Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
01/2002
01/08/2002US6337350 Inhibitors of formation of advanced glycation endproducts (AGEs)
01/08/2002CA2019622C Substituted arylamines and heteroarylamines, their preparation process and pharmaceutical composition containing them
01/03/2002WO2002000614A1 Aryl compounds, their preparation and their use in therapy
01/03/2002WO2002000606A1 Biphenyl compound
01/03/2002WO2002000574A2 Catalysis using phosphine oxide and sulfoxide compounds
01/03/2002WO2000050470A3 Catalysts containing n-pyrrolyl substituted nitrogen donors
01/03/2002US20020002192 For example, 3-benzyl-3-trichloroacetamido-1-(N-phenylamino-carbonyl)-N-(3-(2 -morpholinoethoxy)-phenyl)amino)methylcyclo-hexene; irritable bowel movement; esophageal reflux; counter-acting Erytromycin side effects
01/03/2002US20020002190 Antidiabetic agents increasing the expression of glucokinase (GK) to improve glucose tolerance; increase in glucose exposure coupled through GK in beta-cells to increase insulin secretion and in hepatocytes to increase glycogen deposition
01/03/2002US20020002158 Potentiation of glutamate receptor function; treating central nervous system disorders
01/03/2002US20020002152 Methionine aminopeptidase type 2 inhibitors; n'-((2S,3R)-3-amino-2-hydroxy-5-(isopropylsulfanyl)pentanoyl)-3-chloro benzoyl hydrazide
01/03/2002CA2740931A1 Catalysis using phosphine oxide and sulfoxide compounds
01/02/2002EP1167364A1 Benzopyran-containing compounds and prodrug forms thereof
01/02/2002EP1167348A1 Nitrile derivatives
01/02/2002EP1167342A1 Novel substituted nitrocatechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them
01/02/2002EP1167341A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them
01/02/2002EP1165545A1 Novel compounds
01/02/2002EP1165534A2 Benzoylguanidine derivatives with advantageous properties, method for producing them and their use in the production of medicaments
01/02/2002EP1165533A2 Compounds and methods for treatment of asthma, allergy and inflammatory disorders
01/02/2002EP1165512A2 Method for arylating aza-heterocycles with activated aromatic compounds in the presence of cesium carbonate
01/02/2002EP1165505A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
01/02/2002EP1165504A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF
01/02/2002EP1165502A1 Diaryl derivatives and their use as medicaments
01/02/2002EP1165501A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors
01/02/2002EP1165500A1 Amide derivatives as inhibitors of matrix metalloproteinases,tnf-alpha,and aggrecanase
01/02/2002EP1165497A1 Method of preparing granular n-alkyl-ammonium acetonitrile salts
01/02/2002EP1165495A1 Resorcinol derivatives
01/02/2002EP1165494A2 Hsv primase inhibitors
01/02/2002EP1165487A1 Derivatives of venlafaxine and methods of preparing and using the same
01/02/2002EP1165064A2 Novel inhibitors of formation of advanced glycation endproducts (age's)
01/02/2002EP0873308B1 O-carbamoyl-phenylalaninol compounds and their pharmaceutically useful salts
01/02/2002CN1328999A Piperazine dithioformates compounds, their preparation method and application in cancer-resisting medicine
01/02/2002CN1328824A Compound for curing female sexual disorder
01/02/2002CN1076949C Crop protective products
01/01/2002US6335460 Treating retroviral infections, including human immunodeficiency virus, and aids
01/01/2002US6335445 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
01/01/2002US6335444 Amino alcohol derivative and method for preparing the same
01/01/2002US6335334 Hypertensive agents, anticoagulants; cardiovascular and sexual disorders, angina pectoris, and atherosclerosis
01/01/2002US6335333 Matrix metalloproteinase inhibitors
01/01/2002US6335331 Antihistamines, antiallergens, brochodilator agents and antispasmodic agents
01/01/2002CA2093789C Bi-aromatic compounds and their use in human and veterinary medicine and in cosmetic preparations
01/01/2002CA2010217C Aralkylamine compounds
12/2001
12/27/2001WO2001098303A1 Novel process for the preparation of pyrazolopyrimidinones
12/27/2001WO2001098284A1 Process for the preparation of pyrazolopyrimidinones
12/27/2001WO2001098279A2 Bis-arylsulfones
12/27/2001WO2001098275A2 1-aryl-4-oxo-1,4-dihydro-3-quinolinecarboxamides as antiviral agents
12/27/2001WO2001098272A1 Novel compounds
12/27/2001WO2001098256A1 Thyroid receptor ligands, pharmaceutical compositions comprising them and their use in the treatment of disorders influenced by thyroid hormones
12/27/2001WO2001098253A2 1-amino-alkylcyclohexanes as 5-ht3 and neuronal nicotinicreceptor antagonists
12/27/2001WO2001098251A1 Novel substituted nitrocatechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them
12/27/2001WO2001098250A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them
12/27/2001WO2001097810A2 Use of therapeutic benzamide derivatives
12/27/2001WO2001097808A1 Combinations of depeptidyl peptidase iv inhibitors and other antidiabetic agents for the treatment of diabete mellitus
12/27/2001US20010056106 Substituted phenylamino(methylcyclobutene) derivatives are useful in treating gastrointestinal disorders associated with antagonizing the the motillin receptor
12/27/2001US20010056099 Method of reducing morbidity and the risk of mortality
12/27/2001CA2413299A1 Combinations of dipeptidyl peptidase iv inhibitors and other antidiabetic agents for the treatment of diabetes mellitus
12/27/2001CA2411255A1 Novel compounds
12/27/2001CA2410452A1 1-aryl-4-oxo-1,4-dihydro-3-quinolinecarboxamides as antiviral agents
12/27/2001CA2410447A1 Bis-arylsulfones
12/26/2001CN1328545A Hydrazine derivatives
12/25/2001CA2061875C Purification of 6-aminocapronitrile
12/21/2001CA2351129A1 Novel substituted nitrocatechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them
12/21/2001CA2351125A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them
12/20/2001WO2001096323A1 Serine protease inhibitors
12/20/2001WO2001096298A2 1,2,4-trisubstituted benzenes as inhibitors of 15-lipoxygenase
12/20/2001WO2001096293A1 Vitamin d derivatives
12/20/2001WO2001095883A1 Novel pharmaceutical formulation suitable for nebulisation
12/20/2001WO2001095856A2 Urea derivative useful as an anti-cancer agent and process for preparing same
12/20/2001WO2001087838A8 Cyclohexane derivatives and their use as therapeutic agents
12/20/2001WO2001051456A3 Antibacterial agents
12/20/2001WO2000072834A9 Agent for expression of long-term potentiation of synaptic transmission comprising compound having brain somatostatin activation property
12/20/2001US20010053774 Non-steroidal ligands for the estrogen receptor
12/20/2001DE10027604A1 Solutions of lithium-pyrrolidine in mixture of tetrahydrofuran and hydrocarbon useful for organic chemical synthesis and as polymerization catalysts
12/20/2001CA2411805A1 Serine protease inhibitors
12/20/2001CA2411495A1 1,2,4-trisubstituted benzenes as inhibitors of 15-lipoxygenase
12/19/2001EP1163221A1 Sulfonamide derivatives as 5ht7 receptor antagonists
12/19/2001EP1163213A1 Hydroxamic and carboxylic acid derivatives
12/19/2001EP1163209A1 Compounds and compositions for delivering active agents
12/19/2001EP0813520B1 Arylsulfonylamino hydroxamic acid derivatives
12/19/2001EP0721449B1 Inhibitors of beta-amyloid protein production
12/19/2001EP0720605B1 Aminocyclohexylesters and uses thereof
12/19/2001CN1327468A Organic electroluminescent element
12/19/2001CN1327443A Substituted anilides
12/19/2001CN1327383A Pharmaceutical for treatment of neurological and neuropsychiatric disorders
12/19/2001CN1076345C 2,3-diaminopropionic acid derivatives
12/18/2001US6331640 Diaminopropionic acid derivatives
12/18/2001US6331636 Treatment of central nervous system disorders, diabetes, hypertension, impotency, appetite control
12/18/2001US6331629 Certain 1-(2-naphthyl) and 1-(2-azanaphthyl)-4-(1-phenylmethyl)piperazines; dopamine receptor subtype specific ligands
12/18/2001US6331564 Use of triaryl methane compounds for inhibiting unwanted cellular proliferation associated with inflammatory disease
12/18/2001US6331563 N-Hydroxy-2-(Alkyl, Aryl, or Heteroaryl, Sulfanyl, Sulfinyl or Sulfonyl)-3-Substituted Alkyl, Aryl or Heteroarylamides as Matrix Metalloproteinase inhibitors
12/18/2001US6331542 Protease inhibitors
12/18/2001CA2213815C Pyrrolidinyl hydroxamic acid compounds and their production process
12/13/2001WO2001094354A1 Solutions of lithium pyrrolidine in tetrahydrofuran (thf)/hydrocarbons
12/13/2001WO2001094350A1 6-phenylpyrrolopyrimidinedione derivatives
12/13/2001WO2001094307A1 Propanolaminotetralines, preparation thereof and compositions containing same
12/13/2001WO2001094300A1 Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament
12/13/2001WO2001068599A3 Dosing form for reagents, use of said dosing form in organic chemical synthesis and production of said dosing form
12/13/2001WO2001049275A3 Methods and compositions for mitigating pain using nitrate esters
12/13/2001US20010051747 Diastereomer complex of at least three compounds, at least one is a resolving agent in optically active form, and at least one is an enantiomer in optically active form; rapid separation
12/13/2001US20010051729 Slurry of a sodium aluminum hydride, lithium or titanium containing additive and a Lewis base in solvent; non-pyrophoric; thermal stability
12/13/2001US20010051719 Novel compounds