Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
06/2000
06/21/2000EP1009738A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
06/21/2000EP1009405A1 Pyrrolidine and piperidine modulators of chemokine receptor activity
06/21/2000DE19858779A1 New 3-acylamino-propionic acid and 3-sulfonylamino-propionic acid derivatives useful as endothelin receptor antagonists in treatment of e.g. cardiovascular and renal disorders, migraine and cancer
06/21/2000CN1257496A Block oligomers containing 1-hydrocarbyloxy-2,2,6,6-tetramethyl-4-piperidyl groups as stabilizer for organic materials
06/21/2000CN1257495A Block oligomers containing 1-hydrocarbyloxy-2,2,6,6-tetramethyl-4-piperidyl groups as stabilizers for organic materials
06/21/2000CN1257494A Block oligomers containing 1-hydrocarbyloxy-2,2,6,6-tetramethyl-4-piperidyl groups as stabilizers for organic materials
06/21/2000CN1257493A Block oligomers containing 1-hydrocarbyloxy-2,2,6,6-tetramethyl-4-piperidyl groups a stabilizers for organic materials
06/21/2000CN1257492A Block oligomers containing 1-hydrocarbyloxy-2,2,6,6-tetramethyl-4-piperidyl groups as stabilizers for organic materials
06/21/2000CN1257491A 4-tetrahydropyridylpyrimidine derivatives
06/21/2000CN1257490A Substituted pyridylpyrazoles as herbicides, insecticides and acaricides
06/21/2000CN1257489A Substituted benzopyran derivatives for the treatment of inflammation
06/21/2000CN1257485A Azacyclooctane and heptane derivatives, their preparation and usein therapy
06/21/2000CN1257073A 1-cyclopropyl-6-fluorine-7-(3-methyl piperazine-1-base)-8-methoxy-1,4-dihydrogen-4-oxochinoline-3-carboxylic acid and its salt and preparation process thereof
06/21/2000CN1053666C Benzoheterocylic compounds and process for preparing medicated salt thereof
06/21/2000CN1053660C Process for preparing indole derivatives containing 1,2,4-triazol-1-yl substituents
06/21/2000CN1053659C Pesticidal 1-aryl-5-(substituted alkylideneimino) pyrazoles
06/21/2000CN1053658C Aminostilbazole derivative and medicine
06/21/2000CN1053657C Didepside phthaleins based internal parasite compositions, novel didepside phthaleins and preparation process thereof
06/20/2000US6077857 Heterocyclic compounds containing two amide groups which have hemoregulatory activities, can be used to stimulate hematopoiesis and for the treatment of viral, fungal and bacterial infections
06/20/2000US6077853 Inhibitors of farnesyl-protein transferase
06/20/2000US6077850 Useful for treating cyclooxygenase-2 mediated disorders, such as inflammation and inflammation-related disorders
06/20/2000US6077840 For treating or preventing progesterone-related diseases, for having an abortion, or for orally preventing conception, breast cancer, ovarian cancer, hysteromyoma, endometriosis, meningioma, myeloma, osteoporosis
06/20/2000US6077814 1-Substituted 4-carbamoyl-1,2,4-triazol-5-one derivatives and herbicide
06/17/2000CA2292246A1 New hydrazide derivatives, the procedure for preparing them and the pharmaceutical formulations that contain them
06/15/2000WO2000034437A2 Inhibitors of prenyl-protein transferase
06/15/2000WO2000034271A1 Method for producing pyrazolylbenzoyl derivatives and novel pyrazolylbenzoyl derivatives
06/15/2000WO2000034266A1 Indole derivatives and their use as 5-ht1f agonists
06/15/2000WO2000034265A2 Quinoline-indole antimicrobial agents
06/15/2000WO2000034255A1 Substituted thiazoles for treatment of human diseases involving modulators of p-, l- and e- selectin
06/15/2000WO2000034243A1 N-(2-phenyl-4-piperidinybutyl)-5,6,7,8-tetrahydro-1-naphthalenecarboxamides and their use as neurokinin 1 (nk1) and/or neurokinin 2 (nk2) receptor antagonists
06/15/2000WO2000033844A1 Aryl and heterocyclyl substituted pyrimidine derivatives as anti-coagulants
06/15/2000WO2000033836A1 5-membered heterocycles for the treatment of human diseases involving modulators of selectins
06/15/2000WO2000009107A3 Sulfonamides of n-containing heterocyclic thioesters for vision and memory disorders
06/15/2000WO2000006531A3 Nitric esters and nitrate salts of specific drugs
06/15/2000DE19959619A1 Hindered amine products used as light and heat stabilizers and antioxidants for organic material, especially synthetic polymer, contain partly acylated 2,2,6,6-tetramethylpiperidino groups
06/15/2000DE19857202A1 New benzimidazolyl amidine or nitrile compounds, useful as thrombin inhibitors or antithrombotic agents, for treating deep leg vein thrombosis
06/15/2000CA2354040A1 Aryl and heterocyclyl substituted pyrimidine derivatives as anti-coagulants
06/15/2000CA2353572A1 Method for producing pyrazolylbenzoyl derivatives and novel pyrazolylbenzoyl derivatives
06/15/2000CA2351390A1 Thiourea inhibitors of herpes viruses
06/14/2000EP1007524A1 Indole derivatives as 5-ht1b and 5-ht1d agonists
06/14/2000EP1007522A1 2- 4-[4-(4, 5-dichloro -2-methylimidazol-1-yl) butyl]-1-piperazinyl -5-fluoropyrimidine,preparation and therapeutic use
06/14/2000EP1007521A1 Compounds possessing neuronal activity
06/14/2000EP1007520A1 2-aminopyridines containing fused ring substituents as nos inhibitors
06/14/2000EP1007515A1 Arylpyridazinones as prostaglandin endoperoxide h synthase biosynthesis inhibitors
06/14/2000EP1007513A1 Pesticidal 1-aryl-3-iminopyrazoles
06/14/2000EP1007512A1 Branched alkoxy-subsituted 2-aminopyridines as nos inhibitors
06/14/2000EP1007056A1 Method for the treatment of cystic fibrosis
06/14/2000EP1007051A1 Integrin receptor antagonists
06/14/2000EP1007047A1 Use of mizolastine for preparing a medicine for treating inflammation
06/14/2000EP1007044A1 Quinazolinone-containing pharmaceutical compositions for prevention of neovascularization and for treating malignancies
06/14/2000EP1007037A1 Antithrombotic agents
06/14/2000EP0525057B1 Antimicrobial quinolonyl lactams
06/14/2000CN1256275A Sulfoxide compound and complex of acetone, and production method thereof
06/14/2000CN1053444C Process for refining omeprazole
06/14/2000CN1053438C Benzodiazepin-2-one derivatives, process for their prepn. and pharmaceutical composition containing them
06/14/2000CA2292015A1 Sterically hindered amine compounds
06/13/2000USRE36736 Substituted pyrroles
06/13/2000US6075165 Process for the preparation of polyhalogenated benzotrifluorides, benzotrichlorides and benzoyl chlorides and new trihalogenobenzotrichlorides and -benzoyl chlorides
06/13/2000US6075043 Parasiticidal pyrazoles
06/13/2000US6075041 Cyclic amides
06/13/2000US6075040 Obesity and diabetes
06/13/2000US6075039 5HT receptor binding benzimidazolylpiperidines
06/13/2000US6075034 Spiro[piperidine-4,1'-pyrrolo [3,4-C] pyrrole]derivatives
06/13/2000US6075025 Tricyclic carbamate compounds useful for inhibition of G-protein function and for treatment of proliferative diseases
06/13/2000US6075024 Methods for treating infection using optically pure (S)-lomefloxacin
06/13/2000CA2085878C Bis-benzo or benzopyrido cyclo hepta piperidene, piperidylidene and piperazine compounds and compositions
06/13/2000CA2014062C Pyridine derivatives
06/13/2000CA1341023C Peptide derivatives
06/08/2000WO2000032590A1 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS
06/08/2000WO2000032588A2 Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
06/08/2000WO2000032587A1 Sf2809-i, ii, iii, iv, v and vi substances exhibiting chymase-inhibiting activities
06/08/2000WO2000032579A1 Substituted benzimidazoles and their use as parp inhibitors
06/08/2000WO2000032577A2 Substituted benzo[de]isoquinoline-1,3-diones
06/08/2000WO2000032575A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS
06/08/2000WO2000032574A1 Novel 2-pyridone derivatives, preparation method and therapeutic use
06/08/2000CA2352045A1 Substituted benzo[de]isoquinoline-1,3-diones
06/08/2000CA2347701A1 .beta.-alanine derivatives as .alpha.4 integrin inhibitors
06/07/2000EP1006113A1 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use to inhibit abnormal cell growth
06/07/2000EP1006112A1 3-Hydroxy-2(1H)-pyridinone or 3-hydroxy-4(1H)-pyridinone derivatives useful as reactive oxygen species (ROS) scavengers
06/07/2000EP1006110A1 Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments
06/07/2000EP1005493A1 Antiviral protease inhibitors
06/07/2000EP1005459A1 Substituted isoquinolines as anticonvulsivants
06/07/2000EP1005456A1 Method for producing organic compounds
06/07/2000EP1005455A1 Method for producing substituted-2-nitroguanidine derivatives
06/07/2000EP1005454A1 2-acylaminopropanamines as tachykinin receptor antagonists
06/07/2000EP1005446A1 N-aroylphenylalanine derivatives
06/07/2000EP1005445A1 N-alkanoylphenylalanine derivatives
06/07/2000EP1005361A1 USE OF FVIIa OR FVIIai FOR THE TREATMENT OF ADVERSE CONDITIONS RELATED TO THE FVIIa MEDIATED INTRACELLULAR SIGNALLING PATHWAY
06/07/2000EP1005356A1 Novel antibacterial agents
06/07/2000EP1005343A1 Use of csaid?tm compounds as inhibitors of angiogenesis
06/07/2000EP0773025B1 New stable galenic formulations containing an acid-labile benzimidazol compound, and production process
06/07/2000CN1255918A Synthesis of acridine derivative multidrug-resistant inhibitors
06/07/2000CN1255916A Chemical process for reduction of 1-substituted-3--hydroxymethyl-4-(4-fluorophenyl) tetrahydropyridines
06/07/2000CN1255497A Method for preparing pyrazo [4,3-d] pyrimidine-7-one and its intermediate
06/07/2000CN1255493A Novel dihydro and tetrahydro chinoline compounds, its prepn. method and medicinal compsns.
06/07/2000CN1053190C Quinoxalindione derivs, their prepn. and their used in drugs
06/06/2000US6071948 Treatment of diseases caused by excessive blood vessel growth
06/06/2000US6071935 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use as farnesyl protein transferase inhibitors
06/06/2000US6071932 Carbazolypiperines as GABA uptake inhibitors
06/06/2000US6071931 AT1 -receptor antagonists for preventing and treating postischemic renal failure and for protecting ischemic kidneys