Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
02/2005
02/02/2005EP1501808A1 Tachykinin receptor antagonists
02/02/2005EP1501807A1 Sulfonylquinoxalone acetamide derivatives and related compounds as bradykinin antagonists
02/02/2005EP1501805A1 Substituted pyrazolyl compounds for the treatment of inflammation
02/02/2005EP1501797A1 3-substituted amino-1h-indole-2-carboxylic acid and 3-substituted amino-benzo[b]thiophene-2-carboxylic acid derivatives as interleukin-4 gene expression inhibitors
02/02/2005EP1501796A1 3-substituted amino-1h-indole-2-carboxylic acid and 3-substituted amino-benzo[b]thiophene-2-carboxylic acid derivatives as interleukin-4 gene expression inhibitors
02/02/2005EP1501795A1 Cinnamic acid amides
02/02/2005EP1501787A1 N-biphenylmethyl aminocycloalkanecarboxamide derivatives with a substiituent on the methyl useful as bradykinin antagonists
02/02/2005EP1501515A1 Triaryl-oxy-aryloxy-pyrimidine-2,4,6-trione metalloproteinase inhibitors
02/02/2005EP1501514A2 Protein kinase modulators and methods of use
02/02/2005EP1501467A2 Heterocyclo inhibitors of potassium channel function
02/02/2005EP1297175A4 Methods and compounds for modulating nuclear receptor coactivator binding
02/02/2005EP1292591B1 Substituted bicyclic derivatives for the treatment of abnormal cell growth
02/02/2005EP1286955B1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides
02/02/2005CN1575283A Piperazine derivatives with CCRI receptor antagonist activity
02/02/2005CN1575273A 3, 4-di-substituted cyclobutene-1, 2-diones as CXC-chemokine receptor antagonists
02/02/2005CN1575177A Cxcr3 antagonists
02/02/2005CN1575176A Process for making substituted pyrazoles
02/02/2005CN1575171A Novel anti-diabetic agents
02/02/2005CN1572792A Pyrazolo [4, 3-d] pyrimidine derivatives
02/02/2005CN1187342C Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
02/02/2005CN1187333C Certain substituted caprolactams, pharmaceutical compositions containing them and their use in treating tumors
02/02/2005CN1187326C Novel compounds
02/02/2005CN1187325C Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
02/01/2005US6849739 N-heterocyclic derivatives as NOS inhibitors
02/01/2005US6849713 Topisomerase inhibitor
02/01/2005US6849660 Antimicrobial biaryl compounds
02/01/2005US6849647 Amide compounds and medications containing the same technical field
02/01/2005US6849643 Indazolyl-substituted pyrroline compounds as kinase inhibitors
02/01/2005US6849639 Anticancer agents, antiinflamatory agents, osteoporosis, atherosclerosis
02/01/2005US6849636 Useful for treatment of noninsulin-dependent diabetes, hyperglycemia, obesity, insulin resistance, dyslipidemia, hyperlipidemia, hypertension, Metabolic Syndrome
02/01/2005US6849633 Pyrazole derivative, production process thereof, and pest control agent containing the same as active ingredient
02/01/2005US6849631 Semicarbazides and their uses
02/01/2005US6849629 Heteroaromatic substituted sulfonyl or sulfoxide or thio-pyridazinone derivatives, useful for treating diabetic complications and cardiovascular disorders
02/01/2005US6849622 May be useful for the prophylaxis and treatment of diabetes, particularly type 2 diabetes, and for prophylaxis and treatment of other diseases induced or exacerbated by impaired glucose tolerance
02/01/2005US6849617 Administering Tissue factor pathway inhibitors for prophylaxis of thrombosis and cardiovascular disorders; anticoagulants
02/01/2005US6849367 Photoconductive layer containing azo compound; electrostaticlatent image
02/01/2005CA2166326C Pyridazinone derivatives
01/2005
01/27/2005WO2005007649A1 Improved process for preparing alpha-polymorphic eletriptan hydrobromide
01/27/2005WO2005007648A2 Biaryl piperazinyl-pyridine analogues
01/27/2005WO2005007647A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
01/27/2005WO2005007633A1 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
01/27/2005WO2005007625A2 Heterocyclic amides with anti-tuberculosis activity
01/27/2005WO2005007165A1 Pyrimidine-2, 4-dione derivatives as gonadotropin-releasing hormone receptor antagonists
01/27/2005WO2005007157A1 Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases
01/27/2005WO2004101512A3 Naphthyridine integrase inhibitors
01/27/2005WO2004098518A3 Pyrazole-amide compounds useful as kinase inhibitors
01/27/2005WO2004069794B1 New arylpiperazinyl compounds
01/27/2005WO2004064741A3 Compounds, compositions, and methods
01/27/2005US20050020857 Method for the separation of acids from chemical reaction mixtures by means of ionic fluids
01/27/2005US20050020663 Improved preparation of alpha -polymorphic eletriptan hydrobromide, by salt formation in a solution of 2-butanone and water, distillation, dehydration, desolventizing; purity, white color crystals
01/27/2005US20050020661 Antidiabetic agents
01/27/2005US20050020659 Substituted pyrazole derivatives and related compounds as bradykinin B1 receptor antagonists
01/27/2005US20050020655 Transamination of ondansetron by a Mannich reaction
01/27/2005US20050020654 Novel PPAR agonists, pharmaceutical compositions and uses thereof
01/27/2005US20050020653 Imidazolyl or benzimidazolyl derivatives of triazole compounds substituted at 2 position; anti-fungal agent with broad spectrum activity useful in the treatment of fungal infections in animals, including humans and as agricultural fungicides
01/27/2005US20050020652 For example, 2-(4-{2-[1-(4-tert-Butyl-benzyl)-3-methyl-2-oxo-imidazolidin-4-yl]-ethoxy}-2-methyl-phenoxy)-2-methyl-propionic acid, 2-(4-{3-[1-(4-tert-Butyl-benzyl)-3-methyl-2-oxo-imidazolidin-4-yl]-propyl}-2-methyl-phenoky)-2-methyl-propionic acid; for treating diabetes mellitus
01/27/2005US20050020617 3-substituted oxindole beta3 agonists
01/27/2005US20050020604 5-HT receptor ligands and uses thereof
01/27/2005US20050020601 Novel pyrazinones as CRF1 receptor antagonists
01/27/2005US20050020586 Using 4-imidazoline ester or acid; antiinflammatory agents; microbiocides; bactericides; antitumor agents; autoimmune disease
01/27/2005US20050020578 Oxidoreductase enzyme inhibitors such as (R)-1-[4-(2-methyl-4-phenyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-pyrimidin-2-yl-ethanol, used as antidiabetic agents
01/27/2005US20050020576 Opioid antagonist; analgesics; antiinflammatory agents; side effect reduction
01/27/2005US20050020573 5HT2c receptor modulators
01/27/2005CA2532316A1 Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases
01/27/2005CA2532152A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
01/27/2005CA2532111A1 Improved process for preparing alpha-polymorphic eletriptan hydrobromide
01/27/2005CA2531619A1 Biaryl piperazinyl-pyridine analogues
01/27/2005CA2531508A1 Pyrimidine-2, 4-dione derivatives as gonadotropin-releasing hormone receptor antagonists
01/27/2005CA2529790A1 Heteroaryloxy nitrogenous saturated heterocyclic derivative
01/26/2005EP1500657A1 Substituted pyrazoles as P38 kinase inhibitors
01/26/2005EP1500655A1 New methionine aminopeptidase inhibitor
01/26/2005EP1500653A1 Substituted arylpyrazines
01/26/2005EP1500652A1 Quinazoline derivative and medicine
01/26/2005EP1499623A1 Process for preparing 1,2,3,9-tetrahydro-9-methyl-3-[(2-methyl-1h-imidazol-1-yl)methyl]-4h-carbazol-4-one
01/26/2005EP1499608A1 Substituted imidazole derivatives: gaba a receptor ligands
01/26/2005EP1499599A1 Substituted pyrazine derivatives
01/26/2005EP1499598A1 Chemical compounds with dual activity, processes for their preparation and pharmaceutical compositions
01/26/2005EP1499597A2 Compounds and methods for inducing apoptosis in proliferating cells
01/26/2005EP1499591A1 Carboxylic acid amides
01/26/2005EP1499577A1 2-(2,6-dichlorophenyl)-diarylimidazoles
01/26/2005EP1499319A1 Bicyclo 4.4.0 antiviral derivatives
01/26/2005EP1499305A2 Use of ep4 receptor ligands in the treatment of il-6 involved diseases
01/26/2005EP1379522B1 DIHYDRO-BENZO(b)(1,4)DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS I
01/26/2005EP1373255B1 Process for the preparation of imidazole compounds
01/26/2005EP1296976B1 Novel 1,3-dihydro-2h-indol-one derivatives, method for preparing same and pharmaceutical compositions containing them
01/26/2005EP0844877B1 Use of oxido-squalene cyclase inhibitors to lower blood cholesterol
01/26/2005CN1571783A Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same
01/26/2005CN1571781A 4-imidazolin-2-one compounds
01/26/2005CN1571774A Pyrimidinones as melanin concentrating hormone receptor 1
01/26/2005CN1571667A Inhibitors of dipeptidyl peptidase ó¶
01/26/2005CN1186339C Pyrimidinyl methyl indole derivatives with antibacterial activity
01/26/2005CN1186328C Substd. 5-benzyl-2, 4-diaminopyrimidines
01/26/2005CN1186326C Propane-1, 3-dione derivatives
01/26/2005CN1186322C Proline derivatives and use thereof as drugs
01/25/2005US6846929 A hydroxyphenyl-2-benzotriazoles as light stabilizers having ultraviolet light absorbing activity; stabilizer with heat resistance, photostability, oxidation resistance
01/25/2005US6846928 Compositions useful as inhibitors of protein kinases
01/25/2005US6846840 Alkylating agents possessing both in vitro cytotoxicity and antitumor activity; for therapy of cancer
01/25/2005US6846839 Identifying indolinone compounds that inhibit growth factor stimulated cell proliferation by contacting cells with compounds and with selected growth factors and monitoring inhibitory effect
01/25/2005US6846834 Antiinflammation agents
01/25/2005US6846833 Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same