Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
04/2004
04/01/2004US20040063742 Such as 5-(4-Chlorophenyl)-8-methyl-6,7,8,9-tetrahydro-1-H-pyrrolo(3.2-h)isoquinoline-2,3-dione-3-oxime-(phenyl))urea; kits; drug screening
04/01/2004US20040063725 Binding neuropeptide Y receptors; hypertension, angina, atherosclerosis, depression, anxiety, inflammation, allergies
04/01/2004US20040063717 Employing fatty acid oxidation inhibitor; lowering HbA1c, glucose, total cholesterol and/or triglyceride plasma levels; increasing high density lipoprotein concentration; minimizing side effects; ranolazine
04/01/2004US20040063686 Diabetes, major depression, manic depression, anxiety, schizophrenia, sleep disorders
04/01/2004US20040063679 Amidino and guanidino peptidyl compounds; autoimmune diseases
04/01/2004US20040063671 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
04/01/2004US20040063643 Bombesin antagonists
04/01/2004US20040062706 Reacting selenium with lithium aluminum hydride
04/01/2004CA2499490A1 Amide and sulfonamide ligands for the estrogen receptor
04/01/2004CA2499213A1 Aromatic liver x-receptor modulators
04/01/2004CA2498662A1 Phenol derivatives and their use as rotamase inhibitors
04/01/2004CA2498149A1 3-(3,5-disubstituted-4-hydroxyphenyl)propionamide derivatives as cathepsin b inhibitors
04/01/2004CA2496696A1 Succinic acid semi-amides as anti-corrosive agents
03/2004
03/31/2004EP1403265A1 Industrial process for the synthesis of 5-[bis(carboxymethyl)amino]-3-carboxymethyl-4-cyano-2-thiophene-carboxylic acid tetraesters and use for the synthesis of ranetic acid divalent salts and hydrates thereof
03/31/2004EP1403249A1 Cyclic diamine compounds bearing six-membered cyclic groups
03/31/2004EP1403247A1 N-Alkanoylphenylalanine derivatives
03/31/2004EP1402899A1 Remedies for sepsis
03/31/2004EP1402888A1 The use of substituted carbocyclic compounds as rotamases inhibitors
03/31/2004EP1401918A2 Biodegradable poly(beta-amino esters) and uses thereof
03/31/2004EP1401824A2 Aromatic hydroxamic acid derivatives useful as hdac inhibitors
03/31/2004EP1401821A1 Novel phenylalkyl diamine and amide analogs
03/31/2004EP1015421B1 New phenylamidine derivatives, a process for preparing the same and their use as medicaments
03/31/2004CN1486313A Compounds for use in the treatment of skin conditions
03/31/2004CN1486297A Primary intermediates for oxidative coloration of hair
03/31/2004CN1143854C Novel 2-(iminomethyl) amino-phenyl derivatives,the preparation thereof, application as medicines and pharmaceutical compositions containing same
03/30/2004US6713651 β2-adrenergic receptor agonists
03/30/2004US6713464 Derivatives of 3,3-diphenylpropylamines
03/30/2004CA2278687C 5-aroylnaphthalene derivatives
03/25/2004WO2004024991A1 Organic salts and their use as reagents in electrochemical reactions
03/25/2004WO2004024878A2 Structurally rigid dopamine d3 receptor selective ligands and process for making them
03/25/2004WO2004024703A1 Process for the preparation of 4- (3’-chloro-4’-fluoroanilino) -7-methoxy-6- (3-morpholinopropoxy) quinazoline
03/25/2004WO2004024702A1 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof
03/25/2004WO2004024677A1 N-hydroxyformamidine derivative
03/25/2004WO2003104167A3 Cyanohydrin ethers and esters as high-sensitivity enzyme substrates
03/25/2004WO2003084941A3 Hydroxamic acid derivatives
03/25/2004WO2003082260A3 Tuberculosis treatment using pleuromutilin derivatives
03/25/2004WO2003004480A3 Substituted piperazine and diazepanes as histamine h3 receptor agonists
03/25/2004US20040059134 Introducing in a reactor a5-amino-3-(carboxyalkyl)-4-cyano-2-thiophenecarboxylic acid, potassium carbonate and a quaternaryammonium salt as catalyst acetone solvent and methyl bromo acetate, heating and cooling
03/25/2004US20040059109 Alanine 2, 6-dialkoxyphenyl ester derivatives as hypnotics
03/25/2004US20040059004 10-aryl-11h-benzo[b]fluorene derivatives and analogs for medicinal use
03/25/2004US20040058933 Aryl carbamate derivatives, preperation and use thereof
03/25/2004US20040058932 Novel piperazine derivatives
03/25/2004US20040058916 Central nervous system disorders; psychological disorders; schizophrenia; antiarthritic agents; Alzheimer's disease; anticancer agents
03/25/2004US20040058913 Cyclic diamine compound with condensed-ring groups
03/25/2004US20040058820 Central nervous system disorders; psychological disorders; antiinflammatory agents; multiple sclerosis
03/25/2004CA2498936A1 Structurally rigid dopamine d3 receptor selective ligands and process for making them
03/25/2004CA2496563A1 New carboxamide compounds having mch-antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture
03/24/2004EP1400510A1 Cyclic diamine compounds having fused-ring groups
03/24/2004EP1399431A2 Novel nitriles useful as reversible inhibitors of cysteine proteases
03/24/2004EP1399417A1 Method for producing perfluoroalkanesulfonic acid esters
03/24/2004EP1399414A2 Substituted tetracycline compounds for the treatment of malaria
03/24/2004EP1399159A1 4-substituted-1-(arylmethylidene)thiosemicarbazide, 4-substituted-1-(arylcarbonyl)thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof
03/24/2004EP1399146A1 Novel compounds and compositions as cathepsin inhibitors
03/24/2004EP1292599B1 Solutions of lithium pyrrolidine in tetrahydrofuran (thf)/hydrocarbons
03/24/2004EP1214296B1 Substituted n-phenyl 2-hydroxy-2-methyl-3,3,3-trifluoropropanamide derivatives which elevate pyruvate dehydrogenase activity
03/24/2004EP1161232B1 Hydroxy diphenyl urea sulfonamides as il-8 receptor antagonists
03/24/2004EP1082110B1 Use of compounds for the elevation of pyruvate dehydrogenase activity
03/24/2004CN1484633A N (phenylsulphonyl) glycine derivatives and their therapentic use
03/24/2004CN1142910C Amide compounds
03/23/2004US6710200 Using reporter molecule derivative having aldehyde or ketone group detectable by fluorescence emission, ultraviolet radiation, absorptivity or colorimetric analysis; rearrangements
03/23/2004US6710089 Substituted N-fused-phenyl-N-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
03/23/2004US6710057 Inhibitors of factor xa, as anticoagulants for prophylaxis and treatment of thromboembolic disorders
03/23/2004US6710043 Possess the potentiation of the cholinergic activity
03/23/2004CA2168432C Piperazine compounds used in therapy
03/18/2004WO2004022548A1 Process for producing oxycarbonyl-substituted piperazine derivative
03/18/2004WO2004022534A1 Arylglycine derivatives for use as glycine transport inhibitors
03/18/2004WO2004022529A2 Diarylurea derivatives and their use as chloride channel blockers
03/18/2004WO2004022528A2 Arylglycine derivatives and their use as glycine transport inhibitors
03/18/2004WO2004022526A1 Cathepsin cysteine protease inhibitors
03/18/2004WO2004022523A2 1, 3-diamino-2-hydroxypropane prodrug derivatives
03/18/2004WO2003102202A3 Process for preparing vinylaromatic compounds
03/18/2004WO2003099266A3 Acetamides and benzamides that are useful in treating sexual dysfunction
03/18/2004WO2003097576A3 Diamino-functional chalcones
03/18/2004WO2003018535A3 Novel aminobenzoephenones
03/18/2004US20040054178 Labels for chromatography, spectroscopes
03/18/2004US20040054172 Oxygenated esters of 4-lodo phenylamino benzhydroxamic acids
03/18/2004US20040054009 Useful for potentiating glutamate receptor function in a mammal and therefore useful for treating wide variety of conditions such as psychiatric and neurological disorders
03/18/2004US20040053983 1, 2, 4-tribsubstituted benzenes as inhibitors of 15-lipoxygenase
03/18/2004US20040053953 Treatment of chemokine mediated diseases
03/18/2004US20040053933 Ligands of melanocortin receptors and compositions and methods related thereto
03/18/2004US20040053925 Novel urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and novel use
03/18/2004US20040053916 Cyclohexyl(alkyl)-propanolamines, preparation method and pharmaceutical compositions containing same
03/18/2004US20040053907 Cell adhesion inhibitors
03/18/2004US20040053890 Naphthalene derivatives
03/18/2004US20040053826 Uses of polypeptides
03/18/2004US20040053786 Insecticidal 1,8-naphthalenedicarboxamides
03/18/2004US20040053330 Amino polyols and amino sugars
03/18/2004US20040052828 Provide a cooling sensation to a consumer, which cooling component includes cyclopenten-1-one-2-enamine derivative
03/18/2004CA2497979A1 1, 3-diamino-2-hydroxypropane prodrug derivatives
03/18/2004CA2495939A1 Cathepsin cysteine protease inhibitors
03/18/2004CA2495284A1 Diarylurea derivatives and their use as chloride channel blockers
03/17/2004EP1398030A2 Dipeptidyl peptidase IV effectors
03/17/2004EP1397382A2 Novel estrogen receptor ligand binding domain variants and novel ligands and pharmaceutical compositions
03/17/2004EP1397340A2 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
03/17/2004EP1252151B1 A process for the preparation of quetiapine and intermediates therefor
03/17/2004EP1144365B1 Inhibitors of alpha-4 beta-1 mediated cell adhesion
03/17/2004EP1140839B1 Heterocyclic amides as inhibitors of factor xa
03/17/2004EP1140810B1 Benzenic sulphonamide derivatives and their uses
03/17/2004EP1140802B1 Substituted aryl and heteroaryl derivatives, their production and their use as medicines
03/17/2004CN1483030A Amidoalkyl-piperidine and amidoalkyl-piperazine derivatives for the treatment of nervous system disorders