Patents
Sitemap › C07 - Organic chemistry › C07D - Heterocyclic compounds › C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
09/2000
09/28/2000CA2367861A1 Quinazolines and therapeutic use thereof
09/27/2000EP1038872A1 4-Phenyl-4-heteroarylpiperdine derivatives as opioid receptor ligands
09/27/2000EP1037889A1 Novel compounds
09/27/2000EP1037886A1 Triazine angiogenesis inhibitors
09/27/2000EP1037881A1 Process of preparing substituted pyrimidinones
09/27/2000EP1037880A1 Retinoic acid mimetic anilides
09/27/2000EP1037868A2 $g(a)-HYDROXY, -AMINO, AND HALO DERIVATIVES OF $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS
09/27/2000EP1037639A1 Compounds of heteroaryl substituted imidazole, their pharmaceutical compositions and uses
09/27/2000EP1037635A1 Compounds and methods
09/27/2000EP1037634A1 Novel administration form comprising an acid-labile active compound
09/27/2000EP1037633A1 Antiviral compounds
09/27/2000EP1037607A1 Novel suppository form comprising an acid-labile active compound
09/27/2000CN1268134A Bis-indole derivatives having antimetastatic activity, A process for their preparation and pharmaceutical compositions containing them
09/27/2000CN1268133A 2-Aminopyridines containing fused ring substituents as NOS inhibitors
09/27/2000CN1268132A Cis-substituted fluoromethylpyrrolidine derivatives
09/27/2000CN1268124A Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments
09/27/2000CN1268123A Benzimidazole derivatives
09/27/2000CN1268122A Branched alkoxy- substituted 2-aminopyridines as NOS inhibitors
09/27/2000CN1268116A 3-amidinoaniline derivatives activated blood coagulation factor X inhibitors, and intermediates for producing both
09/27/2000CN1267671A Process for producing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative
09/27/2000CN1056842C Amino acid derivative having anti CCK activity
09/27/2000CN1056834C Novel arylindazoles and their use as herbicides
09/27/2000CN1056832C Fused dihydropyridine derivate, its producing process, and its pharmaceutical composition
09/26/2000US6124472 Eliminating the sulfonic acid residue, with the aid of a base, from a sulfinated pyrrolinecarboxylic acid derivative
09/26/2000US6124464 Mixing a substituted sulfinyl heterocyclic compound containing an imidazole moiety with an alkylamine base or ammonia and a magnesium salt.
09/26/2000US6124463 Treatment of affective disorder, anxiety or depression
09/26/2000US6124331 Selective NPY (Y5) antagonists (tricyclics)
09/26/2000US6124330 N-[4-(Heteroarylmethyl)phenyl]-heteroarylamines
09/26/2000US6124325 Triazole antifungal agents
09/26/2000US6124324 An enzyme inhibitor of reverse transcriptase for the treatment of hiv infection, including mutant, drug-sensitive, drug-resistant, and multi-drug resistant strains of hiv
09/26/2000US6124323 4-substituted piperidine analogs and their use as subtype selective NMDA receptor antagonists
09/26/2000US6124321 An enzyme inhibitor for enhancing memory or treating or preventing alzheimer's disease
09/26/2000US6124320 Treating with non-sedating antihistamines without causing cardiac arrhythmias
09/26/2000US6124318 A neurotrophic drug treating or preventing a disease involving neuronal degeneration such as senile dementia of the alzheimer type
09/26/2000US6124317 2-substituted piperidine analogs and their use as subtype-selective NMDA receptor antagonists
09/26/2000US6124316 Compounds which are specific antagonists of the human NK3 receptor and their use as medicinal products and diagnostic tools
09/26/2000US6124306 Treating human immunodeficiency virus infections
09/26/2000US6124305 Use of N-(substituted glycyl)-2-cyanopyrrolidines in inhibiting dipeptidyl peptidase-IV
09/26/2000US6124302 4,4-disubstituted-3,4-dihydro-2(1H)-quinazolinones useful as HIV reverse transcriptase inhibitors
09/26/2000US6124297 Combatting insects or mites
09/26/2000US6124296 Arylglycinamide derivatives, methods of producing these substances and pharmaceutical compositions containing such compounds
09/26/2000US6124295 Inhibit growth of abnormal cells, such as tumor cells
09/26/2000US6124294 Compounds having high affinity for dopamine d3 receptor; used to treat disorders which respond to dopamine d3 ligands
09/26/2000US6124279 Neurokinin a antagonists, antiasthmatic agents
09/26/2000US6123962 Process for producing stabilized pharmaceutical composition
09/26/2000CA2168016C Benzimidazole derivatives
09/26/2000CA2137832C Inhibitors of angiotensin i chymase(s) including human heart chymase
09/26/2000CA1341102C Tetra-aza macrocycles and metal complexes thereof
09/21/2000WO2000055156A1 Substituted aromatic amidine derivative and medicinal composition comprising the same
09/21/2000WO2000055155A2 Heterocyclic compounds as adenosine deaminase inhibitors
09/21/2000WO2000055154A1 Modified amino-acid amides as cgrp antagonists
09/21/2000WO2000055153A1 Amide derivatives
09/21/2000WO2000055152A1 Aromatic heterocyclic compounds as anti-inflammatory agents
09/21/2000WO2000055144A1 Amine derivatives as protease inhibitors
09/21/2000WO2000055141A1 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, and processes for preparing them
09/21/2000WO2000055139A2 Heterocyclic urea and related compounds useful as anti-inflammatory agents
09/21/2000WO2000055137A1 Compounds and methods for modulation of estrogen receptors
09/21/2000WO2000055126A2 N-cyanomethylamides as protease inhibitors
09/21/2000WO2000055125A2 N-cyanomethyl amides as protease inhibitors
09/21/2000WO2000055120A1 Amide derivatives
09/21/2000WO2000054729A2 Heterocyclic aromatic compounds useful as growth hormone secretagogues
09/21/2000WO2000032577A3 Substituted benzo[de]isoquinoline-1,3-diones
09/21/2000DE19912690A1 New benzimidazolyl amidine or nitrile compounds, useful as thrombin inhibitors or antithrombotic agents, for treating deep leg vein thrombosis
09/21/2000DE19911509A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
09/21/2000DE19911366A1 New 4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors, polyps or respiratory or gastrointestinal diseases
09/21/2000CA2368148A1 Novel compounds and compositions as protease inhibitors
09/21/2000CA2368122A1 Novel compounds and compositions as protease inhibitors
09/21/2000CA2367895A1 Compounds and methods for modulation of estrogen receptors
09/21/2000CA2367461A1 Heterocyclic aromatic compounds useful as growth hormone secretagogues
09/21/2000CA2367352A1 Amine derivatives as protease inhibitors
09/21/2000CA2361939A1 Modified amino acid amides, pharmaceutical compositions containing these compounds and processes for preparing them
09/21/2000CA2361819A1 Amide derivatives
09/20/2000EP1036793A2 A process for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative
09/20/2000EP1036072A1 Thrombin receptor antagonists
09/20/2000EP1036066A1 Substituted pyrimidine and pyridine herbicides
09/20/2000EP1036065A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
09/20/2000EP1036063A1 Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
09/20/2000EP1036062A1 Hydroxamic acid derivatives as matrix metalloprotease (mmp) inhibitors
09/20/2000EP1035852A1 Inhibitors of farnesyl-protein transferase
09/20/2000EP0696288B1 Quinoxalindione derivatives, their preparation and their use in drugs
09/20/2000CN1267302A Benzo (5,6) cycloheptapyridine compounds useful as farnesyl protein transferase inhibitors
09/20/2000CN1267300A Benzo (5,6) cyclohepta (1,2-b) pyridine derivs useful for inhibition of farnesyl protein transferase
09/20/2000CN1267299A Aminooxyamide tricyclic inhibitors of farnesylprotein transferase
09/20/2000CN1267298A Benzo (5,6) cyclohepta (1,2-b) pyridine derivs useful for inhibition of farnesyl-protein transferase
09/20/2000CN1267297A Benzo (5,6) cycloheptapyridine cyclic ureas and lactams useful as farnesyl protein transferase inhibitors
09/20/2000CN1267296A Barbituric acid derivs with antimetastatic and antitumor activity
09/20/2000CN1267295A Processes for preparation of pyridine derivs.
09/20/2000CN1267294A Benzo (5,6) cyclohepta (1,2-b) pyridine derivs. for inhibition of farnesyl-protein transferase
09/20/2000CN1267293A Benzo (5,6) cyclohepta (1,2-b) pyridine derivs. useful for inhibition of farnesyl-protein transferase
09/20/2000CN1267292A Phenyl-substd. tricyclic inhibitors of farnesyl-protein transferase
09/20/2000CN1267291A N-substituted urea inhibitors of farnesyl-protein transferase
09/20/2000CN1267290A Tricyclic sulfonamide inhibitors of farnesyl-protein transferase
09/20/2000CN1267289A Carboxy piperidylacetamide tricyclic compounds useful for inhibition of G-protein function and for treatment of proliferative diseases (farnesyl protein transferase inhibitors)
09/20/2000CN1267288A Tricyclic keto amide derivs. useful as farnesyl protein transferase inhibitors
09/20/2000CN1056605C Compounds as selective human NK 3-receptor antagonists and their use
09/20/2000CN1056602C Esters and amides as PLAZ inhibitors
09/19/2000US6121471 Catalyst and method for amide formation
09/19/2000US6121456 2-(2'Hydroxyphenyl) benzotriazoles and process for their preparation
09/19/2000US6121450 Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors
09/19/2000US6121325 Naphthyl compounds promote release of growth hormone
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