Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
05/2001
05/09/2001EP1097718A1 NPY antagonists for the treatment of female sexual dysfunction
05/09/2001EP1097707A1 Treatment of female sexual dysfunction
05/09/2001EP1097706A1 Phosphodiesterase inhibitors for the treatment of female sexual dysfunction
05/09/2001EP1097382A2 Imidazoline receptor binding compounds
05/09/2001EP1097150A1 Imidazolyl derivatives
05/09/2001CN1294580A Indole derivatives with antiviral activity
05/09/2001CN1294579A Sulfonamide-contg. indole compounds
05/08/2001US6228877 Anticarcinogenic, antitumor and antiproliferative agents
05/08/2001US6228872 Neurotrophic diamide and carbamate agents
05/08/2001US6228847 Inhibitors of nucleoside metabolism
05/08/2001US6228808 Carbamoylphenylsulfonylureas, processes for their preparation and their use as herbicides and plant growth regulators
05/08/2001CA2324484A1 Compounds for the treatment of female sexual dysfunction
05/08/2001CA2323464A1 Compounds for the treatment of female sexual dysfunction
05/08/2001CA2323191A1 Compounds for the treatment of female sexual dysfunction
05/08/2001CA2323183A1 Compounds for the treatment of female sexual dysfunction
05/03/2001WO2001030768A1 Methods and compositions utilizing quinazolinones
05/03/2001WO2001030762A1 Imidazol-4-ylmethanols use as inhibitors of steroid c17-20 lyase
05/03/2001WO2001030333A2 Tissue factor antagonists and methods of use thereof
05/03/2001WO2001030330A2 Method to treat pain utilizing benzimidazole nmda/nr2b antagonists
05/03/2001CA2387869A1 Imidazol-4-ylmethanols use as inhibitors of steroid c17-20 lyase
05/03/2001CA2387857A1 Tissue factor antagonists and methods of use thereof
05/03/2001CA2386441A1 Method to treat pain utilizing benzimidazole nmda/nr2b antagonists
05/02/2001EP1095936A1 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses, and methods and intermediates useful for their preparation
05/02/2001EP1095275A2 Endogenous constitutively activated g protein-coupled orphan receptors
05/02/2001EP1095039A2 New pharmaceutically active compounds
05/02/2001EP1095031A1 Antiviral macrocyclic compounds
05/02/2001EP1095025A2 Benzimidazoles, production thereof and use thereof as medicaments
05/02/2001EP1094826A1 Novel therapeutic agents that modulate alpha-1a adrenergic receptors
05/02/2001EP1094816A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
05/02/2001EP1094810A1 Use of prenyltransferase inhibitors for preparing a medicine for treating pathologies resulting from heterotrimeric g protein membrane fixation
05/02/2001EP0769947B1 Indolinone compounds for the treatment of disease
05/02/2001CN1293671A Substituted bisindolymaleimides for inhibition of cell proliferation
05/02/2001CN1293663A 2,3,4,5-tetrahydro-1H-[1,4] benzodiazepine-3-hydroxamix acids as matrix metal-protease
05/01/2001US6225465 Process for the aminocarbonylation of benzazepines and benzodiazepines
05/01/2001US6225335 3-(4′-bromobenzylindenyl)-2-indolinone and analogues thereof for the treatment of disease
05/01/2001US6225318 4-aminoquinazolone derivatives
05/01/2001US6225312 Piperazine and piperidine compounds
05/01/2001US6225308 Tissue selective compounds in the treatment of prostate cancer or benign prostate hypertrophy
05/01/2001CA2037299C Gamma emitting, cck-a antagonists for pancreatic imaging
04/2001
04/26/2001WO2001029029A1 Tetrahydrobenzindolone derivatives, their preparation and their use as 5-ht7 receptor antagonists
04/26/2001WO2001029028A1 9- (piperazinylalkyl) carbazoles as bax-modulators
04/26/2001WO2001029012A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
04/26/2001WO2001029011A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
04/26/2001WO2001029009A1 4,5-disubstituted-2-aminopyrimidines
04/26/2001WO2001029005A1 Bicyclic vasopressin agonists
04/26/2001WO2001028996A2 Pyrrolidine derivatives, their preparation and their use as inhibitors of neuraminidases
04/26/2001WO2001028987A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/26/2001WO2001028561A1 Gram-positive selective antibacterial compounds, compositions containing such compounds and methods of treatment
04/26/2001WO2001028493A2 Small molecule inhibitors of necrosis
04/26/2001WO2000055139A3 Heterocyclic urea and related compounds useful as anti-inflammatory agents
04/26/2001CA2388859A1 Inhibitors of neuraminidases
04/26/2001CA2387886A1 Bicyclic vasopressin agonists
04/26/2001CA2387034A1 4,5-disubstituted-2-aminopyrimidines
04/26/2001CA2384240A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/25/2001EP1094064A1 5-arylindolederivatives and their use as serotonin(5-ht1)agonists
04/25/2001EP1094063A1 9-(Piperazinylalkyl)carbazoles as Bax-modulators
04/25/2001EP1093372A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS
04/25/2001CN1064965C Novel sulfonamides compound and its use as medicine
04/25/2001CN1064959C N-substituted azabicycloheptane derivatives and preparing process and use thereof
04/24/2001US6222036 Reacting 2-thio-4-dimethyoxymethyl-pyrimidine with acetic acid and catalytic amount of concetrated sulfuric acid to produce 2-thiopyrimidine aldehyde
04/24/2001US6221881 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
04/19/2001WO2001027113A2 PYRAZOLO `4,3-d! PYRIMIDINE DERIVATIVES
04/19/2001WO2001027107A2 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001WO2001027106A1 Substituted pyrroles as antiproliferative agents for the treatment of cancer
04/19/2001WO2001027105A1 Pyrimidine-5-carboxamide compounds, process for producing the same and use thereof
04/19/2001WO2001027103A1 Fab i inhibitors
04/19/2001WO2001027102A1 Substituted diazepanes
04/19/2001WO2001027089A1 Pyrimidine derivatives
04/19/2001WO2001027087A2 Process for making boc-protected 3-aminohydantoins/thiohydantoins and 3-aminodihydrouracils/dihydrothiouracils
04/19/2001WO2001027084A1 Beta disubstituted metalloprotease inhibitors
04/19/2001WO2001027081A1 6-position substituted indoline, production and use thereof as a medicament
04/19/2001WO2001027080A2 5-substituted indolinones and use thereof as kinase and cyclin/cdk complex inhibitors
04/19/2001WO2001026656A2 5-membered heterocycle derivatives and use thereof as monoamine oxidase inhibitors
04/19/2001WO2001026644A2 Mediators of hedgehog signaling pathways, compositions and uses related thereto
04/19/2001WO2000018767A9 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
04/19/2001WO1999032448A8 Substituted pyridine and pyridazine compounds and their pharmaceutical use
04/19/2001DE19949209A1 In 5-Stellung substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel In the 5-position substituted indolinones, their preparation and their use as medicaments
04/19/2001DE19949208A1 New 3-(amino-methylene)-2-indolinone derivatives are kinase inhibitors and cell proliferation inhibitors useful e.g. for treating tumors, metastasis, rheumatoid arthritis or psoriasis
04/19/2001DE19948417A1 Imidazol-Derivate und ihre Verwendung als Arzneimittel Imidazole derivatives and their use as medicaments
04/19/2001CA2388813A1 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001CA2388505A1 5-membered heterocycle derivatives, their preparation and application as medicine
04/19/2001CA2386485A1 Beta disubstituted metalloprotease inhibitors
04/19/2001CA2385071A1 Substituted pyrroles as antiproliferative agents for the treatment of cancer
04/19/2001CA2382605A1 Pyrimidine derivatives
04/18/2001EP1092715A2 Cyano-indole derivatives as inhibitors of serotonin reuptake, method for their preparation and pharmaceutical compositions containing the same
04/18/2001EP1091955A1 Quinolones as serine protease inhibitors
04/18/2001EP1091943A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
04/18/2001EP1091942A1 Potassium channel blocking agents
04/18/2001EP1091941A1 Novel benzimidazoles as corticotropin release factor antagonists
04/18/2001EP1091937A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
04/18/2001CN1291892A Substituted oxoazaheterocyclyl factor Xa inhibitors
04/18/2001CN1064679C Herbicidal thiocarbamoyltetrazolinones
04/17/2001US6218549 Bicyclic aminoimidazoles
04/17/2001US6218547 1-phenyl-benzimidazole compounds and their use as GABA-a receptor modulators
04/17/2001US6218538 Antagonists of n-type neuronal calcium channels useful in the treatment of cerebrovascular ischaemia and pain.
04/17/2001US6218537 Process for making pyridyl and pyrimidine substituted imidazole compounds
04/17/2001US6218431 Substituted biphenyls
04/17/2001US6218424 Heterocyclic ketone and thioester compounds and uses
04/17/2001US6218418 Therapy of cell proliferative disorders associated with an altered cell dependent kinase activity by administering amino pyrazole derivative to mammal
04/17/2001US6218415 Therapy of bone reabsorption by osteoclasts, tumor growth and tumor metastasis, inflammation, cardiovascular disease, nephropathies and retinopathies