Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
10/2004
10/14/2004US20040204410 Such as 1-(4,5-Bis-(4-chloro-phenyl)-2-(2,4-dimethoxy-phenyl)-4,5-dihydro-imidazol-1-yl)-2-methyl-propan-1-one which inhibits the interaction of MDM2 protein with p53-like peptide; antiproliferative agents
10/14/2004US20040204407 5-sulfonamido-substituted indolinone compounds as protein kinase inhibitors
10/14/2004US20040204395 Water-soluble drugs and methods for their production
10/14/2004US20040204386 for uses such as inhibiting the activity of lysophosphatidic acid acyltransferase beta and/or inhibiting the proliferation of a cell (e.g., tumor cell)
10/14/2004US20040204347 administering an effective amount of an inhibitor of the interaction of glutamate with the alpha -amino-3-hydroxy-5-methyl-4-isoxazole-propionate (AMPA) receptor complex to treat demyelinating disorders
10/14/2004US20040204257 System for and a method of manufacturing personal golf putters
10/14/2004US20040202098 Squarylium-metal chelate compounds and optical recording media
10/14/2004DE10315573A1 Substituierte Pyrazole Substituted pyrazoles
10/14/2004DE10315572A1 Substituierte Pyrazole Substituted pyrazoles
10/14/2004DE10315571A1 Pyrazolverbindungen Pyrazole
10/14/2004DE10315569A1 Substituierte Pyrazolverbindungen Substituted pyrazole
10/14/2004DE10315377A1 New carbonyl-substituted carbocyclic or heterocyclic compounds, are factor Xa and factor VIIa inhibitors useful e.g. for treating thrombosis, myocardial infarction, arteriosclerosis, inflammation or tumors
10/14/2004CA2520896A1 Indole acetamides as inhibitors of the hepatitis c virus ns5b polymerase
10/14/2004CA2520894A1 Pyrazolidine-1,2-dicarboxyldiphenylamide derivatives as coagulation factor xa inhibitors for the treatment of thromboses
10/14/2004CA2520281A1 Benzimidazole derivatives and their use for modulating the gabaa recept or complex
10/14/2004CA2519954A1 Benzamide modulators of metabotropic glutamate receptors
10/14/2004CA2519515A1 Benodiazepine spirohydantoin cgrp receptor antagonists
10/14/2004CA2518913A1 Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof
10/14/2004CA2518465A1 Dipeptidyl peptidase inhibitors
10/13/2004EP1466902A1 Androgen receptor antagonists
10/13/2004EP1466603A2 Novel catechols as antimicrobial agents
10/13/2004EP1465891A2 Inhibitors of dipeptidyl peptidase iv
10/13/2004EP1465889A1 Chemokine receptor binding heterocyclic compounds with enhanced efficacy
10/13/2004EP1465888A2 Melanin concentrating hormone receptor ligands: substituted benzoimidazole analogues
10/13/2004EP1465887A1 Novel crystal forms of ondansetron, processes for their preparation, pharmaceutical compositions containing the novel forms and methods for treating nausea using them
10/13/2004EP1465880A1 5-sulphanyl-4h-1,2,4-triazole derivatives and their use as medicine
10/13/2004EP1465875A1 Novel alkansulfonamides as endothelin antagonists
10/13/2004EP1465872A1 4-sulfide/sulfoxide/sulfonyl-1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
10/13/2004EP1465871A1 Pyrazole derivatives for use in diseases associated with the 5-ht2c receptor
10/13/2004EP1465867A1 Ligands of melanocortin receptors and compositions and methods related thereto
10/13/2004EP1465866A2 Protease inhibitors of the coagulation cascade isolated from dysidea sponges
10/13/2004EP1465864A1 Inhibitors of factor xa and other serine proteases involved in the coagulation cascade
10/13/2004EP1465635A2 Melanin concentrating hormone receptor ligands: substituted 2-(4-benzyl-piperazin-1-ylmethyl)- and 2-(4-benzyl-diazepan-1-ylmethyl)-1h-benzoimidazole analogues
10/13/2004EP1465631A2 Pyrimidine a2b selective antagonist compounds, their synthesis and use
10/13/2004EP1465629A1 5-ht3 receptor antagonists and methods of use
10/13/2004EP1397137A4 Hydantion derivatives as inhibitors of matrix metalloproteinases
10/13/2004EP1322309A4 High affinity small molecule c5a receptor modulators
10/13/2004EP1280797B1 Inhibitors of dipeptidyl peptidase iv
10/13/2004EP1165533B1 Compounds and methods for treatment of asthma, allergy and inflammatory disorders
10/13/2004EP1086086B1 Imidazolyl derivatives and their use as somatostatin receptor ligands
10/13/2004CN1537105A Quinazolines as MMP-13 inhibitors
10/13/2004CN1535965A cyanine compound, filter and optical recording material
10/13/2004CN1170842C New amidinobenzylamine derivatives and their use as thrombin inhibitors
10/13/2004CN1170826C Amide compounds
10/12/2004US6803455 Inhibitors of nucleoside metabolism
10/12/2004US6803374 Compounds useful for treating hepatitis C virus
10/12/2004US6803362 Heterocyclic compounds
10/07/2004WO2004085428A1 A new process for preparing olmesartan medoxomil
10/07/2004WO2004085426A1 Novel crystalline forms of candesartan cilexetil
10/07/2004WO2004085425A1 Fused azoles such as 2,5-disubstituted benzimidazoles, benzoxazoles and benzothiazoles as kinase inhibitors
10/07/2004WO2004085409A2 Compounds and libraries of pyridines, pyrazines, imidazo[1,2-a]pyrazines and 1h-imidazo[4,5-b]pyrazin-2-ones and first and second medical uses thereof
10/07/2004WO2004085401A1 1,2,4-substituted 1,2,3,4-tetrahydro-and 1,2 dihydro-quinoline and 1,2,3,4-tetrahydro-quinoxaline derivatives as cetp inhibitors for the treatment of atherosclerosis and obesity
10/07/2004WO2004085392A1 Melatonin derivatives and their use for treating neurological dysfunctions
10/07/2004WO2004084901A1 Methods for treating or preventing an inflammatory or metabolic condition by inhibiting jnk
10/07/2004WO2004084898A1 2-phenoxy- and 2-phenylsulfomamide derivatives with ccr3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders
10/07/2004WO2004084824A2 Biaryl substituted 6-membered heterocyles as sodium channel blockers
10/07/2004WO2004084813A2 Chemical compounds
10/07/2004WO2004075823A3 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament
10/07/2004WO2004026829A3 Heterocyclically substituted indolinones and their use as receptor tyrosine kinase inhibitors
10/07/2004WO2003068757A9 Novel pyridin- and pyrimidin-derivatives
10/07/2004US20040198987 Substituted dihydro 3-halo-1h-pyrazole-5-carboxylates their preparation and use
10/07/2004US20040198986 Chemical compounds
10/07/2004US20040198979 antagonists of urotensin II; (R) N-[4-Chloro-3-(1-methyl-3-pyrrolidinyloxy)-phenyl]-[3-(2-chlorophenoxy)]benzenesulfonamide for example; treating various disease including cardiovascular disorders, gastrointestinal disorders, and psychological disorders
10/07/2004US20040198804 i.e., 3-[3,5-dimethyl-4-[3-oxo-3-(piperazin-1-ylpropyl]-1H-pyrrol-2-ylmethylene]-1,3-dihydroindol-2-one, in which the piperazine may be 4-substituted with methyl or ethyl and salts are tyrosine kinase inhibitors used to treat various kinds of cancer
10/07/2004US20040198802 Antiproliferative agents
10/07/2004US20040198799 Methods of increasing endogenous testosterone levels
10/07/2004US20040198796 Compounds and methods for treating urinary incontinence
10/07/2004US20040198794 Ondansetron forms and processes of making the same
10/07/2004US20040198790 Triazole compound containing a phosphonate group
10/07/2004US20040198787 Efficient process for the preparation of a factor Xa inhibitor
10/07/2004US20040198740 Therapies relating to combinations of aldose reductase inhibitors and cyclooxygenase-2
10/07/2004US20040198739 Prevention reproduction of virus
10/07/2004US20040198735 Sulfonyl heteroaryl triazoles as anti-inflammatory/analgesic agents
10/07/2004US20040198734 2-(4-Aryl or heteroaryl-piperazin-1-ylmethyl)-1H-indole derivatives interacting with the dopamine
10/07/2004US20040198733 Obesity; antidiabetic agents; cardiovascular disorders; antilipemic agentsl circadian rhythm disorders; hypotensive agents; antidepressants; anxiolytic agents
10/07/2004US20040198732 Aminoalkyl-substituted aromatic bicyclic compounds, methods for their preparation and their use as pharmaceuticals
10/07/2004US20040198731 Antidiabetic agents; cardiovascular disorders; anticholesterol agents; antidepressants; schizophrenia; antilipemic agents; circidian rhythm disorders
10/07/2004US20040198730 Pyridylfurans and pyrroles as raf kinase inhibitors
10/07/2004US20040198720 3-(Arylamino)methylene-1, 3-dihydro-2H-indol-2-ones as kinase inhibitors
10/07/2004US20040198700 Administering to a patient an azetidinone compound containing at least 3 phenyl rings fo rprevention of a vascular condition, diabetes, obesity, stroke, lowering a concentration of a sterol or stanol in plasma of a mammal, preventing demyelination or treating Alzheimer's disease
10/07/2004US20040197705 Cyanide compound, optical filter, and optical recording material
10/07/2004CA2520440A1 Methods for treating or preventing an inflammatory or metabolic condition by inhibiting jnk
10/07/2004CA2520405A1 1,2,4-substituted 1,2,3,4-tetrahydro-and 1,2 dihydro-quinoline and 1,2,3,4-tetrahydro-quinoxaline derivatives as cetp inhibitors for the treatment of atherosclerosis and obesity
10/07/2004CA2519677A1 Biaryl substituted 6-membered heterocycles as sodium channel blockers
10/07/2004CA2518909A1 Heterocyclic compounds and methods of use
10/06/2004EP1464678A1 Cyanine compound, optical filter, and optical recording material
10/06/2004EP1464645A1 Indole derivative
10/06/2004EP1464641A1 4-Phenyl-piperazinyl, -piperidinyl and tetrahydropyridyl derivatives as dopamine D4 antagonists
10/06/2004EP1464335A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist
10/06/2004EP1463724A1 Pyrrolidone carboxamides
10/06/2004EP1463716A1 Pyrrolidine and piperidine derivates as nk1 antagonists
10/06/2004EP1463714A2 Vanilloid receptor ligands and their use in treatments
10/06/2004EP1463506A1 Substituted quinazoline derivatives as inhibitors of aurora kinases
10/06/2004EP1463505A2 3-(phenyl-alkoxy)-5-(phenyl)-pyridine derivatives and related compounds as kinase inhibitors for the treatment of cancer
10/06/2004EP1185521B1 Substituted 1-aza-2-imino-heterocycles and their use as activators of nicotinic acetylcholine receptors
10/06/2004EP1165516B1 Heterocyclic urea and related compounds useful as anti-inflammatory agents
10/06/2004EP1144403B1 Substituted pyrazoles as p38 kinase inhibitors
10/06/2004EP1064270B1 Disubstituted pyrazolines and triazolines as factor xa inhibitors
10/06/2004EP1032424B9 Combination of an aldose reductase inhibitor and a glycogen phosphorylase inhibitor
10/06/2004EP1027336B1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors