Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
08/2002
08/01/2002WO2002058679A2 Antiangiogenic compounds and an assay for inhibitors of cell invasion
08/01/2002WO2002058656A1 Novel couplers for use in oxidative hair dyeing
08/01/2002WO2002058655A1 Novel couplers for use in oxidative hair dyeing
08/01/2002WO2002058654A1 Primary intermediates for oxidative coloration of hair
08/01/2002WO2002058653A1 Primary intermediates for oxidative coloration of hair
08/01/2002WO2002058632A2 Primary intermediates for oxidative coloration of hair
08/01/2002WO2002046139A3 1,7 and 1,9-diarylpolymethine salts
08/01/2002WO2002040461A3 Aminoalkoxybiphenyl carboxamides as histamine-3 receptor ligands and their therapeutic applications
08/01/2002WO2002012190A3 Non-imidazole aryloxypiperidines as h3 receptor ligands
08/01/2002WO2002002505A3 Compounds to treat alzheimer's disease
08/01/2002WO2001098279A3 Bis-arylsulfones
08/01/2002WO2001078697A3 Method and compositions for the treatment of allergic conditions using pgd2 receptor antagonists
08/01/2002US20020103239 Such as N-hydroxy-2-(((4-phenoxyphenyl)-sulfonyl)methyl) benzamide which inhibits matrix metalloprotease activity
08/01/2002US20020103238 Such as 3-benzyl-2-cyclopenten-1-one; for treatment of gastrointestinal disorders such as irritable bowel syndrome or esophageal reflux, and inhibiting side effects with administration of erythromycin
08/01/2002US20020103220 Such as N-(4-chlorobenzyl)-6-(4-morpholinylmethyl)-4-oxo-1-phenyl-1,4- dihydro-3-quinolinecarboxamide for treatment of herpes virus; viral DNA polymerase inhibitors
08/01/2002US20020103205 Muscarinic antagonists
08/01/2002US20020103198 Acylamino cyclopropane derivatives
08/01/2002US20020103194 Secondary amine, imine, amidine, guanidine, or other nitrogen functional group compounds; for treatment or prevention of diseases in which treatment is mediated by muscarinic receptor agonism such as cognitive decline and Alzheimer's disease
08/01/2002US20020103192 Perfluoroalkylketones, ketooxazoles, ketoamides, ketoesters, and diketones, and their dihydroxy derivatives, such as 7-((1,1'-biphenyl)-3-yloxy)-1-(1,3-oxazol-2-yl)-1-heptanone
08/01/2002US20020103191 Antitumor dibenzofluorene derivatives
08/01/2002US20020103164 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
08/01/2002US20020103163 Acetylenic sulfonamide thiol TACE inhibitors
08/01/2002CA2461450A1 Process for preparing higher primary alkanols
08/01/2002CA2435883A1 Benzylamine analogue
08/01/2002CA2435829A1 Trisubstituted carbocyclic cyclophilin binding compounds and their use
08/01/2002CA2435647A1 Urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and use
08/01/2002CA2435633A1 Antiangiogenic compounds and an assay for inhibitors of cell invasion
08/01/2002CA2433836A1 Novel couplers for use in oxidative hair dyeing
08/01/2002CA2431634A1 Primary intermediates for oxidative coloration of hair
08/01/2002CA2431611A1 Primary intermediates for oxidative coloration of hair
07/2002
07/31/2002EP1226128A1 New pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical agents containing these compounds
07/31/2002EP1226116A1 Processes for the preparation of sumatriptan and related compounds
07/31/2002EP1226112A2 Retro-anandamides, high affinity and stability cannabinoid receptor ligands
07/31/2002EP1226107A1 N-benzyl-p-phenylenediamine-derivatives containing colouring agents for keratin fibres and novel n-benzyl-p-phenylenediamine-derivatives
07/31/2002EP1225886A2 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
07/31/2002EP0719267B1 Second messenger cell signaling inhibitors
07/31/2002CN1088459C 1,4-disubstituted piperazines
07/31/2002CN1088457C Photochromic naphthopyran compounds
07/31/2002CN1088359C Medicine for curing cerebrovascular disturbance with psychonosema
07/30/2002US6426347 1-phenyl-4-benzylpiperazines dopamine receptor subtype specific ligands
07/30/2002US6426171 Photoresist monomer, polymer thereof and photoresist composition containing it
07/25/2002WO2002057298A2 C-terminal modified oxamyl dipeptides as inhibitors of the ice/ced-3 family of cysteine proteases
07/25/2002WO2002057261A2 Diaminothiazoles and their use as inhibitors of cyclin-dependent kinase
07/25/2002WO2002057260A1 Compounds for use in the treatment of skin conditions
07/25/2002WO2002057242A2 Urea derivatives as integrin alpha 4 antagonists
07/25/2002WO2002057236A1 Phenyl derivatives
07/25/2002WO2002057233A1 Mch antagonists and their use in the treatment of obesity
07/25/2002WO2002057230A1 Il-8 receptor antagonists
07/25/2002WO2002057218A1 Alanine 2,6-dialkoxyphenyl ester derivatives as hypnotics
07/25/2002WO2002057215A2 Sodium channel modulators
07/25/2002WO2002057211A1 Symmetrically disubstituted aromatic compounds and pharmaceutical compositions for inhibiting poly (adp-ribose) glycohydrolase, and methods for their use
07/25/2002WO2002056886A1 Angiogenesis inhibitors contaiing urea derivative as the active ingredient
07/25/2002WO2002056874A2 Lipid-based nitric oxide donors
07/25/2002WO2002044119A3 Synthesis of 2-aryl-1-naphthol derivatives via a tandem palladium catalyzed arylation and dehydrogenation
07/25/2002WO2002032874A3 Substituted heterocyclic compounds for treating multidrug resistance
07/25/2002WO2002002519A3 THROMBIN OR FACTOR Xa INHIBITORS
07/25/2002WO2001040188A9 Curcumin analogues for treating cancer
07/25/2002US20020099241 For use in protecting plants against infestation by phytopathogenic microorganisms
07/25/2002US20020099215 For therapy and prophylaxis of P-glycoprotein-mediated multidrug resistance
07/25/2002US20020099089 Administering compounds such as trans-3-(naphth-2-yl)-but-2-enoic acid-N-(2-carboxy-phenyl)-amide or like for therapy of conditions associated with increased telomerase activity, e.g. tumour diseases
07/25/2002US20020098148 Radiolabelled substituted carbonylaminobenzene derivatives which bind androgen recepotr
07/25/2002DE10102322A1 New disubstituted and trisubstituted benzene derivatives useful as coagulation inhibitors for the treatment of thromboembolic diseases
07/25/2002CA2443080A1 Lipid-based nitric oxide donors
07/25/2002CA2434939A1 Urea derivatives as integrin alpha 4 antagonists
07/25/2002CA2434636A1 Symmetrically disubstituted aromatic compounds and pharmaceutical compositions for inhibiting poly (adp-ribose) glycohydrolase, and methods for their use
07/25/2002CA2434296A1 Diaminothiazoles and their use as inhibitors of cyclin-dependent kinase
07/25/2002CA2433879A1 C-terminal modified oxamyl dipeptides as inhibitors of the ice/ced-3 family of cysteine proteases
07/24/2002EP1224165A1 Novel compounds
07/24/2002EP1223921A2 Tissue factor antagonists and methods of use thereof
07/24/2002EP1102743B1 Amide derivatives which are useful as cytokine inhibitors
07/24/2002EP0846109B1 Quinone compound, its production and use
07/24/2002CN1360577A Hydroxamic acid derivs. as matrix metalloprotease inhibitors
07/23/2002US6423717 Nervous system disorders
07/23/2002US6423714 Cyclohexene derivatives useful as antagonists of the motilin receptor
07/23/2002US6423710 Cyclic AMP-specific phosphodiesterase inhibitors
07/23/2002US6423690 Antibacterial agents
07/18/2002WO2002055519A2 Novel process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2r, 4r)-4-hydroxy -6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide
07/18/2002WO2002055496A1 Aryl piperidine and piperazine derivatives as inducers of ldl-receptor expression
07/18/2002WO2002031025A3 Biodegradable poly(beta-amino esters) and uses thereof
07/18/2002WO2002012224A3 Bicyclic compounds as h3 receptor ligands
07/18/2002WO2001072728A3 Novel piperazine derivatives
07/18/2002WO2001056974A3 Inha inhibitors and their use as antibacterials
07/18/2002US20020095055 Reacting a tertiary or secondary amine with hydrogen peroxide in presence of a recyclable heterogeneous layered double hydroxide exchanged with one of the anions of transition metal oxides as a catalyst in a solvent
07/18/2002US20020095054 Process to produce oxazolidinones
07/18/2002US20020095038 Novel method for the preparation of piperazine and its derivatives
07/18/2002US20020094979 Use of 5HT-6 antagonists
07/18/2002CA2538995A1 Novel process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2r,4r)-4-hydroxy -6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide
07/17/2002EP1222179A1 Process for preparing piperazine-substituted aliphatic carboxylates
07/17/2002EP1222163A1 2'-substituted 1,1'-biphenyl-2-carbonamides, method for the production thereof, use thereof as a medicament and pharmaceutical preparations containing said compounds
07/17/2002EP1222152A1 A method for preparing and screening one or more compounds
07/17/2002EP1039902A4 Inhibitors of gap junction communication
07/17/2002EP0939629A4 Thiol sulfonamide metalloprotease inhibitors
07/17/2002CN1359375A Novel piperazinylalkyl thiopyrimidine derivatives, pharmaceutical compositions containing the same, and a process for the preparation of same
07/17/2002CN1359373A 6[(aryl and heteroaryl)oxy] methyl] naphthalene-2-carboximidamide derivatives, preparation and therapeutic application thereof
07/17/2002CN1359371A Benzamide derivatives for the treatment of diseases mediated by cytokines
07/17/2002CN1358715A Process for one-stage catalysis synthesing N-alkyl cycloimine from hexanolactam
07/17/2002CN1087659C Hexanolactam hydrogenation for preparing hexamet hylene radical imine catalyst and its application
07/16/2002US6420561 Piperazinyl or piperidinyl acid derivatives for treatment of rheumatic diseases, arthritis due to gout and antiinflammatory agents
07/16/2002US6420560 H1—histamine receptor antagonists
07/16/2002US6420556 Multistage reaction for hypotensive agents or cardiotonic agents