Patents
Sitemap › C07 - Organic chemistry › C07D - Heterocyclic compounds › C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
08/2000
08/22/2000US6107485 In one step, by reacting n-substituted amidine (or its hydrochloride salt) with a beta-keto ester in the presence of a base under conditions of high pressure
08/22/2000US6107369 Crosslinked thick film with no pin hole is formed by curing a curable monomer and tris-pyrrolidonyl triazine crosslinker
08/22/2000US6107330 Inhibitor for narcotic analgesic dependence/resistance acquisition
08/22/2000US6107329 Hypotensive agents; cardiovascular disorders
08/22/2000US6107324 5-HT2A receptor inverse agonists
08/22/2000US6107312 Bactericide
08/22/2000US6107308 Antihistamine; leutriene antagonist
08/22/2000US6107301 1N-alkyl-N-arylpyrimidinamines and derivatives thereof
08/22/2000US6107299 Insecticides; miticides
08/22/2000US6107297 2,4-Dithi(oxo)-pyrimidin-5-yl compounds bearing a tricyclic substituent useful as P2 purinoceptor antagonists
08/22/2000US6107295 Arylalkanoyl pyridazines
08/22/2000US6107291 Antiinflammatory agent
08/22/2000US6107253 1-(pyridyl)-pyrazols and their use as herbicides
08/22/2000CA2085987C Piperidyl-substituted indoles
08/17/2000WO2000047577A1 Phenyl urea and phenyl thiourea derivatives as orexin receptor antagonists
08/17/2000WO2000047576A1 Cinnamide derivatives as orexin-1 receptors antagonists
08/17/2000WO2000047574A1 Heteroaryl-substituted quinolin-2-one derivatives useful as anticancer agents
08/17/2000WO2000047573A1 Heterocyclic derivatives as inhibitors of factor xa
08/17/2000WO2000047571A1 Piperidine and piperazine derivatives as inhibitors of the abeta fibril formation
08/17/2000WO2000047562A1 Spirocyclic ketones and their use as tachykinin antagonists
08/17/2000WO2000047559A2 5-ht1f agonists
08/17/2000WO2000047558A1 Amide compounds and medicinal use thereof
08/17/2000WO2000047554A2 INHIBITORS OF FACTOR Xa
08/17/2000WO2000047553A2 ALKENYL AND ALKYNYL COMPOUNDS AS INHIBITORS OF FACTOR Xa
08/17/2000WO2000047212A1 Quinazoline derivatives as angiogenesis inhibitors
08/17/2000WO2000027819A3 Antrhranilic acid amides and the use thereof as medicaments
08/17/2000WO2000012076A9 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
08/17/2000CA2362392A1 Heterocyclic derivatives as inhibitors of factor xa
08/17/2000CA2362389A1 Piperidine and piperazine derivatives as inhibitors of the abeta fibril formation
08/17/2000CA2362375A1 Alkenyl and alkynyl compounds as inhibitors of factor xa
08/17/2000CA2362272A1 Spirocyclic ketones and their use as tachykinin antagonists
08/17/2000CA2361428A1 Inhibitors of factor xa
08/17/2000CA2360164A1 5-ht1f agonists
08/16/2000EP1028111A1 Amide derivatives or salts thereof
08/16/2000EP1027338A2 New carboxylic acid derivatives, carrying amido side-chains; production and use as endothelin receptor antagonists
08/16/2000EP1027336A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
08/16/2000EP1027335A1 Ortho-hydroxypyridinone derivatives as iron chelating and antioxidant agents
08/16/2000EP1027332A1 Novel lactam metalloprotease inhibitors
08/16/2000EP1027328A1 Substituted anilides
08/16/2000EP1027052A1 Novel combination
08/16/2000EP1027048A2 Selective cyclooxygenase-2 inhibitors against premature labor
08/16/2000EP1027042A1 Inhibitors of farnesyl protein transferase
08/16/2000EP1027041A1 Novel cyanoaziridines for treating cancer
08/16/2000EP0842171B1 Herbicidal sulphonylamino(thio)carbonyl triazolinones with heterocyclyloxy substituents
08/16/2000EP0755374B1 Process for peptide segment condensation
08/16/2000CN1263528A N-triazolyl-2-indolecarboxamides and their use as CCK-A agonists
08/16/2000CN1263527A Cis-disubstituted aminocycloalykyl-pyrrolidine derivatives
08/16/2000CN1263526A Triazine derivatives, their production and use
08/16/2000CN1263101A New derivative of erythromycin, its preparation method and medicinal application
08/16/2000CN1055469C Optically pure salts of pyridinylmethyl sulfinyl-1H-benzimidazole compounds, its preparing method and use
08/16/2000CN1055465C Optical active 2-imidazoline-5-thione derivatives and preparating method and use thereof
08/15/2000US6103936 Reacting aldehyde, sulfide, sulfone, or sulfoxide with formamide in presence of acid catalyst, and optionally a dehydrating agent
08/15/2000US6103910 D-proline derivatives
08/15/2000US6103905 Quinoline-indole antimicrobial agents, uses and compositions related thereto
08/15/2000US6103902 Carbamoylation process
08/15/2000US6103752 Therapeutic heterocyclic compounds
08/15/2000US6103744 Administering to the patient a dopamine autoreceptor agonists for the treatment of schizophrenia, parkinson,s disease, tourette,s syndrom, alcoholism and drug addiction
08/15/2000US6103738 Quinoline and quinazoline compounds useful in therapy
08/15/2000US6103737 Aryl- and arylamino- substituted heterocycles as corticotropin releasing hormone antagonists
08/15/2000US6103732 Endothelin receptor inhibitors; hypotensive agents, cardiotonic agents; acute myocardial infarct, pulmonary hypertension, raynaud's syndrome, atherosclerosis; asthma; cardiovascular disorders
08/15/2000US6103731 Imidazol[1,5-c]quinazolines; a new class of GABA brain receptor
08/15/2000US6103720 Ketobenzamides as calpain inhibitors
08/15/2000US6103719 Neurokinin-a- or neurokinin-b tachnkinin antagonistic properties; substance p antagonism; respiratory, gastrointestinal, nervous system, skin disorders;
08/15/2000US6103718 Selective cyclic nucleotide phosphodiesterase (pde) inhibitors (specifically of type 4) which are effective bronchial therapeutics; bronchodilators; respiratory system disorders
08/15/2000CA2196215C 1,4-dihydropyridine compound and pharmaceutical composition containing the same
08/15/2000CA2105385C Treatment of cognitive disorders
08/10/2000WO2000046221A1 Sulfamato hydroxamic acid metalloprotease inhibitor
08/10/2000WO2000046220A1 Triazole and tetrazole derivatives, and their therapeutic use
08/10/2000WO2000046219A1 Alpha-azacyclomethyl quinoline derivatives for treating urinary incontinence
08/10/2000WO2000046214A1 Substituted 4-amino-2-aryltetrahydroquinazolines, their preparation, their use and pharmaceutical compositions comprising them
08/10/2000WO2000046208A1 Substituted pyrazole carboxylic acids used to combat anaemias
08/10/2000WO2000046199A2 Indole derivatives as anti-inflammation agents
08/10/2000WO2000046198A1 Anti-inflammatory indole derivatives
08/10/2000WO2000046196A1 Indole derivatives and their use as mcp-1 antagonists
08/10/2000WO2000046195A1 Anti-inflammatory indole derivatives
08/10/2000WO2000046194A1 Cyclic amine derivatives and uses thereof
08/10/2000WO2000046187A2 Antizyme modulators and their use
08/10/2000WO2000046181A1 Carboxylic acid derivatives, process for their preparation and their use as rotamase enzyme activity inhibitors
08/10/2000WO2000045894A2 Use of pyrazole carboxamides
08/10/2000WO2000045814A1 Methods and compositions to enhance white blood cell count
08/10/2000WO2000028975A3 Improved chemical process and pharmaceutical formulation
08/10/2000WO2000027822A3 Tricyclic pyrazole derivatives
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/10/2000DE19905255A1 New carboxylic acid derivatives are rotamase inhibitors useful as neuroprotective agents for treating e.g. Parkinson's disease, amyotrophic lateral sclerosis, Alzheimer's disease, Huntington's disease
08/10/2000DE19905254A1 New ether compounds, useful for treating neurological diseases e.g. Parkinson's disease, amyotrophic lateral sclerosis and Alzheimer's disease
08/10/2000DE19904710A1 Substituierte 4-Amino-2-aryl-tetrahydrochinazoline, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate Substituted 4-amino-2-aryl-tetrahydroquinazolines, their preparation, their use and pharmaceutical compositions containing them
08/10/2000DE19904406A1 Substituierte Pyrazolcarbonsäuren Substituted pyrazole
08/10/2000DE19904397A1 Verwendung von Pyrazol-Carbonsäureamiden Use of pyrazole carboxamides
08/10/2000CA2362259A1 Antizyme modulators and their use
08/10/2000CA2362230A1 Sulfamato hydroxamic acid metalloprotease inhibitor
08/10/2000CA2362077A1 Cyclic amine derivatives and uses thereof
08/10/2000CA2361816A1 Substituted pyrazole carboxylic acids used to combat anaemias
08/10/2000CA2361636A1 Use of pyrazole carboxamides
08/10/2000CA2357013A1 Anti-inflammatory indole derivatives
08/10/2000CA2356898A1 Indole derivatives and their use as mcp-1 antagonists
08/10/2000CA2355734A1 Indole derivatives as anti-inflammation agents
08/09/2000EP1026160A1 Nitrogenous fused-ring compounds, process for the preparation of the same, and drugs
08/09/2000EP1026151A1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides and insecticides
08/09/2000EP1025847A1 Neovascularization promoters and neovascularization potentiators
08/09/2000EP1025091A1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system
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