Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
09/2004
09/23/2004WO2004052304A3 Antibacterial compounds having a (pyrrole carboxamide)-(benzamide)-(imidazole carboxamide) motif
09/23/2004WO2004030637A3 Treatment of obesity and other disorders associated with excessive food intake
09/23/2004US20040186295 G protein-coupled receptors activators such as 2-[2-(3-chlorophenyl)-2H-tetrazol-5-yl]pyridine, used as analgesics, anxiolytic, antidepressants, and for prophylaxis of psychological disorders
09/23/2004US20040186161 Prodrugs of a 3-(pyrrol-2-ylmethylidene)-2-indolinone derivatives
09/23/2004US20040186160 for treating an abnormal condition associated with protein kinase activity such as cell proliferation, differentiation apoptosis and inhibiting protein kinase signal transduction
09/23/2004US20040186159 used to treat glaucomatous optic neuropathy and/or lower and control intraocular pressure (IOP) associated with normal-tension glaucoma, ocular hypertension, and/or glaucoma in warm blooded animals, including man
09/23/2004US20040186156 useful for solid tumors and leukemia; auto-immune diseases such as psoriasis, alopecia and multiple sclerosis; cardiovascular diseases such as stenoses, arterioscleroses and restenoses; infectious diseases caused by unicellular parasites; nephrological diseases, neurodegenerative diseases
09/23/2004US20040186154 treating or preventing a hypercholesterolemia-related or an inflammation-related condition ; apical sodium co-dependent bile acid transport inhibitor and an amount of a cyclooxygenase-2 (COX-2) selective inhibitor or its prodrug; kits
09/23/2004US20040186153 Pharmaceutical use of N-carbamoylazole derivatives
09/23/2004US20040186151 E.g., 2-[3-(4'-Methoxyphenyl)-propionylamino]-2-(4'-n-butoxy-3'-carboxyphenyl)-2-ethyl[4-(4'-nitrophenyl)]imidazole; inhibitors of protein tyrosine phosphatases; antidiabetic, -carcinogenic, -inflammation agents; antiallergens; infections; modulation of growth hormones/factors; Alzeimer's; obesity
09/23/2004US20040186146 E.g., R-N-2-[4-(pyrrolidin-1'-yl)methylphenyl]propionyl-methanesulfonamide; inhibition of chemotaxis of neutrophils induced by interleukin-8; antiinflammatory agents; psoriasis, ulcerative cholitis, glomerular nephritis, acute respiratory insufficiency, idiopathic fibrosis, and rheumatoid arthritis
09/23/2004US20040186140 Cyclic derivatives as modulators of chemokine receptor activity
09/23/2004US20040186129 2-Aroylimidazole compounds for treating cancer
09/23/2004US20040186125 E.g , 3-cyclohexyl-2-furan-3-yl-1Hindole-5-carboxylic acid; hepatitis C viricides that target RNA dependent RNA polymerases (Ns5B) in mammals, an enzyme essential to viral replication; used in conjunction with an mmunomodulatory agent, such as beta -, delta - gamma -, and omega -interferon
09/23/2004US20040186119 glycogen synthase kinase (GSK-3) inhibitors; for treatment of diabetes and alzheimer's disease
09/23/2004US20040186118 Chk-, Pdk- and Akt-inhibitory pyrimidines, their production and use as pharmaceutical agents
09/23/2004US20040186114 Cytokine inhibitors
09/23/2004US20040186111 Therapeutic agents useful for treating pain
09/23/2004US20040186110 Nitrogenous heterocylic compounds
09/23/2004US20040186106 such as (S)-N-{{(1R, 2R)-2-{4-{[2-(4-Methyl-piperazin-1-yl)-benzimidazol-1-yl]methyl}-phenyl}-cyclohex-1-yl} carbonyl}-phenylglycinamide; for treatment of ischemic brain disorders
09/23/2004US20040186098 Method for preventing and treating hearing loss using sensorineurotrophic compounds
09/23/2004US20040186088 Mercapto-cycloalkyl or heterocyclyl ring-sulfonyl-aryl or heteroaryl derivatives; preventing the cleavage Of tumor necrosis factor- alpha from cell membranes in mammal; treating autoimmune diseases, inflammation, inflammatory bowel disease, Crohn's disease, asthma, sepsis and septic shock
09/23/2004US20040186076 Pharmaceutical complex
09/23/2004US20040185352 Photothermographic element comprising improved base precursors and methods for their use
09/23/2004DE10311065A1 New 1-(cyclic amino-alkyl)-pyrimidin-2(1H)-one derivatives, are selective dopamine D3 receptor ligands useful for treating CNS disorders, especially schizophrenia or depression
09/23/2004DE10310278A1 New N-(benzazinyl)-(hetero)aralkylamine derivatives, are inhibitors of factor Xa and/or related serine proteases, useful e.g. as antithrombotic agents and intermediates
09/23/2004CA2518986A1 Imino ether derivative compounds and drugs containing the compounds as the active ingredient
09/23/2004CA2517885A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors
09/23/2004CA2515289A1 Weak base salts
09/22/2004EP1460066A1 Piperazine compounds
09/22/2004EP1458713A1 Indolinone derivatives useful as protein kinase inhibitors
09/22/2004EP1458712A2 Novel compounds
09/22/2004EP1458711A1 Use of oxindole derivatives in the treatment of dementia related diseases, alzheimer s disease and conditions associated with glycogen synthase kinase-3
09/22/2004EP1458710A1 Heteroaryl substituted pyrrole modulators of metabotropic glutamate receptor-5
09/22/2004EP1458707A2 New compounds
09/22/2004EP1458693A1 Amorphous and crystalline forms of losartan potassium and process for their preparation
09/22/2004EP1458691A2 Benzodiazepine derivatives, preparation thereof and use thereof
09/22/2004EP1458687A2 Pyrimidine compounds
09/22/2004EP1458685A2 Substituted phenyl derivatives
09/22/2004EP1458394A1 Use of oxindole derivatives in the treatment of dementia related diseases, alzheimer s disease and conditions associated with glycogen synthase kinase-3
09/22/2004EP1458393A1 Substituted diketopiperazines as oxytocin antagonists
09/22/2004EP1458386A1 Aroyl pyrrole heteroeryl and methanols useful for treating a central nervous system disorder
09/22/2004EP1458383A2 Heteroaryl substituted pyrazole modulators of metabotropic glutamate receptor-5
09/22/2004EP1458381A1 Triazoles as oxytocin antagonists
09/22/2004EP1458380A1 Cis-2,4,5- triphenyl-imidazolines and their use in the treatment of tumors
09/22/2004EP1458379A1 Hydroxyphenyl-pyrazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
09/22/2004EP1458375A2 Compositions for decreasing activity of hormone-sensitive lipase
09/22/2004EP1458374A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/22/2004EP1379527B1 Epindolidione pigments
09/22/2004EP1169320B1 Farnesyl transferase inhibitors having a pyrrole structure and process for preparation thereof
09/22/2004EP1140860B1 Pyrimidine compounds
09/22/2004EP0914321B1 Indole derivatives for the treatment of osteoporosis
09/22/2004EP0830347B1 Novel substituted piperazine derivatives having tachykinin receptor antagonists activity
09/22/2004CN1531527A Carbazole derivatives and their use as neuropeptide Y5 receptor ligands
09/22/2004CN1167699C Extraction process of chlorhematin as iron-replenishing agent
09/22/2004CN1167698C New N-triazolyl methyl piperazine derivative using as neurokinin receptor antagonistic agent
09/22/2004CN1167687C Arylpyridazinones as prostaglandin endoperoxide H synthase biosynthesis inhibitors
09/22/2004CN1167686C Novel benzimidazole derivatives and pharmaceutical compsns. comprising these compounds
09/22/2004CN1167683C Aromatic pyrozole compound, its preparation, agricultural composition containnig it and use thereof
09/22/2004CN1167680C Fused-ring compounds and use thereof as drugs
09/22/2004CN1167422C Quinazoline derivatives as angiogenesis inhibitors
09/21/2004US6794506 Treatment of inflammatory diseases, such as asthma, alzheimer's disease, atherosclerosis, aids dementia, diabetes, inflammatory bowel disease, rheumatoid arthritis, tissue transplantation, tumor metastasis
09/21/2004US6794406 For therapy and prophylaxis of arteriosclerosis and hypercholesterolaemia
09/21/2004US6794404 Viral polymerase inhibitors
09/21/2004US6794395 Substituted indolinones, their manufacture and their use as medicaments
09/21/2004US6794379 Antiinflammatory agents; autoimmune disease; skin disorders
09/21/2004US6794359 Vertebrate intestinal protein which absorbs cholesterol, its inhibitors and mehtod of identifying the same
09/21/2004CA2114017C Amide tetrazole acat inhibitors
09/16/2004WO2004079434A2 Vapor deposited electro-optic films self-assembled through hydrogen bonding
09/16/2004WO2004078943A2 Alternative heterocycles for dna recognition
09/16/2004WO2004078752A1 Arylvinylazacycloalkane compounds and methods of preparation and use thereof
09/16/2004WO2004078744A2 Urea derivatives and their use as vanilloid receptor antagonists in the treatment of pain
09/16/2004WO2004078733A1 Quinazolines useful as modulators of ion channels
09/16/2004WO2004078732A1 N-aryl heteroaromatic products, compositions containing same and use thereof
09/16/2004WO2004078731A1 Quinoline-carboxylic acids and the derivatives thereof, a focused library
09/16/2004WO2004078722A1 Organic compound and organic electroluminescence device
09/16/2004WO2004078116A2 P38 inhibitors and methods of use thereof
09/16/2004WO2004050653A3 Oxime ester photoinitiators with heteroaromatic groups
09/16/2004WO2004046101A3 Cyanoguanidines and cyanoamidines as erbb2 and egfr inhibitors
09/16/2004WO2004026264A3 Novel aromatic compounds possessing antifungal or antibacterial activity
09/16/2004WO2003094839A3 Pyrimidinone compounds, compositions and methods
09/16/2004WO2003028729A3 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
09/16/2004US20040181076 Reaction of carbazolone, forrmaldehyde and amine compound in nonaqueous solution and bonding to water, solvent
09/16/2004US20040181062 Benzimidazole cyclooxygenase-2 inhibitor
09/16/2004US20040181059 Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
09/16/2004US20040180945 in particular, strains of the HIV that have developed cross resistance to other anti-HIV drugs
09/16/2004US20040180925 such as (S)-1-[2-(2-Pyrazinylamino)ethylamino]acetyl-2-pyrrolidinecarbonitrile dimethanesulfonate
09/16/2004US20040180914 5-Cyano-2-aminopyrimidine derivatives
09/16/2004US20040180912 for promoting the release of parathyroid hormone, e.g. for preventing or treating bone conditions which are associated with increased calcium depletion or resorption or in which stimulation of bone formation and calcium fixation in the bone is desirable
09/16/2004US20040180906 Anti-inflammatory medicaments
09/16/2004US20040180901 Arylpiperazines and arylpiperidines and their use as metalloproteinase inhibiting agents
09/16/2004US20040180896 P38 inhibitors and methods of use thereof
09/16/2004US20040180892 control of cardiovascular homeostasis is achieved through a combination of both direct neuronal control and systemic neurohormonal activation
09/16/2004US20040180891 Pyrazole derivatives useful in the treatment of hyper-proliferative disorders
09/16/2004US20040180888 Phenylindoles for the treatment of HIV
09/16/2004US20040180887 N-aroyl cyclic amine derivatives as orexin receptor antagonists
09/16/2004US20040180885 Indole derivatives, process for preparation of the same and use thereof
09/16/2004US20040180882 Small molecule modulators of hepatocyte growth factor (scatter factor) activity
09/16/2004US20040180878 Phenylsulfonyl-1,3-dihydro-2h-indole-2-one derivatives, their preparation and their therapeutic use
09/16/2004DE20320528U1 Neue Kristallformen von Ondansetron und Arzneimittel, welche die neuen Formen enthalten New crystal forms of ondansetron and pharmaceutical compositions containing the new forms