| Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397) |
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| 09/10/2008 | EP1965807A2 S1p receptor modulating compounds and use thereof |
| 09/10/2008 | EP1965790A2 Metabolites of wortmannin analogs and methods of using the same |
| 09/10/2008 | EP1685107B1 1,4-dihydropyridine compounds, pharmaceutical compositions, and methods for the treatment of cardiovascular disease |
| 09/10/2008 | EP1646389B1 Pyrimidine-2,4-dione derivatives as gonadotropin-releasing hormone receptor antagonists |
| 09/10/2008 | EP1597240B1 Bicyclic heterocycles, medicaments containing said compounds, use thereof, and method for the production thereof |
| 09/10/2008 | EP1438053B1 Pyrimidine derivatives, pharmaceutical agent containing said compounds, use and method for making same |
| 09/10/2008 | EP1427708B1 Amino-phthalazinone derivatives as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them |
| 09/10/2008 | EP1362856B1 Water-soluble triazole fungicide |
| 09/10/2008 | EP1323710B1 Nitrogenous five-membered ring compounds |
| 09/10/2008 | CN101263125A Quinazoline derivatives useful in cancer treatment |
| 09/10/2008 | CN101263124A Quinazoline derivatives useful in cancer treatment |
| 09/10/2008 | CN101263121A Histone deacetylase inhibitors |
| 09/10/2008 | CN101260104A Inhibition of phosphoinositide 3-kinase beta |
| 09/09/2008 | US7423176 Bicyclic aromatic sulfinyl derivatives |
| 09/09/2008 | US7423156 Optionally fused oxazolyl- or thiazolyl-aminophenylbenzoyl(cyclo)alkanoic acid derivatives, e.g., trans-(1R,2R)-2-({3'-fluoro-4'-,[(6-fluoro-1,3-benzothiazol-2-yl)amino]-1,1'-biphenyl-4-yl}carbonyl)cyclopentanecarboxylic acid; diacylglycerol O-acyltransferase type 1 inhibitors |
| 09/09/2008 | US7423154 Asymmetric process for the preparation of diarylethylpiperazines derivatives and novel asymmetric diarylmethylamines as intermediates |
| 09/09/2008 | US7423150 Substituted benzazoles and methods of their use as inhibitors of Raf kinase |
| 09/09/2008 | US7423148 Small molecule PI 3-kinase inhibitors and methods of their use |
| 09/09/2008 | US7423058 Inhibitors of hepatitis C virus NS3 protease |
| 09/09/2008 | US7423052 Piperidine compounds for use as orexin receptor antagoinst |
| 09/09/2008 | US7423050 2,4,6-trifluoro-N-[6-[(1-methyl-4-piperidinyl)carbonyl]-2-pyridinyl]-benzamide (hemisuccinate/hydrochloride salt); migraine; inhibit peptide extravasation, while avoiding significant vasoconstrictive activity; improved solubility |
| 09/09/2008 | US7423039 (4-phenylpiperazin-1-yl)acylpiperidine derivatives, preparation thereof and application of same in therapeutics |
| 09/09/2008 | US7423030 1-amino-phthalazine derivatives, the preparation and the therapeutic use thereof |
| 09/09/2008 | CA2460865C Quinoline derivatives as neuropeptide y antagonists |
| 09/09/2008 | CA2419696C Compounds, antibodies, reagent kits, methods of producing antibodies, and methods of detecting analytes |
| 09/09/2008 | CA2252163C D-proline derivatives |
| 09/09/2008 | CA2225756C Substituted cyanophenyl uracils |
| 09/09/2008 | CA2211646C Substituted phenyl compounds as endothelin antagonists |
| 09/04/2008 | WO2008106047A2 Carbamate compounds |
| 09/04/2008 | WO2008105515A1 Novel hydroxamic acid derivative |
| 09/04/2008 | WO2008105442A1 Sulfonamide derivative |
| 09/04/2008 | WO2008105058A1 Sulfonamides |
| 09/04/2008 | WO2008104754A1 Novel pyrimidine derivatives 698 |
| 09/04/2008 | WO2008104597A2 Sulfonyltryptophanols |
| 09/04/2008 | WO2008104580A1 New use of glutaminyl cyclase inhibitors |
| 09/04/2008 | WO2008104203A2 18f fluoro-benzoyl labelled biological active coumpounds as diagnositic imaging agents as well as benzotriazol-1-yloxy-benzoyl, 2,5-dioxo-pyrrolidin-1-yloxy) benzoyl and trimethylammonio-benzoyl precursers |
| 09/04/2008 | WO2008104077A1 Small molecule inhibitors of protein arginine methyltransferases (prmts) |
| 09/04/2008 | WO2008084067A3 Pharmaceutically active dihydrobenzofurane-substituted benzimidazole derivatives |
| 09/04/2008 | WO2008080965A3 Hiv inhibiting 5,6-substituted pyrimidines |
| 09/04/2008 | US20080214835 Processes for preparing darifenacin hydrobromide |
| 09/04/2008 | US20080214811 Xanthene dyes |
| 09/04/2008 | US20080214650 crystalline polymorphic dosage forms of anticholesterol agents; statins; small particle size distribution |
| 09/04/2008 | US20080214640 3'-{[1-(3,4-Dimethylphenyl)-3-methyl-5-oxo-1,5-dihydropyrazol-4-ylidene]hydrazino}-2'-hydroxybiphenyl-3-carboxylic acid or a salt; treatment of thrombocytopenia; may be coadministered with a colony stimulating factor, cytokine, chemokine, or an interleukin or cytokine receptor agonist or antagonist |
| 09/04/2008 | US20080214617 antitumor agents; anticancer agents; structurally related to the leptomycin family; Leptolstatin |
| 09/04/2008 | US20080214564 Macrolide compound in solid form, process for preparation thereof, and pharmaceutical composition containing the same |
| 09/04/2008 | US20080214545 4-{3-tert-butyl-5-[({[4-(pyridin-4-yloxy)phenyl]amino}carbonyl)amino]-1H-pyrazol-1-yl}-N-(2-pyrrolidin-1-ylethyl)benzamide; antiproliferatives; angiogenesis inhibitors |
| 09/04/2008 | US20080214524 e.g. N-[2-(3-fluorophenyl)ethyl]-N'-isoquinolin-5-ylurea; opioid receptor inhibitor; analgesic, antiinflammatory agent; inflammatory thermal hyperalgesia, urinary incontinence and bladder overactivity |
| 09/04/2008 | US20080214519 Chromane Substituted Benzimidazole Derivatives as Acid Pump Antagonists |
| 09/04/2008 | CA2679514A1 18f fluoro-benzoyl labelled biologically active compounds as diagnostic imaging agents as well as benzotriazol-1-yloxy-benzoyl, 2,5-dioxo-pyrrolidin-1-yloxy-benzoyl and trimethylammonio-benzoyl precursers |
| 09/04/2008 | CA2679446A1 New use of glutaminyl cyclase inhibitors |
| 09/04/2008 | CA2679263A1 Sulfonamide compound |
| 09/03/2008 | EP1964834A1 Sulphonyltryptophanols |
| 09/03/2008 | EP1964569A2 3'-or 2'-hydroxymethyl substituted nucleoside derivatives for treatment of viral infections |
| 09/03/2008 | EP1963312A1 Beta-secretase modulators and methods of use |
| 09/03/2008 | EP1963311A1 Chromane substituted benzimidazoles and their use as acid pump inhibitors |
| 09/03/2008 | EP1963310A2 Methods of preparing a vegf-r inhibitor |
| 09/03/2008 | EP1963286A1 Pyrazinecarboxamide derivatives and plant disease controlling agents containing the same |
| 09/03/2008 | EP1963285A1 Bradykinin 1 receptor antagonists |
| 09/03/2008 | EP1963282A1 Sulfoximine-substituted pyrimidines , their preparation and use as drugs |
| 09/03/2008 | EP1963281A2 Heterocyclic derivatives as modulators of ion channels |
| 09/03/2008 | EP1963274A1 Benzoylpyrazole compounds and herbicides containing them |
| 09/03/2008 | EP1963273A2 Substituted isoquinoline-1,3(2h,4h)-diones, 1-thioxo-1,4-dihydro-2h-isoquinoline-3-ones and 1,4-dihydro-3(2h)-isoquinolones and use thereof as kinase inhibitors |
| 09/03/2008 | EP1963260A1 Process for the production of ezetimibe and intermediates used in this proces |
| 09/03/2008 | EP1962849A1 Quinoline derivatives useful in the treatment of mglur5 receptor-mediated disorders |
| 09/03/2008 | EP1761497B1 Azadecalin glucocorticoid receptor modulators |
| 09/03/2008 | EP1730112B1 3-((hetero)arylsulfonyl)-8'[ (aminoalkyl)oxy]quinolines as 5-ht6 receptor antagonists for the treatment of cns disorders |
| 09/03/2008 | EP1718613B1 Pyridine derivatives and their use as cb2 receptor modulators |
| 09/03/2008 | EP1626720B1 4-(2-phenylsulfanyl-phenyl)-piperidine derivatives as serotonin reuptake inhibitors |
| 09/03/2008 | EP1465626B1 Pharmaceutical compositions (kit) comprising dihydropyridinone compounds and an immunoregulatory (or an antiinflammatory) agent and their uses |
| 09/03/2008 | EP1303505B1 Phenyl-substituted 5,6-dihydropyrone derivatives for use as pesticides and herbicides |
| 09/03/2008 | EP1042293B9 Substituted pyridine and pyridazine compounds and their pharmaceutical use |
| 09/03/2008 | CN101258150A Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes |
| 09/03/2008 | CN101258146A Pharmaceutical dosage forms and compositions comprising lecozotan |
| 09/03/2008 | CN101255155A Arylvinylazacycloalkane compounds and methods of preparation and use thereof |
| 09/03/2008 | CN101255132A 6-aryl-3-substituted methylene-pyridinone derivatives and uses thereof |
| 09/03/2008 | CN101255131A Heterocyclic derivatives as opioid modulators |
| 09/03/2008 | CN100415724C Pyrimidine derivatives |
| 09/03/2008 | CN100415720C Quinoline derivative and quinazoline derivative, and medicinal composition containing the same |
| 09/03/2008 | CN100415719C 2,5-disubstituted 3-mercaptopentanoic acid |
| 09/03/2008 | CN100415717C Diarylmethylidene piperidine derivatives and their use as delta opioid receptor agonists |
| 09/03/2008 | CN100415716C 1-(1,2-disubstituted piperidyl)-4-substituted diethylenediamine derivative |
| 09/02/2008 | US7420089 for hepatitis C; histone deacetylase inhibitors; N-hydroxy-4-{[(naphthyl-carbonylamino]alkoxy}benzamides; anticarcinogenic agent; acute promyelocytic leukemia; cell-cycle arrest in late G1 phase or at the G2/M transition |
| 09/02/2008 | US7420070 Resolution with acid; salt formation, cyclization |
| 09/02/2008 | US7420055 Antagonists of the chemokine receptor 9 (CCR9); inhibit TECK ligand; antiinflammatory agents and immunoregulators; inflammatory bowel disease; (2-phenylsulfonamidophenyl)-pyridinyl-methanones; N-[4-chloro-2(pyridine4-carbonyl)-phenyl]4-morpholin-4-yl-benzenesulfonamide |
| 09/02/2008 | US7420001 N-({4'-[(1-benzofuran-2-ylcarbonyl)amino]-1,1'-biphenyl-4-yl}sulfonyl)glycine; metalloproteinase inhibitors; arthritis, macular degeneration, graft versus host disease, cancer, osteoarthritis |
| 09/02/2008 | US7419999 Gamma lactams as prostaglandin agonists and use thereof |
| 09/02/2008 | US7419994 4-(substituted cycloalkylmethyl) imidazole-2-thiones, 4-(substituted cycloalkenylmethyl) imidazole-2- thiones, 4-(substituted cycloalkylmethyl) imidazol-2-ones and 4-(substituted cyloalkenylmethyl) imidazol-2-ones and related compounds |
| 09/02/2008 | US7419986 Antidepressant azaheterocyclylmethyl derivatives of heterocycle-fused benzodioxans |
| 09/02/2008 | US7419984 for uses such as inhibiting the activity of lysophosphatidic acid acyltransferase beta and/or inhibiting the proliferation of a cell (e.g., tumor cell) |
| 09/02/2008 | US7419983 Gonadotropin-releasing hormone receptor antagonists and methods related thereto |
| 09/02/2008 | US7419980 Treating conditions improved by monoamine reuptake; 1-[1-(2-naphthyl)-2-piperazin-1-ylethyl]cyclobutanol; sexual disorders, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders, hot flashes |
| 09/02/2008 | US7419976 Diazepanes derivatives useful as IFA inhibitors |
| 09/02/2008 | US7419975 Organic compounds |
| 09/02/2008 | US7419967 e.g. hexahydrofuro[2,3-b]furan-3-yl N-((1S,2R)-1-benzyl-3-(cyclopentyloxy)[(3-[2-(dimethylamino)ethyl]aminophenyl)sulfonyl]amino-2-hydroxypropyl)carbamate; against human immunodeficiency virus, chronic and acute viral infections |
| 09/02/2008 | US7419966 Viricides; human t-cell leukemia, lymphoma virus |
| 09/02/2008 | CA2466728C Azetidinyl diamines useful as ligands of the nociceptin receptor orl-1 |
| 09/02/2008 | CA2294351C Compounds useful for inhibition of farnesyl protein transferase |
| 09/02/2008 | CA2248338C 2-amino-4-bicycloamino-1,3,5-triazines as herbicides and plant growth regulators |
| 09/02/2008 | CA2160447C Amino(thio)ether derivatives |
| 08/28/2008 | WO2008103693A2 Chemical linkers with single amino acids and conjugates thereof |