Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
01/2000
01/19/2000EP0971709A1 Novel compounds useful as neuro-protective agents
01/19/2000EP0672038B1 Herbicides
01/19/2000CN1242006A Guanidinyl heterocycle compounds useful as alpha-2 adrenoceptor agonists
01/19/2000CN1242001A Guanidinylamino heterocycle compounds useful as alpha-2 adrenoceptor agonists
01/18/2000US6015904 Stable reagents for the preparation of radio pharmaceuticals
01/13/2000WO2000001680A1 New 2-aminothiazol-fused 2-aminoindans and 2-aminotetralins and their use
01/13/2000WO2000001679A1 Retinoid-associated receptor regulators
01/13/2000WO1999018941A3 Ih-MODULATORS
01/13/2000DE19830430A1 New sulfur-substituted sulfonylamino-carboxylic acid N-arylamide derivatives useful as guanylate cyclase activators in treatment of e.g. cardiovascular disorders, asthma and diabetes
01/13/2000CA2332178A1 Retinoid-associated receptor function regulating agent
01/12/2000EP0970091A1 Process for the preparation of heteroaryl-zinc halides
01/12/2000EP0970090A1 Substituted 4-arylmethylene-2-imino-2,3-dihydrothiazoles and derivatives and their pharmaceutical use
01/12/2000EP0970077A1 Improved method for producing thiazolidinediones, and new thiazolidinediones
01/12/2000EP0970064A1 Process for the preparation of benzothiazolone compounds
01/12/2000EP0970063A1 Process for the preparation of substituted thiazolidinedione
01/12/2000EP0970062A2 Pyrrolidine and thiazole derivatives with metallo-beta-lactamase inhibitory properties
01/12/2000EP0970060A1 Lta 4 hydrolase inhibitors
01/12/2000EP0970046A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
01/12/2000CN1241182A Process for preparation of thiazole derivs.
01/12/2000CN1048240C Process for preparing 7-substed-9-substed. amino-6-demethyl-6-deoxytetracyclines
01/11/2000US6013837 Aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
01/11/2000US6013658 Animal growth regulators
01/11/2000US6013649 Bond disorders; autoimmune diseases; antitumor agents
01/06/2000WO2000000485A1 Epothilon derivatives, their preparation process, intermediate products and their pharmaceutical use
01/06/2000WO2000000482A1 1-(benzothiazol-2-yl)-4-(1-phenylmethyl)piperazines: dopamine receptor subtype specific ligands
01/06/2000WO2000000477A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000WO2000000473A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000WO2000000470A1 Amino acid derivatives and drugs containing the same as the active ingredient
01/06/2000WO2000000465A1 Hydrazine derivatives
01/06/2000WO2000000458A1 Substituted propionyl derivatives and intermediates thereof
01/06/2000CA2336625A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000CA2336162A1 Amino acid derivatives and pharmaceutical composition comprising, as active ingredients, them
01/06/2000CA2336150A1 1-(benzothiazol-2-yl)-4-(1-phenylmethyl)piperazines: dopamine receptor subtype specific ligands
01/06/2000CA2335921A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
01/06/2000CA2335245A1 Hydrazine derivatives
01/05/2000EP0968198A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR INHIBITING $g(b)-AMYLOID PEPTIDE
01/05/2000EP0968182A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
01/05/2000EP0968179A1 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
01/05/2000EP0776884B1 Substituted amide derivative
01/05/2000EP0664792B1 Fibrinogen receptor antagonists
01/05/2000CN1240439A Aminophenol derivates with fungicidal property
01/05/2000CN1240436A Method for producing 2-chloro-5-aminomethylthiazole
01/05/2000CN1240428A Diphenyl alkyl-tetrahydropyridines, process for their preparation, and pharmaceutical compositions containing them
01/05/2000CN1240419A Aromatic amine derivatives having NOS inhibitory effect
01/04/2000US6011175 Inhibition of farnesyltransferase
01/04/2000US6011045 Inhibitors of bone resorption; anticancer agents
01/04/2000US6011036 Heterocyclic compounds having antidiabetic hypolipidemic antihypertensive properties process for their preparation and pharmaceutical compositions containing them
12/1999
12/29/1999WO1999067230A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION
12/29/1999WO1999067209A1 Hydroximic acid derivatives, process for their preparation and intermediates therefor
12/29/1999WO1999067201A1 Hydroxamic acid derivatives as inhibitors of the production of human cd23 and of the tnf release
12/29/1999WO1999066944A1 Methods for identifying novel multimeric agents that modulate receptors
12/29/1999WO1999066925A1 Protease inhibitors
12/29/1999WO1999054326A8 Dihydropyrimidines
12/29/1999WO1999031079A3 Methods for the esterification of alcohols and compounds useful therefor as potential anticancer agents
12/29/1999EP0967211A1 Ferredoxin:NADP reductase inhibitors as herbicides
12/29/1999EP0966490A2 Catalyst compositions for the polymerization of olefins
12/29/1999EP0966465A1 Inhibitors of impdh enzyme
12/29/1999EP0966454A1 Disubstituted bicyclic heterocycles, their production and use as medicaments
12/29/1999EP0966443A1 Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of mip-1-alpha binding to its ccr1 receptor
12/29/1999EP0612314B1 2-pyrazinylethylamine derivatives and their use as pharmaceuticals
12/29/1999CN1239889A Novel compounds useful as neuro-protective agents
12/29/1999CA2342778A1 Inhibitors of .alpha.4.beta.1 mediated cell adhesion
12/29/1999CA2335876A1 Protease inhibitors
12/29/1999CA2335513A1 Hydroxamic acid derivatives as inhibitors of the production of human cd23 and of the tnf release
12/29/1999CA2319650A1 Methods for identifying novel multimeric agents that modulate receptors
12/28/1999US6008365 Adrenoreceptor agonists and dopamine da2-receptor agonists, useful in the treatment of obstructive airway diseases
12/28/1999US6008363 Process for producing guanidine derivatives, intermediates therefor and their production
12/28/1999US6008237 Potent agonists of peroxidsome proliferator activated receptor; for controlling or preventing of diabetes, hyperglycemia, hyperlipidemia, hypercholesterolemia, atherosclerosis, obesity, vascular restenosis
12/28/1999US6008204 Antidotes for preventing certain undesired side effects of retinoids
12/28/1999US6008176 As textile detergent builders in powder detergent formulations and as calcium sequestrants in oral hygiene products
12/28/1999US6007865 For inhibiting and reversing nonenzymatic cross-linking (protein aging), treating kidney damage and treating complications of diabetes, preventing food spoilage
12/28/1999US6007827 Method of depigmenting or bleaching mammalian skin using L-2-oxothiazolidine-4-carboxylic acid
12/23/1999WO1999065913A2 Epothilone minor constituents
12/23/1999WO1999065886A1 Benzazole compounds and their use
12/23/1999WO1999065885A1 Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof
12/23/1999WO1999065884A1 Carbon substituted aminothiazole inhibitors of cyclin dependent kinases
12/23/1999WO1999065872A1 Diarylselenide compounds and their use in human or veterinary medicine and in cosmetics
12/23/1999WO1999065871A2 Thiolesters and uses thereof
12/23/1999WO1999065870A2 Sulfonamide inhibitors of aspartyl protease
12/23/1999WO1999065484A1 New use
12/23/1999WO1999065315A1 Biocidal composition and its use
12/23/1999DE19826988A1 Epothilon-Nebenkomponenten Epothilone secondary components
12/23/1999CA2336189A1 Epothilone minor constituents
12/23/1999CA2335464A1 Novel thiolesters and uses thereof
12/23/1999CA2332325A1 Carbon substituted aminothiazole inhibitors of cyclin dependent kinases
12/23/1999CA2330977A1 Benzazole compounds and their use
12/22/1999EP0965585A1 Anti-amnesic thiazolidine derivatives
12/22/1999EP0964851A1 C-terminal ketone hydroxamic acid inhibitors of matrix metalloproteinases and tnfa secretion
12/22/1999EP0939628A4 Thiol sulfone metalloprotease inhibitors
12/22/1999EP0792261B1 O-benzyl oxime ether derivatives and their use as pesticides
12/22/1999EP0733033B1 Pharmaceutically active substituted aromatic compounds
12/22/1999EP0635018B1 4-(1H-2-METHYLIMIDAZO[4,5-c]PYRIDINYLMETHYL)PHENYLSULPHONAMIDE DERIVATIVES AS ANTAGONISTS OF PAF
12/22/1999CN1239474A Substituted pyridines and biphenyls as anti-hypercholesterinemic, anti-hyperlipoproteinemic and anti-hyperglycemic agents
12/21/1999US6005142 Process for preparing benzyl-substituted rhodanine derivatives
12/21/1999US6005141 Use of glycine-N,N-diacetic acid derivatives as biodegradable complexing agents for alkaline earth metal ions and heavy metal ions and process for the preparation thereof
12/21/1999US6005115 Forms A and B of N-[[[2-[[[2-[(diaminomethylene)amino]-4-thiazolyl]methyl ]thio]ethyl]ami no]methylene]-4-bromo-benzenesulfonamide
12/21/1999US6004994 Antiinflammatory agents, cyclooxygenase inhibitors and analgesics
12/21/1999US6004952 Micacocidin derivatives
12/21/1999US6004903 2-Anylocyclohexanediones having improved herbicidal properties
12/21/1999US6004543 L-2-oxothiazolidine-4-carboxylic acid derivatives and use thereof for skincare