Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
04/2002
04/24/2002CN1083444C Process for preparing N-alkyl ammonium acetonitrile compounds
04/24/2002CN1083419C Pentanoic acid derivatives, its preparation, medicinal materials having same and use thereof
04/23/2002US6376665 Antiarthritic agents, antiinflammatory agents
04/23/2002US6376514 Piperidine-derived compounds containing a quinolyl group that inhibits p-glycoprotein transport protein activity; for treating cancer and other diseases
04/23/2002US6376506 Sulfamide-metalloprotease inhibitors
04/23/2002US6376495 Antidiabetic piperazine derivatives, processes for their preparation and compositions containing them
04/23/2002US6376494 Cycloalkyl-substituted aryl-piperazines, piperidines and tetrahydropyridines as serotonergic agents
04/18/2002WO2002031025A2 Biodegradable poly(beta-amino esters) and uses thereof
04/18/2002WO2002030929A1 Novel pleuromutilin derivatives
04/18/2002WO2002030915A2 Aryl-indane compounds for use as inhibitors of p-glycoprotein mediated transport
04/18/2002WO2002030881A1 Sulfonylguanidine
04/18/2002WO2002030880A2 N-substituted amino acid derivatives (factor xa inhibitors)
04/18/2002WO2002030870A2 Substituted c-cyclohexylmethylamine derivatives
04/18/2002WO2002012166A3 Triamine derivative melanocortin receptor ligands and methods of using same
04/18/2002WO2002006207A3 Novel coupling components for oxidation colouring agents
04/18/2002WO2001087830A3 Substituted thioacetamides
04/18/2002US20020045777 Used to treat hypercholesterolemia, hyperlipemia, arteriosclerosis, vascular diseases, mycoses, gallstones, hyperproliferative disorders, and treatment and/or prophylaxis of impaired glucose tolerance and diabetes.
04/18/2002US20020045753 E.g., (S)-N-(4-(4-((3,4-dihydro-6-hydroxy-2,5,7,8-tetramethyl-2H-1-benzopyran-2 -yl)-carbonyl)-1-piperazinyl)phenyl)-2-thiophenecarboximidamide , or a salt thereof.
04/18/2002US20020045751 Thyromimetic organic compounds
04/18/2002US20020045749 Antibacterial agents
04/18/2002US20020045629 Sleep, eating and brain disorders, wakefulness promoters; Parkinson's disease, antiischemic agents, stroke, chronic fatigue syndrome; antidepressants; schizophrenia, nervous system disorders; multiple sclerosis, cognition activators
04/18/2002US20020045626 Benzylpiperazinyl and piperidinyl ethanone derivatives: dopamine receptor subtype specific ligands
04/18/2002DE10048716A1 Use of sulfonylguanidine derivatives, mostly new compounds, for treating e.g. pain and neurodegeneration, have affinity for the gabapentin binding site
04/18/2002CA2424107A1 Sulfonylguanidines
04/18/2002CA2423935A1 Substituted c-cyclohexylmethylamine derivatives
04/17/2002EP1196406A1 Amino ceramide-like compounds and therapeutic methods of use
04/17/2002EP1196404A1 Piperazine derivatives as modulators of chemokine receptor activity
04/17/2002EP1196403A1 Antipsychotic cyclic n-aralkyl amines
04/17/2002EP1196389A1 N-heterocyclic derivatives with neuronal activity
04/17/2002EP1196371A1 Quaternary bis-ammonium salt precursors and their uses as prodrugs having an antiparasitic activity
04/17/2002CN1345317A (1-phenacy-3-phenyl-3-piperidylethyl)piperidine derivatives, method for production thereof and pharmaceutical compositions containing the same
04/17/2002CN1345309A Diaryl derivatives and their use as medicaments
04/17/2002CN1345308A Acetylenic alpha-amino acid based sulfonamide hydroxamic acid TACE inhibitors
04/17/2002CN1345307A N-(2-phenyl-4-amino-butyl)-1-naphthamides as neurokinin-1 receptor antagonists
04/17/2002CN1345305A Method of preparing granular N-alkyl-ammonium acetonitrile salts
04/17/2002CN1345303A Oxamic acids and derivatives as thyroid receptor ligands
04/17/2002CN1345302A Production of acrylic monomers
04/17/2002CN1344717A Quaternary ammonium salt compound of piperazine with pain relieving effect
04/17/2002CN1082959C Substituted benzothienylpiperazines, their use as medicaments and processes for their preparation
04/17/2002CN1082953C Process to prepare oxazolidinones
04/17/2002CN1082790C Herbicides
04/16/2002US6372778 Sulfonamide inhibitors of aspartyl protease
04/16/2002US6372762 Heterocyclic compounds for nervous system disorders
04/16/2002US6372758 Sulfamato hydroxamic acid metalloprotease inhibitor
04/16/2002US6372752 Enzyme inhibitors, respiratory system disorders, tuberculosis and mycobacterium bactericides
04/16/2002US6372734 Crystalline dibenzothiazepine derivative and its use as an antipsychotic agent
04/16/2002CA2009690C Phenylhydrazones, the manufacture thereof and therapeutic and cosmetic compositions prepared therefrom
04/11/2002WO2002028829A2 Peptide deformylase inhibitors
04/11/2002WO2002028816A1 Substituted 5-amino-1-pentene-3-ol derivatives
04/11/2002WO2002028815A1 Pharmaceutical compounds
04/11/2002WO2002028810A2 Retinoids for the treatment of emphysema
04/11/2002WO2001066247A3 A nickel-rhenium catalyst for use in reductive amination processes
04/11/2002WO2001044161A3 Method for producing combinatorial libraries of aryl-substituted amines
04/11/2002WO2001036374A3 Bis-basic compounds for use as tryptase inhibitors, method for producing the same and their use as medicaments
04/11/2002US20020042524 Process for cis-1{2-[4-(6-methoxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenoxy] ethyl}pyrrolidine
04/11/2002US20020042517 Omega-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
04/11/2002US20020042511 New derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
04/11/2002US20020042443 Estrogen agonist / antagonist metabolites
04/11/2002US20020042414 Antiallergens
04/11/2002US20020042410 Central nervous system disorders therapy
04/11/2002US20020042406 Ring opening metathesis of alkenes
04/11/2002US20020042399 Analgesics; skin disorders
04/11/2002US20020042376 Antiinflammatory agents; autoimmune disease; antiischemic agents
04/11/2002US20020042357 Polypharmacophoric agents
04/11/2002DE10141565A1 Cyclobutanone compounds useful in liquid crystal media, especially for plasma-addressed displays, comprises substituted trans-cyclohexylene, p-phenylene and-or other cyclic groups,
04/11/2002DE10048714A1 5-Amino-1-penlen-3-ol-Derivate 5-amino-1-penlen-3-ol derivatives
04/11/2002DE10046993A1 Substituierte Zimtsäureguanidide, Verfahren zur ihrer Herstellung, ihre Verwendung als Medikament sowie sie enthaltendes Medikament Substituted Zimtsäureguanidide, processes for their preparation, their use as a medicament and they drug-containing
04/11/2002CA2419777A1 Pharmaceutical compounds
04/10/2002EP1195376A1 Azoamidine compounds and their use as polymerization initiators
04/10/2002EP1194422A1 Biaryl compounds
04/10/2002EP1194415A2 Novel piperazinylalkylthiopyrimidine derivatives, pharmaceutical compositions containing the same, and a process for their preparation
04/10/2002EP1194405A1 Sulfur-containing thyroxane derivatives and their use as hair growth promotors
04/10/2002EP1194403A1 Indanyl-substituted benzole carbonamide, method for the production of the same, use thereof as a medicament and pharmaceutical preparations containing the same
04/10/2002EP0739351B1 Monomeric diols and phosphate linked oligomers formed therefrom
04/10/2002CN1344266A Novel compounds
04/10/2002CN1344259A Processes and intermediates for prepn. of 1,3-diazin-b 6-ones and uracils
04/10/2002CN1344250A 间苯二酚衍生物 Resorcinol derivatives
04/10/2002CN1344247A Multicyclic compounds which inhibit beukocyte adhesion mediated by VLA-4
04/09/2002US6369265 Heterocoupling reaction, mixing in a liquid an aryl halide, bonding to aromatic rings, grignard reaction, metal compound and heterocyclic carbene
04/09/2002US6369226 Substituted benzamide inhibitors of rhinovirus 3C protease
04/09/2002US6369194 Alpha-beta-diketo compounds produced by reacting an alpha-keto acid or acid chloride with a ylide such as (cyanomethylene)phosphoranes, oxidizing the cyano diketo phoshorane and reacting with a nucleophile
04/09/2002US6369073 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase
04/09/2002CA2120229C Methylpiperazinoazepine derivatives, their preparation and their use
04/09/2002CA2090321C Therapeutically useful 2-aminotetralin derivatives
04/04/2002WO2002026720A2 PIPERAZINE BASED INHIBITORS OF FACTOR Xa
04/04/2002WO2002026683A1 Tandem acyl-claisen rearrangement in the preparation of chiral products
04/04/2002WO2002010178A8 Adamantyl groups containing phosphane ligands, the production and use thereof in catalytical reactions
04/04/2002WO2002004407A3 7-substituted tetracycline compounds
04/04/2002WO2001090717A3 Linker arms for nanocrystals and compounds thereof
04/04/2002WO2001090716A3 Linker arms for nanocrystals and compounds thereof
04/04/2002WO2001085694A3 Substituted diamide derivatives useful as motilin antagonists
04/04/2002WO2001047898A3 Substituted piperazine derivatives and their use as inhibitors of the microsomal triglyceride transfer protein (mtp)
04/04/2002US20020040162 Contrast media for angiography
04/04/2002US20020040061 Compounds such as 1-(3-(2-hydroxybenzoylamino)propyl)-2-pyrrolidinone; dosage forms of bioactive agents or drugs
04/04/2002US20020040060 2'-methyl-biphenyl-2-carboxylic acid-(3,5-bis-trifluoromethyl-benzyl)-methyl-amide, for example; treating disease related to neurokinin 1 receptor
04/04/2002US20020040025 Aryl substituted pyridines, pyrimidines, pyrazines and triazines and the use thereof
04/04/2002US20020040024 A phenoxy substituted piperidine derivative, useful for treating or preventing histamine H3 receptor activity
04/04/2002US20020039998 Administering to human therapeutically effective amount of a combination of drug which is metabolized by cytochrome p450 monooxygenase or pharmaceutically acceptable salt thereof and ritonavir
04/04/2002DE10044792A1 Substituierte Phenylcyclohexancarbonsäureamide und ihre Verwendung Substituted Phenylcyclohexancarbonsäureamide and their use
04/03/2002EP1192945A2 Use of an estrogen agonist/antagonist for treating osteoarthritis