577882A1 Epoxidized esters of vegetable oil fatty acids as reactive diluents
02/09/2006CA2576112A1 Piperidine derivatives as histamine h3 receptor ligands
02/09/2006CA2575936A1 Quinoline derivatives as neurokinin receptor antagonists
02/09/2006CA2574966A1 Isoindoline compounds and methods of their use
02/09/2006CA2573223A1 Aromatic compound
02/08/2006EP1622895A2 1-aryl-3-(indol-5-yl)-prop-2-en-1-ones, compositions comprising the same and use thereof
02/08/2006EP1622893A1 New alicyclic-amine-substituted 4-carboxamido-benzimidazoles as parp-inhibitors and antioxidants
02/08/2006EP1622886A2 Substituted amino carboxylic acids as inhibitors of protein tyrosine phosphatase-1b
02/08/2006EP1622876A1 Cannabinoid receptor ligands and uses thereof
02/08/2006EP1622872A1 1,2,4-substituerte 1,2,3,4-tetrahydro-and 1,2 dihydro-quinoline and 1,2,3,4-tetrahydro-quinoxaline derivatives as cetp inhibitors for the treatment of atherosclerosis and obesity
02/08/2006EP1622871A1 Cyclic amine derivatives, processes for their preparation, and pharmaceutical compositions containing them