Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
06/2000
06/06/2000US6071921 4-phenyl-7-arylquinoazolines; angiogenisis inhibitors and/or vascular permeability reducing effects in warm-blooded animals; anticarcinogenic and -arthritic agents; rheumatic diseases; vascular endothelium growth factor inhibitors
06/06/2000US6071917 Analgesics; antiinflammatory agents; especially for the treatment of asthma, cerebral traumatic shock and allergic rhinitis; competitive binding at receptors
06/06/2000US6071915 Arylsubstituted piperazines useful in the treatment of benign prostatic hyperplasia
06/06/2000US6071912 Inhibit human factor xa and are therefore useful as pharmacological agents for the treatment of disease-states characterized by thrombotic activity; amino-, oxy- and thia-substituted triazines
06/06/2000US6071909 Phenylbenzimidazole derivatives as ligands for GABA receptors
06/06/2000US6071908 Radiation-activated cytotoxin therapy of neoplastic disease
06/06/2000US6071907 Tricyclic compounds useful as FPT inhibitors
06/06/2000US6071903 2,3,4,5-tetrahydro-1H-[1,4]-benzodiazepine-3-hydroxyamic acids
06/06/2000US6071900 Heterocyclic compounds and their use
06/06/2000US6071895 Polar-substituted hydrocarbons
06/06/2000US6071860 For selective control of broad-leaved and grass weeds in crops of useful plants
06/02/2000WO2000031074A2 Indole derivatives and their use as serotonin receptor ligands
06/02/2000WO2000031072A1 Process for making 5-substituted pyrazoles using dithietanes
06/02/2000WO2000031068A1 Polyhydroxylated heterocyclic derivatives as anti-coagulants
06/02/2000WO2000031067A1 Propanoic acid derivatives as integrin inhibitors
06/02/2000WO2000031066A1 Substituted n-pyrazolyl-phenoxynicotinic acid-(thio)amides that can be used as herbicides
06/02/2000WO2000031065A1 Compounds having cytokine inhibitory activity
06/02/2000WO2000031064A1 Enantioselective alkylation of tricyclic compounds
06/02/2000WO2000031063A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS
06/02/2000WO2000031062A1 Cycloalkyl-substituted aminomethylpyrrolidine derivatives
06/02/2000WO2000031061A1 2-oxoimidazole derivatives
06/02/2000WO2000031047A1 Substituted 4-amino-2-aryl-cyclopenta[d]pyrimidines, their production and use and pharmaceuticalreparations containing same
06/02/2000WO2000031039A1 Substituted benzo[de]isoquinoline-1,3-diones
06/02/2000WO2000031038A1 Quinoline derivatives as nk-2 and nk-3 receptor ligands
06/02/2000WO2000031037A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
06/02/2000WO2000031034A1 Insecticidal photostable acid salt derivatives of n-benzyl-4-benzhydrolpiperidines
06/02/2000WO2000009105A3 Small molecule carbamates or ureas for vision and memory disorders
06/02/2000CA2351865A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
06/02/2000CA2351725A1 Substituted pyrazoles as p38 kinase inhibitors
06/02/2000CA2351526A1 Indole derivatives and their use as serotonin receptor ligands
06/02/2000CA2351497A1 Cycloalkyl-substituted aminomethylpyrrolidine derivative
06/02/2000CA2351348A1 Substituted benzo[de]isoquinoline-1,3-diones
06/02/2000CA2350969A1 Compounds having cytokine inhibitory activity
06/02/2000CA2350081A1 Process for making 5-substituted pyrazoles using dithietanes
06/02/2000CA2291880A1 Novel derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one, and compositions and methods for inhibiting abnormal cell growth comprising said derivatives
05/2000
05/31/2000EP1004592A1 Derivatives of erythromycin, their process of preparation and their application as medicaments
05/31/2000EP1004581A2 Process for the preparation of thalidomide
05/31/2000EP1004580A2 Imides as inhibitors of TNF alpha
05/31/2000EP1004578A2 5-oxo-pyrrolidine-2-carboxylic acid hydroxamide derivatives
05/31/2000EP1004572A2 Amines as inhibitors of TNF alpha
05/31/2000EP1004306A2 Estrogen agonists/antagonists
05/31/2000EP1003821A1 Anisotropic retardation layers for display devices
05/31/2000EP1003743A1 3,3-disubstituted piperidines as modulators of chemokine receptor activity
05/31/2000EP1003738A1 Bicyclic compounds as ligands for 5-ht1 receptors
05/31/2000EP1003737A1 Phenyl urea and phenyl thiourea derivatives as hfgan72 antagonists
05/31/2000EP1003736A1 Substituted 4-benzoyl-pyrazoles
05/31/2000EP1003734A2 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONIST
05/31/2000EP1003726A1 Nitrophenyl-sulfonyl-imidazoles and use thereof for controlling vegetable and animal pests
05/31/2000EP1003724A1 Substituted quinoline derivatives with antiviral action
05/31/2000EP1003723A1 2-acylaminopropanamines as tachykinin receptor antagonists
05/31/2000EP1003721A1 Benzylidene-1,3-dihydro-indol-2-one derivatives as receptor tyrosine kinase inhibitors, particularly of raf kinases
05/31/2000EP1003541A1 Inhibitors of hiv reverse transcriptase
05/31/2000EP1003540A1 $g(b)2-ADRENERGIC RECEPTOR AGONISTS
05/31/2000EP1003514A1 Cyclic amine modulators of chemokine receptor activity
05/31/2000EP1003512A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
05/31/2000EP1003511A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS
05/31/2000EP1003504A2 Indole derivatives and their use as mcp-1 antagonists
05/31/2000EP1003374A4 Inhibitors of farnesyl-protein transferase
05/31/2000EP1003374A1 Inhibitors of farnesyl-protein transferase
05/31/2000DE19955340A1 CCR-3-Rezeptor-Antagonisten CCR-3 receptor antagonists
05/31/2000CN1255162A Protease inhibitors
05/31/2000CN1255124A Substituted isoquinoline derivatives and their use as anticonulsants
05/31/2000CN1255119A Protease inhibitors
05/31/2000CN1255042A Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them
05/31/2000CN1254596A Process for preparing composition to kill internal parasites
05/31/2000CN1052984C New erythromycin derivative and its preparing process and application in medicine
05/30/2000US6069254 Carboxamide derivatives of piperidine for the treatment of thrombosis disorders
05/30/2000US6069251 Highly selective partial agonists or antagonists at brain dopamine receptor subtypes or prodrugs; diagnosis and treatment schizophrenia; antidepressants; certain movement disorders such as parkinsonism.
05/30/2000US6069162 Indolyl and benzofuranyl carboxamides as inhibitors of nitric oxide production
05/30/2000US6069157 Parasiticidal compounds
05/30/2000US6069156 Indole derivatives as cGMP-PDE inhibitors
05/30/2000US6069152 Nervous system disorders; cardiovascular disorders; gastrointestinal disorders
05/30/2000US6069151 Controlling tumor necrosis factor
05/30/2000US6069143 Anticoagulants
05/30/2000US6069114 Herbicides for selectively controlling broad-leaved weeds and grass weeds in crops of useful plants
05/30/2000US6068856 Oral pharmaceutical composition with delayed release of active ingredient for pantoprazole
05/30/2000CA2206104C Adamantyl substituted oxindoles as pharmaceuticals agents
05/30/2000CA1341008C A - unsaturated amines, their production and use
05/25/2000WO2000029403A1 Novel pyrimidine derivatives and processes for the preparation thereof
05/25/2000WO2000029397A1 New piperazine and piperidine compounds
05/25/2000WO2000029386A1 Pyrimidinedione derivatives useful as alpha 1a adrenoceptor antagonists
05/25/2000WO2000029382A1 Certain substituted caprolactams, pharmaceutical compositions containing them and their use in treating tumors
05/25/2000WO2000029380A1 Tetrahydroisoquinoline derivatives as lhrh antagonists
05/25/2000WO2000029377A1 4-aroyl-piperidin-ccr-3 receptor antagonists iii
05/25/2000WO2000028975A2 Improved chemical process and pharmaceutical formulation
05/25/2000WO2000018361A3 Method of treating hair loss using sulfonamides
05/25/2000WO2000011951A3 Use of 5-amino-pyrazol-derivatives for combating micro-organisms
05/25/2000DE19854081A1 New 2-phenoxy-N-pyrazolyl-nicotinamide derivatives, useful as pre- or post-emergence, total or selective herbicides
05/25/2000DE19853278A1 New 4-amino-2-aryl-cyclopentapyrimidine derivatives are activators of soluble guanylate cyclase, useful for treating or preventing e.g. thrombosis and restenosis
05/25/2000CA2351644A1 Pyrimidine derivatives and processes for the preparation thereof
05/25/2000CA2351187A1 Tetrahydroisoquinoline derivatives as lhrh antagonists
05/25/2000CA2350722A1 4-aroyl-piperidin-ccr-3 receptor antagonists iii
05/24/2000EP1002797A1 4,5-DIHYDRO- 1H]-BENZ g]INDAZOLE-3-CARBOXYLIC ACID DERIVATIVES
05/24/2000EP1002796A2 Novel quinoxalindione derivatives, their production and use in medicaments
05/24/2000EP1002795A1 HIV Replication inhibiting pyrimidines
05/24/2000EP1002123A1 Enzymatic kinetic resolution of an intermediate useful for preparing substituted tricyclics
05/24/2000EP1001948A1 Bisimino-substituted phenyl compounds and their use as pesticides
05/24/2000EP1001945A1 QUINOLINE AND QUINOXALINE COMPOUNDS WHICH INHIBIT PLATELET-DERIVED GROWTH FACTOR AND/OR p56?lck TYROSINE KINASES
05/24/2000EP1001939A1 Heterocyclic substituted 4-benzoyl-pyrazole as herbicides
05/24/2000EP1001934A1 Indole compounds as cox-2 inhibitors