Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
03/1999
03/30/1999US5889163 Method for producing azo dye compounds
03/30/1999US5889059 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
03/30/1999US5889037 Prevention, therapy tissue damage from lipid peroxidation
03/30/1999US5889035 1-(Arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-3-(heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics
03/30/1999US5889032 Heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
03/30/1999US5889025 Antidiabetic compounds having hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
03/30/1999US5889014 Heterocyclic compounds for inhibiting phosphodiesterase IV
03/30/1999US5889004 4-heteroaryl-1-piperazinealkylthiols and derivatives thereof and their therapeutic utility
03/30/1999US5888940 Desiccating plants
03/30/1999CA2144313C 4-hydroxy-2-cyclopentenone derivative and carcinostatic and osteogenesis promoter containing the same
03/24/1999EP0903348A1 Epothilone derivatives, preparation and utilization
03/24/1999EP0902782A1 Urea derivatives as inhibitors of impdh enzyme
03/24/1999EP0667855B1 Substituted arylalkynyl- and heteroarylalkynyl-n-hydroxyurea inhibitors of leukotriene biosynthesis
03/24/1999CN1211571A Process for producing chloroacetylaminothiazoleacetic acid derivatives
03/24/1999CN1042631C Substituted salicylic acids, its medicinal composition and use
03/24/1999CN1042630C Substituted AZA (cyclo) alkanes and its preparing process, use and pesticide composition containing same
03/23/1999US5886188 Method to convert 5-carboxanilido-haloalkylthiazoles to a single form
03/23/1999US5886044 IL-8 receptor antagonists
03/23/1999US5886043 Antiarthritic agents, antitumor agents, antiinflammatory agents
03/23/1999US5886036 Treating hiv infections
03/23/1999US5886024 Thiophene-containing butonic acid derivatives as matrix metalloprotease inhibitors
03/23/1999US5886014 Benzimidazole derivatives, their preparation and their therapeutic use
03/23/1999US5885990 Fibrinolysis promoting action; thrombolysis action
03/23/1999CA2247735A1 Novel 5-membered ring heterocycles, their preparation, their use and pharmaceutical preparations comprising them
03/23/1999CA2022611C Optical resolution method for 3s-(3-carboxybenzyl)-6-(5-fluoro-2-benzothiazolyl)methoxy-4s-chromanol
03/18/1999WO1999012906A1 Heterocyclic compounds as pesticides
03/18/1999WO1999012902A1 N-heterocyclic methylpropylamine derivatives, process for producing the same and germicides
03/18/1999WO1998058911A3 Prostaglandin agonists
03/18/1999WO1998057937A3 Inhibitors of factor xa with a neutral p1 specificity group
03/17/1999EP0902013A1 Novel amidine derivatives, their preparation and their use as medicaments with LTB-4 antagonistic effect
03/17/1999EP0902007A1 Chalcone derivatives and drugs containing the same
03/17/1999EP0901789A1 Method of treating tourette's syndrome
03/17/1999CN1211321A Methods for measurment and treatment predicated on presence of advanced glycosylation endproducts in tobacco and its combustion byproducts
03/17/1999CN1211242A Biologically active benzothiazolone ethananines
03/17/1999CN1042536C Preparation of cephalosporin antibiotic using synisomer of thiazolyl intermediate cis-isomer
03/17/1999CN1042532C Substituted phenyltrifluoethoxypropionic acid and its use
03/16/1999US5883248 Quaternary ammonium intermediates
03/16/1999US5883247 Acylation with aminothiazole derivative activated as mixed anhydride of thiophosphoric acid
03/16/1999US5883110 Organic molecules capable of inhibiting protein tyrosine phosphatase activity, and the use of such molecules to treat various disease states including diabetes mellitus, glioma, melanoma, kaposi's sarcoma, hemangioma, ovarian cancer, breast
03/11/1999WO1999011658A1 Meta-benzamidine derivatives as serin protease inhibitors
03/11/1999WO1999011657A1 1-amino-7-isoquinoline derivatives as serine protease inhibitors
03/11/1999WO1999011638A1 Substituted 1-aryl-3- heteroaryl-thioureas and substituted 1-aryl-3-heteroaryl-isothioureas as antiatherosclerotic agents
03/11/1999WO1999011637A1 Protease inhibitors
03/11/1999WO1999011636A1 Process for the preparation of 5-hydroxymethylthiazoles
03/11/1999WO1999011629A1 Novel carboxylic acid derivatives, their production and their use as mixed eta/etb endothelin-receptor antagonists
03/11/1999DE19738578A1 Carboxylic acid derivatives useful as endothelin A and B antagonists also active as renin and angiotensin inhibitors
03/11/1999CA2302361A1 Protease inhibitors
03/11/1999CA2302350A1 Novel carboxylic acid derivatives, their production and their use as mixed eta/etb endothelin-receptor antagonists
03/11/1999CA2294089A1 Process for the preparation of 5-hydroxymethylthiazoles
03/10/1999EP0900566A1 Novel tripeptide compounds and anti-aids drugs
03/10/1999EP0900210A1 Antivirally active heterocyclic azahexane derivatives
03/10/1999EP0900209A1 Thiazoline acid derivatives
03/10/1999EP0900198A1 New vitamin d derivatives with carbo- or heterocyclic substituents at c-25, a process for their production, intermediate products and their use for producing medicaments
03/10/1999EP0900197A1 Beta-thiopropionyl-aminoacid derivatives and their use as beta-lactamase inhibitors
03/10/1999EP0900080A1 Novel indole and benzothiazole derivatives
03/10/1999EP0677039B1 Cyclobutane derivatives as inhibitors of squalene synthetase and protein farnesyltransferase
03/10/1999CN1210523A Process for producing 5-hydroxyoxazolidinones
03/10/1999CN1210522A 2,4-diamino-1,3,5-iriazines, processes for their preparation and their use as herbicides and plant-growth regulators
03/10/1999CN1210520A Naphthol derivatives and process for preparation thereof
03/09/1999US5880288 Contacting solution of alkyl 4-halo-2-chloroacetoacetate in acetonitrile with thioacetamide, adding amine, heating to reflux
03/09/1999US5880287 Polyoxyhydrocarbyl related products and methods for fluorescence assays
03/09/1999US5880147 Amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prohylactic use
03/09/1999US5880135 Antagonist activity with respect to corticotropin releasing hormone
03/09/1999US5879657 Radiolabeled platelet GPIIb/IIIa receptor antagonists as imaging agents for the diagnosis of thromboembolic disorders
03/09/1999US5879412 Compositions and processes for dyeing keratin fibers with an oxidation base, a coupler, a cationic direct dye, and an oxidizing agent
03/04/1999WO1999010330A1 Heterocyclic ketones as npy y5 antagonists
03/04/1999WO1999010313A1 N-aroylphenylalanine derivatives
03/04/1999WO1999010312A1 N-alkanoylphenylalanine derivatives
03/04/1999WO1999009980A1 Method for treating pain
03/04/1999WO1999009979A1 Method for treating neuropathic pain
03/04/1999WO1999009829A1 Method for treating pain
03/04/1999WO1998053790A3 Compounds that inhibit the binding of vascular endothelial growth factor to its receptors
03/04/1999CA2302504A1 Method for treating pain
03/04/1999CA2302442A1 Method for treating neuropathic pain
03/04/1999CA2302294A1 Method for treating pain
03/04/1999CA2301821A1 Heterocyclic ketones as npy y5 antagonists
03/04/1999CA2300121A1 N-alkanoylphenylalanine derivatives
03/03/1999EP0724570B1 Amidino derivatives useful as nitric oxide synthase inhibitors
03/03/1999CN1209803A Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method therefor
03/03/1999CN1209802A Synthesis and use of retinene derivative having negative hormone and/or antagonist activities
03/02/1999US5877334 Of protease inhibitor
03/02/1999US5877207 Synthesis and use of retinoid compounds having negative hormone and/or antagonist activities
03/02/1999US5877196 N- 4-(imidazolyl or pyrazolyl)phenyl(oxy, sulfinyl, sulfenyl or sulfonyl)alkyl!carboxamides, sulfonamides or phosphoramides having antiarrhythmic properties
03/02/1999US5877193 Use of N-(4-aryl-thiazol-2-yl)-sulfonamides
03/02/1999US5876749 Pharmaceutical composition
02/1999
02/25/1999WO1999009018A1 BENZOTHIAZOLONE DERIVATIVES HAVING SELECTIVE β2 RECEPTOR AGONIST ACTIVITY
02/25/1999WO1999009017A1 Solid and liquid-phase synthesis of benzoxazoles and benzothiazoles and their use
02/25/1999WO1999009009A1 Method for producing organic compounds
02/25/1999WO1999009008A1 Method for producing substituted-2-nitroguanidine derivatives
02/25/1999WO1999009002A1 Phenol derivatives
02/25/1999WO1998052915A3 Leukotriene b4 derivatives, in particular oximo-ltb4 antagonists
02/25/1999DE19833750A1 New thiazolyl-alkadienol and -epoxide derivatives
02/25/1999CA2301227A1 Solid and liquid-phase synthesis of benzoxazoles and benzothiazoles and their use
02/25/1999CA2301172A1 Method for the producing substituted-2-nitroguanidine derivatives
02/25/1999CA2300808A1 Method for the producing substituted-2-nitroguanidine derivatives
02/24/1999EP0897912A1 Amidino derivatives useful as nitric oxide synthase inhibitors
02/24/1999EP0897652A1 Organometallic complexes for use in electroluminescent devices
02/24/1999CN1042224C Process for producing 2-iminothiazoline derivatives and process for producing their intermediates
02/23/1999US5874473 Substituted cycloalkanecarboxylic acid derivatives as matrix metalloprotease inhibitors
02/23/1999US5874472 Aminoacid derivatives as no synthase inhibitors