Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
09/2004
09/08/2004CN1165303C DNA binding indole derivatives, their prodrugs and immunoconjugates as anticancer agents
09/07/2004US6787652 Lowering lipids and serum cholesterol without generating adverse cardiac effects; 4,5-dihydro-3,5-dioxo-1,2,4-triazine derivatives
09/07/2004US6787651 Substituted indoles, pharmaceutical compounds containing such indoles and their use as PPAR-γ binding agents
09/07/2004US6787561 Benzimidazole compounds
09/07/2004US6787558 Neuropeptide y receptor antagonists, for treating arthritis, cardiovascular diseases, diabetes, renal failure, eating disorders and obesity
09/07/2004US6787556 Benzoic acid derivatives for the treatment of diabetes mellitus
09/07/2004US6787555 Such as 4-(4-fluorophenyl)-5-(2-phenylmethylamino)pyrimidin-4-yl)-1-ethoxymethyl -(1,2,3)triazole for inhibition of release of inflammatory interleukins; for treatment of osteoarthritis, rheumatoid arthritis, and congestive heart failure
09/07/2004US6787550 Indole derivatives and their use for the treatment of osteoporosis amongst other applications
09/07/2004US6787546 Heterocycle derivatives and drugs
09/07/2004US6787543 Preparation of tachykinin antagonists; substituted nitrogen-containing heterocycles
09/07/2004US6787542 Aryl phenylheterocyclyl sulfide derivatives and their use as cell adhesion-inhibiting anti-inflammatory and immune-suppressive agents
09/07/2004US6787540 Compounds useful as reversible inhibitors of cysteine proteases
09/07/2004US6787538 Hormone replacement therapy; agonists, antagonists; antiestrogens with little to no intrinsic estrogenicity
09/07/2004CA2140146C Process for preparing indole derivatives containing a 1,2,4-triazol-1-yl substituent
09/02/2004WO2004074279A1 Methods of making 6-[(4,5-dihydro-1h-imidazol-2-yl)amino-]-7-methyl-1h-benzimidazole-4-carbonitrile and its preferred salt form
09/02/2004WO2004074274A1 Substituted n-aryl nitrogen heterocycles
09/02/2004WO2004074258A1 Novel sulphated imidazole derivatives, method for production thereof, novel intermediates obtained, application thereof as medicaments and pharmaceutical compositions comprising the above
09/02/2004WO2004074257A1 Non-nucleoside reverse transcriptase inhibitors
09/02/2004WO2004074250A1 Novel compounds and compositions containing the same
09/02/2004WO2004074244A2 Pyrimidine compounds
09/02/2004WO2004074243A2 Heterocyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands
09/02/2004WO2004073634A2 Phenylenediamine urotensin-ii receptor antagonists and ccr-9 antagonists
09/02/2004WO2004058730A3 Triazole derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1
09/02/2004WO2004050637A3 2-(2-hydroxybiphenyl-3-yl)-1h-benzoimidazole-5-carboxamidine derivatives as factor viia inhibitors
09/02/2004WO2004049797A3 Pesticidal sulphonylaminopyrazoles
09/02/2004WO2004039352A3 Amorphous form of losartan potassium
09/02/2004WO2004035569A3 Novel compounds with antibacterial activity
09/02/2004WO2004014851A3 Tyrosine kinase inhibitors
09/02/2004WO2003101954A3 Nf-kb inhibitors and uses thereof
09/02/2004US20040171881 N,N'-substituted-1,3-diamino-2-hydroxypropane derivatives
09/02/2004US20040171848 Fluoropyrrolidines as dipeptidyl peptidase inhibitors
09/02/2004US20040171843 Process for preparing losartan potassium with improved flow ability
09/02/2004US20040171799 Method of the solid phase synhesis of pyrrole-imidazole polyamide
09/02/2004US20040171649 Intermediates for anthranilic amide insecticides and blood coagulation factor Xa inhibitors
09/02/2004US20040171634 Anticancer, antitumor agents, antiarthritic agents
09/02/2004US20040171630 both receptor-type and non-receptor type tyrosine kinases; to treat angiogenesis, cancer, tumor growth, atherosclerosis, age related macular degeneration, diabetic retinopathy, inflammatory diseases,
09/02/2004US20040171617 treatment for disorders and diseases, such as chronic inflammation, tissue breakdown and cancer
09/02/2004US20040171614 Novel gamma secretase inhibitors
09/02/2004US20040171606 antagonism/inhibition, of the D3 receptor; substance abuse.
09/02/2004US20040171543 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
09/02/2004US20040171520 Melanocortin receptor-specific peptidomimetics
09/02/2004US20040171490 Preventing infestation of plants by phytopathogenic microorganisms; horticulture, agriculture
09/02/2004US20040171099 Using luciferin derivatives for analyzing metabolic activity in animals, cells or in cell-free reaction formulations
09/02/2004US20040171075 Modulation of protein functionalities
09/02/2004DE10307142A1 Substituierte N-Aryl-Stickstoffheterocyclen Substituted N-aryl nitrogen heterocycles
09/02/2004CA2767153A1 Phenylenediamine urotensin-ii receptor antagonists and ccr-9 antagonists
09/02/2004CA2517002A1 Methods of making 6-[(4,5-dihydro-1h-imidazol-2-yl)amino-]-7-methyl-1h-benzimidazole-4-carbonitrile and its preferred salt form
09/02/2004CA2516590A1 Substituted n-aryl nitrogen heterocycles
09/02/2004CA2515570A1 Heterocyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands
09/01/2004EP1452527A1 Azabicyclo compound, matrix metalloprotease inhibitor, and skin preparation
09/01/2004EP1452526A1 Indole compound and medicinal use thereof
09/01/2004EP1452525A1 Amide derivatives and drugs
09/01/2004EP1452524A1 "2-oxo-1-pyrrolidine derivative and its pharmaceutical uses"
09/01/2004EP1451185A1 Indole-2-carboxamides as factor xa inhibitors
09/01/2004EP1451177A1 Substituted 2-pyrrolidine-2-yl-1h-indole derivatives for the treatment of migraine
09/01/2004EP1451160A2 Pyrazole-amides and-sulfonamides
09/01/2004EP1451154A2 Inhibitors of cytosolic phospholipase a2
09/01/2004EP1451153A1 Nk1 antagonists
09/01/2004EP1450901A2 (1-phenyl-2-heteroaryl)ethyl-guanidine compounds as inhibitors of mitochondrial f1f0 atp hydrolase
09/01/2004EP1450808A1 Quinazoline derivatives for the treatment of t cell mediated diseases
09/01/2004EP1450800A2 SUBSTITUTED AMINO METHYL FACTOR Xa INHIBITORS
09/01/2004EP1450794A1 Novel dipeptidyl peptidase iv (dp-iv) inhibitors as anti-diabetic agents
09/01/2004EP1450791A1 Hydrazonopyrazole derivatives and their use as therapeutics
09/01/2004EP1292594B1 Quinazoline derivatives for the treatment of tumours
09/01/2004EP1060165B1 Method for preparing an n-substituted heterocyclic derivative using a phase-transfer catalyst
09/01/2004EP0944621B1 2-imidazolinylaminoindole compounds useful as alpha-2 adrenoceptor agonists
09/01/2004CN1525968A Compositions for prevention or treatment of hepatopathy
09/01/2004CN1525960A Lorenz Gisela
09/01/2004CN1525957A Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
08/2004
08/31/2004US6784293 Solution and solid-phase synthesis of boc-protected 3-aminohydantoins/thiohydantoins and 3-aminodihydrouracils/ dihydrothiouracils
08/31/2004US6784197 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
08/31/2004US6784195 Extracellular signal regulated kinase (erk); anticancer agents and protein kinase inhibitors
08/31/2004US6784182 Serine protease inhibitors
08/31/2004US6784181 Ligands for the delta receptor
08/31/2004US6784167 17-beta-hydroxysteroid dehydrogenase-II inhibitors
08/26/2004WO2004072068A1 Vanilloid receptor ligands and their use in treatments
08/26/2004WO2004072064A1 Synthesis of 2-butyl-3-(2'-(1-trityl-1h-tetrazol-5-yl)biphenyl-4-yl)-1,3-diazaspirol[4,4]-non-ene-4-one
08/26/2004WO2004072063A1 Heteroaryl substituted pyrolls useful as inhibitors of protein kinases
08/26/2004WO2004072062A2 Indolylmaleimide derivatives
08/26/2004WO2004072047A1 Indoles, benzimidazoles or naphhimidazoles as histone deacetylase (hdac) inhibitors
08/26/2004WO2004072025A2 Substituted n-arylheterocycles, method for production and use thereof as medicaments
08/26/2004WO2004071460A2 Cyclic derivatives as modulators of chemokine receptor activity
08/26/2004WO2004071454A2 Substituted azetidine compounds as inhibitors of dipeptidyl peptidase iv
08/26/2004WO2004071448A2 Substituted azole derivatives as inhibitors of protein tyrosine phosphatases
08/26/2004WO2004071447A2 Substituted azole derivatives as therapeutic agents
08/26/2004WO2004071390A2 Piperazine-2-carboxamide derivatives
08/26/2004WO2004043354A3 Ophthalmic compositions for treating ocular hypertension
08/26/2004WO2004018461A3 Antibacterial benzoic acid derivatives
08/26/2004US20040167341 Pyrrolidines as dipeptidyl peptidase inhibitors
08/26/2004US20040167333 For therapy of eosinophil-dependent inflammatory diseases
08/26/2004US20040167224 Nitrogen containing heterocyclic compounds and medicines containing the same
08/26/2004US20040167201 Pyrrolidine melanocortin-specific compounds
08/26/2004US20040167198 Vasculostatic agents and methods of use thereof
08/26/2004US20040167194 Methods of making 6-[(4,5-Dihydro-1H-imidazol-2-yl)amino-]-7-methyl-1H-benzimidazole-4-carbonitrile and its preferred salt form
08/26/2004US20040167193 Fungicides
08/26/2004US20040167158 Heterocyclic compounds for the treatment of migraine
08/26/2004US20040167142 Pyrimidinone compounds
08/26/2004US20040167141 Anticancer agents; antidiabetic agents; Alzheimer's disease
08/26/2004US20040167122 Central nervous system disorders; anxiolytic agents; neurodegenerative disorders; obsessive compulsive disorders; schizophrenia; antidepressants; alzheimer's disease; neuropathic pain; stroke
08/26/2004US20040167121 Indazolinone compositions useful as kinase inhibitors