| Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
|---|
| 09/19/2000 | US6121308 Indole and benzimidazole antithrombotic compounds, such as 1-methyl-2-(n-(4-amidinophenyl)-aminomethyl)-5-(n-(hydroxycarbonylmethyl) -quinoline-8-sulphonylamino)-indole |
| 09/19/2000 | US6121307 Side effect reduction; administering to treat depression |
| 09/19/2000 | US6121286 Antileukotriene activity and antihistaminic activity, for treating asthma; compounds such as 6-methoxy-3-(2-(3-(2-quinolylmethoxy)benzyl)tetrazolyl)quinolin-2-one |
| 09/19/2000 | US6121284 Specified 1-(alkyl or cycloalkyl)-2-methyl-3-(alkoxycarbonyl)-4-(substituted pyridyl or aryl)-5-oxo-1,4,5,6,7,8-hexahydroquinoline compounds; treating sickle cell anemia, psychoses, depression |
| 09/19/2000 | US6121283 N-substituted-6-(2-(4-trifluoromethylphenyl)phenylcarbonyl-amino) -1,2,3,4-tetrahydroisoquinolines; treating disorders including obesity, hyperlipidemia, and diabetes; microsomal triglyceride transfer protein (mtp); apolipoprotein b (apo-b) |
| 09/19/2000 | US6121281 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use |
| 09/19/2000 | US6121280 Azabicyclic rotomase inhibitors |
| 09/19/2000 | US6121279 Phosphodiesterase inhibitor for treating respiratory system disorders |
| 09/19/2000 | US6121272 Bidentate metalloprotease inhibitors |
| 09/19/2000 | US6121267 Substituted piperazines and piperidines as central nervous system agents |
| 09/19/2000 | US6121266 Pyridazines as interleukin-1β converting enzyme inhibitors |
| 09/19/2000 | US6121262 Neurokin (tachykinin) antagonists |
| 09/19/2000 | US6121260 Appetite stimulation with dosage of neuropeptide y (npy) receptor agonist |
| 09/14/2000 | WO2000053596A2 Imidazole compounds as histamine h3 ligands |
| 09/14/2000 | WO2000053594A1 Aminomethylpyrrolidine derivatives having aromatic substituents |
| 09/14/2000 | WO2000053582A1 HETEROCYCLIC COMPOUNDS HAVING EFFECT OF ACTIVATING NICOTINIC ACETYLCHOLINE α4β2 RECEPTOR |
| 09/14/2000 | WO2000053544A1 Process for producing carboxylic acid derivative and condensing agent comprising quaternary ammonium salt |
| 09/14/2000 | WO2000044722A8 Chondrongenesis promotors and indolin-2-one derivatives |
| 09/14/2000 | WO2000031074A3 Indole derivatives and their use as serotonin receptor ligands |
| 09/14/2000 | WO2000024717A3 Isoquinoline derivatives |
| 09/14/2000 | WO2000004012A8 COMPOUNDS SPECIFIC FOR THE HUMAN α1d ADRENERGIC RECEPTOR AND USES THEREOF |
| 09/14/2000 | WO1999063999A8 H1-histamine receptor antagonists |
| 09/14/2000 | DE19911039A1 Abgewandelte Aminosäureamide, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung Modified amino acid amides, pharmaceutical compositions containing them and methods for their preparation |
| 09/14/2000 | CA2366260A1 Heterocyclic compounds having effect of activating .alpha.4.beta.2 nicotinic acetylcholine receptors |
| 09/14/2000 | CA2362319A1 Imidazole compounds as histamine h3 ligands |
| 09/13/2000 | EP1035115A1 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists |
| 09/13/2000 | EP1035110A1 Benzylaminodiacetamide derivatives, compositions containing the same, process for their preparation and uses |
| 09/13/2000 | EP1034174A1 Azaring-ether derivatives and their use as nicotinic ach receptor modulators |
| 09/13/2000 | EP1034173A2 Method for producing 8-methoxy-quinoline carboxylic acids |
| 09/13/2000 | EP1034167A1 Alpha-alkylthio substituted pyrimidine ethers and thioethers as viral reverse transcriptase inhibitors |
| 09/13/2000 | EP1034164A1 Substituted beta-alanine derivatives as cell adhesion inhibitors |
| 09/13/2000 | EP1033965A2 Agents and method for producing semi-permanent colorations of keratin fibers |
| 09/13/2000 | EP0983248A4 Analogs of duocarmycin and cc-1065 |
| 09/13/2000 | EP0764166B1 Corticotropin releasing factor antagonists |
| 09/13/2000 | EP0607193B1 Triazole antifungal agents |
| 09/13/2000 | CN1266433A Benzpyrido cycloheptane compounds useful for inhibition of franesyl protein transferase |
| 09/13/2000 | CN1266431A Aroyl-piperazine derivatives, their preparation and their use as tachykinin antagonists |
| 09/13/2000 | CN1266428A Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same |
| 09/13/2000 | CN1266057A Novel cyano-indole serotonin reextracted inhibitor compound, its preparation process and medicinal compositions having same |
| 09/13/2000 | CN1056370C 4-aryloxy (arylthio or arylamino) pyrimidine derivative with herbicide active, and preparation process thereof |
| 09/13/2000 | CN1056369C Pyridazinone derivatives or their salts, processes of their production, and anti-shock agents containing them |
| 09/12/2000 | US6117999 Chemical intermediate for nelfinavir |
| 09/12/2000 | US6117995 Oxidation of the corresponding heterocyclic amine compound |
| 09/12/2000 | US6117886 Excellent antileukotriene activity and antihistaminic activity, and is useful for the prevention and treatment of, for example, asthma. |
| 09/12/2000 | US6117885 Biphenyl-substituted quinoline derivatives |
| 09/12/2000 | US6117884 4-substituted quinoline derivatives having fungicidal activity |
| 09/12/2000 | US6117883 Useful for modulating a muscarinic receptor. |
| 09/12/2000 | US6117882 5-HT4 agonists and antagonists |
| 09/12/2000 | US6117868 Treatment of gastrointestinal ulcers or gastritis caused by microbial infection |
| 09/12/2000 | US6117866 For inhibiting platelet aggregation or clot formation and reocclusion of an artery or vein in a mammal following fibrinolytic therapy or angioplasty; for treating stroke, transient ischemia attacks, or myocardial infarction |
| 09/12/2000 | CA2105384C Treatment of addiction to drugs and substances of abuse |
| 09/08/2000 | WO2000052007A1 4-heterocyclysulfonamidyl-6-methoxy-5-(2-methoxy-phenoxy)-2-pyridyl-pyrimidine derivatives, their preparation and use as endothelin receptor antagonists |
| 09/08/2000 | WO2000052005A1 Febrifugine and isofebrifugine and processes for the preparation of both |
| 09/08/2000 | WO2000051991A1 4-AMINO-QUINAZOLINE AND QUINOLINE DERIVATIVES HAVING AN INHIBITORY EFFECT ON SIGNAL TRANsSDUCTION MEDIATED BY TYROSINE KINASES |
| 09/08/2000 | WO2000051990A1 Antiviral 2,4-pyrimidinedione derivatives and process for the preparation thereof |
| 09/08/2000 | WO2000051988A1 Nitroxyderivatives having antiinflammatory, analgesic and antithrombotic activity |
| 09/08/2000 | WO2000051987A2 Inhibitors of advanced, post-amadori glycosylation reactions |
| 09/08/2000 | WO2000051986A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers |
| 09/08/2000 | WO2000051985A1 Fluorides of 4-substituted piperidine derivatives |
| 09/08/2000 | WO2000051984A1 2-aryl indole derivatives as antagonists of tachykinins |
| 09/08/2000 | WO2000051614A1 Inhibitors of prenyl-protein transferases |
| 09/08/2000 | WO2000051611A1 Inhibitors of prenyl-protein transferase |
| 09/08/2000 | WO2000051610A1 Pyrrolidine modulators of chemokine receptor activity |
| 09/08/2000 | WO2000051609A1 3-alkyl substituted pyrrolidine modulators of chemokine receptor activity |
| 09/08/2000 | WO2000051608A1 3-thienyl and 3-furanyl pyrrolidine modulators of chemokine receptor activity |
| 09/08/2000 | WO2000051607A1 3-cyclopropyl and 3-cyclobutyl pyrrolidine modulators of chemokine receptor activity |
| 09/08/2000 | WO2000051547A2 Inhibitors of prenyl-protein transferase |
| 09/08/2000 | WO2000023060A3 Method of treating immunological disorders mediated by t-lymphocytes |
| 09/08/2000 | WO2000012497B1 Quinazoline derivatives as medicaments |
| 09/08/2000 | CA2362778A1 Inhibitors of prenyl-protein transferase |
| 09/08/2000 | CA2362495A1 Inhibitors of prenyl-protein transferases |
| 09/08/2000 | CA2362493A1 Inhibitors of prenyl-protein transferase |
| 09/08/2000 | CA2361164A1 Nitroxyderivatives having antiinflammatory, analgesic and antithrombotic activity |
| 09/08/2000 | CA2330541A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers |
| 09/07/2000 | DE19910403A1 Medicaments containing hydroxy-benzo-cyclopentabenzazepine-dione derivatives, useful as cellular hyperproliferation inhibitors, especially antitumor agents |
| 09/06/2000 | EP1033366A2 Amide derivatives useful as Neuropeptide Y (NPY) antagonists |
| 09/06/2000 | EP1032570A1 Isoquinoline derivatives and their therapeutical use |
| 09/06/2000 | EP1032569A1 Imidazole derivatives, preparation and therapeutic application thereof |
| 09/06/2000 | EP1032561A1 Substituted oximes as neurokinin antagonists |
| 09/06/2000 | EP1032559A1 Aminoalkylphenol derivatives and related compounds |
| 09/06/2000 | EP1032556A1 Pharmaceutically active compounds and methods of use |
| 09/06/2000 | EP1032424A1 Combination of an aldose reductase inhibitor and a glycogen phosphorylase inhibitor |
| 09/06/2000 | EP1032393A1 QUINOLINE-CONTAINING $g(a)-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS |
| 09/06/2000 | EP0593766B1 Pyridonecarboxylic acid derivative |
| 09/06/2000 | CN1265659A Substituted cyclobutylamine derivatives |
| 09/06/2000 | CN1265652A 2-acrylaminopropanamines as tachykinin receptor antagonists |
| 09/06/2000 | CN1265591A Coumpound |
| 09/06/2000 | CN1265585A (Imidazol-5-yl) methyl-2-quinolinone derivatives as inhibitors of smooth muscle cell proliferation |
| 09/06/2000 | CN1265394A Compound as intermediates for use in preparation of optically active 2-imidazoline-5-one or 2-imidazoline-5-thionone derivatives |
| 09/06/2000 | CN1056144C New use of 6-heterocyclic-4-amino-3,4,5-tetrahydrobenz (CD) indoles compound |
| 09/06/2000 | CN1056143C Piperidine derivatives and its use |
| 09/06/2000 | CN1056140C Biphenyl derivatives, their preparation and theirt use for treatment of hypertension and cardiac disease |
| 09/05/2000 | US6114590 Catalyzing the halogenation with potassium fluoride in the presence of a quaternary phosphonium salt or a crown ether |
| 09/05/2000 | US6114542 Ethers of polyalkyl or polyalkenyl N-hydroxyalkyl succinimides and fuel compositions containing the same |
| 09/05/2000 | US6114536 Indolin-2-one derivatives |
| 09/05/2000 | US6114535 Process and intermediates for the manufacture of pyridine-2,3-dicarboxylate compounds |
| 09/05/2000 | US6114532 Anticoagulant |
| 09/05/2000 | US6114530 Isoquiolinamines and phthalazinamines useful in treating stress related disorderes such as post traumatic stress disorder as well as depression, headache and anxiety |
| 09/05/2000 | US6114420 Triazine derivatives containing 2,2,6,6-tetramethyl-4-piperidyl groups |
| 09/05/2000 | US6114374 2-and 2,5-substituted phenylketoenols |