Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
07/1999
07/01/1999WO1999032111A1 INHIBITION OF p38 KINASE ACTIVITY USING SUBSTITUTED HETEROCYCLIC UREAS
07/01/1999WO1999032106A1 Inhibition of raf kinase using substituted heterocyclic ureas
07/01/1999CA2315720A1 Inhibition of p38 kinase activity using substituted heterocyclic ureas
07/01/1999CA2311428A1 Anilide derivative, production and use thereof
07/01/1999CA2309973A1 Thiazole-derivatives having microbicidal and plant immunizing activities
07/01/1999CA2300197A1 Thiourea and benzamide compounds, compositions and methods of treating or preventing inflammatory diseases and atherosclerosis
06/1999
06/30/1999EP0926140A1 Method for preparing 2-mercaptothiazole
06/30/1999EP0925300A1 Pharmaceutically active compounds and methods of use
06/30/1999CN1221410A Novel substituted 2,4-thiazolidine diketone derivatives, method for preparation thereof and pharmaceutical compositions containing the same
06/30/1999CN1043891C Fluorobenzothiazolyloxyacetamides and preparation method and use as weed killer
06/29/1999US5917016 Useful as photocleavable linking groups in solid phase synthesis
06/24/1999WO1999031096A1 Piperazine derivatives useful as hypoglycemic agents
06/24/1999WO1999031092A1 Benzamine derivatives
06/24/1999WO1999031079A2 Methods for the esterification of alcohols and compounds useful therefor as potential anticancer agents
06/24/1999WO1999031065A1 N-benzyl-3-indenylacetamides derivatives for treating neoplasia
06/24/1999WO1999031061A1 Integrin receptor antagonists
06/24/1999CA2313651A1 Benzamine derivatives
06/23/1999EP0923583A1 Method for producing epothilones, and intermediate products obtained during the production process
06/23/1999EP0923530A1 Inhibition of matrix metalloproteases by substituted biaryl oxobutyric acids
06/23/1999EP0923529A1 Subsitute 4-arylbutyric acid derivatives as matrix metalloprotease inhibitors
06/23/1999EP0923371A1 Pharmaceutical compositions comprising tyrphostins
06/22/1999US5914423 Difluorobutenes and difluorobutanes
06/22/1999US5914344 Substituted carboxanilide derivative and plant disease control agent comprising same as active ingredient
06/22/1999US5914332 Retroviral protease inhibiting compounds
06/22/1999CA1340604C Process for the preparation of 7-[2-(2-aminothiazol-4-y1)-2-hydroxyiminoacetamido]-3-cephem compounds
06/17/1999WO1999029700A2 Cyclohexadiene-derivatives as pesticides
06/17/1999WO1999029670A2 Aminocarbonyltetralin and dihydronaphtalene derivates as thrombin inhibitors
06/17/1999WO1999029660A1 Adamantane derivatives
06/17/1999WO1999029311A1 Hiv/fiv protease inhibitors having a small p3 residue
06/17/1999DE19755268A1 Benzamidinderivate Benzamidine derivatives
06/17/1999CA2312889A1 Adamantane derivatives
06/16/1999EP0922032A1 Herbicidal pyridinyl and pyrazolylphenyl ketones
06/16/1999EP0921798A1 Novel treatment of leptine resistance
06/16/1999CN1219929A Urea derivatives as inhibitors of IMPDH enzyme
06/16/1999CN1219927A Phenylalkylcarboxylic acid derivatives
06/16/1999CN1043609C Process for preparing pharmaceutical composition containing benzothiazole compounds
06/15/1999US5912360 Dioxolane intermediates
06/15/1999US5912352 Catalytic reduction of hydrazide to hydrazine derivative in presence of complex hydride; acyl migration; hydrogenation; catalyst selectivity
06/15/1999US5912259 Nonsteroid antiinflammatory agents for nervous system disorders
06/15/1999US5912243 Novel compounds for controlling nematodes, insect or acarid pests
06/10/1999WO1999028324A1 A process for the reduction of oxiranyl epothilones to olefinic epothilones
06/10/1999WO1999028306A1 Benzenesulfonamide compounds
06/10/1999WO1999027890A2 A process for the preparation of ring-opened epothilone intermediates which are useful for the preparation of epothilone analogs
06/10/1999DE19754490A1 Durch einen Aminocarbonylrest substituierte Bicyclen, ihre Herstellung und ihre Verwendung als Arzneimittel By an aminocarbonyl radical substituted bicyclic compounds, their preparation and their use as medicaments
06/10/1999CA2311929A1 A process for the reduction of oxiranyl epothilones to olefinic epothilones
06/10/1999CA2309969A1 Benzenesulfonamide compounds
06/09/1999EP0920414A1 Matrix metalloproteinase inhibitors
06/09/1999EP0920306A2 Chemokine receptor antagonists and methods of use therefor
06/09/1999EP0647636B1 Benzothiazole compound, process for producing the same, and use thereof
06/09/1999EP0615549B1 Process for the preparation of pharmaceutically active thiazolidine or oxazolidine compounds by a yeast reductase
06/08/1999US5910592 Substituted thiazolidinedione derivatives
06/08/1999CA1340588C Amino acid derivatives
06/03/1999WO1999026927A2 Metabotropic glutamate receptor antagonists for treating central nervous system diseases
06/03/1999WO1999026909A2 Alpha-hydroxy, -amino and -fluoro derivatives of beta-sulphonyl hydroxamic acids as matrix metalloproteinases inhibitors
06/03/1999WO1999026615A1 Cyclic amino acid derivatives as cell adhesion inhibitors
06/03/1999WO1999010312B1 N-alkanoylphenylalanine derivatives
06/03/1999WO1999005096A3 Urokinase inhibitors
06/03/1999WO1999002502A3 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
06/03/1999CA2311131A1 Metabotropic glutamate receptor antagonists for treating central nervous system diseases
06/03/1999CA2310401A1 Alpha-hydroxy, -amino and -halo derivatives of beta-sulfone hydroxamates as matrix metalloproteinase inhibitors
06/03/1999CA2309338A1 Cyclic amino acid derivatives as cell adhesion inhibitors
06/02/1999EP0919542A2 Phthalic acid diamide derivatives, agricultural and horticultural insecticides, and a method for application of the insecticides
06/02/1999EP0918760A1 Biologically active benzothiazolone ethanamines
06/02/1999EP0918759A1 Novel thiazolidone-2 derivatives, 4-diketone substituted, method for obtaining them and pharmaceutical compositions containing same
06/02/1999EP0918748A1 Fungicides
06/02/1999EP0918747A1 INHIBITORS OF THE PRODUCTION OF s-CD23 AND THE SECRETION OF TNF
06/02/1999EP0625138B1 Novel amidine derivatives, their preparation and their use as medicaments with ltb4 antagonistic effect
06/02/1999CN1218461A Alkylaminobenzothiazole and -benzoxazole derivatives
06/02/1999CN1218460A Substituted 4-hydroxy-phenylalcanoic acid derivatives with activity to ppar-'gamma'
06/02/1999CN1218045A Imide derivatives or salts thereof
06/01/1999US5908931 Preorganized hexadentate ligands useful in radiographic imaging agents
05/1999
05/27/1999WO1999025702A1 Herbicidal n-alkenyl heteroarylyloxyacetamides
05/27/1999WO1999025701A1 NOVEL HETEROCYCLICALLY SUBSTITUTED α-HYDROXYCARBOXLIC ACID DERIVATIVES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS
05/27/1999WO1999025358A1 Cyclopentane heptan(ene)oic acid, 2-heteroarylalkenyl derivatives as therapeutic agents
05/27/1999CA2310630A1 Cyclopentane heptan(ene)oic acid, 2-heteroarylalkenyl derivatives as therapeutic agents
05/27/1999CA2308746A1 Novel heterocyclically substituted .alpha.-hydroxycarboxylic acid derivatives, method for producing the same and their use as endothelin receptor_antagonists
05/26/1999EP0917462A1 Cell adhesion inhibitors
05/25/1999CA1340554C Derivatives of pyrido-benzothiazine with high anti-microbial activity
05/20/1999WO1999024460A2 Dipeptide nitriles
05/20/1999WO1999024416A1 Aminothiazole inhibitors of cyclin dependent kinases
05/20/1999WO1999024415A1 Retinoid receptor agonists
05/20/1999WO1999024411A1 Receptor with an affinity for compounds of the oxazoline class
05/20/1999WO1999024035A1 Benzothiazole protein tyrosine kinase inhibitors
05/20/1999DE19751200A1 New epothilone derivatives
05/20/1999DE19750529A1 New heterocyclic alpha-hydroxycarboxylic acid derivatives useful for treating hypertension, chronic coronary insufficiency, asthma, prostate cancer etc.
05/20/1999DE19748818A1 Optically active, smectic liquid crystal mixture, containing a temperature stable polyfluorinated cyclohexane derivative useful of the fabrication of switching and display devices
05/20/1999CA2309603A1 Receptor with an affinity for compounds of the oxazoline class
05/20/1999CA2309331A1 Agent acting on retinoid receptor
05/20/1999CA2309319A1 Benzothiazole protein tyrosine kinase inhibitors
05/19/1999EP0916651A1 Phenylalkylcarboxylic acid derivatives
05/19/1999EP0915868A1 Carbanilides used as pesticides
05/19/1999EP0915858A1 Intermediates for the preparation of 2-imidazoline-5-ones
05/19/1999EP0915847A1 Substituted sulfonamides as selective beta3 agonists for the treatment of diabetes and obesity
05/19/1999EP0915825A2 Substituted tetrahydronaphthalene and dihydronaphthalene derivatives having retinoid and/or retinoid antagonist-like biological activity
05/19/1999CN1216978A New vitamin-D derivatives with carbo- or heterocyclic substitutents at C-25, process for the prodn. intermediate products and their use for producing medicaments
05/19/1999CN1216767A Novel 5-membered ring heterocycles, their prepn. their use and pharmaceutical preparations comprising them
05/18/1999US5905158 Sunscreening compositions comprising natural products of a marine hydroid, and derivative thereof
05/18/1999US5905080 Central nervous system, psychological, eating disorders; cognition activators, parkinson*s disease
05/18/1999US5905077 Inhibitors of HIV protease useful for the treatment of AIDS
05/18/1999CA1340543C Pharmaceutically active compounds