Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
09/2000
09/05/2000US6114368 Triazolyl disulphides
09/05/2000US6114365 Arylmethyl-carbonylamino-thiazole derivatives, process for their preparation, and their use as antitumor agents
09/05/2000US6114361 5-oxo-pyrrolidine-2-carboxylic acid hydroxamide derivatives
09/05/2000US6114360 Pyrrole compounds
09/05/2000US6114357 Hemoregulatory compounds
09/05/2000US6114354 N-substituted azaheterocyclic compounds
09/05/2000US6114349 Substituted quinoline derivatives with antiviral action
09/05/2000US6114346 Treating sleep disorders using desloratadine
09/05/2000US6114334 Piperazine derivatives as therapeutic agents
09/05/2000US6114333 2-Pyrimidineamine derivatives and processes for their preparation
09/05/2000US6114329 5-HT4 receptor antagonists useful in the treatment of gastroinstestinal, cardiovascular and CNS disorders
09/05/2000US6113946 Self-assembling polynucleotide delivery system comprising dendrimer polycations
09/05/2000US6113527 3,3-bis-hydroxymethyl-7-(cis-4-isopropyl-cyclohexyl)-1-phenyl -1,7-diaza-spiro-(3.5)nonane-2-one, for example; agonists of the orphanin fq (ofq) receptor; useful in the treatment of psychiatric, neurological and physiological disorders
08/2000
08/31/2000WO2000050872A2 A system for cell-based screening
08/31/2000WO2000050470A2 Catalysts containing n-pyrrolyl substituted nitrogen donors
08/31/2000WO2000050419A1 Substituted bicyclic heterocycles and the use thereof as thrombin inhibitors
08/31/2000WO2000050417A1 Anti-cancer dihydroquinazoline derivatives
08/31/2000WO2000050416A1 6-substituted heteroquinolinecarboxylic acid derivatives and addition salts thereof and processes for the preparation of both
08/31/2000WO2000050408A1 Pyridazin-3-one derivatives and medicines containing the same
08/31/2000WO2000050406A1 Isoquinoline derivatives and isoquinoline combinatorial libraries
08/31/2000WO2000050405A1 Quinoline derivatives as tyrosine kinase inhibitors
08/31/2000WO2000050403A1 N-[2-hydroxy-3-(1-piperidinyl)propoxy]pyridine-1-oxide-3-carboximidoyl chloride and its use in the treatment of insulin resistance
08/31/2000WO2000050401A1 3-phenylpyridine derivatives and their use as nk-1 receptor antagonists
08/31/2000WO2000050400A1 2-aminopyridines containing fused ring substituents
08/31/2000WO2000050399A1 Inhibitors of cellular niacinamide mononucleotide formation and their use in cancer therapy
08/31/2000WO2000050398A2 Phenyl- and pyridinyl derivatives as neurokinin 1 antagonists
08/31/2000WO2000050397A1 Substituted piperidinedione derivatives and herbicide
08/31/2000WO2000050396A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
08/31/2000WO2000050395A1 Sulfonamide-containing indole compounds
08/31/2000WO2000050037A1 Nitrosated and nitrosylated proton pump inhibitors, compositions and methods of use
08/31/2000WO2000012074A3 Use of piperidines and/or piperazines as inhibitors of p38-alpha kinase
08/31/2000WO2000007996A3 Pyrazoles as estrogen receptor modulators
08/31/2000WO2000001375A3 Calcium channel blockers
08/31/2000DE19908567A1 New 4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors, polyps or respiratory or gastrointestinal diseases
08/31/2000DE19907813A1 Substituierte bicyclische Heterocyclen, deren Herstellung und deren Verwendung als Arzneimittel Substituted bicyclic heterocycles, their preparation and their use as medicaments
08/31/2000DE10008367A1 New 1-alkoxy-substituted hindered 2,2,6,6-tetramethylpiperidine group-containing amines useful as stabilizers for (thermoplastic) polymers, coatings, color photographic materials and printing inks
08/31/2000DE10008042A1 Neurokinin-1-Rezeptorantagonisten Neurokinin-1 receptor antagonists
08/31/2000CA2371876A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
08/31/2000CA2364754A1 6-substituted heteroquinolinecarboxylic acid derivatives and addition salts thereof and processes for the preparation of both
08/31/2000CA2364708A1 Anti-cancer dihydroquinazoline derivatives
08/31/2000CA2363628A1 Catalysts containing n-pyrrolyl substituted nitrogen donors
08/30/2000EP1031570A1 Immuno-modulator exhibiting anti-microbial and anti-mycobacterial activities, method for producing the same and pharmaceutical preparation for treating mycobacterioses as well as lung chronic and non specific conditions, sexually transmitted diseases and the resulting immuno-deficiency
08/30/2000EP1031569A1 Processes for producing 7-isoindolinequinolonecarboxylic derivatives and intermediates therefor, salts of 7-isoindolinequinolonecarboxylic acids, hydrates thereof, and composition containing the same as active ingredient
08/30/2000EP1031564A1 Inhibitors of cellular nicotinamide mononucleotide formation and their use in cancer therapy
08/30/2000EP1031563A1 Sulfonyl derivatives
08/30/2000EP1030844A1 Compounds which inhibit tryptase activity
08/30/2000EP1030843A1 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000EP1030838A1 Method of synthesis of pyrrole amides
08/30/2000EP1030836A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
08/30/2000EP1030665A1 Therapeutic uses of quinoline derivatives
08/30/2000EP1030662A2 Treatment of t-helper cell type 2 mediated immune diseases with retinoid antagonists
08/30/2000EP0769010B1 2-[1',2',4'-triazol-3'-yloxymethylene]-anilides and their use as pest-control agents
08/30/2000CN1265098A Heterocyclic derivatives which inhibit factor XA
08/30/2000CN1265034A Treatment of hepatic cirrhosis
08/30/2000CN1265033A Certain diarylimidaozle derivatives, new class of NPY speific ligands
08/29/2000US6110947 An analgesic agent for treating stroke, abdominal pain; as antiinflammatory, diuretic, anesthetic or neuroprotective agents
08/29/2000US6110945 An antiinflammatory agent inhibiting the binding of integrins to their ligands; in the prophylaxis for treating immune or inflammatory disorders
08/29/2000US6110941 Compounds analogous to thalidomide from the class comprising piperidine-2,6-diones
08/29/2000US6110939 As a substance p antagonists treating tachykinin-mediated disease, asthma, central nervous system disorder
08/29/2000US6110938 1-(arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-4-(heteroaryl)piperidines and related compounds useful as antipsychotics and analgesics
08/29/2000US6110934 Substituted benzamide derivatives and their use as anticonvulsants
08/29/2000US6110927 Treatment of atrial fibrillation
08/29/2000US6110924 Barbituric acid derivatives, processes for their production and pharmaceutical agents containing these compounds
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/29/2000US6110871 2-((phenyl, pyridyl or pyrazolyl)(oxy or thio)), 6-((substituted)phenyl)-cyanopyridines; herbicidal activity with the necessary selectivity and enhanced soil degradation
08/29/2000CA2012628C New fluoro-4 benzoic derivatives, process for their preparation and pharmaceutical compositions containing them
08/24/2000WO2000049021A2 16-halogen-epothilone derivatives, method for producing them and their pharmaceutical use
08/24/2000WO2000049015A1 Pyridine compounds and their pharmaceutical use
08/24/2000WO2000048994A1 Thioamide derivatives
08/24/2000WO2000048989A1 Mevinolin derivatives
08/24/2000WO2000048584A2 Aroyl aminoacyl pyrroles for use in the treatment of neuropathic pain
08/24/2000WO2000015992A3 Tube for lining pipes and channels, and a method and device for the production thereof
08/24/2000WO2000002887B1 Ligands for metals and metal-catalyzed processes
08/24/2000DE19908765A1 New, chemically and metabolically stable 16-halo or cyano-epothilone derivatives are cell division regulators useful e.g. for treating malignant tumors or chronic inflammatory disease
08/24/2000CA2361390A1 Aroyl aminoacyl pyrroles for use in the treatment of neuropathic pain
08/24/2000CA2361278A1 16-halogen-epothilone derivatives, method for producing them and their pharmaceutical use
08/23/2000EP1029853A1 Heteroaromatic bicyclic derivatives useful as anticancer agents
08/23/2000EP1029851A1 Piperazine compounds and medicinal use thereof
08/23/2000EP1028958A1 Arylpiperazines as serotonin reuptake inhibitors and 5-ht1d alpha antagonists
08/23/2000EP1028957A1 Piperidine derivatives and their use as tachykinin antagonists
08/23/2000EP1028956A1 Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom
08/23/2000EP1028955A1 Pyrimidinone compounds and pharmaceutical compositions containing them
08/23/2000EP1028954A1 Substituted imidazoles useful in the treatment of inflammatory diseases
08/23/2000EP1028953A1 Aromatic heterocyclic compounds as anti-inflammatory agents
08/23/2000EP1028949A1 Carbamoylphenylsulfonyl ureas, method for their production and their application as herbicides and plant growth regulators
08/23/2000EP1028948A1 Phenyl-alkyl-imidazoles as h3 receptor antagonists
08/23/2000EP1028945A1 Substituted pyridine compounds as anti-inflammatory agents
08/23/2000EP1028943A2 Orally-active nipecotamide glycolamide esters for the treatment of thrombosis disorders
08/23/2000EP0667859B1 Molecule labelling using 2-hydraninopyridine derivatives
08/23/2000EP0658159B1 Arylidene and heteroarylidene oxindole derivatives as tyrosine kinase inhibitors
08/23/2000CN1264385A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same
08/23/2000CN1264378A Quinoline-4-carboxamide derivatives as NK-2 and NK-3 receptor antagonists
08/23/2000CN1264377A Substituted pyrazoles as P38 kinase inhabitors
08/23/2000CN1264376A 3(5)-Heteroaryl substituted pyrazoles as P38 kinase inhibitors
08/23/2000CN1264375A Crystal modification of N-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use
08/23/2000CN1264367A Nitrophenyl-sulfonyl-imidazoles and use thereof for controlling vegetable and animal pests
08/23/2000CN1264300A Arylsubstituted piperazines useful in the threatement of bening prostatic hyperlasia
08/23/2000CN1055684C Method for preparing substituted pyridine
08/22/2000USRE36831 Iron-pyridone complexes for anemia