Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
10/1999
10/21/1999WO1999052874A1 Difluoroalkene derivatives, process for producing the same, and agricultural or horticultural pest control agent
10/21/1999WO1999052493A2 Compounds that inhibit the binding of integrins to their receptors
10/21/1999WO1999026927A3 Metabotropic glutamate receptor antagonists for treating central nervous system diseases
10/21/1999DE19817459A1 New heterocyclic amide derivatives useful as cysteine protease inhibitors for treating neurodegenerative diseases, neuronal damage, stroke, cranial trauma, Alzheimer's disease, etc.
10/21/1999DE19817264A1 New dihydropyrimidine derivatives and their corresponding mesomers useful as antiviral agents
10/20/1999EP0950656A1 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
10/20/1999EP0950049A1 Diphenyl alkyl-tetrahydropyridines, process for their preparation, and pharmaceutical compositions containing them
10/20/1999EP0832078B1 N-hydroxyureas as antiinflammatory agents
10/20/1999EP0778821B1 Ortho-substituted aromatic ether compounds and their use in pharmaceutical compositions for pain relief
10/20/1999CN1232392A Pharmaceutical compositions comprising tyrphostins
10/20/1999CN1045766C N-aminoalkylcarbonyloxyalkylpyrrole insecticidal, acaricidal and molluscicidal agents
10/19/1999US5969145 Process for the production of epothilones and intermediate products within the process
10/19/1999US5968970 Treatment of hiv
10/19/1999US5968962 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
10/19/1999US5968942 Inhibitors of hiv protease
10/19/1999US5968908 Restricted 9-cis retinoids
10/14/1999WO1999051607A2 Process for purification of a cephalosporin derivative
10/14/1999WO1999051579A1 Fungicide compositions comprising a hydroximic or hydrazonic group
10/14/1999WO1999051572A1 Sulfonamide derivatives
10/14/1999WO1999051564A1 Propanolamine derivatives
10/14/1999CA2327290A1 Sulfonamide derivatives
10/14/1999CA2324940A1 Fungicide compositions comprising a hydroximic or hydrazonic group
10/13/1999EP0949242A1 Aromatic amine derivatives having nos inhibitory effect
10/13/1999EP0949238A1 Substituted propionyl derivatives
10/13/1999EP0948492A1 Process for the preparation of heteroaryl-phenylalanines
10/13/1999EP0948491A1 Aminothiazole derivatives useful in the preparation of beta-lactam antibiotics
10/13/1999EP0783486B1 Novel prostaglandin synthase inhibitors
10/13/1999CN1231665A Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/13/1999CN1231661A Aralkyl and aralkylidene heterocyclic lactams and imides
10/13/1999CN1045597C Alkylenediamine derivatives having heterocyclic group and medicinal composition thereof
10/12/1999US5965774 Substituted anilide derivative
10/12/1999US5965741 Ortho-substituted aromatic ether compounds and their use in pharmaceutical compositions for pain relief
10/12/1999US5965740 Alpha-substituted benzyl heterocyclic derivatives, intermediates for producing the same and pesticides containing the same as active ingredient
10/12/1999US5965736 Luciferins able to react with a phosphatase enzyme; detection of enzyme conjugates; use with charge-coupled devices, e.g. including charge-coupling device cameras and luminometers; durability; efficiency; immunoassays
10/12/1999US5965613 Fungicides for use in agriculture and horticulture; the compounds also have insecticidal and acaricidal activity
10/12/1999US5965601 Novel compounds for inhibiting replication of a retrovirus; treating hiv
10/12/1999US5965589 Thiazolidinedione derivatives, their production and use
10/12/1999US5965584 Pharmaceutical composition
10/12/1999US5965546 1-[(2-pyrimidinyloxy)alkyl]4-(heteroaryl)piperazines and related compounds and their therapeutic utility
10/12/1999US5965539 Peptidomimetics; anti-cancer drugs
10/12/1999US5965054 Comprising salts consisting of alkyl substituted, nitrogen-containing heterocyclic delocalized aromatic cations, and their perfluoro derivatives; high energy, high voltage
10/12/1999CA1340785C Platelet activating factor antagonists
10/07/1999WO1999050245A1 Indole derivatives with antiviral activity
10/07/1999WO1999050225A1 Aminocyclohexyl ether compounds and uses thereof
10/07/1999CA2326166A1 Indole derivatives with antiviral activity
10/06/1999EP0946539A1 Sulphonamide derivatives, process for their preparation, and their use as medicaments
10/06/1999EP0946532A1 Preparation of thiazoles
10/06/1999EP0946531A1 Process for the preparation of thiazole derivatives
10/06/1999EP0946530A1 Method for producing 2-chloro-5-aminomethylthiazole from 2-chloro-5-methylthiazole via 2-chloro-5-chloromethylthiazole
10/06/1999EP0946528A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS
10/06/1999EP0946518A1 Modulators of proteins with phosphotyrosine recognition units
10/06/1999EP0946501A1 Prevention of loss and restoration of bone mass by certain prostaglandin agonists
10/06/1999EP0946499A1 N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
10/06/1999EP0946203A1 Tricyclic functional dyes for contrast enhancement in optical imaging
10/06/1999EP0946097A1 Composition and use
10/06/1999EP0839133B1 4,9-ethano-benzo(f)isoindole derivatives as farnesyl transferase inhibitors
10/06/1999CN1230884A Thiol sulfone metalloprotease inhibitors
10/05/1999US5962640 Methods for preparing novel dipeptide compounds or pharmacuetically acceptable salts thereof
10/05/1999US5962529 Metalloproteinase inhibitors
10/05/1999US5962495 Estrogen sensitive diseases; breast cancer; prostate tumors
10/05/1999US5962489 Fungicides
10/05/1999US5962470 Heterocyclic compounds having anti-diabetic activity and their use
09/1999
09/30/1999WO1999048880A1 Benzothiazolone-7-sulfonamide derivatives
09/30/1999WO1999048879A1 Thiocarboxamide derivatives and their use as inhibitors of alpha-4 integrins
09/30/1999WO1999048862A1 Resins for antifouling agents against periphytons, process for the preparation of the resins, and antifouling agents against periphytons containing the same
09/30/1999WO1999006340A3 Sulfonylamino substituted hydroxamic acid derivatives as metalloprotease inhibitors
09/29/1999EP0945431A2 Process and intermediates for the preparation of phenylacetic derivatives
09/29/1999EP0944604A1 Guanidinyl heterocycle compounds useful as alpha-2 adrenoceptor agonists
09/29/1999EP0944601A1 Guanidinylamino heterocycle compounds useful as alpha-2 adrenoceptor agonists
09/29/1999EP0944580A2 N-(aryl/heteroaryl) amino acid esters, pharmaceutical compositions, and methods for inhibiting beta-amyloid peptide release and/or its synthesis
09/29/1999EP0944314A1 Methyl substituted fungicides and arthropodicides
09/29/1999EP0811005B1 Herbicidal benzoyl derivatives
09/29/1999CN1230183A Process for prepn. of nizatidine
09/29/1999CN1230114A Novel treatment of leptine resistance
09/29/1999CN1230110A Cell adhesion inhibitors
09/28/1999US5959118 Process for the preparation of 5-hydroxymethylthiazoles
09/28/1999US5958957 Modulators of molecules with phosphotyrosine recognition units
09/28/1999US5958954 2,2-dialkyl-4-aryl-substituted benzopyran and benzothiopyran derivatives
09/28/1999US5958931 Phenyl-substituted 5H-thiazolo 3,2-A!pyrimidine derivative glutamate receptor antagonists
09/28/1999US5958926 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
09/28/1999US5958923 Treatment of nervous system disorders
09/28/1999US5958910 Use of N-(4-aryl-thiazol-2-yl)-sulfonamides
09/28/1999US5958839 Herbicidal compounds
09/28/1999US5958683 Screening method using the RZR receptor family
09/23/1999WO1999047529A1 Heterocyclic signal transduction inhibitors, compositions containing them
09/23/1999WO1999047520A1 Process for the preparation of nitroguanidine derivatives
09/23/1999WO1999047508A1 Benzenesulfonamide-derivatives and their use as medicaments
09/23/1999WO1999047501A2 Nonnucleoside inhibitors of reverse transcriptase for the treatment of hiv-infection
09/23/1999WO1999047500A1 Method for producing lactams using oligophosphate catalysts
09/23/1999WO1999047497A2 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
09/23/1999DE19813821A1 New epothilone derivatives
09/23/1999DE19811880A1 Preparation of lactam by gas phase cyclizing hydrolysis of aminonitrile, useful e.g. as solvent and in polyamide production
09/23/1999CA2323783A1 Benzenesulfonamide-derivatives and their use as medicaments
09/23/1999CA2323616A1 Method for producing lactams using oligophosphate catalysts
09/23/1999CA2323418A1 Nonnucleoside inhibitors of reverse transcriptase for the treatment of hiv-infection
09/23/1999CA2322742A1 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
09/23/1999CA2321678A1 Process for the preparation of nitroguanidine derivatives
09/23/1999CA2319493A1 Heterocyclic signal transduction inhibitors, compositions containing them
09/22/1999EP0942756A2 Optical diagnostic agents for diagnosis of neurodegenerative diseases by means of near infra-red radiation (nir radiation)
09/22/1999CN1229082A Amine compound and its acid addition salt