Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
04/2006
04/27/2006WO2006042955A1 Pyridine derivatives and the preparation and the therapeutic use thereof
04/27/2006WO2006012256A3 Fkbp binding composition and pharmaceutical use thereof
04/27/2006WO2005101989A3 Piperidine derivatives as modulators of chemokine receptor ccr5
04/27/2006WO2005090320A3 Triazole derivatives and method of using the same to treat hiv infections
04/27/2006US20060089503 Processes for producing optically active 2-thiomethyl-3-phenylpropionic acid derivative and for producing intermediate therefor
04/27/2006US20060089382 Substituted 3-cyanoquinolines as mek inhibitors
04/27/2006US20060089379 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
04/27/2006US20060089371 Phenyl or heteroaryl amino alkane derivatives as ip receptor antagonist
04/27/2006US20060089369 pyrimidine and pyridine derivatives; diabetes, neurodegenerative disorders, obesity, atherosclerotic cardiovascular disease, hypertension, polycystic ovary syndrome, syndrome X, ischemia, traumatic brain injury, bipolar disorder, immunodeficiency, cancer
04/27/2006US20060089363 Antibacterial agents
04/27/2006US20060089360 Inflammatory or neuropathic pain and diseases involving sensory nerve function such as asthma, rheumatoid arthritis, osteoarthritis, inflammatory bowel disorders, urinary incontinence, migraine and psoriasis; 6-(1H-indol-5-yl)-N-(4-(trifluoromethyl)phenyl)-4-pyrimidinamine
04/27/2006US20060089356 Substituted imidazoles as cannabinoid receptor modulators
04/27/2006US20060089354 ligands for receptor localization studies; for inhibiting binding of vanilloid ligand to a capsaicin receptor; Phosphoric acid dibenzyl ester 4-(4-tert-butyl-phenylamino)-7-(3-trifluoromethyl-pyridin-2-yl)-quinazolin-2-ylmethyl ester; to treat neuropathic pain, itch, urinary incontinence, cough, obesity
04/27/2006US20060089346 Optionally fused aryl-substituted azepanones, oxazepanone or thiazepanones substituted with a dipeptide group, e.g., N2-[(3,5-difluorophenyl)acetyl]-N1-[(2R,3R)-2-(2,5-difluorophenyl)-4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-3-yl]-L-alaninamide; secretase inhibitors for treating Alzheimer's disease
04/27/2006US20060089262 Substituted (thioxo)carbonylamino phenyl uraciles
04/27/2006DE102004051277A1 Heterocyclische Carbonylverbindungen Heterocyclic carbonyl
04/27/2006CA2584422A1 1-(hetero)aryl-3-amino-pyrollidine derivatives for use as mglur3 receptor antagonists
04/27/2006CA2584342A1 Improved inhibitors for the soluble epoxide hydrolase
04/27/2006CA2584328A1 Phosphodiesterase 4 inhibitors
04/27/2006CA2583267A1 Novel b1 bradykinin receptor antagonists
04/27/2006CA2583158A1 Triazoles and their use as bradykinin b1 receptor antagonists
04/27/2006CA2583153A1 1,5-diheterocycle-1h-triazole derivative
04/27/2006CA2582778A1 Pyridine derivatives and the preparation and the therapeutic use thereof
04/26/2006EP1650206A1 Phenylazole compounds, production process, and antioxidants
04/26/2006EP1650203A1 Process of preparation of benzimidazol-2-yl quinolinone derivatives
04/26/2006EP1650192A1 Quinolone derivative or salt thereof
04/26/2006EP1648885A1 Novel compounds
04/26/2006EP1648884A2 Pyrazolyl-indole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
04/26/2006EP1648881A1 Substituted indole ligands for the orl-1 receptor
04/26/2006EP1648870A2 Sulfonic acid derivatives of polycyclic dyes used for analytical applications
04/26/2006EP1648867A1 Ppar active compounds
04/26/2006EP1648866A1 Process and intermediate compounds useful in the preparation of statins, particularly atorvastatin
04/26/2006EP1648458A1 2-'4(phenylamino)-piperidin-1-yl]-n-phenyl-acetamine derivtives and related compounds as neuropeptide y5 (npy5) ligands for the treatement of obesity
04/26/2006EP1648447A1 Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases
04/26/2006EP1648426A2 Benzimidazole derivatives and their use as protein kinases inhibitors
04/26/2006CN1764655A Aromatic sulfone hydroxamates and their use as protease inhibitors
04/26/2006CN1764651A Quinazoline derivatives as antitumor agents
04/26/2006CN1764650A 2, 3, 6-trisubstituted-4-pyrimidone derivatives
04/26/2006CN1764649A Benzyl-pyridazinons as reverse transcriptase inhibitors
04/26/2006CN1764647A Tetrahydroisoquinolyl acetamide derivatives for use as orexin receptor antagonists
04/26/2006CN1764641A Viral polymerase inhibitors
04/26/2006CN1764635A carboxylic acid compounds
04/26/2006CN1764380A N-phenyl- (4-pyridyl)- azinyl!amine derivatives as plant protection agents.
04/26/2006CN1763028A Novel ascorbic acid compounds, methods of synthesis and application use thereof
04/26/2006CN1763027A Novel ascorbic acid compounds, methods of synthesis and application use thereof
04/26/2006CN1762355A (imidazol-5-yl)methyl-2-quinolinone derivatives as inhibitors of smooth muscle cell proliferation
04/26/2006CN1253441C Protease inhibitors
04/25/2006US7034069 High molecular weight hydroxyphenylbenzotriazole uv-absorbers for thin film applications
04/25/2006US7034051 Fused bicyclic carboxamide derivatives and methods of their use
04/25/2006US7034049 3(5)-amino-pyrazole derivatives, process for their preparation and their use as antitumor agents
04/25/2006US7034047 Triazole derivative
04/25/2006US7034043 Cell adhesion inhibitors
04/25/2006US7034039 Fused heterocyclic compounds
04/25/2006US7034035 Having a high residual activity, greater activity at lower application rates, curative activity, and a broader spectrum of efficacy; heterocyclic aromatic amides having a hydroxy group adjacent to the amide functionality
04/25/2006US7034034 Substituted 2-cyclohexyl-4-phenyl-1H-imidazole derivatives
04/25/2006US7034031 Modulators of TNF-α signaling
04/25/2006US7034022 Proteases, kinases enzyme inhibitors; cardiovascular disorders; central nervous system disorders; antiinflammatrory agents; bone disorders; infections
04/25/2006US7034021 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses
04/25/2006US7034018 Substituted pyrrole mannich bases to combat pain and allergic reactions
04/25/2006CA2167291C Substituted 2-phenylpyridines with herbicidal action
04/20/2006WO2006042150A1 Diaminoalkane aspartic protease inhibitors
04/20/2006WO2006041872A2 Thrombin receptor antagonists
04/20/2006WO2006041405A1 Substituted amino-pyrimidones and uses thereof
04/20/2006WO2006041121A1 Remedies/preventives for chronic skin disease
04/20/2006WO2006041120A1 Pharmaceutical composition
04/20/2006WO2006040666A1 Substituted n-alkylpyrimidinones
04/20/2006WO2006040650A1 4-methoxyacridine-1-carboxamide derivatives and the phenazine and oxanthrene analogs as pde4-inhibitors for the treatment of asthma and chronic pulmonary disease (copd)
04/20/2006WO2006040646A1 Benzimidazole or indole amides as inhibitors of pin1
04/20/2006WO2006040526A1 Quinazoline derivatives for use against cancer
04/20/2006WO2006040182A1 Heterocyclic compounds suitable for treating disorders that respond to modulation of the dopamine d3 receptor
04/20/2006WO2006040176A1 Azabicycloheptyl compounds suitable for treating disorders that respond to modulation of the dopamine d3 receptor
04/20/2006WO2006040113A2 Heterocyclic diamide insecticidal agents
04/20/2006WO2006025979A9 Modulators of nuclear receptors
04/20/2006WO2006018708A3 Pyrrolidine derivatives as muscarinic receptor antagonists
04/20/2006WO2006013393A3 Quinoline derivatives as neurokinin receptor antagonists
04/20/2006WO2005117882A8 Hydroxamic acid derivatives as metalloprotease inhibitors
04/20/2006WO2005113513A3 Aryl sulfonamides
04/20/2006WO2005040155A8 Pyrimidin-2-amine derivates and their use as a2b adenosine receptor antagonists
04/20/2006US20060084693 e.g. 4-{2-[4-(5-cyano-1H-indol-3-yl)butylamino]ethoxy}benzofuran-2-carboxylic acid methyl ester; serotonin 5 HT1A and 5HT1D receptors agonist and antagonist, serotonin reuptake inhibitor; neuroleptic and hypotensive agent;
04/20/2006US20060084688 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
04/20/2006US20060084680 ((1S)-5-{2-[(3-methyl-7-propyl-1,2-benzisoxazol-6-yl)oxy]ethoxy}-2,3-dihydro-1H-inden-1-yl)acetic acid; diabetes, obesity, hyperlipidemia, and atherosclerotic diseases; hyperglycemia, hyperinsulinemia, impaired glucose tolerance, dyslipidemia, hypertriglyceridemia, and insulin resistance
04/20/2006US20060084658 Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound
04/20/2006US20060084651 Chemical compounds
04/20/2006US20060084616 enzyme inhibitors such as beta-1'-nicotinamide-2'-deoxyribose, used for treating diseases and conditions associated with CD38, related enzymes and cyclic-adenosine-diphosphate-ribose (cADPR)
04/20/2006US20060083679 Agents with selective K-opioid receptor affinity
04/20/2006US20060083676 For marking and identifying metabotropic glutamate receptor sites and for imaging an organ; in particular non-competitive mGlu1 receptor ligands
04/20/2006CA2584261A1 Pharmaceutical composition
04/20/2006CA2584169A1 Remedies/preventives for chronic skin disease
04/20/2006CA2583983A1 Heterocyclic compounds suitable for treating disorders that respond to modulation of the dopamine d3 receptor
04/20/2006CA2583333A1 Azabicycloheptyl compounds suitable for treating disorders that respond to modulation of the dopamine d3 receptor
04/20/2006CA2582639A1 Thrombin receptor antagonists
04/20/2006CA2582202A1 Diaminoalkane aspartic protease inhibitors
04/20/2006CA2580497A1 Substituted n-alkylpyrimidinones
04/20/2006CA2580419A1 Novel insecticides
04/19/2006EP1647545A1 Antiviral protease inhibitors
04/19/2006EP1646627A1 Chemical compounds containing tocopherol and at least one additional pharmaceutical active substance
04/19/2006EP1646626A1 Pyrrole-2, 5-dione derivatives as liver x receptor modulators
04/19/2006EP1646624A1 Indoles useful in the treatment of inflammation
04/19/2006EP1646615A1 Pyrimidine derivatives as modulators of atp-binding cassette transporters
04/19/2006EP1646613A1 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors