Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
12/1998
12/30/1998WO1998058916A1 NEW β-AMINO AND β-AZIDOCARBOXYLIC ACID DERIVATIVES, THE PRODUCTION THEREOF AND THE USE THEREOF AS ENDOTHELIN RECEPTOR ANTAGONISTS
12/30/1998WO1998058915A2 Pyrimidin-2,4,6-trion derivatives and their use as metalloprotease-inhibitors
12/30/1998WO1998058677A1 Pharmaceutical formulations containing voriconazole
12/30/1998EP0887348A1 Bis-Indole derivatives having antimetastatic activity, a process for their preparation and pharmaceutical compositions containing them
12/30/1998EP0887346A2 Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists
12/30/1998EP0887344A1 Quinolines and quinazolines useful in therapy
12/30/1998EP0886635A1 2-amino-5,6-dichlorobenzimidazole derivatives having antiviral activity
12/30/1998EP0705258B1 Azolyl-cyclic amine derivatives with immunomodulatory activity
12/30/1998CN1203599A Substitued pyrrolidinone, thiazolidinone or oxazolidinone as herbicides
12/30/1998CN1203228A Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
12/30/1998CA2294259A1 Barbituric acid derivatives with antimetastatic and antitumor activity
12/30/1998CA2294113A1 Pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical preparations containing these compounds
12/30/1998CA2294050A1 New .beta.-amino and .beta.-azidocarboxylic acid derivatives, the production thereof and the use thereof as endothelin receptor antagonists
12/29/1998US5854273 Bisimide compounds
12/29/1998US5854268 Azetidine, pyrrolidine and piperidine derivatives
12/29/1998US5854265 Biheteroaryl inhibitors of farnesyl-protein transferase
12/29/1998US5854264 Inhibitors of farnesyl-protein transferase
12/29/1998US5854263 1- (1,4-benzodioxanyl)alkyl!-3-(heteroaryl) pyrrolidines and related compounds and their therapeutic utility
12/29/1998US5854249 Opioid diarylmethylpiperazines and piperidines
12/29/1998US5854243 3-heteroaryl-1-pyrrolidinealkylthiols and derivatives thereof and their therapeutic utility
12/29/1998CA2036427C Acyl compounds
12/29/1998CA2002859C Method of treating epithelial disorders
12/24/1998DE19726427A1 Pyrimidin-2,4,6-trion-Derivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel Pyrimidine-2,4,6-trione derivatives, processes for their preparation and medicaments containing these compounds
12/23/1998WO1998057966A1 Novel aryloxy substituted pyrimidine imidazole compounds
12/23/1998WO1998057954A1 Aroyl-piperazine derivatives, their preparation and their use as tachykinin antagonists
12/23/1998WO1998057951A1 NOVEL GUANIDINE MIMICS AS FACTOR Xa INHIBITORS
12/23/1998WO1998057937A2 Inhibitors of factor xa with a neutral p1 specificity group
12/23/1998WO1998057642A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998WO1998057641A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998WO1998057639A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998WO1998057638A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998EP0885890A1 Sulfonylureidopyrazole derivatives
12/23/1998EP0885887A2 Sulfonamide inhibitors of HIV-Aspartyl protease
12/23/1998EP0885215A1 Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
12/23/1998EP0885214A1 Cyclic imido-1,3,5-triazine crosslinking agents
12/23/1998EP0885212A1 Quinoxalinediones
12/23/1998EP0885201A1 2-amino-4-bicycloamino-1,3,5-triazines as herbicides and plant growth regulators
12/23/1998EP0885199A1 Kappa agonist compounds and pharmaceutical formulations thereof
12/23/1998EP0885189A2 Method for the synthesis of poly-pyrrole and poly-imidazole carboxamides on a solid support
12/23/1998EP0719304B1 Cyanine dyes and process for the production
12/23/1998EP0527851B1 1h-substituted-1,2,4-triazole compounds for treatment of cardiovascular disorders
12/23/1998CN1202902A Thrombin inhibitors
12/23/1998CN1202895A Mercaptoalkylpeptidyl compounds having an imidazole substituent and their use as inhibitors of matrix metalluproteinass (MMP) and/or tumour necrosis factor (TNF)
12/23/1998CN1202886A 3-spiro-indolin-2-one derivatives, its preparing method and its medicinal compounds
12/23/1998CN1041311C Method for preparing benzopyran and related LTB4 antagonists
12/23/1998CN1041308C Process for preparing substituted maleimides
12/23/1998CA2430623A1 Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
12/23/1998CA2294590A1 Alpha 1a adrenergic receptor antagonists
12/23/1998CA2294349A1 Alpha 1aadrenergic receptor antagonists
12/23/1998CA2294344A1 Alpha 1a adrenergic receptor antagonists
12/23/1998CA2294137A1 Novel aryloxy substituted pyrimidine imidazole compounds
12/23/1998CA2293408A1 Alpha 1a adrenergic receptor antagonists
12/23/1998CA2292883A1 Aroyl-piperazine derivatives, their preparation and their use as tachykinin antagonists
12/23/1998CA2291442A1 Novel guanidine mimics as factor xa inhibitors
12/23/1998CA2290982A1 Inhibitors of factor xa with a neutral p1 specificity group
12/22/1998US5852210 Cinnamic acid derivatives
12/22/1998US5852195 Pyranone compounds useful to treat retroviral infections
12/22/1998US5852192 Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
12/22/1998US5852049 Aromatic ethers derived from indoles which are useful as medicaments
12/22/1998US5852043 HIV protease inhibitors
12/22/1998US5852039 Pharmaceutical composition containing quinoline or quinazoline derivatives
12/22/1998US5852028 Pyrimidine carboxylates and related compounds and methods for treating inflammatory conditions
12/22/1998US5852022 Antipsychotic agents, composition and method of use
12/22/1998US5852019 Pyrimidinylpyrazole derivatives
12/22/1998US5852017 2,3(1H,4H)-quinoxalinediones
12/22/1998US5852016 Quinoxaline derivatives useful in therapy
12/22/1998US5852011 Benzimidazole derivatives
12/22/1998US5852010 Inhibitors of farnesyl-protein transferase
12/22/1998US5852008 Heteroatom substituted benzoyl derivatives that enhance synaptic response mediated by receptors
12/22/1998US5851999 FLK-1 is a receptor for vascular endothelial growth factor
12/22/1998CA1340283C Substituted sulfonyldiamides, process for their preparation, and their use as herbicides and plant growth regulators
12/17/1998WO1998056788A1 Imidazolyl-cyclic acetals
12/17/1998WO1998056771A2 Piperazine derivatives and their use as anti-inflammatory agents
12/17/1998WO1998056767A1 Pesticidal 1-aryl-3-iminopyrazoles
12/17/1998WO1998056764A1 Method for producing nitroguanidine derivatives
12/17/1998WO1998056376A1 Novel heteroaryl compounds for the modulation of protein tyrosine enzyme related cellular signal transduction
12/17/1998CA2293681A1 Method for producing nitroguanidine derivatives
12/17/1998CA2293400A1 Novel heteroaryl compounds for the modulation of protein tyrosine enzyme related cellular signal transduction
12/16/1998EP0884314A2 Metal alkoxides
12/16/1998EP0883402A1 Novel cycloalkyl substituded imidazoles
12/16/1998CN1202161A Macrocyclic compounds as metalloprotease inhibitors
12/16/1998CN1202159A Pyrazin-2-one derivatives, their use, and intermediates for their production
12/16/1998CN1202158A Heterrocyclically substituted salicyclic acid derivatives
12/16/1998CN1202157A Pyridazin-3-one derivatives, their use, and intermediates for their production
12/16/1998CN1202107A Selective 'beta'3 adrenergic agonists
12/15/1998US5849919 Fused benzeneoxyacetic acid derivatives which have PGI2 receptor anonist activity
12/15/1998US5849910 Process for the preparation of unsymmetrical 4,6-bis aryloxy-pyrimidine compounds
12/15/1998US5849893 Nucleic acid-binding oligomers possessing C-branching for therapy and diagnostics
12/15/1998US5849780 1-benzenesulfonyl-1-1,3-dihydroindol-2-one derivatives, their preparation and pharmaceutical compositions in which they are present
12/15/1998US5849778 N-pyrazolyl anilines as pesticides
12/15/1998US5849764 Antagonists of gonadotropin releasing hormone
12/15/1998US5849758 Herbicidal 2, 6-disubstituted pyridines and 2, 4-disubstituted pyrimidines
12/15/1998US5849746 Substituted 1,4-piperazine-heteroaryl derivatives as 5-HT1D receptor agonists
12/15/1998US5849744 Pyrrolyl tetrahydrobenzoquinoxaline diones, their preparation and use as glutamate receptor antagonist
12/15/1998US5849743 Quinoxalines and drugs prepared therefrom
12/15/1998US5849741 Fused pyridazine compounds
12/15/1998US5849739 5-arylindole derivatives
12/15/1998US5849665 Synergistic composition and process for selective weed control
12/15/1998US5849361 Methine dyes based on formylaminopyridones
12/15/1998CA2092653C Substituted pyrrolidine derivatives as hiv protease inhibitors