Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
12/2000
12/28/2000WO2000043373A3 Kinase inhibitors
12/28/2000DE19928306A1 New 4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors, polyps or respiratory or gastrointestinal diseases
12/28/2000CA2375211A1 Antiviral agents
12/28/2000CA2375182A1 5-cyano-2-aminopyrimidine derivatives
12/28/2000CA2373921A1 Novel benzimidazole derivatives and pharmaceutical compositions comprising these compounds
12/27/2000EP1062216A1 Inhibitors of phospholipase a2
12/27/2000EP1062210A1 1,2-diazepane derivatives as interleukin-1beta converting enzyme inhibitors
12/27/2000EP1062208A1 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
12/27/2000EP1062205A2 Inhibitors of phospholipase enzymes
12/27/2000EP1061936A1 Cyclic dipeptides and azetidinone compounds and their use in treating cns injury and neurodegenerative disorders
12/27/2000EP0823900B1 Quinazoline derivatives
12/27/2000EP0821671B1 Arylsulfonyl hydroxamic acid derivatives as mmp and tnf inhibitors
12/27/2000EP0639050B1 Synergistic composition and process for selective weed control
12/27/2000CN1278258A Azaring-ether derivatives and their use as nicotinic ach receptor modulators
12/27/2000CN1278251A Novel carboxylic acid derivatives which carry amide side chains, prodn. of same, and use as endothelin receptor antagonists
12/27/2000CN1278244A Dipeptide nitriles
12/27/2000CN1059902C Estrogen excitant/antagonist
12/26/2000US6166219 Treatment of diabetes and related disorders
12/26/2000US6166205 2-Aryl-4-(1-[4-heteroaryl]piperazin-1-yl)methylimidazoles: dopamine . D.sub4 receptor subtype ligands
12/26/2000US6166060 Antihistamines; sleep disorders; central nervous system disorders
12/26/2000US6166037 A blocking agent for blocking the entry of hiv into target cells of a patient to prevent infection of the patient by hiv
12/26/2000US6166027 Treatment of high blood pressure and cardiac insufficiency, angina pectoris, arrhythmias, thromboembolic diseases, ischaemias, myocardial infarction, cerebral stroke, restenoses, coronary angioplasties, arteriosclerosis
12/26/2000US6166023 1,5- and 3-O-substituted 1H-indazoles having anti-asthmatic, anti-allergic, anti-inflammatory, immunomodulating and neuroprotective action, process for their preparation and their use as medicaments
12/26/2000US6166015 Pyrrolidine derivatives-CCR-3 receptor antagonists
12/26/2000US6166005 Heterocyclic metalloprotease inhibitors
12/26/2000US6165996 Compounds with chelation affinity selectivity for first transition series elements: use in medical therapy and diagnosis
12/26/2000US6165980 Distamycin derivatives, wherein the distamycin formyl group is substituted by a benzoyl group bearing alkylating group a bis-halo-ethylamino or a n-alkyl-n-haloethyl-amino group, while amidine group is substituted by various nitrogen groups
12/26/2000US6165944 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides
12/21/2000WO2000077519A1 Solid phase synthesis of n,n-disubstituted diazacycloalkylcarboxy derivatives
12/21/2000WO2000077027A2 Serine protease inhibitors
12/21/2000WO2000076984A2 Novel compounds, their use and preparation
12/21/2000WO2000076983A1 1-(4-arylsulfonyl)-3-substituted-5-aryl-2-pyrazolines as inhibitors of cyclooxygenase-2
12/21/2000WO2000076980A1 Novel nitrogen-contaiing heterocyclic derivatives or salts thereof
12/21/2000WO2000076971A2 Serine protease inhibitors
12/21/2000WO2000076970A2 Serine protease inhibitors
12/21/2000WO2000076969A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits using isoindoline derivatives
12/21/2000WO2000076966A2 Indolinylamide derivatives and the use thereof as antiviral drugs
12/21/2000WO2000076521A1 Antiviral indoleoxoacetyl piperazine derivatives
12/21/2000WO2000076503A1 1-(4-sulfamylaryl)-3-substituted-5-aryl-2-pyrazolines as inhibitors of cyclooxygenase-2
12/21/2000WO2000053579A3 Solid phase synthesis of 4-aminoproline derivatives and/or combinatorial libraries thereof
12/21/2000WO2000049001A3 Phenoxy-, phenylthio-, phenylamino-, benzyloxy-, benzylthio- or benzylaminopyrimidine insectidices and acaricides
12/21/2000DE19927415A1 Indolinylharnstoffderivate Indolinylharnstoffderivate
12/21/2000CA2383008A1 Compounds
12/21/2000CA2377153A1 1-(4-sulfamylaryl)-3-substituted-5-aryl-2-pyrazolines as inhibitors of cyclooxygenase-2
12/21/2000CA2375920A1 Compounds
12/21/2000CA2373394A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits using isoindoline derivatives
12/21/2000CA2340663A1 Antiviral indoleoxoacetyl piperazine derivatives
12/20/2000EP1061075A2 Substituted triazoles, imidazoles and pyrazoles as herbicides
12/20/2000EP1061074A1 Novel process and intermediates
12/20/2000EP1060170A1 Optically active substituted 2,4-diamino-1,3,5-triazines as herbicides
12/20/2000EP1060166A1 Five-membered, benzo-condensed heterocycles used as antithrombotic agents
12/20/2000EP1060165A1 Method for preparing n-substituted heterocyclic derivatives using a phase-transfer catalyst
12/20/2000EP0543858B1 Benzimidazole derivatives, process for their preparation and application
12/20/2000CN1277605A Arylpyridazinones as prostaglandin endoperoxide H synthase biosynthesis inhibitors
12/20/2000CN1277604A Heteraryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
12/19/2000US6162927 (2s,3r,4s)-2-(2,2-dimethylpentyl)-4-(7-methoxy-1,3-benzodioxol-5-yl)-1-(n,n-di(n-butyl)aminocarbonylmethyl)-pyrrolidine-3-carboxylic acid, or salt or ester thereof, in pure form; adminstering to treat hypertension, other diseases
12/19/2000US6162922 4'-((2-alkyl or alkoxy-4-oxo-1,3-diazaspiro(4.4)non-1-en-3-yl)methyl)(1,1'-bip henyl)-2-car bonitrile and its salts using phase transfer catalysis.
12/19/2000US6162822 Bisimide compounds
12/19/2000US6162819 Pyrazole derivatives, their preparation and their use in pharmaceuticals
12/19/2000US6162818 Respiratory system disorders; crohn's disorder; cardiovascular disorders
12/19/2000US6162812 Pharmaceutical compositions containing HIV protease inhibitors and methods of their use
12/19/2000US6162804 Tyrosine kinase inhibitors
12/19/2000US6162800 N-(pyrimidinyl)-aspartic acid analogs as interleukin-1β converting enzyme inhibitors
12/19/2000US6162442 Use of aqueous L-Tryptophan and/or L-Threonine salt solutions
12/18/2000CA2311872A1 Processes and intermediates for preparing (indole-2-carbonyl)-amides
12/14/2000WO2000075135A1 Biaryl inhibitors of prenyl-protein transferase
12/14/2000WO2000075119A2 Substituted 2-aryl-1,2,4-triazine-3,5-di(thi)ones used as herbicides
12/14/2000WO2000075117A1 Compositions and methods for inhibiting cell death
12/14/2000CA2375942A1 Substituted 2-aryl-1,2,4-triazine-3,5-di(thi)ones
12/14/2000CA2375843A1 Compositions and methods for inhibiting cell death
12/13/2000CN1276370A Process for preparing anticancer compound, and intermediate
12/12/2000US6160118 Process for the synthesis of substituted piperazinones via Mitsunobu reaction
12/12/2000US6160001 Halobenzimidazoles and their use as microbicides
12/12/2000US6159998 Administered as vasodilators, analgesics, anesthetics, sedatives, and anitspasmodic agents
12/12/2000US6159978 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
12/12/2000US6159969 Uracil derivatives, and antitumor effect potentiator and antitumor agent containing the same
12/12/2000US6159964 Vitronectin receptor antagonists
12/12/2000CA2011949C Ultraviolet absorbing lenses and methods of making the same
12/07/2000WO2000073300A1 Amino heterocycles useful as pharmaceutical agents
12/07/2000WO2000073299A1 Sulfonamide compounds with pharmaceutical activity
12/07/2000WO2000073279A1 4-phenyl-pyrimidine derivatives
12/07/2000WO2000073275A1 Substituted phenylcyclohexane carboxylic acid amides that have an adenosine uptake inhibiting effect
12/07/2000WO2000073264A1 Cell proliferation inhibitors
12/07/2000DE19925593A1 Substituierte 2-Aryl-1,2,4-triazin-3,5-di(thi)one Substituted 2-aryl-1,2,4-triazine-3,5-di (thi) ones
12/07/2000CA2375186A1 Substituted phenylcyclohexane carboxylic acid amides that have an adenosine uptake inhibiting effect
12/07/2000CA2371395A1 Amino heterocycles useful as pharmaceutical agents
12/07/2000CA2371092A1 Cell proliferation inhibitors
12/06/2000EP1057819A1 Phthalazine derivatives and remedies for erectile dysfunction
12/06/2000EP1057814A1 Tetrahydrobenzindole derivatives
12/06/2000EP1057484A1 Cell death inhibitors
12/06/2000EP1056742A1 Anti-viral pyrimidine derivatives
12/06/2000EP1056733A1 Histamine h3 receptor ligands
12/06/2000EP1056729A1 N-[(substituted five-membered di- or triaza diunsaturated ring)carbonyl]guanidine derivatives for the treatment of ischemia
12/06/2000EP1056725A1 Inhibition of raf kinase using aryl and heteroaryl substituted heterocyclic ureas
12/06/2000EP1056719A2 Inhibitors of phospholipase enzymes
12/06/2000EP1056714A1 Phenylalanine derivatives as inhibitors of alpha4 integrins
12/06/2000EP0597088B1 Novel imidazole derivatives, their preparation and therapeutic applications
12/06/2000CN1275977A Heterocyclic thioesters and ketones
12/06/2000CN1275912A Novel amide derivatives
12/06/2000CN1059210C Process for preparation of 6-heterocyclic-4-amino-1,3,4,5-tetrahydrbenz [cd] indoles and acid additive salt used as medicine