Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
11/2004
11/04/2004US20040220174 for example, 1-(4-methoxyphenyl)-7-oxo-6-[5-(2-oxo-1-piperidinyl)2-pyridinyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide; use as anticoagulant agent for treatment of thromboembolic disorders
11/04/2004US20040220173 central nervous system disorders; psychological disorders; Parkinson's disease; Huntington's disease ; sleep disorders
11/04/2004US20040220169 anticoagulants; factor x inhibitor; N-[1-(5-chloro-1H-benzimidazol-2-yl)ethyl]-3-methyl-4-(2,5-dihydropyrrol-1-ylcarbonyl)benzamide
11/04/2004US20040220148 5-Membered ring heterocycles as inhibitors of leucocyte adhesion and as VLA-4 antagonists
11/04/2004US20040220112 administering 2-(N-Methylsulfonamido-2-aminophenyl)-N-methyl-N-[(1S)-1-phenyl-2-(1-pyrrolidinyl)ethyl]acetamide as an anti-pruritic agent; antihyperalgesics; analgesics; central nervous system side effect reduction
11/04/2004CA2526897A1 4-anilino-quinazoline derivatives as antiproliferative agents
11/04/2004CA2522803A1 Substituted pyrimidinones and pyrimidinthiones as crf antagonists
11/04/2004CA2522682A1 Indazole derivatives as jnk inhibitors
11/04/2004CA2522565A1 Hydroxamic acids useful in the treatment of hyper-proliferative disorders
11/04/2004CA2522562A1 2-phenyl-benzimidazol and 2-phenyl-imidazo-`4,5!-pyridine derivatives as checkpoint kinase cds1 (chk2) inhibitors for the treatment of cancer
11/04/2004CA2522476A1 Biaryl substituted thiazoles, oxazoles and imidazoles as sodium channel blockers
11/04/2004CA2522079A1 Quinazoline derivatives for treatment of cancer
11/03/2004EP1472245A2 Heteroaryl compounds useful as inhibitors of gsk-3
11/03/2004EP1472234A1 Quinazolinone derivatives and their use as cb agonists
11/03/2004EP1472230A2 Ansamycins having improved pharmacological and biological properties
11/03/2004EP1472226A1 Heterocyclic amide compounds as apolipoprotein b inhibitors
11/03/2004EP1472221A2 Substituted indoles, method for production and use thereof for the inhibition of pain
11/03/2004EP1472201A2 Method for the separation of acids from chemical reaction mixtures by means of ionic fluids
11/03/2004EP1471915A2 2,4-pyrimidinediamine compounds and their uses
11/03/2004EP1471910A2 Substituted quinazolin-4-ylamine analogues as modulators of capsaicin receptors
11/03/2004EP1471908A1 Process for preparing losartan potassium with improved flowability
11/03/2004EP1232153B1 Imidazole derivatives and their use as raf kinase inhibitors
11/03/2004EP1189883B1 Substituted pyrrolidines as cell adhesion inhibitors
11/03/2004CN1543462A Crystals including a malic acid salt of a 3-pyrrole substituted 2-indolinone, and compositions thereof
11/03/2004CN1543461A Melanocortin receptor ligands
11/03/2004CN1543460A Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests
11/03/2004CN1543459A Quinoline derivatives and quinazoline derivatives having azolyl group
11/03/2004CN1543455A 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same
11/03/2004CN1543453A 6-(aryl-amido or aryl-amidomethyl)-naphthalen-2-yloxy-acidic derivatives as inhibitors of plasminogen activator inhibitor type-1 (PAI-1)
11/03/2004CN1543346A Novel compounds
11/03/2004CN1543311A Selective substituted aryl ketone and safener based herbicides
11/03/2004CN1542002A Inhibitors of metalloproteinase, pharmaceutical compositions containing them, their pharmaceutical application and methods and intermediate compounds for their preparation
11/03/2004CN1541532A Herbicidal synergistic composition, and method of controlling weeds
11/03/2004CN1173972C Azaring-ether derivatives and their use as nicotinic ach receptor modulators
11/03/2004CN1173956C Novel piperazinylalkyl thiopyrimidine derivatives, pharmaceutical compositions containing the same, and a process for the preparation of same
11/03/2004CN1173946C Method for preparing an N-[(aliphatic or aromatic) carbonyl]-2-aminoacetamide compound and a cyclyzed compound
11/02/2004US6812243 Indole derivatives and their use for the treatment of malignant and other diseases based on pathological proliferation
11/02/2004US6812240 8-azaprostaglandin carbonate and thiocarbonate analogs as therapeutic agents
11/02/2004CA2315614C Pyrazoles
11/02/2004CA2301787C New derivatives of benzo[3,4]cyclobuta[1,2-c]pyrrole, the procedure for preparing them and the pharmaceutical compounds that contain them
11/02/2004CA2115536C Heterocyclically substituted phenyl-cyclohexane-carboxylic acid derivatives
10/2004
10/28/2004WO2004092346A2 Small molecule inhibition of a pdz-domain interaction
10/28/2004WO2004092162A1 Inhibitors of serine proteases, particularly hcv ns3-ns4a protease
10/28/2004WO2004092161A1 Inhibitors of serine proteases, particularly hcv ns3-ns4a protease
10/28/2004WO2004092160A1 Bromide and its crystal
10/28/2004WO2004092159A1 Method for synthesising 5-chloro-1-aryl-4-(4, 5-dicyano-1h-imidazol-2-yl)-3-alkyl-1h-pyrazole derivatives
10/28/2004WO2004092140A1 Biaryl substituted pyrazoles as sodium channel blockers
10/28/2004WO2004092132A1 [b]-fused bicyclic proline derivatives and their use for treating arthritic conditions
10/28/2004WO2004092130A2 N-containing heteroaromatic compounds as modulators of ppars and methods of treating metabolic disorders
10/28/2004WO2004078732B1 N-aryl heteroaromatic products, compositions containing same and use thereof
10/28/2004WO2004075823A8 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament
10/28/2004WO2004058721A3 Pyrazole derivatives modulators of hepatocyte growth factor (scatter factor) activity
10/28/2004US20040215023 Crystal and process for producing the same
10/28/2004US20040215019 Substituted isoindoles and the e use thereof
10/28/2004US20040214928 For therapy of proliferative disorders and neurological disorders
10/28/2004US20040214890 1,3-diamino-2-hydroxypropane derivatives are useful as inhibitors of the beta-secretase enzyme that are useful in the treatment of Alzheimer's disease and other diseases characterized by deposition of A beta peptide in a mammal
10/28/2004US20040214874 Inhibition of protein-tyrosine kinase cmet to block cancer cell proliferation, oral bioavailibility; 2-(2,6-dichlorophenyl)-4-phenyl-5-(pyrimidin-4yl)-1H-imidazoles
10/28/2004US20040214857 Substituted benzimidazoles and imidazo-[4,5]-pyridines
10/28/2004US20040214845 Barbiturates as integrin antagonists and their use for treating inflammatory diseases
10/28/2004US20040214843 Such as spiro(cyclohexane-1-4'-(3',4'-dihydro)quinazolin)-2'(1'H)-one for treatment of T-cell-related diseases, autoimmune diseases, osteoarthritis, multiple sclerosis, osteoporosis, asthma and cancer
10/28/2004US20040214841 Quinazoline derivatives for treatment of tumours
10/28/2004US20040214832 Piperazine derivative renin inhibitors
10/28/2004US20040214821 Benzimidazole compounds for modulating IgE and inhibiting cellular proliferation
10/28/2004US20040214820 3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them
10/28/2004US20040214818 Alzheimer's disease; Parkinson's disease; Huntington's disease; cognition activators; learning enhancement; central nervous system disorders
10/28/2004US20040214817 Diaminotriazoles useful as inhibitors of protein kinases
10/28/2004US20040214814 Pyrazole compounds useful as protein kinase inhibitors
10/28/2004US20040214107 optical and electro-optical apparatus comprising recording layer consists of organic pigments and stabilizer agents, and reflection layers formed on light transmitting substrates; sensitivity for red light
10/28/2004CA2522596A1 Process for synthesizing insecticide compounds
10/28/2004CA2522195A1 [b]-fused bicyclic proline derivatives and their use for treating arthritic conditions
10/28/2004CA2521678A1 Inhibitors of serine proteases, particularly hcv ns3-ns4a protease
10/28/2004CA2521135A1 N-containing heteroaromatic compounds as modulators of ppars and methods of treating metabolic disorders
10/28/2004CA2520804A1 Biaryl substituted pyrazoles as sodium channel blockers
10/27/2004EP1471057A1 Pyrimidinylacetic acid derivatives useful for the treatment of diseases mediated by CRTH2
10/27/2004EP1471049A1 Novel thyroid hormone receptor ligand, medicinal compositions containing the same and use thereof
10/27/2004EP1470137A1 Edg receptor agonists
10/27/2004EP1470136A1 Method for the separation of acids from chemical reaction mixtures by means of ionic fluids
10/27/2004EP1470128A1 Intermediates for preparing glycogen phosphorylase inhibitors
10/27/2004EP1470121A1 Pyrimidine derivatives as rho-kinase inhibitors
10/27/2004EP1470119A1 Benzothiophene compounds having antiinfective activity
10/27/2004EP1470114A1 Peptide nucleic acid oligomers from 1-benzenesulfonyl-3-amino acid side chain-4-(2-nucleobase(acetyl))-piperazin-2-ones
10/27/2004EP1469854A1 Condensed heterocyclic compounds
10/27/2004EP1244457B1 Use of modulators of annexin for the manufacture of a medicament for the treatment and/or prevention of arthritis and arthritic diseases
10/27/2004EP1212269B1 Methods for preparing n- (aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds
10/27/2004EP1150952B1 Indole derivatives and their use as mcp-1 receptor antagonists
10/27/2004EP0957100B1 Diamine derivatives and pharmaceutical containing the same
10/27/2004CN1541215A HIV inhibiting pyrimidines derivatives
10/27/2004CN1541206A Substituted dihydro 3-hylo-1H-pyrazoloe-5-carboxylates their prepn. and use
10/27/2004CN1541205A Diamide invertebrate pest control agents contg. non-aromatic heterocyclic ring
10/27/2004CN1541098A Combination therapy for treatment of cancer
10/27/2004CN1541086A Dyeing compson. for kerationous fibres comprising particular dicationic diazo dye
10/27/2004CN1539825A Compounds useful to treat retroviral infections
10/27/2004CN1172672C Alpha-ketoamide multicatalytic protease inhibitors
10/26/2004US6809201 Intercalator suitable for electrochemical detection of double strand DNAs and a process for preparing thereof
10/26/2004US6809199 (Halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
10/26/2004US6809107 Neurodegenerative diseases
10/26/2004US6809102 For therapy of proliferative diseases, such as cancer; to interrupt mitosis
10/26/2004US6809098 Compounds
10/26/2004US6809092 1,3,4,5-tetrahydro-2h-2-benzazepin-2-yl derivatives; cysteine protease inhibitors
10/26/2004CA2132514C Antiproliferative quinazolines