Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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11/02/2000 | EP1048655A1 1,2-dihydro-2-oxoquinoline derivatives |
11/02/2000 | EP1048652A1 Aromatic compounds having cyclic amino or salts thereof |
11/02/2000 | EP1047692A1 Methods of synthesizing and screening inhibitors of bacterial nad synthetase enzyme, compounds thereof and methods of treating bacterial and microbial infections with these inhibitors |
11/02/2000 | EP1047691A1 Quinolinepiperazine and quinolinepiperidine derivatives, their preparation and their use as combined 5-ht1a, 5-ht1b and 5-ht1d receptor antagonists |
11/02/2000 | EP1047690A1 Heterocyclic ether and thioether compounds useful in controlling chemical synaptic transmission |
11/02/2000 | EP1047689A1 Substituted guanidine derivatives |
11/02/2000 | EP1047684A1 Substituted alpha,beta-anellated butyrolactones |
11/02/2000 | EP1047678A1 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders |
11/02/2000 | EP1047675A1 Chemokine receptor antagonists and methods of use therefor |
11/02/2000 | EP1047673A1 Novel heterocyclic compounds |
11/02/2000 | EP1047425A1 Integrin receptor antagonists |
11/02/2000 | EP1047418A1 Inhibition of raf kinase using substituted heterocyclic ureas |
11/02/2000 | EP0808312B1 Indole derivatives as 5-ht receptor antagonist |
11/02/2000 | CA2371308A1 Tri-aryl acid derivatives as ppar receptor ligands |
11/02/2000 | CA2371274A1 Selective npy (y5) antagonists |
11/02/2000 | CA2370241A1 Tetrahydroisoquinolinyl-indole derivatives for the treatment of depression |
11/02/2000 | CA2367695A1 Heteroaryl diazacycloalkanes, their preparation and use |
11/01/2000 | CN1272108A Indole derivatives as 5-HT1B and 5-HT1D agonists |
11/01/2000 | CN1058010C Novel quinoline carboxylic acid derivatives having 7-(4-aminomethyl-3-oxime) pyrrolidine substituent and process for preparing thereof |
10/31/2000 | US6140504 Substituted intermediate compounds for the preparation of n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides |
10/31/2000 | US6140372 Acyl derivatives of melatonin and of melatoninergic analogues and their use as medicinal products |
10/31/2000 | US6140361 For inhibiting binding of human immunodeficiency virus rev protein to rev responsive elements (rre) |
10/31/2000 | US6140357 Small molecule inhibitors of rotamase enzyme activity |
10/31/2000 | US6140352 Carbazolyl-substituted ethanolamines as selective β-3 agonists |
10/31/2000 | US6140351 Ortho-anthranilamide derivatives as anti-coagulants |
10/31/2000 | US6140349 Cyclic amine modulators of chemokine receptor activity |
10/31/2000 | US6140345 For treating psychoses and pain |
10/31/2000 | US6140344 For treating pathological conditions such as asthma, rhinitis, eczema and parasitic infections featuring tissue eosinophilia |
10/31/2000 | US6140342 Cholesteryl ester transfer protein inhibitor; used to elevate certain plasma lipid levels, including high density lipoprotein-cholesterol and to lower certain other plasma lipid levels, such as ldl-cholesterol and triglycerides |
10/31/2000 | US6140339 Monomeric and dimeric arylisoquinoline alkaloids and derivatives thereof |
10/31/2000 | US6140338 For treating acute inflammatory diseases, chronic inflammatory diseases, acquired immune deficiency syndrome, cancer, ischemic reflow disorder and/or arteriosclerosis |
10/31/2000 | US6140335 Use of mizolastine for treating inflammatory diseases associated with 5-lipoxygenase |
10/26/2000 | WO2000063207A1 Pesticidal indazole or benzotriazole derivatives |
10/26/2000 | WO2000063204A2 Substituted azoles |
10/26/2000 | WO2000063203A1 Piperidine-indole compounds having 5-ht6 affinity |
10/26/2000 | WO2000063186A1 Process and intermediates for preparing benzodiazepines |
10/26/2000 | WO2000063183A1 Process for the preparation of substituted pyrimidines |
10/26/2000 | WO2000063172A1 N-substituted piperidine derivatives |
10/26/2000 | WO2000063171A1 Tricyclic compounds |
10/26/2000 | WO2000063168A1 Synthesis of azetidine derivatives |
10/26/2000 | WO2000063140A1 Template directed solid-state organic synthesis |
10/26/2000 | WO2000062782A1 Novel synthesis and crystallization of piperazine ring-containing compounds |
10/26/2000 | WO2000039082A3 1,2-annelated quinoline derivatives |
10/26/2000 | WO2000035886A3 (hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors |
10/26/2000 | WO2000035865A3 Tubulin-binding agents |
10/26/2000 | WO2000021508A3 Novel therapeutic use of compounds with beta-3-agonist activity |
10/26/2000 | WO2000004012A9 COMPOUNDS SPECIFIC FOR THE HUMAN α1d ADRENERGIC RECEPTOR AND USES THEREOF |
10/26/2000 | DE19918211A1 New 2-carbocyclyl-benzimidazole-carboxamide derivatives, are PARP inhibitors useful e.g. for treating neurodegenerative disease, epilepsy, ischemia, tumors, inflammation or diabetes |
10/26/2000 | CA2370417A1 Substituted azoles |
10/26/2000 | CA2370285A1 Process for the preparation of substituted pyrimidines |
10/26/2000 | CA2370265A1 Pesticidal indazole or benzotriazole derivatives |
10/26/2000 | CA2368815A1 Novel synthesis and crystallization of piperazine ring-containing compounds |
10/25/2000 | EP1045846A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof |
10/25/2000 | EP1045845A1 N-oxides of heterocyclic compounds with tnf and pde-iv inhibiting activity |
10/25/2000 | EP1045844A1 Inhibitors of farnesyl-protein transferase |
10/25/2000 | EP1045843A1 Inhibitors of farnesyl-protein transferase |
10/25/2000 | EP1045842A2 Methods of use and compositions for benzylidene- and cinnamylidene-anabaseines |
10/25/2000 | EP1045839A2 Novel amines as pharmaceutical agents |
10/25/2000 | EP1045837A1 Monomeric and dimeric arylisoquinoline alkaloids and derivatives thereof |
10/25/2000 | EP1045836A1 Pyridones as src family sh2 domain inhibitors |
10/25/2000 | EP1045835A1 Catalyst and method for amide formation |
10/25/2000 | EP1045834A1 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders |
10/25/2000 | EP1045833A1 2,3-substituted indole compounds as cox-2 inhibitors |
10/25/2000 | EP1045693A1 Aminophenoxyacetic acid derivatives as neuroprotectants |
10/25/2000 | EP0720601B1 Gastrin and cck receptor ligands |
10/25/2000 | CN1271357A bisethers of 1-oxa, aza and thianaphthalen-2-ones as phospholamban inhibitors |
10/25/2000 | CN1271355A Heterocyclic compounds and antitumor agent containing the same as active ingredient |
10/25/2000 | CN1271354A Compounds possessing neuronal activity |
10/25/2000 | CN1271349A Substituted quinazoline derivatives and their use as tyrosine kinase inhibitors |
10/25/2000 | CN1271348A Method for producing (hetero) aromatic hydroxylamines |
10/25/2000 | CN1271346A Method for producing substituted 2-nitroguanidine derivative |
10/25/2000 | CN1271345A Method for producing substituted 2-nitroguanideine derivatives |
10/25/2000 | CN1271284A Vitronectin receptor antagonist |
10/25/2000 | CN1270959A 4-phenyl pyridine derivatives |
10/24/2000 | US6137002 Glycoprotein IIb/IIIa antagonists |
10/24/2000 | US6136844 5-aroylpyrrol-2-ylmethylarene derivatives |
10/24/2000 | US6136834 Tetrazole compounds and pharmaceutical agents containing such derivative |
10/24/2000 | US6136826 Aminopiperidine compounds substituted with alkanoyl |
10/24/2000 | US6136823 Pyridonecarboxylic acid derivatives or salts thereof and drugs containing the same as the active ingredient |
10/24/2000 | US6136822 Quinolinone derivative, method for preparing the same, and anti-allergic agent |
10/24/2000 | US6136812 Methods of administering AMPA receptor antagonists to treat dyskinesias associated with dopamine agonist therapy |
10/24/2000 | US6136800 Steroids |
10/24/2000 | US6136344 Oral pharmaceutical dosage form |
10/19/2000 | WO2000061608A2 Low-molecular inhibitors of complement proteases |
10/19/2000 | WO2000061580A1 Substituted bicyclic heteroaryl compounds as integrin antagonists |
10/19/2000 | WO2000061579A1 New endothelin converting enzyme inhibitors, their production and their use |
10/19/2000 | WO2000061577A1 Prodrugs of thrombin inhibitors |
10/19/2000 | WO2000061576A1 Triarylimidazoles |
10/19/2000 | WO2000061575A1 Process for the production of indole derivatives and intermediates therefor |
10/19/2000 | WO2000061564A1 Antiviral pyrimidinedione derivatives and process for the preparation thereof |
10/19/2000 | WO2000061563A1 Antiviral pyrimidinedione derivatives and process for the preparation thereof |
10/19/2000 | WO2000061562A1 Neurotrophic substituted pyrimidines |
10/19/2000 | WO2000061561A1 Cyanoguanidine compounds |
10/19/2000 | WO2000061551A2 Pyrimidine-2-one derivatives as integrin receptor ligands |
10/19/2000 | WO2000061549A2 Pharmaceutical compounds |
10/19/2000 | WO2000061541A2 Pharmaceutical compounds |
10/19/2000 | WO2000061537A2 Pharmaceutical compounds |
10/19/2000 | WO2000007996A8 Pyrazoles as estrogen receptor modulators |
10/19/2000 | DE19917504A1 New hydroxy-indole derivatives, useful in treatment of degenerative joint disease, viral and parasitic infections, bronchial, dermatological, neurodegenerative and prostate disorders, etc. |
10/19/2000 | DE19916719A1 Neue ECE-Inhibitoren, ihre Herstellung und Verwendung New ECE inhibitors, their preparation and use |