Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
03/2004
03/17/2004CN1482121A Process for preparing N-formyl morpholine
03/16/2004US6706923 Perfluoroalkyl-substituted amines, acids, amino acids and thioether acids
03/16/2004US6706765 Aminoguanidines and alkoxyguanidines as protease inhibitors
03/16/2004US6706745 Biphenylamidine derivatives
03/16/2004US6706742 Alpha-amino-acid compounds
03/16/2004US6706716 Compounds specific for the human α1d adrenergic receptor and uses thereof
03/16/2004US6706715 Reversible inhibitors of the blood clotting enzyme factor viia
03/16/2004US6706712 Cyclic derivatives as modulators of chemokine receptor activity
03/16/2004US6706710 Form of (R)-N-[5-methyl-8-(4-methylpiperazin-1-yl)-1,2,3,4-tetrahydro-2-naphthyl]-4-morpholinobenzamide
03/11/2004WO2004021500A1 Nonaqueous electrolyte and nonaqueous-electrolyte secondary battery
03/11/2004WO2004020422A1 1, 4- substituted piperidine derivatives and use thereof as base-inhibitors in treatment of alzheimer's disease
03/11/2004WO2004020401A1 Synthesis of sulfonamide derivatives
03/11/2004WO2004019946A1 Inhibitors for excessive accumulation of sodium ion in cells
03/11/2004WO2004019926A1 Preventive and/or therapeutic agent for heart failure
03/11/2004WO2004009578A3 Pentacyclic oxepines and derivatives thereof, process for their preparation and pharmaceutical compositions containing them
03/11/2004WO2004000789A9 Amide linker peroxisome proliferator activated receptor modulators
03/11/2004WO2003078420A3 Process for making chiral 1,4-disubstituted piperazines
03/11/2004WO2003006444A3 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
03/11/2004WO2003002524A3 Urea derivatives with antiproteolytic activity
03/11/2004US20040049083 Arylpiperazines having activity at the serotonin 1A receptor
03/11/2004US20040049038 N-substituted with a methylene-bridged nonaromatic ring system, e.g., N-(2-(benzyloxy)-5,6,7,8,9,10-hexahydro-6,9-methanobenzo(a)(8)annulen-11-yl)-N'-(2,2,2-trifluoroethyl)-sulfamide; preventing or treating Alzheimer's Disease
03/11/2004US20040049033 Acylated aminothiol compound
03/11/2004US20040048897 Il-8 receptor antagonists
03/11/2004US20040048891 Aniline derivatives or salts thereof and cytokine production inhibitors containing the same
03/11/2004US20040048875 Compounds and methods for treatment of asthma, allergy and inflammatory disorders
03/11/2004US20040048872 Sedatives, anticonvulsants, hypnotics and general anesthetics.
03/11/2004US20040048856 Monoamine reuptake inhibitors for treatment of CNS disorders
03/11/2004US20040048851 Amidinophenylalanine derivatives as thrombin inhibitors
03/11/2004DE10238865A1 New carboxamides are melanin-concentrating hormone receptor antagonists, useful for treating e.g. metabolic diseases, diabetes, eating disorders, cardiovascular disease, emotional disorders, reproductive and memory disorders
03/11/2004CA2497109A1 Nonaqueous electrolyte and nonaqueous electrolyte secondary battery
03/10/2004EP1395567A1 4 (phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain anxiety or gastrointestinal disorders
03/10/2004EP1395561A1 Carbamate and oxamide compounds as inhibitors of cytokine production
03/10/2004EP1395551A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases
03/10/2004EP1395548A1 Derivatives of diphenylurea, diphenyloxalic acid diamide and diphenylsulfuric acid diamide and their use as medicaments
03/10/2004EP1395265A2 Combretastatin a-3 prodrug
03/10/2004EP1395256A2 Prodrugs via acylation with cinnamate
03/10/2004EP1303249B1 Antimycotic nail varnish composition
03/10/2004CN1481376A Oxybenzamides derivatives as factor xa inhibitors
03/10/2004CN1481358A Carboxylic acid amide derivatives and their use in treatment of thromboembolic diseases and tumours
03/10/2004CN1481238A Aniline derivatives or salts thereof and cytokine prodn inhibitors contg. same
03/10/2004CN1480438A Stable ethene in hibitory compound and its prepn method
03/10/2004CN1141301C Prepn of acetyl morphine
03/09/2004US6703507 Nonaqueous liquid comprising the ammonium salt of a sulfonated or carboxylated phosphite ligand; use as a media for chemical reactions, including those using transition metal catalysts
03/09/2004US6703403 Method for improving pharmacokinetics
03/09/2004US6703368 Peptide-containing α-ketoamide cysteine and serine protease inhibitors
03/04/2004WO2004018461A2 Antibacterial benzoic acid derivatives
03/04/2004WO2004018442A1 Crystalline and amorphous forms of (s) -repaglinide and the processes for preparation thereof
03/04/2004WO2004018436A2 Compounds derived from aryl carbamates, preparation thereof and uses of same
03/04/2004WO2004018414A2 Antibacterial agents
03/04/2004WO2003075907A3 Small molecule entry inhibitors
03/04/2004WO2002098856A3 Piperazine oxyquinoline (naphthaline) platelet adenosine diphosphate receptor antagonists
03/04/2004WO2002038540A9 Activity-dependent cysteine protease profiling reagent
03/04/2004US20040044250 Transition-metal-catalyzed carbon-nitrogen bond-forming methods using carbene ligands
03/04/2004US20040044202 Functionalized monomers for synthesis of rubbery polymers
03/04/2004US20040044081 Hypotensive agents; cardiovascular disorders; anticholesterol agents; antiarrhythmia agents
03/04/2004US20040044061 Analgesics; side effect reduction
03/04/2004US20040044049 Compounds for inhibiting insulin secretion and methods related thereto
03/04/2004US20040044047 Alpha and beta-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
03/04/2004US20040044037 Sleep disorders; antidepressants; analgesics; central nervous system disorders
03/04/2004US20040044009 Drug abuse; cental nervous system disorders; cognition activators
03/04/2004US20040044008 Dietetics; antilipemic agents; non-insulin dependent diabetes; cardiovascular disorders
03/04/2004US20040044004 Calcium channel inhibitors comprising benzhydril spaced from piperazine
03/03/2004EP1392779A1 Fluorinated-photoinitiators in dual cure resins
03/03/2004EP1392667A1 Method for the production of biperidin
03/03/2004EP1392660A1 Substituted benzoylcyclohexenones and their use as herbicidal agents
03/03/2004EP1392644A1 Cinnamide derivatives as kcnq potassium channel modulators
03/03/2004EP1392639A1 Pyruvate derivatives
03/03/2004EP1392637A2 Modulators of peroxisome proliferator activated receptors
03/03/2004EP1392315A1 Methods of treating alzheimer's disease
03/03/2004EP1392280A2 Arylsulfonamide ethers, and methods of use thereof
03/03/2004EP1124797B1 N-arylsulfonyl amino acid omega amides
03/03/2004EP0938317B1 Compositions for reducing respiratory depression
03/03/2004CN1478472A 细胞粘连抑制剂 Cell adhesion inhibitor
03/03/2004CN1140459C Method of removing N-nitrosomorpholine and its application
03/02/2004US6700007 Method for preparing alkoxyamines from nitroxides
03/02/2004US6699990 Colorfastness; waterproofing; oxidative color hair dyes
03/02/2004US6699898 Method of treating coronary artery disease or other cetp-mediated disorders in a subject by administering a therapeutically effective amount of a compound of one of claims
03/02/2004US6699893 Glucocorticoid receptor modulators
03/02/2004US6699891 Npyy5 antagonists
03/02/2004US6699867 4-(4-Methyl-piperazin-1-ylmethyl)-4,5-dihydrothiazol-2-ylamine
03/02/2004US6699467 As carriers for delivering active agents such as peptides, drugs by administration, such as oral, subcutaneous, sublingual, and intranasal administration
02/2004
02/26/2004WO2004016576A1 Fused benzene derivative and use
02/26/2004WO2003097575A3 Amino-functional chalcones
02/26/2004WO2003097574A3 Aminoalkoxy-functional chalcones
02/26/2004WO2003057144A3 Change inhibitors of dipeptidyl peptidase iv
02/26/2004WO2002098869A3 1,4-disubstituted benzo-fused cycloalkyl urea compounds
02/26/2004WO2002096869A3 Piperazine mono(dithio)carbamate ester compounds and analogs thereof
02/26/2004WO2002083067A9 Prodrugs via acylation with cinnamate
02/26/2004WO2002057211A8 Symmetrically disubstituted aromatic compounds and pharmaceutical compositions for inhibiting poly (adp-ribose) glycohydrolase, and methods for their use
02/26/2004US20040039203 Reacting an aminoguanidine derivative with an aldehyde to form an intermediate, reacting intermediate with an aromatic acid derivative in presence of alkali metal alcoholate
02/26/2004US20040039061 Suppress expression and induction of inflammatory cytokines, cell adhesion molecule gene and virus and suppressors for nuclear factor kappa beta (nf-kb)
02/26/2004US20040039053 Administering to a patient a (3-halomethylphenoxy) (4-halophenyl) acetic acid derivatives or salt, free of its (+) stereoisomer to treat the type II diabetes, gout, insulin resistance and atherosclerosis
02/26/2004US20040039020 Novel pharmaceutical formulation suitable for nebulisation
02/26/2004US20040038989 (S)-3-(4-Phenyl-1-piperazinyl)-1,2-propanediol cyclic acetals, useful as intermediates for the preparation of levodropropizine
02/26/2004US20040038983 3-aza- and 1,4-diaza-bicyclo[4.3.0]nonanes, and methods of use thereof
02/26/2004US20040038941 Compounds for the treatment of inflammatory disorders
02/26/2004US20040038858 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours
02/26/2004US20040037022 Aminoalcohol derivatives
02/26/2004CA2495383A1 Fused benzene derivative and use
02/25/2004EP1391199A1 Carboxylic acid derivatives and drugs containing the same as the active ingredient