Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
09/1999
09/22/1999CN1229080A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229079A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229078A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/21/1999CA2165137C Process for the manufacture of related intermediates including cistofur
09/21/1999CA2122712C A reduction method for substituted 5-methylene-thiazolidinediones
09/16/1999WO1999046253A1 Heterocyclyl anthracyclinone derivatives
09/16/1999WO1999046232A1 Carboxylic acid derivatives and drugs containing the same as the active ingredient
09/16/1999WO1999045914A1 Alkyl amine derivative and local anesthetic agent using the same
09/16/1999WO1999034785A3 Treatment of dyskinesias
09/16/1999CA2321832A1 Heterocyclyl anthracyclinone derivatives
09/15/1999EP0941990A2 Process for the preparation of azamethines and azamethines obtained thereby
09/15/1999EP0941215A1 Glyoxylic acid amides and their use as pesticides
09/15/1999EP0941086A1 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
09/15/1999EP0749421B1 Sulphonamide derivatives as aspartyl protease inhibitors
09/15/1999EP0741697B1 Amino acid derivatives and their use as phospholipase a2 inhibitors
09/15/1999CN1228771A 1,3-diheterocyclic metalloprotease inhibitors
09/15/1999CN1228420A Process for producing intermecliates used in process for producing-2-iminothiazoline derivatives
09/14/1999US5952386 Excellent insecticidal activity for the control of noxious insects
09/14/1999US5952375 Compounds and methods for synthesis and therapy
09/14/1999US5952362 2-imidazoline, 2-oxazoline, 2-thiazoline, and 4-imidazole derivatives of methylphenyl, methoxyphenyl, and aminophenyl alkylsulfonamides and ureas and their use
09/14/1999US5952360 Admisnistering to a mammal certain phenyl oxazoles or phenyl thiazoles
09/14/1999US5952359 Thiazoles and their agricultural compositions
09/14/1999US5952356 Treating diabetes in a mammal with an active material and a glucosidase inhibitor
09/14/1999US5952346 Inhibits the actions of the alzheimer's protein amyloid (beta/a4) in isolated endothelial cells; quinoline derivatives
09/14/1999US5952345 Synthesis and use of retinoid compounds having negative hormone and/or antagonist activities
09/14/1999US5952316 2-amino-1,3-propanediol compound and immunosuppressant
09/14/1999US5952311 Photosensitizing chemical means for killing tumor cells, wherein tumoricidal activity is activated by absorbing light or energy within a specific wavelength range, and energy donating chemical means for activating photosensitizer
09/14/1999US5952306 Integrin receptor antagonists
09/14/1999CA2144125C Use of sulfonic acids as antiageing agents in a cosmetic or dermatologic composition
09/14/1999CA1340749C Preparation and use of fluorescent benzothiazole derivatives
09/10/1999WO1999045004A1 Nitrate salt of anti-ulcer medicine
09/10/1999WO1999045000A1 Process for producing 4-thiazolylmethyl derivative
09/10/1999WO1999044993A1 Acryronitrile-based compound, method for producing the same and pest controlling agent comprising the same
09/10/1999WO1999029670A3 Aminocarbonyltetralin and dihydronaphtalene derivates as thrombin inhibitors
09/10/1999CA2322493A1 Nitrate salt of anti-ulcer medicine
09/08/1999EP0940139A2 Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
09/08/1999EP0939629A1 Thiol sulfonamide metalloprotease inhibitors
09/08/1999EP0939628A1 Thiol sulfone metalloprotease inhibitors
09/08/1999CN1227842A Penems and their derivatives
09/07/1999US5948804 Anaesthetic premedication
09/07/1999US5948803 Improve the insulin resistance and have potent hypoglycemic effect and lipid-lowering effect
09/07/1999US5948780 Administering a metalloproteinase inhibitor
09/07/1999US5948436 Protease inhibitor
09/07/1999CA1340721C 1,4-dihydro-quinoline-and naphthyridine-3-carboxylic acid antibacterial agents
09/02/1999WO1999043664A1 Heterocyclic diarylmethylene derivatives, methods of preparing them and their uses in therapeutics
09/02/1999WO1999043656A1 Propylamine derivatives and use thereof
09/02/1999WO1999043653A1 Synthesis of epothilones, intermediates thereto and analogues therof
09/02/1999WO1999043644A1 N-sulphonyl and n-sulphinyl phenylglycinamide___________________
09/02/1999WO1999043285A2 Sulphonamide derivatives
09/02/1999WO1999043212A2 Wood preservatives
09/02/1999WO1999024460A3 Dipeptide nitriles
09/02/1999CA2322139A1 Sulphonamide derivatives
09/02/1999CA2320838A1 N-sulphonyl and n-sulphinyl phenylglycinamide___________________
09/02/1999CA2320829A1 Heterocyclic diarylmethylene derivatives, methods of preparing them and their uses in therapeutics
09/01/1999EP0938676A1 Combinatorial process for preparing thiazolidinone libraries
09/01/1999EP0638564B1 Benzothiazolesulfonamide derivative, process for producing the same, and use thereof
09/01/1999CN1227540A Hydroxamic and carboxylic acid derivatives having MMP and TNF inhibitory activity
09/01/1999CN1227225A Thiazole derivatives
08/1999
08/31/1999US5945532 Method for manufacture of cephalosporin and intermediates thereof
08/31/1999US5945451 Fluorobutenyl(thio)ethers used as pesticides
08/26/1999WO1999042466A2 β-LACTAM-LIKE CHAPERONE INHIBITORS
08/26/1999WO1999042455A1 Antiviral agents
08/26/1999WO1999042437A1 Method for the production of 1,3-disubstituted 2-nitroguanidines
08/26/1999WO1999042436A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
08/26/1999WO1999029700A3 Cyclohexadiene-derivatives as pesticides
08/26/1999WO1999026909A3 Alpha-hydroxy, -amino and -fluoro derivatives of beta-sulphonyl hydroxamic acids as matrix metalloproteinases inhibitors
08/26/1999CA2355117A1 .beta.-lactam-like chaperone inhibitors
08/26/1999CA2320469A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
08/25/1999EP0937708A2 sulphonamide derivatives
08/25/1999EP0936895A1 Sunscreening compositions comprising natural products of a marine hydroid, and derivatives thereof
08/25/1999EP0749430B1 Thiazolidinedione derivatives as anti-hyperglycemic agents
08/25/1999CN1226889A Substituted sulphonyl amino (thio) carbonyl compounds and their use as herbicides
08/24/1999US5942632 Novel 4,5-bis(protected-amino), 2-(protected-carboxy)-1,3-dioxolane compounds that can be used to prepare hiv protease inhibitors by coupling to a solid support via an ester or an amide linkage
08/24/1999US5942530 Method for treating pain
08/24/1999US5942522 1-benzyl-3-ethoxycarbonyl-4-dimethylaminoethoxy-6-methyl-2-(1h) -quinolinone; antiviral against dna containing viruses, such as herpes group viruses
08/24/1999CA2176974C Phenyl heterocycles as cyclooxygenase-2 inhibitors
08/19/1999WO1999041224A1 Biaryl-acetic acid derivatives and their use as cox-2 inhibitors
08/19/1999WO1999021845A3 4-aminothiazole derivatives, their preparation and their use as inhibitors of cyclin-dependent kinases
08/19/1999DE19806717A1 New urethane, thiourethane and dithiourethane derivatives used to inhibit cholesterol biosynthesis and in treatment of e.g. hyperlipidemia, cell proliferation diseases, mycosis etc.
08/19/1999DE19806715A1 New urethane derivatives are used to inhibit cholesterol biosynthesis and to treat e.g. hyperlipidemia, cell proliferation diseases, mycosis etc.
08/19/1999DE19806713A1 New urethane derivatives are used to inhibit cholesterol biosynthesis and to treat e.g. hyperlipidemia, cell proliferation diseases, mycosis etc.
08/19/1999DE19806469A1 Preparation of 2-nitroguanidine derivatives useful as insecticides and acaricides
08/19/1999CA2318966A1 Biaryl-acetic acid derivatives and their use as cox-2 inhibitors
08/18/1999CN1226245A Compounds with pharmacologically active, preparation method and use thereof
08/18/1999CN1226244A Carbanilides used as pesticides
08/18/1999CN1226240A Intermediates for preparation of 2-imidazoline-5-ones
08/18/1999CN1044705C (1-phenyl-1-heterocyclyl) alkane derivatives and their preparation method and use
08/17/1999US5939563 Fungicides
08/17/1999US5939560 Inhibitors of DP-mediated processes, compositions and therapeutic methods thereof
08/12/1999WO1999040087A2 Inhibition of human telomerase by a g-quadruplex-interaction compound
08/12/1999WO1999040076A1 Thiazole compounds, production process, pest control agent, and antifungal agent
08/12/1999WO1999040072A1 Five-membered, benzo-condensed heterocycles used as antithrombotic agents
08/12/1999WO1999039710A1 Use of 2-amino-6- trifluoromehthoxy- benzothiazole for preventing or treating cerebellum dysfunction
08/12/1999CA2319494A1 5-membered heterocyclic condensed benzoderivatives, the preparation thereof and their use as pharmaceuticals
08/11/1999EP0934992A1 Light-emitting material for organo-electroluminescence device and organic electroluminescence device
08/11/1999EP0934938A1 Substituted benzoylaminothiazole derivatives and drugs containing the same
08/11/1999EP0934937A1 Azole derivatives as superoxide radical inhibitor
08/11/1999EP0934316A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
08/11/1999EP0934302A2 Aminophenol derivates
08/11/1999EP0934291A1 Protease inhibitors