Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
09/2000
09/12/2000US6118007 Preparation process of nitroguanidine derivatives
09/12/2000US6118001 Anticancer agent; antiarthritic agent
09/12/2000US6117987 Alkyl or aryl substituted dihydronaphthalene derivatives having retinoid and/or retinoid antagonist like biological activity
09/12/2000US6117893 Heterocyclic compounds having anti-diabetic activity and their use
09/12/2000US6117870 Cyclic amide derivatives
09/08/2000WO2000051998A1 Compounds useful as reversible inhibitors of cathepsin s
09/08/2000WO2000051997A1 Polycyclic thiazole systems and their utilization as anorectics
09/08/2000WO2000051996A1 Polycyclic thiazole-2-ylides amines, method for the production thereof and their utilization as medicaments
09/08/2000WO2000051995A1 Polycyclic 2-amino-thiazole systems, method for the production thereof and medicament containing said compounds
09/08/2000WO2000051994A1 Polycyclic 2-amino-dihydrothiazole systems, method for the production thereof and their utilization as medicament
09/08/2000WO2000051993A2 Dihetero-substituted metalloprotease inhibitors
09/08/2000WO2000051979A1 C16 unsaturated fp-selective prostaglandins analogs
09/08/2000WO2000051977A1 Aldehyde intermediates for the preparation of prostaglandin derivatives
09/08/2000WO2000051602A1 Utilization of polycyclic 2-amino-thiazole systems in the production of medicaments for prophylaxis or treatment of obesity
09/08/2000WO2000027341A3 Novel method of treatment
09/08/2000CA2366954A1 Dihetero-substituted metalloprotease inhibitors
09/08/2000CA2364903A1 Polycyclic thiazole systems and their utilization as anorectics
09/08/2000CA2364902A1 Polycyclic thiazole-2-ylides amines, method for the production thereof and their utilization as medicaments
09/08/2000CA2364900A1 Polycyclic 2-amino-thiazole systems, method for the production thereof and medicament containing said compounds
09/08/2000CA2364899A1 Polycyclic 2-amino-dihydrothiazole systems, method for the production thereof and their utilization as medicament
09/08/2000CA2362554A1 Utilization of polycyclic 2-amino-thiazole systems in the production of medicaments for prophylaxis or treatment of obesity
09/08/2000CA2360740A1 Compounds useful as reversible inhibitors of cathepsin s
09/06/2000EP1032556A1 Pharmaceutically active compounds and methods of use
09/06/2000EP1032395A1 Cyclopentane heptan(ene)oic acid, 2-heteroarylalkenyl derivatives as therapeutic agents
09/06/2000EP0824514B1 Dihalopropene compounds, insecticides containing them as active ingredients, and intermediates for their production
09/06/2000EP0649843B1 Thiazoline derivative
09/06/2000CN1265675A Benzyl compounds which inhibit leukocyte adhesion mediated by VLA-4
09/06/2000CN1265669A Compounds which inhibit leukocyte adhesion mediated by VLA-4
09/06/2000CN1265657A Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4
09/06/2000CN1265647A Acrylic metalloprotease inhibitor
09/06/2000CN1265645A Urokinase inhibitors
09/05/2000US6114578 Process for the preparation of benzothiazolone compounds
09/05/2000US6114533 2,4-pentadienoic acid derivatives having retinoid-like biological activity
09/05/2000US6114532 Anticoagulant
09/05/2000US6114526 Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
09/05/2000US6114365 Arylmethyl-carbonylamino-thiazole derivatives, process for their preparation, and their use as antitumor agents
08/2000
08/31/2000WO2000050413A1 Novel process of preparing a benzothiazolone compound
08/31/2000WO2000050392A1 2-mercaptocarboxylic acid derivatives
08/31/2000WO2000040558A8 Aspartic protease inhibitors
08/31/2000WO2000019994A9 Estrogen receptor ligands
08/31/2000WO2000012074A3 Use of piperidines and/or piperazines as inhibitors of p38-alpha kinase
08/31/2000DE19908539A1 Polycyclische 2-Amino-Dihydrothiazolsysteme, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Polycyclic 2-amino-Dihydrothiazolsysteme, processes for their preparation and their use as medicaments
08/31/2000DE19908538A1 Polycyclische 2-Amino-Thiazol Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen Polycyclic 2-amino-thiazole systems, methods for their preparation and medicaments containing these compounds
08/31/2000DE19908537A1 Verwendung von polycyclischen 2-Amino-Thiazol Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas Use of 2-amino-thiazole polycyclic systems for the production of medicaments for the prophylaxis or treatment of obesity
08/31/2000DE19908536A1 Polycyclische Thiazol-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Polycyclic thiazol-2-ylidene amines, process for their preparation and their use as medicaments
08/31/2000DE19908533A1 Polycyclische Thiazol-Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen Polycyclic thiazole systems, processes for their preparation and pharmaceutical compositions containing these compounds
08/31/2000DE19908447A1 Verfahren zur Herstellung von 2-Chlor-5-chlormethylthiazol A process for the preparation of 2-chloro-5-chloromethylthiazole
08/31/2000CA2360456A1 Novel process of preparing a benzothiazolone compound
08/30/2000EP1031566A1 Process for the preparation of 2-chloro-5-chloromethyl-thiazole
08/30/2000EP1031563A1 Sulfonyl derivatives
08/30/2000EP1030850A2 Azoline derivatives
08/30/2000CN1265096A Hydrazine derivatives
08/30/2000CN1055924C Novel aminoalkyl benzoxazolinones and benzothizolinones and pharmaceutical compsns. and method for preparing same
08/29/2000US6110949 A serine protease inhibitor treating non-insulin-dependent diabetes mellitus
08/29/2000US6110948 Treating of malignant tumor, tuberculosis, diabetes, blood dyscrasia, endocrine disease, infectious disease, or acquired immunodeficiency syndrome
08/29/2000US6110946 An enzyme inhibitors of retroviral aspartate protease for the treatment of aids
08/29/2000US6110938 1-(arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-4-(heteroaryl)piperidines and related compounds useful as antipsychotics and analgesics
08/29/2000US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor
08/29/2000US6110929 Immunomodulators which induce cytokine biosynthesis, including interferon and/or tumor biosynthesis, necrosis factor and inhibit t-helper-type 2 immune response; for treatment of viral and neoplastic diseases
08/29/2000CA2035832C Thiazolidine derivatives with anti-diabetic activity, their preparation and their use
08/23/2000EP1029861A1 Benzisothiazol-piperazinyl derivative and its use as neuroleptic
08/23/2000EP1029851A1 Piperazine compounds and medicinal use thereof
08/23/2000EP1028942A2 Dipeptide nitriles
08/23/2000EP1028716A1 Method for treating and preventing heart failure and ventricular dilatation
08/23/2000EP0836596B1 Hydrazine derivatives
08/23/2000EP0820447B1 Process for making 2-aryl benz(ox, thi, imid)azoles and 2-aminoaryl aminobenz(ox, thi, imid)azoles
08/23/2000EP0805795B1 Novel aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
08/23/2000CN1264385A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same
08/22/2000US6107622 Chevron correction and autofocus optics for laser scanner
08/22/2000US6107329 Hypotensive agents; cardiovascular disorders
08/22/2000US6107318 Psychological disorders
08/22/2000US6107317 N-(substituted glycyl)-thiazolidines, pharmaceutical compositions containing them and their use in inhibiting dipeptidyl peptidase-IV
08/22/2000CA2176973C Phenyl heterocycles as cyclooxygenase-2 inhibitors
08/17/2000WO2000047579A1 Substituted benzthiazolylalkylamino-1,3,5-triazines as herbicides
08/17/2000WO2000047552A1 Tyrosine alkoxyguanidines as integrin inhibitors
08/17/2000WO2000033837A3 Myt1 kinase inhibitors
08/17/2000WO2000012076A9 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
08/17/2000DE19905609A1 Substituierte Benzthiazolylalkylamino-1,3,5-triazine Benzthiazolylalkylamino substituted-1,3,5-triazines
08/17/2000CA2362372A1 Tyrosine alkoxyguanidines as integrin inhibitors
08/16/2000EP1028125A1 Dipeptide compounds having fungicidal activity and their agronomic use
08/16/2000EP1028111A1 Amide derivatives or salts thereof
08/16/2000EP1027713A1 Nonaqueous electrolyte for electrical storage devices
08/16/2000EP0805802B1 Substituted phenyl compounds as endothelin antagonists
08/16/2000EP0738259B1 Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them
08/15/2000US6103937 Producing unsaturated nitrogen containing compounds such as enamides, enamines and aryl amineslamides using as catalyst nickel and an organophosphine or carbene ligand
08/15/2000US6103921 Preparation of 3-chloro-1-thiocyanato-2-propene, by reacting 1,3-dichloropropene and a thiocyanate salt
08/15/2000US6103907 Phenylalkylcarboxylic acid compounds and compositions for treating hyperglycemia
08/15/2000US6103742 Administering to said patient a therapeutically effective amount of an insulin sensitivity enhancer in combination with a statin compound to treat diabetes
08/15/2000US6103725 High affinity to the dopamine d4 receptor; antagonists; antipsychotic agents, e.g. schizophrenia, with reduced side-effects; antipsychotic agents; anxiolytic and antiemetic agents; motoric functions, addiction, sleep, feeding
08/15/2000CA2136553C 7-(2-aminoethyl)-benzothiazolones
08/10/2000WO2000046184A1 N2-phenylamidine derivatives
08/10/2000WO2000045635A1 Thiazole derivatives and combinatorial libraries thereof
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/09/2000EP1026163A1 Process for producing substituted alkylamines or salts thereof
08/09/2000EP1026149A1 Amidocarboxylic acid derivatives
08/09/2000EP1025090A1 Vitronectin receptor antagonists
08/09/2000EP1025085A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
08/09/2000EP0823068B1 Color-providing compounds
08/09/2000CN1262620A Beta-Alkoxyacrylates against malaria
08/08/2000US6100406 Benzothiazolylthio or thiadiazolylthio substituted phenols as multifunctional additives for lubricants