Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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06/06/2000 | US6071921 4-phenyl-7-arylquinoazolines; angiogenisis inhibitors and/or vascular permeability reducing effects in warm-blooded animals; anticarcinogenic and -arthritic agents; rheumatic diseases; vascular endothelium growth factor inhibitors |
06/06/2000 | US6071917 Analgesics; antiinflammatory agents; especially for the treatment of asthma, cerebral traumatic shock and allergic rhinitis; competitive binding at receptors |
06/06/2000 | US6071915 Arylsubstituted piperazines useful in the treatment of benign prostatic hyperplasia |
06/06/2000 | US6071912 Inhibit human factor xa and are therefore useful as pharmacological agents for the treatment of disease-states characterized by thrombotic activity; amino-, oxy- and thia-substituted triazines |
06/06/2000 | US6071909 Phenylbenzimidazole derivatives as ligands for GABA receptors |
06/06/2000 | US6071908 Radiation-activated cytotoxin therapy of neoplastic disease |
06/06/2000 | US6071907 Tricyclic compounds useful as FPT inhibitors |
06/06/2000 | US6071903 2,3,4,5-tetrahydro-1H-[1,4]-benzodiazepine-3-hydroxyamic acids |
06/06/2000 | US6071900 Heterocyclic compounds and their use |
06/06/2000 | US6071895 Polar-substituted hydrocarbons |
06/06/2000 | US6071860 For selective control of broad-leaved and grass weeds in crops of useful plants |
06/02/2000 | WO2000031074A2 Indole derivatives and their use as serotonin receptor ligands |
06/02/2000 | WO2000031072A1 Process for making 5-substituted pyrazoles using dithietanes |
06/02/2000 | WO2000031068A1 Polyhydroxylated heterocyclic derivatives as anti-coagulants |
06/02/2000 | WO2000031067A1 Propanoic acid derivatives as integrin inhibitors |
06/02/2000 | WO2000031066A1 Substituted n-pyrazolyl-phenoxynicotinic acid-(thio)amides that can be used as herbicides |
06/02/2000 | WO2000031065A1 Compounds having cytokine inhibitory activity |
06/02/2000 | WO2000031064A1 Enantioselective alkylation of tricyclic compounds |
06/02/2000 | WO2000031063A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS |
06/02/2000 | WO2000031062A1 Cycloalkyl-substituted aminomethylpyrrolidine derivatives |
06/02/2000 | WO2000031061A1 2-oxoimidazole derivatives |
06/02/2000 | WO2000031047A1 Substituted 4-amino-2-aryl-cyclopenta[d]pyrimidines, their production and use and pharmaceuticalreparations containing same |
06/02/2000 | WO2000031039A1 Substituted benzo[de]isoquinoline-1,3-diones |
06/02/2000 | WO2000031038A1 Quinoline derivatives as nk-2 and nk-3 receptor ligands |
06/02/2000 | WO2000031037A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists |
06/02/2000 | WO2000031034A1 Insecticidal photostable acid salt derivatives of n-benzyl-4-benzhydrolpiperidines |
06/02/2000 | WO2000009105A3 Small molecule carbamates or ureas for vision and memory disorders |
06/02/2000 | CA2351865A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists |
06/02/2000 | CA2351725A1 Substituted pyrazoles as p38 kinase inhibitors |
06/02/2000 | CA2351526A1 Indole derivatives and their use as serotonin receptor ligands |
06/02/2000 | CA2351497A1 Cycloalkyl-substituted aminomethylpyrrolidine derivative |
06/02/2000 | CA2351348A1 Substituted benzo[de]isoquinoline-1,3-diones |
06/02/2000 | CA2350969A1 Compounds having cytokine inhibitory activity |
06/02/2000 | CA2350081A1 Process for making 5-substituted pyrazoles using dithietanes |
06/02/2000 | CA2291880A1 Novel derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one, and compositions and methods for inhibiting abnormal cell growth comprising said derivatives |
05/31/2000 | EP1004592A1 Derivatives of erythromycin, their process of preparation and their application as medicaments |
05/31/2000 | EP1004581A2 Process for the preparation of thalidomide |
05/31/2000 | EP1004580A2 Imides as inhibitors of TNF alpha |
05/31/2000 | EP1004578A2 5-oxo-pyrrolidine-2-carboxylic acid hydroxamide derivatives |
05/31/2000 | EP1004572A2 Amines as inhibitors of TNF alpha |
05/31/2000 | EP1004306A2 Estrogen agonists/antagonists |
05/31/2000 | EP1003821A1 Anisotropic retardation layers for display devices |
05/31/2000 | EP1003743A1 3,3-disubstituted piperidines as modulators of chemokine receptor activity |
05/31/2000 | EP1003738A1 Bicyclic compounds as ligands for 5-ht1 receptors |
05/31/2000 | EP1003737A1 Phenyl urea and phenyl thiourea derivatives as hfgan72 antagonists |
05/31/2000 | EP1003736A1 Substituted 4-benzoyl-pyrazoles |
05/31/2000 | EP1003734A2 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONIST |
05/31/2000 | EP1003726A1 Nitrophenyl-sulfonyl-imidazoles and use thereof for controlling vegetable and animal pests |
05/31/2000 | EP1003724A1 Substituted quinoline derivatives with antiviral action |
05/31/2000 | EP1003723A1 2-acylaminopropanamines as tachykinin receptor antagonists |
05/31/2000 | EP1003721A1 Benzylidene-1,3-dihydro-indol-2-one derivatives as receptor tyrosine kinase inhibitors, particularly of raf kinases |
05/31/2000 | EP1003541A1 Inhibitors of hiv reverse transcriptase |
05/31/2000 | EP1003540A1 $g(b)2-ADRENERGIC RECEPTOR AGONISTS |
05/31/2000 | EP1003514A1 Cyclic amine modulators of chemokine receptor activity |
05/31/2000 | EP1003512A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS |
05/31/2000 | EP1003511A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS |
05/31/2000 | EP1003504A2 Indole derivatives and their use as mcp-1 antagonists |
05/31/2000 | EP1003374A4 Inhibitors of farnesyl-protein transferase |
05/31/2000 | EP1003374A1 Inhibitors of farnesyl-protein transferase |
05/31/2000 | DE19955340A1 CCR-3-Rezeptor-Antagonisten CCR-3 receptor antagonists |
05/31/2000 | CN1255162A Protease inhibitors |
05/31/2000 | CN1255124A Substituted isoquinoline derivatives and their use as anticonulsants |
05/31/2000 | CN1255119A Protease inhibitors |
05/31/2000 | CN1255042A Diaryl ethers and processes for their preparation and herbicidal and desiccant compositions containing them |
05/31/2000 | CN1254596A Process for preparing composition to kill internal parasites |
05/31/2000 | CN1052984C New erythromycin derivative and its preparing process and application in medicine |
05/30/2000 | US6069254 Carboxamide derivatives of piperidine for the treatment of thrombosis disorders |
05/30/2000 | US6069251 Highly selective partial agonists or antagonists at brain dopamine receptor subtypes or prodrugs; diagnosis and treatment schizophrenia; antidepressants; certain movement disorders such as parkinsonism. |
05/30/2000 | US6069162 Indolyl and benzofuranyl carboxamides as inhibitors of nitric oxide production |
05/30/2000 | US6069157 Parasiticidal compounds |
05/30/2000 | US6069156 Indole derivatives as cGMP-PDE inhibitors |
05/30/2000 | US6069152 Nervous system disorders; cardiovascular disorders; gastrointestinal disorders |
05/30/2000 | US6069151 Controlling tumor necrosis factor |
05/30/2000 | US6069143 Anticoagulants |
05/30/2000 | US6069114 Herbicides for selectively controlling broad-leaved weeds and grass weeds in crops of useful plants |
05/30/2000 | US6068856 Oral pharmaceutical composition with delayed release of active ingredient for pantoprazole |
05/30/2000 | CA2206104C Adamantyl substituted oxindoles as pharmaceuticals agents |
05/30/2000 | CA1341008C A - unsaturated amines, their production and use |
05/25/2000 | WO2000029403A1 Novel pyrimidine derivatives and processes for the preparation thereof |
05/25/2000 | WO2000029397A1 New piperazine and piperidine compounds |
05/25/2000 | WO2000029386A1 Pyrimidinedione derivatives useful as alpha 1a adrenoceptor antagonists |
05/25/2000 | WO2000029382A1 Certain substituted caprolactams, pharmaceutical compositions containing them and their use in treating tumors |
05/25/2000 | WO2000029380A1 Tetrahydroisoquinoline derivatives as lhrh antagonists |
05/25/2000 | WO2000029377A1 4-aroyl-piperidin-ccr-3 receptor antagonists iii |
05/25/2000 | WO2000028975A2 Improved chemical process and pharmaceutical formulation |
05/25/2000 | WO2000018361A3 Method of treating hair loss using sulfonamides |
05/25/2000 | WO2000011951A3 Use of 5-amino-pyrazol-derivatives for combating micro-organisms |
05/25/2000 | DE19854081A1 New 2-phenoxy-N-pyrazolyl-nicotinamide derivatives, useful as pre- or post-emergence, total or selective herbicides |
05/25/2000 | DE19853278A1 New 4-amino-2-aryl-cyclopentapyrimidine derivatives are activators of soluble guanylate cyclase, useful for treating or preventing e.g. thrombosis and restenosis |
05/25/2000 | CA2351644A1 Pyrimidine derivatives and processes for the preparation thereof |
05/25/2000 | CA2351187A1 Tetrahydroisoquinoline derivatives as lhrh antagonists |
05/25/2000 | CA2350722A1 4-aroyl-piperidin-ccr-3 receptor antagonists iii |
05/24/2000 | EP1002797A1 4,5-DIHYDRO- 1H]-BENZ g]INDAZOLE-3-CARBOXYLIC ACID DERIVATIVES |
05/24/2000 | EP1002796A2 Novel quinoxalindione derivatives, their production and use in medicaments |
05/24/2000 | EP1002795A1 HIV Replication inhibiting pyrimidines |
05/24/2000 | EP1002123A1 Enzymatic kinetic resolution of an intermediate useful for preparing substituted tricyclics |
05/24/2000 | EP1001948A1 Bisimino-substituted phenyl compounds and their use as pesticides |
05/24/2000 | EP1001945A1 QUINOLINE AND QUINOXALINE COMPOUNDS WHICH INHIBIT PLATELET-DERIVED GROWTH FACTOR AND/OR p56?lck TYROSINE KINASES |
05/24/2000 | EP1001939A1 Heterocyclic substituted 4-benzoyl-pyrazole as herbicides |
05/24/2000 | EP1001934A1 Indole compounds as cox-2 inhibitors |