Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
02/2004
02/10/2004US6689909 Substituted N-phenyl 2-hydroxy-2-methyl-3,3,3-trifluoropropanamide derivatives which elevate pyruvate dehydrogenase activity
02/10/2004US6689896 Thyromimetic organic compounds
02/10/2004US6689882 Reacting a morpholine with a substituted benzene, wherein morpholine is used as a reactant and as the only one solvent
02/10/2004US6689771 Amide derivatives as inhibitors of matrix metalloproteinases, TNF-α, and aggrecanase
02/10/2004US6689174 N-benzyl-p-phenylenediamine-derivatives containing coloring agents for keratin fibres and novel n-benzyl-p-phenylenediamine-derivatives
02/05/2004WO2004011449A2 Method for the production of phenylalanine derivatives
02/05/2004WO2004011418A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc-chemokine receptor ligands
02/05/2004WO2004011410A1 Chemical compounds
02/05/2004WO2004011004A1 Formulation of liposomal derivatives of phenylalanine
02/05/2004WO2004010942A2 Substituted heterocyclic compounds as modulators of the ccr5 receptor
02/05/2004WO2003075857A3 Amino-methyl substituted tetracycline compounds
02/05/2004WO2003051348A3 Composition, synthesis and therapeutic applications of polyamines
02/05/2004US20040024215 Such as 4'-trifluoromethyl-biphenyl-2-carboxylic acid(4-(4-(alpha-methyl-benzyl)-piperazin-1-yl)-phenyl)-amide; apoprotein B-100 (apoB-100) and microsomal triglyceride transfer protein (MTP)
02/05/2004US20040024209 Drugs such as 4-(3-Bromo-4-fluorobenzyl)morpholine used as viricides against herpes viruses
02/05/2004US20040024205 Monomethylation of nitrogeneous heterocycles
02/05/2004US20040024067 Deacetylase inhibitors
02/05/2004US20040024059 Novel pleuromutilin derivatives
02/05/2004US20040024057 Nitrosated nonsteroidal antiinflammatory compounds, compositions and methods of use related applications
02/05/2004US20040023945 Cyclic amp-specific phosphodiesterase inhibitors
02/05/2004US20040023806 Agrochemicals in agriculture for controlling acarids and insects and for preventing the infestation of crop plants by phytopathogenic fungi.
02/05/2004US20040022856 Carriers for drug delivery
02/05/2004US20040022831 For therapy of mycosis of the nail
02/05/2004DE10238048A1 Verfahren zur Herstellung von Phenylalanin-Derivaten Process for the preparation of phenylalanine derivatives
02/05/2004DE10234058A1 Neue substituierte Benzoesäureamide, deren Herstellung und deren Verwendung als Arzneimittel New substituted benzamides, their preparation and their use as medicaments
02/05/2004DE10234057A1 Neue Carbonsäureamide, deren Herstellung und deren Verwendung als Arzneimittel New carboxamides, their preparation and their use as medicaments
02/05/2004DE10233632A1 Formulierungen von Phenylalanin-Derivaten Formulations of phenylalanine derivatives
02/05/2004CA2494668A1 Chemical compounds
02/04/2004EP1386916A1 Process for the monomethylation of nitrogen containing heterocycles
02/04/2004EP1385625A2 A nickel-rhenium catalyst for use in reductive amination processes
02/04/2004EP1385508A1 Dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
02/04/2004EP1115697B1 Unsaturated hydroximic acid derivatives as parp inhibitors
02/04/2004CN1473158A Radiopharmaceuticals for diagnosing alzheimer's disease
02/04/2004CN1137118C Water soluble azoles as broad-spectrun antifungals
02/03/2004US6686502 Compounds and methods for treatment of asthma, allergy and inflammatory disorders
02/03/2004US6686484 Anticoagulants; serine protease inhibitor
02/03/2004US6686467 Inhibitors of the production of cytokines such as tumour necrosis factor (hereinafter tnf), for example tnf alpha , and various members of the interleukin (hereinafter il) family, for example il-1, il-6 and il-8
02/03/2004US6686424 Preparation of functionalized alkoxyamine initiator and its use
02/03/2004US6686360 N-benzylpiperazine compounds
02/03/2004US6686353 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
02/03/2004US6686350 Cell adhesion inhibitors
02/03/2004CA2355987C Bicyclic amide derivatives and their use as muscle relaxants
02/01/2004CA2434481A1 Process for the methylation of nitrogenated heterocyclics
01/2004
01/29/2004WO2004009603A1 Dihydro-dibenzo[b,e]oxepine based selective estrogen receptor modulators, compositions and methods
01/29/2004WO2004009578A2 Pentacyclic oxepines and derivatives thereof, process for their preparation and pharmaceutical compositions containing them
01/29/2004WO2004009552A1 Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs
01/29/2004WO2004009531A1 Acetylenic compounds useful in treating inflammatory disorders
01/29/2004WO2004009086A1 Selective estrogen receptor modulators containing a phenylsulfonyl group
01/29/2004WO2004009034A2 Thiomolybdate analogues and uses thereof
01/29/2004WO2003066035A3 Compounds for inhibiting insulin secretion and methods related thereto
01/29/2004US20040019216 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
01/29/2004US20040019117 Anti tubercular drug: compostions and methods
01/29/2004US20040019103 Method of enhancing cellular production of molecular chaperon, hydroxylamine derivatives useful for enhancing the chaperon production and the preparation thereof
01/29/2004US20040019087 Thiomolybdate analogues and uses thereof
01/29/2004US20040019086 Aminediols for the treatment of Alzheimer's disease
01/29/2004US20040019043 Thiomolybdate analogues and uses thereof
01/29/2004US20040019039 Substituted piperazines and diazepanes
01/29/2004US20040019023 Administering 9,10-secopregna-5,7,10(19),16- tetraene derivative to a patient for treating skin diseases such as psoriasis
01/29/2004DE10232525A1 Neue Anthracen-Derivate und deren Verwendung als Arzneimittel Novel anthracene derivatives and their use as medicaments
01/29/2004CA2493127A1 Thiomolybdate analogues and uses thereof
01/29/2004CA2492907A1 Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs
01/28/2004EP1384719A1 Inhibitors of the glucosyl ceramide synthase enzyme useful for the treatment of cancers, sphingolipidosis and microbial infections
01/28/2004EP1383760A1 Biarylcarboxamide compounds as apolipoprotein b inhibitors
01/28/2004EP1383753A1 Piperazine-benzamide derivatives useful as apob-100 and/or mtp inhibitor
01/28/2004EP1383752A2 Deuterated 3-piperidinopropiophenone and medicaments containing said compounds
01/28/2004EP1383750A2 Urea derivatives as integrin alpha 4 antagonists
01/28/2004EP1383748A2 Novel compounds and compositions as cathepsin inhibitors
01/28/2004EP1383731A1 Biaryl compounds as serine protease inhibitors
01/28/2004EP1383730A2 Anticholinergic compounds and methods of use
01/28/2004EP1000016B1 Isocyanoalkyl carbonic acid derivatives, their conversion into secondary amidoalkyl carbonic acid derivatives by isocyanide-multicomponent reactions, as well as these secondary amidoalkyl carbonic acid derivatives.
01/28/2004CN1471516A Process for the preparation of 1,5-disubstituted-3-amino-1,2,4-triazoles and substituted aminoguamidines as intermediate compounds
01/28/2004CN1471509A 9-substituted minocycline compounds
01/28/2004CN1471506A Method for preparing carbonyl alpha-substituted nitrogen compounds
01/28/2004CN1136192C Aryl and hetaryl-sulfonamide derivatives, their preparation and use as endo thelin antagonists
01/28/2004CN1136187C 1-amino-alkylcyclohexane NMDA receptor antagonists
01/27/2004US6683215 N-(4-carbamimidoyl-phenyl)-glycine derivatives
01/27/2004US6683201 Analine derivatives as OSC inhibitors
01/27/2004US6683184 Piperazine derivatives and process for the preparation thereof
01/27/2004US6683099 Substituted N,N-disubstituted cycloalkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
01/27/2004US6683078 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors
01/27/2004US6683074 Cyclic amine derivatives-CCR-3 receptor antagonists
01/27/2004CA2214720C Arylsulfonylamino hydroxamic acid derivatives
01/22/2004WO2004007471A1 N-phenyl-(2r,5s)dimethylpiperadine derivative
01/22/2004WO2004007470A1 Novel anthracene derivatives and the use thereof as a medicament
01/22/2004WO2004007439A1 Biaryl derivatives
01/22/2004WO2004007437A1 Urea-substituted and urethane-substituted acylureas, methods for the production thereof and their use as medicaments
01/22/2004WO2004006878A1 Merocyanine derivatives for cosmetic use
01/22/2004WO2003072030A3 Methods for preventing or treating cardiac arrhythmia
01/22/2004WO2003049690A3 Hiv integrase inhibitors
01/22/2004US20040014971 N-(4-(4-(2-oxo-1-phenyl-2-((2,2,2-trifluoroethyl)amino)ethyl)-1 -piperazinyl)-phenyl)-4'-(trifluoromethyl)-(1,1'-biphenyl)-2-carboxamide for treatment of obesity, diabetes, and cardiovascular disorders; decreases apoplioprotein secretion
01/22/2004US20040014966 Such as 2-(phenylsulfonyl)-5-(1-piperazinyl)phenylamine which is a 5-HT receptor ligand; for performing positron emission tomography, nuclear magnetic resonance
01/22/2004US20040014796 Antiinflammatory agents; rheumatic diseases; antitumor agents
01/22/2004US20040014784 Substituted propargylamines
01/22/2004US20040014783 Antiinflammatory agents; autoimmune diseases; rheumatic diseases; anticholesterol agents; cardiovascular disorders
01/22/2004US20040014745 Amide compounds
01/22/2004CA2493373A1 Urea-substituted and urethane-substituted acylureas, methods for the production thereof and their use as medicaments
01/21/2004EP1382333A2 Use of beta 3 adrenergic receptor agonists in the treatment of dysuria
01/21/2004EP1381594A1 Urea compounds useful as anti-inflammatory agents
01/21/2004EP1381591A2 Certain salts of discodermolide acid, pharmaceutical compositions containing them and their use in treating tumors
01/21/2004EP1381590A1 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands
01/21/2004EP1381357A2 Glycyrrhetinic acid derivatives, progesterone and progesterone derivatives and their use for the manufacture of a medicament to inhibit 11beta-hydroxysteroid dehydrogenase activity