Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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12/17/2003 | EP1370255A2 Cdc25 phosphatase inhibitors |
12/17/2003 | EP1109805B1 Inhibitors of bacterial nad synthetase |
12/17/2003 | EP1000047B1 1-(n-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of the phenyl ring |
12/17/2003 | CN1462268A Substituted cinnamic acid guanidides, method for the production thereof, their use as medicament, and medicine containing these compounds |
12/17/2003 | CN1131229C Salt of naphthyridine carboxylic acid derivative |
12/17/2003 | CN1131222C Benzamide derivs and their use as APOB-100 secretion inhibitors |
12/17/2003 | CN1131221C Drug dependence remedies |
12/17/2003 | CN1131220C Process for one-stage catalysis synthesing N-alkyl cyclomine from hexanolactam |
12/17/2003 | CN1131212C Phenyl-and pyridinyl derivatives |
12/16/2003 | US6664394 As inactivator of antigen- specific T cells is useful in the prophylaxis or therapy of autoimmune diseases, disorders involving an autoimmune component or neoplastic diseases |
12/16/2003 | US6664272 Such as 1,5-Bis-(2, 4-difluorophenyl)penta-1,4-diene-3 -one; administering to inhibit tissue factor and vascular endothelial growth factor (VEGF) production in cancerous tissue |
12/16/2003 | US6664259 Il-8 receptor antagonists |
12/16/2003 | US6664258 Spirocyclic dopamine receptor subtype ligands |
12/16/2003 | CA2195125C Difluorostatone antiviral agents |
12/11/2003 | WO2003102202A2 Process for preparing vinylaromatic compounds |
12/11/2003 | WO2003101974A1 Aralkyl-alcohol peiperazine derivatives and their uses as antidepressant |
12/11/2003 | WO2003101935A1 Monomer compound comprising several cationic groups, process for making the same, and polymers comprising units deriving therefrom |
12/11/2003 | WO2003101931A2 Preparation of 4-(n, n-disubstitutedamino) butyraldehyde acetals |
12/11/2003 | WO2003101927A1 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes, and parkinson's disease |
12/11/2003 | WO2003057666A3 Inhibitors of dipeptidyl peptidase iv |
12/11/2003 | WO2002083067A3 Prodrugs via acylation with cinnamate |
12/11/2003 | WO2002062778A3 Anti-thrombotic compounds, production and use thereof as medicaments |
12/11/2003 | WO1999065855A3 Combinatorial libraries of geminally substituted amines |
12/11/2003 | US20030229121 Antihistamines, antiallergens, skin disorders, antiinflammatory agents |
12/11/2003 | US20030229094 Acetamides and benzamides that are useful in treating sexual dysfunction |
12/11/2003 | US20030229072 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binning agents |
12/11/2003 | US20030229050 Insecticidal anthranilamides |
12/11/2003 | US20030228986 Polyol ester derivatives of polyamines and use in turbine oils to improve cleanliness |
12/11/2003 | US20030228978 Catalysts containing per-ortho aryl substituted aryl or heteroaryl substituted nitrogen donors |
12/11/2003 | CA2487957A1 An improved process for the preparation of 4-(n, n-disubstitutedamino) butyraldehyde acetals |
12/11/2003 | CA2486803A1 Process for preparing vinylaromatic compounds |
12/10/2003 | EP1368325A1 New asymmetric process for the preparation of diarylmethylpiperazines derivatives and novel asymmetric diarylmetylamines as intermediates |
12/10/2003 | EP1368299A2 Substituted c-cyclohexylmethylamine derivatives |
12/10/2003 | EP1083889B1 Tetrahydronaphtalene compounds and their use for the treatment of neurodegenerative diseases |
12/10/2003 | EP0971885B1 Process for preparing indane-like compounds |
12/10/2003 | EP0970046B1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors |
12/10/2003 | EP0933346B1 NOVEL p-TERPHENYL COMPOUNDS |
12/10/2003 | CN1130403C In situ block copolymer formation during polymerization of vinyl axomatic monomer |
12/09/2003 | US6660859 Arylpiperzine derivatives are useful for treatment of anxiety, depression, hypertension, cognitive disorders, sexual dysfunction, brain trauma, memory loss, eating disorders, obesity, substance abuse, and obsessive-compulsive diseases |
12/09/2003 | US6660751 Sulfonamide derivatives as 5-HT7 receptor antagonists |
12/09/2003 | US6660739 Heterocyclic amides as inhibitors of factor Xa |
12/09/2003 | US6660466 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent |
12/09/2003 | CA2269394C A process for the preparation of esters of [2-[4-[(4-clorophenyl)phenylmethyl]-1-piperazinyl]-ethoxy]acetic acid |
12/09/2003 | CA2264985C 6,8-dimercarptooctanoic acid derivatives substituted in 6-s and/or 8-s by the radical (3-methylthiopropanoyl) and pharmaceutical compositions used to treat cancerous tumors |
12/04/2003 | WO2003099819A2 Oxophenyl-cyclohexyl-propanolamine derivatives, production and use thereof in therapeutics |
12/04/2003 | WO2003099776A1 Calcium receptor modulating arylalkylamines |
12/04/2003 | WO2003099769A1 Anilino liver x-receptor modulators |
12/04/2003 | WO2003099281A2 Administration of a partial fatty acid inhibitor such as ranolazine for the treatment of diabetes |
12/04/2003 | WO2003099274A1 Hepatitis c virus inhibitors |
12/04/2003 | WO2003099266A2 Acetamides and benzamides that are useful in treating sexual dysfunction |
12/04/2003 | WO2003072062A3 Amino-substituted (e)-2,6-dialkoxystyryl 4-substituted benzylsulfones for treating proliferative disorders |
12/04/2003 | WO2003066604A3 Novel aryl- and heteroarylpiperazines |
12/04/2003 | WO2003057169A3 4-dedimethylamino tetracycline compounds |
12/04/2003 | WO2003034989A3 α-HYDROXYARYLBUTANAMINE INHIBITORS OF ASPARTYL PROTEASE |
12/04/2003 | WO2003024946A3 Oxamate derivatives containing a variously substituted nitrogen heterocycle |
12/04/2003 | WO2003020686A3 Method for producing 4-amino-1-naphthol ethers |
12/04/2003 | US20030225302 Aromatic amides, their preparation process and their use as pesticides |
12/04/2003 | US20030225285 Oxidizing a protected aminoalcohol to a chiral protected aminoaldehyde and diastereoselectively forming the aminoepoxide from said aminoaldehyde with an organometallic methylene-adding reagent in an appropriate solvent |
12/04/2003 | US20030225272 Novel mmp-2/mmp-9 inhibitors |
12/04/2003 | US20030225228 A catalyst for the polymerization of olefins, contains a titanium zirconium or hafnium complex of a dianionic bidentate ligand, (at least one of donor atoms of the ligand is a nitrogen atom substituted by a pyrrolyl group) |
12/04/2003 | US20030225179 Carbocyclic oxo, amines used as photoinitiators, formed by reacting 1-(4-(bis-(2-hydroxyethyl)-amino))-2-methyl-2-morpholino-1-propanone with caprolactone in the presence of catalysts; inks |
12/04/2003 | US20030225158 Compounds that modulate PPAR activity and methods for their preparation |
12/04/2003 | US20030225152 Such as 3-phenylaminomethylene-1,3-dihydroindol-2-one; use treating cancer, blood vessel proliferative disorders, fibrotic disorders, mesangial cell proliferative disorders and metabolic diseases |
12/04/2003 | US20030225130 Triphenylalkene derivatives and their use as selective estrogen receptor modulators |
12/04/2003 | US20030225086 Polycyclic aryl and heteroaryl substituted 1,4-quinones useful for selective inhibition of the coagulation cascade |
12/04/2003 | US20030225084 Have an affinity for the gabapentin binding site and can be used to treat conditions such as pain, epilepsy, migraine and others. |
12/04/2003 | US20030225076 Mitogen ERK Kinase ("MEK") enzyme inhibitors |
12/04/2003 | US20030225071 N-heterocyclic amides and carbamates |
12/04/2003 | US20030225065 Use of 4-(1,4-diazepan-1-yl)- or 4-piperazin-1-yl-2-aminophenyl phenyl sulfones for treatment of disorders of the central nervous system. |
12/04/2003 | US20030225059 Cyclohexyl derivatives and their use as therapeutic agents |
12/04/2003 | US20030224940 Alpha-sulfin-and alpha-sulfonamino acid amide derivatives |
12/04/2003 | CA2486644A1 Anilino liver x-receptor modulators |
12/04/2003 | CA2486564A1 Acetamides and benzamides that are useful in treating sexual dysfunction |
12/03/2003 | EP1366030A2 Melanin concentrating hormone receptor ligands |
12/03/2003 | EP1366018A1 Omega-aminoalkylamides of r-2-aryl-propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells |
12/03/2003 | EP1366015A1 Benzene-1 2-diol mannich bases ligands polymers and method of selective metal ions removal |
12/03/2003 | EP1366010A2 Method for producing vinyl, aryl and heteroaryl acetic acids and derivatives thereof |
12/03/2003 | EP1178953B1 Aromatic amides |
12/03/2003 | CN1460101A Novel compounds inhibiting factor Xa activity |
12/03/2003 | CN1460097A NF-kB inhibitor containing substituted benzoic acid derivative as active ingredient |
12/03/2003 | CN1129581C Cyanophenyl derivatives |
12/02/2003 | US6656971 Non-peptidic small organic compounds having an affinity for cyclophilin (CyP)-type immunophilins; inhibiting their peptidyl-prolyl isomerase activity; treating variety of medical conditions |
12/02/2003 | US6656965 HIV protease inhibitors based on amino acid derivatives |
12/02/2003 | US6656954 Such as N-hydroxy-2-(((4-phenoxyphenyl)-sulfonyl)methyl) benzamide which inhibits matrix metalloprotease activity |
12/02/2003 | US6656943 1-phenyl-4-benzlpiperazines: dopamine receptor subtype specific ligands |
12/02/2003 | US6656737 Reacting 9-anthracenemethanol, pyridine, and p-nitrophenyl chloroformate; reacting the product with an amine, especially piperazine, to form a product that can be used to determine the total amount of isocyanate in a sample |
12/02/2003 | US6656498 Cationic liposomes for gene transfer |
12/02/2003 | CA2244785C Pentafluorobenzenesulfonamides and analogs |
11/27/2003 | WO2003097623A1 Aralkyl-ketone piperazine derivatives and their uses as new antalgic or ataractic agent |
11/27/2003 | WO2003097589A1 Method for the production of sulphamic acid halogenides |
11/27/2003 | WO2003097576A2 Diamino-functional chalcones |
11/27/2003 | WO2003097575A2 Amino-functional chalcones |
11/27/2003 | WO2003097574A2 Aminoalkoxy-functional chalcones |
11/27/2003 | WO2003096989A2 Anti tubercular drug: compositions and methods |
11/27/2003 | WO2003014064A8 Naphthylurea and naphthylacetamide derivatives as vanilloid receptor 1 (vr1) antagonists |
11/27/2003 | WO2003009850A1 Substituted piperazines as modulators of the melanocortin receptor |
11/27/2003 | WO2002100813A3 Modulators of peroxisome proliferator activated receptors |
11/27/2003 | WO2002057242A3 Urea derivatives as integrin alpha 4 antagonists |
11/27/2003 | US20030220496 3-(optionally hydroxyl)-4-(cyclopropylcarbonyl)-cumene intermediate |
11/27/2003 | US20030220493 Selectively inhibit binding to the alpha -1a adrenergic receptor; chemical intermediates |