Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
09/2004
09/16/2004CA2517844A1 Quinazolines useful as modulators of ion channels
09/16/2004CA2512243A1 N-aryl heteroaromatic products, compositions containing same and use thereof
09/15/2004EP1457490A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity
09/15/2004EP1456203A1 Ethylene diamine derivatives and their use as orexin-receptor antagonists
09/15/2004EP1456201A1 Benzhydryl derivatives
09/15/2004EP1456200A1 Lactams as tachykinin antagonists
09/15/2004EP1456182A1 Pyrimidine derivatives as modulators of insuline-like growth factor-1 receptor (igf-i)
09/15/2004EP1456181A1 Methods for preparing sodium-hydrogen exchanger type-1 inhibitors
09/15/2004EP1456180A1 3,4-diarylpyrazoles and their use in the therapy of cancer
09/15/2004EP1456178A1 7-sulfonyl-3-benzazepine derivatives as modulators of the dopamine receptor and their use for the treatment of cns disorders
09/15/2004EP1456172A1 Pyrrolidine-2-ones as factor xa inhibitors
09/15/2004EP1455579A1 Pyrazoles-pyrimidine fungicides
09/15/2004EP1363902B1 Chemical compounds
09/15/2004EP1212317B1 Indole derivatives and their use for the treatment of osteoporosis amongst other applications
09/15/2004EP0990653B1 2-oxoimidazole derivatives
09/15/2004EP0889726B1 Novel cycloalkyl substituted imidazoles
09/15/2004EP0693072B9 Method for the synthesis of 4- and/or 5-(di)substituted 2-aminoimidazoles from 2-aminoimidazoles and aldehydes
09/15/2004CN1529704A 3-(4-amidopyrrol-2-2ylmethlidene)-2-indolinone derivatives as protein kinase inhibitors
09/15/2004CN1529703A 新的吲哚衍生物 The new indole derivatives
09/15/2004CN1529595A 4,5-hydro-1H-pyrazole derivative having protent CB1-antagonistic
09/15/2004CN1528750A Pyrimidine derivatives and preparing method thereof
09/15/2004CN1528742A Compound for treating asthma, irritability an a inflammation and its intermediate
09/15/2004CN1166645C Bicyclic heterocyles, medicaments contg. these compounds, their use and methods for prodn. thereof
09/15/2004CN1166643C 4-phenyl-pyrimidine derivatives
09/15/2004CN1166638C Novel benzo-[3,4] cyclobutano [1,2-C] pyrroles compound, its prepn. and medicine composition containing the same
09/15/2004CN1166636C Arylpiperazinyl-cyclohexyl indole derivatives for the treatment of depression
09/15/2004CN1166633C New alpha-amino acid sulfuryl compounds, its preparing method and medicinal composition containing them
09/15/2004CN1166363C Use of moxonidine for postmyocardial infarction treatment
09/14/2004US6790957 Converting tertiary hydroxy group of a triazole antifungal compound into a phosphate group to improve aqueous solubility
09/14/2004US6790860 Pyrrolidine derivatives
09/14/2004US6790852 Heterocyclic nitrogen compounds such as 2-(2,6-dichlorophenyl) -4-(3-bromophenyl)-5-(2-(3- hydroxypropylamino)pyrimidin-4-yl) -n-h-imidazole, used as tyrosine kinase inhibitors; anticarcinogenic or antitumor agents
09/14/2004US6790845 Having an attached non-aromatic heterocyclic ring
09/14/2004US6790810 Tetrazolinone derivatives
09/10/2004WO2004076457A1 Solvent-free process for the preparation of pyrrolo (3,4c) pyrrole compounds
09/10/2004WO2004076456A1 Solvent-free process for the preparation of diketopyrrolopyrrole derivatives
09/10/2004WO2004076442A1 Polymorphs of losartan
09/10/2004WO2004076429A1 Ethynyl derivatives serving as factor xa inhibitors
09/10/2004WO2004076424A1 Heterocyclic kinase inhibitors
09/10/2004WO2004076412A2 Aminoheteroaryl compounds as protein kinase inhibitors
09/10/2004WO2004076410A2 Polymorphs of pyrrole substituted 2-indolinone protein kinase inhibitors
09/10/2004WO2004076407A2 Pyrrolidine derivatives as oxytocin antagonists
09/10/2004WO2004076406A2 Losartan potassium polymorphs and process for the preparation thereof
09/10/2004WO2004075895A1 Ocular hypotensive agent
09/10/2004WO2004075840A2 Selective non-steroidal glucocorticoid receptor modulators
09/10/2004WO2004075823A2 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament
09/10/2004WO2004052847A3 Tricyclic steroid hormone nuclear receptor modulators
09/10/2004WO2004050643A3 Non-nucleoside reverse transcriptase inhibitors
09/10/2004WO2004047769A3 Benzimidazoles and analogs thereof as antibacterials
09/10/2004WO2004022523A3 1, 3-diamino-2-hydroxypropane prodrug derivatives
09/10/2004WO2003087092A3 Inhibitors of serine proteases, particularly hepatitis c virus ns3 - ns4 protease
09/10/2004WO2003061652A8 3-(imidazolyl)-2-alkoxypropanoic acids as tafia inhibitors
09/10/2004CA2517391A1 Ethynyl derivatives serving as factor xa inhibitors
09/10/2004CA2517256A1 Aminoheteroaryl compounds as protein kinase inhibitors
09/10/2004CA2516900A1 Polymorphs of pyrrole substituted 2-indolinone protein kinase inhibitors
09/10/2004CA2516684A1 Selective non-steroidal glucocorticoid receptor modulators
09/10/2004CA2516660A1 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament
09/09/2004US20040176603 Substituted nitrogen-containing heterobicycles, the preparation thereof and their use as pharmaceutical compositions
09/09/2004US20040176594 Drugs that inhibit phosphorylation kinases as an antigrowth or antiproliferation agent
09/09/2004US20040176443 Capsaicin receptor ligands
09/09/2004US20040176433 treatment of tumor necrosis factor mediated disorders; asthma; inflammatory bowel disease; arthritis
09/09/2004US20040176428 treatment of Type 2 diabetes mellitus, obesity and lipid disorders; coadministration with HMG CoA reductase inhibitors
09/09/2004US20040176400 Fused pyrimidines as antagonists of the corticotropin releasing factor (crf)
09/09/2004US20040176399 A2B adenosine receptor antagonists
09/09/2004US20040176396 anti-protoazoal; poultry feed; therapy for cytokine mediated disease i.e. osteoarthritis, cerebral malaria, chronic pulmonary inflammatory disease, silicosis, pulmonary sarcosis, bone resorption diseases, reperfusion injury, graft v. host rejection
09/09/2004US20040176389 Piperazine oxime dervatives having nk-1 receptor antagonistic activity
09/09/2004US20040176388 example compound: cis-1-[(2-chloro-3-trifluoromethylphenyl)acetyl]-6-(3,4,5-trimethylpiperazin-1-yl)indole; treatment of CNS and other disorders
09/09/2004US20040176385 treating cancer by inhibiting phosphotidylinositol 3-kinase; in combination with other known agents to modulate cellular proliferation
09/09/2004US20040176382 treatment of inflammation, proliferative diseases, and certain cardiovascular disorders as well as Alzheimer's disease;
09/09/2004US20040176379 agonist effect from one or more of a somatostatin subtype receptor; diabetes mellitus, hyperlipidemia, insulin insensitivity, Syndrome X; inhibiting the proliferation of helicobacter pylori
09/09/2004US20040176377 inhibitors of glycogen synthase kinase-3 beta; treatment of diabetes or neurodegenerative diseases such as Alzheimer's disease; 6-(2-butylamino-pyrimidin-4-yl)-3-oxo-2,3-dihydro-pyridazine-4-carboxylic acid (3-pyridin-3-yl-propyl)-amide, as example
09/09/2004US20040176363 N-Acylpiperazine derivatives; cardiovascular disorders; anticoagulants
09/09/2004US20040176358 Compositions and methods relating to novel compounds and targets thereof
09/09/2004US20040176348 Arylvinylazacycloalkane compounds and methods of preparation and use thereof
09/09/2004US20040176325 P38 MAP kinase inhibitors comprising indazole derivatives; antiinflammatory and antiproliferative agents; autoimmune, bone, and neurodegenerative disorders; viricides, infections
09/09/2004US20040176271 2-amino-4-aryl or heteroaryl pyridines or pyrimidines; Janus kinases (JAK)
09/09/2004DE10308907A1 Ethynylderivate Ethynylderivate
09/09/2004DE10306250A1 Substituierte N-Arylheterozyklen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Substituted N-Arylheterozyklen, processes for their preparation and their use as medicaments
09/08/2004EP1454902A1 N- (substituted five-membered di-or triaza diunsaturated ring)carbonyl guanidine derivateives for the treatment of ischemia
09/08/2004EP1454901A1 Piperazine compounds and pharmaceutical compositions containing them.
09/08/2004EP1454898A1 Novel phenylalanine derivative
09/08/2004EP1453826A1 Amorphous form of 2-n-butyl-3-[[2-(1h-tetrazol-5-yl)[1,1'-biphenyl]-4-yl]methyl]-1,3-diazaspiro[4,4'] non-1-en-4-one
09/08/2004EP1453823A1 2-guanidino-4-heterocyclylquinazolines
09/08/2004EP1453811A2 Peroxisome proliferator activated receptor agonists
09/08/2004EP1453800A2 Protein kinase inhibitors
09/08/2004EP1453789A2 N,n'-substituted-1,3-diamino-2-hydroxypropane derivatives
09/08/2004EP1453516A2 Novel tri-substituted pyrimidines, method for production and use thereof as medicament
09/08/2004EP1453515A2 Method to treat cystic fibrosis
09/08/2004EP1453503A2 Ep4 receptor agonist, compositions and methods thereof
09/08/2004EP1453502A2 Pharmaceutical formulations comprising indolinone derivatives
09/08/2004EP1345603A4 (halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
09/08/2004EP1289972B1 Serine protease inhibitors
09/08/2004EP1201664B1 Benzimidazole compounds and drugs containing the same
09/08/2004EP1089994B1 Novel form of irbesartan, methods for obtaining said form and pharmaceutical compositions containing same
09/08/2004EP0993456B1 2-substituted 4,5-diaryl imidazoles
09/08/2004EP0623126B1 Imidazole derivatives and their use as cytokine inhibitors
09/08/2004CN1527829A Pyrazole derivatives as HIV reverse transcriptase inhibitors
09/08/2004CN1527710A Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands
09/08/2004CN1527709A Therapeutic combinations for cardiovascular and inflammatory indications
09/08/2004CN1527701A Tablets quickly disintegrated in oral cavity
09/08/2004CN1165546C New derivative of erythromycin, its preparation method and medicinal application