Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
02/2005
02/10/2005US20050032869 Antitumor, anticarcinogenic, antiproliferative, and antimetastasis agents; tyrosine kinase inhibitors; autoimmune, nervous system, neurodegenerative, and skin disorders; neurofibromatosis, atherosclerosis, graft versus host disease, glomerulonephritiis, hyperplasia; angiogenesis inhibitors
02/10/2005US20050032868 Selected substituted pyrazole derivatives and related compounds as bradykinin B1 receptor antagonists
02/10/2005US20050032862 Preparing a novel crystal form by sonication and temperature oscillation of a suspension; filtered and dried faster; treating cardiovascular disorders
02/10/2005US20050032810 Novel anthelmintic and insecticidal compositions
02/10/2005US20050032809 5-HT receptor ligands and uses thereof
02/10/2005US20050032805 Antimicrobial biaryl compounds
02/10/2005US20050032792 Peptidyl spiroheterocyclic, amidino and guanidino compounds; reversible inhibitors of the cysteine protease cathepsin S, K, F, L and B; useful in the treatment of autoimmune and other related diseases
02/10/2005US20050032791 Derivatives of sulphonamides, their preparation and use as medicaments
02/10/2005US20050032790 For example, 1-(2-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4,4'-bispiperidine; for treatment of thrombosis, emphysema, cirrhosis; antiarthritic agents, anticancer agents, antihistamines
02/10/2005US20050032772 Compounds useful as reversible inhibitors of cysteine proteases
02/10/2005US20050032752 8-Azaprostaglandin carbonate and thiocarbonate analogs as therapeutic agents
02/10/2005US20050031993 Cyanine compound, optical recording material, and optical recording medium
02/10/2005US20050031899 Carbazole derivative, organic semiconductor element, light emitting element, and electronic device
02/10/2005DE10331675A1 Hetarylsubstituierte Pyrazolidindion-Derivate Hetarylsubstituierte pyrazolidindione derivatives
02/10/2005CA2534649A1 Bicyclic imidazol derivatives against flaviviridae
02/10/2005CA2534451A1 Angiotensin ii receptor blocker derivatives
02/10/2005CA2534038A1 Inhibitors of akt activity
02/10/2005CA2533901A1 Piperazine derivatives and their use as therapeutic agents
02/10/2005CA2533474A1 2-aminophenyl-4-phenylpyrimidines as kinase inhibitors
02/10/2005CA2533102A1 Method for characterising polypeptides by maldi-tof mas spectrometry
02/10/2005CA2532965A1 3, 4-disubstituted 1h-pyrazole compounds and their use as cyclin dependent kinases (cdk) and glycogen synthase kinase-3 (gsk-3) modulators
02/09/2005EP1505125A1 Cyanine compound, optical recording material, and optical recording medium
02/09/2005EP1505064A1 2-Aminopyrimidine derivatives
02/09/2005EP1505063A1 Benzimidazole derivatives
02/09/2005EP1505061A1 Compound exhibiting pgd 2 receptor antagonism
02/09/2005EP1504008A1 7-aminoimidazotriazones
02/09/2005EP1503996A1 Aryl ketone pyrrolo-triazine compounds useful as kinase inhibitors
02/09/2005EP1503994A1 Substituted (thioxo)carbonylamino phenyl uraciles
02/09/2005EP1503993A2 Compounds, methods and compositions
02/09/2005EP1503991A1 Hexahydro-pyridazine-3-carboxylic acid derivatives, pharmaceutical compositions containing same and preparation methods thereof
02/09/2005EP1503988A2 Fredericamycin derivatives
02/09/2005EP1503761A1 Substituted piperazines as melanocortin receptor ligands
02/09/2005EP1503754A1 Beta-agonist compounds comprising nitric oxide donor groups and reactive oxygen species scavenger groups and their use in the treatment of respiratory disorders
02/09/2005EP1430047B1 Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same
02/09/2005EP1430034B1 Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same
02/09/2005EP1414816B1 Stable polymorph of flibanserin, technical process for its preparation and the use thereof for preparing medicaments
02/09/2005EP1349839B1 Phenylethenyl or phenylethinyl derivatives as glutamate receptor antagonists
02/09/2005EP1105376B1 Oxindole derivatives as growth hormone releasers
02/09/2005CN1578773A Methods and compositions of novel triazine compounds
02/09/2005CN1578663A Inhibitors of histone deacetylase
02/09/2005CN1576275A Substituted bicyclic derivatives for the treatment of abnormal cell growth
02/09/2005CN1575816A Compounds for the treatment of female sexual dysfunction
02/09/2005CN1188408C Process for extracting heme from animal blood
02/09/2005CN1188407C Imidazole derivatives with farnesyl transferase to inhibite activity and preparing method thereof
02/09/2005CN1188399C New pyrazolone compound and eye plastic lens made therefrom
02/08/2005US6852752 Urea compounds, compositions and methods of use and preparation
02/08/2005US6852749 Pyrazolidinol compounds
02/08/2005US6852748 Derivatives of 6,7-dihydro-5H-imidazo(1,2- alpha )imidazole-3- sulfonyl)-pyrrolidine-2-carboxylic acid amide which exhibit good inhibitory effect upon the interaction of CAMs and Leukointegrins and are thus useful in the treatment
02/08/2005US6852745 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
02/08/2005US6852743 Preventives for the recurrence of cerebrovascular failure and agents for ameliorating troubles following cerebrovascular failure and inhibiting progress thereof
02/08/2005US6852726 Such as 1-(4,5-dihydro-1H-imidazol-2-ylmethyl)-3-methanesulfonyl-2-methyl-1H-indole for preventing/treating disorders modulated by alpha-1A/L adrenoceptors such as urinary incontinence and sexual disorders
02/08/2005US6852725 Imidazolyl derivatives
02/08/2005US6852717 Inhibit the release of inflammatory cytokines such as interleukin-1 and tumor necrosis factor; for use in therapy of diseases and pathological conditions involving inflammation such as chronic inflammatory disease
02/08/2005US6852712 Controlling cell differentiation; antiinflammatory agents
02/08/2005CA2112081C Imidazole compounds, their preparation and use
02/08/2005CA2097208C The sulphate salt of a substituted triazole, pharmaceutical compositions thereof, and their use in therapy
02/03/2005WO2005009993A1 Novel compounds
02/03/2005WO2005009992A1 Cyclohexanecarboxylic acid compound
02/03/2005WO2005009978A1 2-aminopyrimidine and 2-aminopyridine-4-carbamates for use in the treatment of autoimmune diseases
02/03/2005WO2005009975A2 Benzimidazole derivatives as mek inhibitors
02/03/2005WO2005009973A1 5-membered heterocycle-based p38 kinase inhibitors
02/03/2005WO2005009968A1 Quinoline derivates and their use in therapy
02/03/2005WO2005009957A1 Tyrosine kinase inhibitors
02/03/2005WO2005009435A1 Aminopyrazole compounds and use as chk1 inhibitors
02/03/2005WO2004106307A3 Novel imidazole derivatives, the production thereof, and the use of the same as a medicament
02/03/2005WO2004075840A3 Selective non-steroidal glucocorticoid receptor modulators
02/03/2005US20050027121 Heterocyclic carboxy amines such as (2R)-1-[3,5-Bis(trifluoromethyl)benzoyl]-4-[4-((3S)-3-ethylmorpholino)-2-butynyl]-2-[(1H-indol-3-yl)methyl]piperazine, used as substance P and neurokinin antagonist for prophylaxis of diseases
02/03/2005US20050026989 treatment or prophylaxis of cardiovascular disease, metabolic disease, cancerous disease, or fibrotic disease; arrhythmias, life-threatening cardiac ventricular fibrillation, myocardial infarction, angina pectoris; ischemic states of the heart, diabetes
02/03/2005US20050026987 CBI analogues of the duocarmycins and CC-1065
02/03/2005US20050026985 Such as N-{5-[1-(4-tert-butylphenyl)-3-pyridin-2-yl-1H-pyrazol-5-yl]pentanoyl}tyrosinamide; useful for the treatment of mammalian infertility
02/03/2005US20050026981 Stable oral solid drug composition
02/03/2005US20050026975 Such as ethyl 4-chloroacetamido-N-(3,4-dichlorobenzyl)indole-2-carboxylate use in the treatment of disease mediated by monocyte chemoattractant protein-1
02/03/2005US20050026970 Antiproliferative agents, enzyme inhibitor for treating cancer, restenosis, psoriasis, autoimmune disease, atherosclerosis, osteoarthritis, rheumatoid arthritis, heart failure, chronic pain, and neuropathic pain; chemical synthesis
02/03/2005US20050026968 Heterocyclic amides with anti-tuberculosis activity
02/03/2005US20050026963 Pyrazole substituted directly, or by a bridge, with a heteroaryl group containing N adjacent to the point of connection of the heteroaryl useful in the treatment of psychiatric and mood disorders such as, schizophrenia, anxiety, depression, bipolar disorder, circadian rhythm and sleep disorders
02/03/2005US20050026936 1,4-Dideoxy-1-C-(4-hydroxypyrrolo[3,2-d]pyrimidin-7-yl)-1,4-imino-D-ribitol derivatives or salts; parasite purine nucleoside, -hydrolase, -phosphorylase and/or phosphoribosyl transferase inhibitors; antiprotozoa, anticarcinogenic, antiinflammatory, and immunosuppressant agents; autoimmune diseases
02/03/2005US20050026929 2-Phenyl-4-(piperidin-1-ylcarbonyl)-oxazole derivatives; capsase activators; cancer, autoimmune diseases, rheumatoid arthritis, inflammatory bowel disease, or psoriasis
02/03/2005US20050026927 Pyrazole derivatives as psychopharmaceuticals
02/03/2005US20050026923 For therapy of viral diseases
02/03/2005US20050026914 Pyrimidine or pyridine carbamate compounds as for example 1,1-dimethylethyl 4-(4-((4-((((2,6-dimethylphenyl)oxy)carbonyl)(4-(methyloxy)phenyl)amino)-2-pyrimidinyl)amino)phenyl)-1-piperazinecarboxylate; for the treatment of protein tyrosine kinase-associated disorders
02/03/2005US20050026911 Benzotriazapinone salts and methods for using same
02/03/2005US20050026905 2-Phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
02/03/2005US20050026903 Pyrazole compound; gastrointestinal disorders; central nervous system disorders
02/03/2005US20050026174 Alternative heterocycles for DNA recognition
02/03/2005US20050025774 Such as N-(2-ethoxybenzyl)-5-hydroxy-1-methyl-2-(4-methylphenyl)-6-oxo-1,6-dihydropyrimidine-4-carboxamide; for preventing, treating or delaying AIDS
02/03/2005CA2770493A1 Cyclohexanecarboxylic acid compound
02/03/2005CA2533397A1 Substituted pyridin-2-ylamine analogues
02/03/2005CA2532980A1 2-aminopyrimidine and 2-aminopyridine-4-carbamates for use in the treatment of autoimmune diseases
02/03/2005CA2532400A1 Tyrosine kinase inhibitors
02/03/2005CA2532248A1 Novel compounds
02/03/2005CA2532231A1 Aminopyrazole compounds and use as chk1 inhibitors
02/03/2005CA2532154A1 Quinoline derivates and their use in therapy
02/03/2005CA2532064A1 Hydroxypyridine cgrp receptor antagonists
02/03/2005CA2531490A1 Substituted pyrimidin-4-ylamina analogues as vanilloid receptor ligands
02/03/2005CA2528586A1 Cyclohexanecarboxylic acid compound
02/02/2005EP1501841A2 Non nucleoside reverse transcriptase inhibitors
02/02/2005EP1501826A2 Substituted indoles as alpha-1 agonists
02/02/2005EP1501825A2 Substituted imidazolylmethyl pyridine and pyrazine derivatives: gaba a receptor ligands
02/02/2005EP1501822A1 Phthalazinone derivatives
02/02/2005EP1501809A1 Triazole derivatives as tachykinin receptor antagonists